![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-2_7de353ee3e6da7d439f1ec3aa8996b73.svg) | 3,5,7,8-Tetrahydro-2-[4-(trifluoromethyl)phenyl]-4H-thiopyrano[4,3-d]pyrimidin-4-one | IC50 | 106.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-2_bba0e8ca6afb314c59542be5b90d2370.svg) | Olaparib | IC50 | 3.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-2_5bde39defdeb9b3639f2a3e58f77f3b5.svg) | Veliparib | IC50 | 17.5 [1], 70.0 [2], 137.0 [3] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-2_5bde39defdeb9b3639f2a3e58f77f3b5.svg) | Veliparib | Ki | 5.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-2_f2b198c2d504e236c39c9f094ca41530.svg) | IWR-1-endo | IC50 | 18700.0 [1], 25000.0 [2], 35000.0 [3], 170000.0 [4] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-2_9d37a00818f71911ddc7ae7fb3af75a7.svg) | N~2~,N~2~-Dimethyl-N~1~-(6-oxo-5,6-dihydrophenanthridin-2-YL)glycinamide | IC50 | 33.5 [1], 382.0 [2] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-2_4ce1e392071f9a35d153ee0e21369703.svg) | Rucaparib | IC50 | 28.2 [1], 138.0 [2] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-2_67f6ced2b72cac0cc2b4d65f0d199019.svg) | Niraparib | IC50 | 2.1 [1], 15.3 [2] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-2_9702119f8d8353419fd0adaa755f86bb.svg) | Nvp-tnks656 | IC50 | 19000.0 [1], 32000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-2_028a11317906182ba0740511a9b10018.svg) | 4,4'-Oxydibenzamide | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-2_4026fc6979250bfc1845fabc7c54a0f6.svg) | 2-(Azetidin-3-yl)-1H-benzimidazole-4-carboxamide | Ki | 11.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-2_5990b92b8b207aaa055fb0a86512c4bc.svg) | 2-[4-(4-Fluorobenzoyl)piperidin-1-yl]-N-[(4-oxo-3,5,7,8-tetrahydropyrano[4,3-d]pyrimidin-2-yl)methyl]-N-(thiophen-2-ylmethyl)acetamide | IC50 | 19000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-2_59fb4f7f48babb39c7b1fc9f7648ba3f.svg) | 2-[4-(4-Fluorobenzoyl)piperidin-1-yl]-N-[(4-oxo-3,5,7,8-tetrahydropyrano[4,3-d]pyrimidin-2-yl)methyl]-N-propylacetamide | IC50 | 19000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-2_9640d72ce10399f21864841df59636d7.svg) | N-[(4-Oxo-3,5,7,8-tetrahydropyrano[4,3-d]pyrimidin-2-yl)methyl]-3-phenyl-N-(thiophen-2-ylmethyl)propanamide | IC50 | 19000.0 [1], 56400.0 [2] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-2_e51f5257e4b0add6e02102390d50f025.svg) | 3-(3-Hydroxyphenyl)-N-[(4-oxo-3,5,7,8-tetrahydropyrano[4,3-d]pyrimidin-2-yl)methyl]-N-(thiophen-2-ylmethyl)propanamide | IC50 | 19000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-2_4667a5d9a8b83caa371123bbce4c495e.svg) | N-[(4-Oxo-3,5,7,8-tetrahydropyrano[4,3-d]pyrimidin-2-yl)methyl]-3-phenyl-N-(thiophen-3-ylmethyl)propanamide | IC50 | 10400.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-2_d6e687c802ab565b500c07fcbfa3d912.svg) | 2-[4-(4-Fluorobenzoyl)piperidin-1-yl]-N-[(4-oxo-3,5,7,8-tetrahydropyrano[4,3-d]pyrimidin-2-yl)methyl]acetamide | IC50 | 3100.0 [1], 3150.0 [2] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-2_046f3de6eb4d2d97f4263a9f01986ecc.svg) | 2-[4-(4-Fluorobenzoyl)piperidin-1-yl]-N-[(4-oxo-3,5,7,8-tetrahydropyrano[4,3-d]pyrimidin-2-yl)methyl]-N-(pyridin-2-ylmethyl)acetamide | IC50 | 19000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-2_e4d6a30808f19ef02288b0b5233ffa46.svg) | 2-[4-(4-Fluorobenzoyl)piperidin-1-yl]-N-(2-methylpropyl)-N-[(4-oxo-3,5,7,8-tetrahydropyrano[4,3-d]pyrimidin-2-yl)methyl]acetamide | IC50 | 19000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-2_1dfd9162a8d3412bf049216cb53b22fb.svg) | N-Benzyl-2-[4-(4-fluorobenzoyl)piperidin-1-yl]-N-[(4-oxo-3,5,7,8-tetrahydropyrano[4,3-d]pyrimidin-2-yl)methyl]acetamide | IC50 | 19000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-2_e436b7d5bd8c4c655e3fc8afe19f99cc.svg) | Talazoparib | Ki | 0.85 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-2_979b4880256c881f24510e2d72655f5e.svg) | Bmn-673 8R,9S | IC50 | 4.1 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-2_35aec792bbfc6c95d4c64c30a66ec983.svg) | 4-Methoxybenzamide | IC50 | 77000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-2_dea69defff582730421352373662e055.svg) | 2-(4-Nitrophenyl)quinazolin-4-ol | IC50 | 2064.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-2_0736bd1a9c6d0fc2d5d01fcfa8a8fe5a.svg) | 2-(4-Chlorophenyl)quinazolin-4-ol | IC50 | 2600.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-2_b7c1de4a3b880cd0247e145bc7a0dcfe.svg) | 2-(4-Bromophenyl)-3,4-Dihydroquinazolin-4-One | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-2_aa0974474c3754d928b4d05f08aff109.svg) | 3-(4-Oxo-3,4-dihydroquinazolin-2-yl)propanoic acid | IC50 | 125.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-2_b96387d19fb60c745fd82c5b553f23f0.svg) | 2-(4-Fluorophenyl)quinazolin-4-ol | IC50 | 4688.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-2_0d917f12b4f21e18825c944259cad2ab.svg) | 2-(4-Methylphenyl)-4H-chromen-4-one | IC50 | 27800.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-2_ac816ce46bba81cb1254651c45ab97a7.svg) | 1H-Benzimidazole-7-carboxamide, 2-(1-propyl-4-piperidinyl)- | Ki | 5.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-2_f0ddb6875e45fa0e6cdffc2a25da2c26.svg) | 5-[[4-(4-Methoxyphenyl)-5-pyridin-4-yl-1,2,4-triazol-3-yl]sulfanylmethyl]-3-(4-methylphenyl)-1,2,4-oxadiazole | IC50 | 19000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-2_dd84fc74b732278dbf24a662d15b01bc.svg) | 2-[2-Fluoro-4-[(2S)-2-pyrrolidinyl]phenyl]-1H-benzimidazole-7-carboxamide | Ki | 1.5 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-2_da759c45c4a5813431ec3296123568ca.svg) | 4-[[3-[(6S)-3-(1,1-Difluoroethyl)-6-methyl-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine-7-carbonyl]phenyl]-difluoromethyl]-2H-phthalazin-1-one | IC50 | 30.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-2_895ffca54a4e36e44050383b60daf9be.svg) | 8-Chloro-2-{3-[4-(4-fluorophenyl)-1,2,3,6-tetrahydropyridin-1-yl]propyl}-3,4-dihydroquinazolin-4-one | IC50 | 500.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-2_c9872e8acd53bbab0db191c61a53399c.svg) | CID 16665853 | Ki | 3.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-2_7260fe64bd7e1b45b18038522ee7fe7a.svg) | 5-(2-Oxo-2-phenylethoxy)isoquinolin-1(2H)-one | IC50 | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-2_85e553e8c353d11a071114967cb3946f.svg) | 1H-Benzimidazole-7-carboxamide, 2-[4-(2-pyridinyl)phenyl]- | Ki | 2.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-2_58e01c0bb8eff75743ac57fac59fc826.svg) | 2-(4-Nitrophenyl)-4H-chromen-4-one | IC50 | 8300.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-2_41feab3c9fd34f20ec15f681338460cd.svg) | 4-Quinazolinol, 5,6,7,8-tetrahydro-2-(4-methyl-1-piperazinyl)- | IC50 | 3600.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-2_7362302d52d88fc7bdf6b3491a4eb693.svg) | 8-Methoxy-2-(4-nitro-phenyl)-3H-quinazolin-4-one | IC50 | 928.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-2_5750baca8423e7c362467cf03d973560.svg) | 8-Methoxy-2-phenyl-quinazolin-4-ol | IC50 | 1539.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-2_8d5a3e82a8dab0474b51e286a372e735.svg) | 8-Methyl-2-[4-(Trifluoromethyl)phenyl]-3h-Quinazolin-4-One | IC50 | 3098.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-2_90e980d4e7b3fc3c5f4944bc4e1ac8f4.svg) | 8-Methoxy-2-[4-(Trifluoromethyl)phenyl]-3,4-Dihydroquinazolin-4-One | IC50 | 570.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-2_472c3cf9d774b2094ec1f932ca6c063b.svg) | Morpholin-4-Yl[4-(Tetrazolo[1,5-A]quinoxalin-4-Ylamino)phenyl]methanone | IC50 | 5011.87 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-2_736cd1a1103a1e8463eac5db2b41e4a4.svg) | 3-(4-Cyanophenyl)quinoxaline-5-carboxamide | IC50 | 8.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-2_3740a0a21ff3ca353bc2d4cc0ce3c9e8.svg) | 4'-Isopropylflavone | IC50 | 34900.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-2_0c910e9df8f26d2b4069eb5d31297518.svg) | 2-(4-Pyridine-3-ylphenyl)-1H-benzimidazole-4-carboxamide | Ki | 8.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-2_9f55c70eef839ae3878767dd7b8cd018.svg) | 2-(4-Tert-Butylphenyl)-2,3-dihydroquinazoline-4(1H)-one | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-2_dd293d72769226a0e0dafb5851d2a4b7.svg) | 4-[(3Ar,4r,7s,7as)-1,3-Dioxooctahydro-2h-4,7-Methanoisoindol-2-Yl]-N-(Quinolin-8-Yl)benzamide | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-2_2320f07b06d1a98ce6485951a52cffb3.svg) | 3H-Pyridazino(3,4,5-de)quinazolin-3-one, 8-((1,3-dihydro-2H-isoindol-2-yl)methyl)-1,2-dihydro- | IC50 | 1.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-2_1429faacc2c24ca8da9bfe6f7406325a.svg) | N-(2-Methoxyphenyl)-4-{[3-(4-Oxo-3,4-Dihydroquinazolin-2-Yl)propanoyl]amino}benzamide | IC50 | 931.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-2_5644794b80cfe89001355cea696d6311.svg) | 2-[4-(Trifluoromethyl)phenyl]-3h-Quinazolin-4-One | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-2_a2fd086bc2f670526a1094b10470e6bf.svg) | 2-[4-[6-[(3R,5S)-3,5-Dimethylpiperazin-1-yl]-4-methylpyridin-3-yl]phenyl]-7-methyl-3H-pyrrolo[2,3-d]pyrimidin-4-one | IC50 | 990.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-2_147a1fcfb265b0bc85e54f7504e39337.svg) | 2-(4-Chlorophenyl)-8-methyl-3H-quinazolin-4-one | IC50 | 6350.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-2_a144654689895dbd7a7e997224632a58.svg) | 2-(4-Fluorophenyl)-8-methyl-3H-quinazolin-4-one | IC50 | 683.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-2_62abb697f03c7dd7e787dc8ff611fb32.svg) | Benzyl N-[[4-(8-methyl-4-oxo-3H-quinazolin-2-yl)phenyl]methyl]carbamate | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-2_bc93841ce4a01297d80930c4cbcdcaf9.svg) | 2-(4-Bromophenyl)-8-methyl-3H-quinazolin-4-one | IC50 | 10529.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-2_8bb392e7b15962b1319cb492d6db09e2.svg) | 2-(4-Chlorophenyl)-8-methoxy-3H-quinazolin-4-one | IC50 | 6022.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-2_42cb637297ccd2eab77731f4608ef765.svg) | 2-[4-(Trifluoromethyl)phenyl]-3,5,6,8-tetrahydrothiopyrano[3,4-d]pyrimidin-4-one | IC50 | 479.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-2_3d10ce0b6f310e22c87dc816048c24b4.svg) | 3-(4-Methoxyphenyl)-5-[[4-(4-methoxyphenyl)-5-methyl-1,2,4-triazol-3-yl]sulfanylmethyl]-1,2,4-oxadiazole | IC50 | 19000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-2_0dd6b42450002fd52f56aacfb4c7815b.svg) | 3-(3,4-Dimethoxyphenyl)-5-[[4-(4-methoxyphenyl)-5-methyl-1,2,4-triazol-3-yl]sulfanylmethyl]-1,2,4-oxadiazole | IC50 | 19000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-2_75b8c4d44ff8d7dae7a9265f975784da.svg) | 4-Tert-Butyl-N-(5,6-Dihydro[1,3]thiazolo[2,3-C][1,2,4]triazol-3-Yl)benzamide | IC50 | 19000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-2_aee167f244ed6999c4420a7616495cc6.svg) | 4-(4-Carbamoylphenoxy)benzoic acid | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-2_ede58385aeeb47ca11424e85b710e9e0.svg) | 2-(4-(Pyridin-4-yl)phenyl)-1H-benzimidazole-4-carboxamide | Ki | 1.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-2_410af0ab6e7320aee9a24ec4c166c008.svg) | 4-[(2-Fluorophenyl)methoxy]benzamide | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-2_c18e776e19bcb8483ae899b1f9dd2f26.svg) | 2-[4-[3-[(4-Oxo-3H-phthalazin-1-yl)methyl]benzoyl]piperazin-1-yl]pyridine-3-carbonitrile | IC50 | 1.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-2_cc06a47ef1cd90f88c44822007ee39ab.svg) | N-{4-[(2-Chlorophenyl)(Pyrimidin-4-Yl)carbamoyl]phenyl}-4-Methoxybenzamide | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-2_035cd7f13f54718b51887c460245840e.svg) | 2-[(2s)-2-Methylpyrrolidin-2-Yl]-1h-Benzimidazole-7-Carboxamide | Ki | 2.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-2_c96f4e4ded1c3075d17804cb7f6bdc91.svg) | 2-(3-Methylpyrrolidin-3-yl)-1H-1,3-benzodiazole-4-carboxamide | Ki | 2.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-2_cb243c4c9d219ed4e85461ee69100fe0.svg) | 6-Fluoro-2-[(2R)-2-methylpyrrolidin-2-yl]-1H-1,3-benzodiazole-4-carboxamide | Ki | 4.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-2_fbc186dc6ed96f500ea5b572e86e159c.svg) | 1-[3-[4-(2-Chlorophenyl)-5-pyrimidin-4-yl-1,2,4-triazol-3-yl]cyclobutyl]-2-oxo-3H-benzimidazole-5-carbonitrile | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-2_c48de2c6fb83618d6a143a3027a797c5.svg) | Tert-butyl (3S)-3-[[5-[(2,4-dioxoquinazolin-1-yl)methyl]-2-fluoropyridin-3-yl]carbamoyl]pyrrolidine-1-carboxylate | IC50 | 8.6 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-2_d470a6c99a1c192a34826a64c60927e8.svg) | Parp-2-IN-1 | IC50 | 11.5 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-2_95177cb843f49b362e1e633856924d84.svg) | (3S)-N-[5-[(2,4-Dioxoquinazolin-1-yl)methyl]-2-fluoropyridin-3-yl]-1-phenylpyrrolidine-3-carboxamide | IC50 | 4.1 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-2_0e5c6f966621e708166560794c9a8764.svg) | (E)-3-[4-[[4-[2-Fluoro-5-[(4-oxo-3H-phthalazin-1-yl)methyl]benzoyl]piperazin-1-yl]methyl]phenyl]-N-hydroxyprop-2-enamide | IC50 | 2.53 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-2_50a4076ef1fd113c952cbec98b2371b9.svg) | 4-[[4-[2-Fluoro-5-[(4-oxo-3H-phthalazin-1-yl)methyl]benzoyl]piperazin-1-yl]methyl]-N-hydroxybenzamide | IC50 | 31.52 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-2_c2238aca996cd99a4b05730df4710559.svg) | 6-Fluoro-2-(4,5,6,7-tetrahydrofuro[2,3-c]pyridin-2-yl)-1H-benzimidazole-4-carboxamide | IC50 | 144.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-2_95addead49ae4636717f1f000f3f7b37.svg) | 2-(4-Fluorophenyl)-8-methoxyquinazolin-4(3H)-one | IC50 | 1562.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-2_2d7962cdae8647afd55af5b543f9687f.svg) | Pamiparib | IC50 | 0.5 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-2_a10c50ab8009e8d3673b27e944edd523.svg) | 3-[(4-Oxo-3H-quinazolin-2-yl)sulfanyl]-N-[4-(5-phenyl-1,3,4-oxadiazol-2-yl)cyclohexyl]propanamide | IC50 | 2450.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-2_e06144509445fbdd2338f861f2b5f9d7.svg) | N-[trans-4-(4-Cyanophenoxy)cyclohexyl]-3-[(4-Oxo-3,4-Dihydroquinazolin-2-Yl)sulfanyl]propanamide | IC50 | 1760.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-2_0f682577c6d9fb9509805784a2a28980.svg) | Benzyl N-{[4-(4-Oxo-3,4-Dihydroquinazolin-2-Yl)phenyl]methyl}carbamate | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-2_a08cd9b05982a7d9e21c6b0eafcb79a6.svg) | 2-(4-((Pyridin-4-Yl)methyl)piperazin-1-Yl)-3,4,5,6,7,8-Hexahydroquinazolin-4-One | IC50 | 4200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-2_2e14cc7d0095f864892bafb0383bb66b.svg) | 4-[3-(4-Oxo-3H-quinazolin-2-yl)propanoylamino]-N-quinolin-8-ylbenzamide | IC50 | 6900.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-2_841732ebe8b3ab4c3c60886e582b565f.svg) | 4-[3-(8-Methyl-4-oxo-3H-quinazolin-2-yl)propanoylamino]-N-quinolin-8-ylbenzamide | IC50 | 11600.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-2_c1053641f14dc4fde8706c5a7eac6956.svg) | 2-(4-(Trifluoromethyl)phenyl)-7,8-dihydro-3H-thiopyrano[3,2-D]pyrimidin-4(6H)-one | IC50 | 4080.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-2_98b2062b6bf4308499c3cdd361da78ca.svg) | N-(Cyclopropylmethyl)-2-[4-(4-fluorobenzoyl)piperidin-1-yl]-N-[(4-oxo-3,5,7,8-tetrahydropyrano[4,3-d]pyrimidin-2-yl)methyl]acetamide | IC50 | 19000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-2_c09a72abbb6370cec52613215e3a54f0.svg) | N-Ethyl-2-[4-(4-fluorobenzoyl)piperidin-1-yl]-N-[(4-oxo-3,5,7,8-tetrahydropyrano[4,3-d]pyrimidin-2-yl)methyl]acetamide | IC50 | 19000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-2_92d484c2c7a4b8732ded9bf091cd7a90.svg) | 3-(8-Methyl-4-oxo-3H-quinazolin-2-yl)propanoic acid | IC50 | 145.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-2_05e64afc459a4c88f61c372beb46ac40.svg) | 2-(4-Bromophenyl)-8-methoxy-3H-quinazolin-4-one | IC50 | 259.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-2_e1e8daed121d37f1b2d0a78dc90b702f.svg) | 6-Fluoro-2-(4,5,6,7-tetrahydrothieno[3,2-c]pyridin-2-yl)-1H-benzimidazole-4-carboxamide | IC50 | 73.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-2_3ff19b3fab763c9b50a51244273159a0.svg) | 6-Fluoro-2-(4,5,6,7-tetrahydrothieno[2,3-c]pyridin-2-yl)-1H-benzimidazole-4-carboxamide | IC50 | 124.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-2_5fcb6392834df18bd89ad490c8df29fc.svg) | (3S)-1-(2-Cyclopropylethyl)-N-[5-[(2,4-dioxoquinazolin-1-yl)methyl]-2-fluoropyridin-3-yl]pyrrolidine-3-carboxamide | IC50 | 1.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-2_0c6afb87ab1d19c74a7888ee8a17a824.svg) | Tert-butyl (3S)-3-[[2-chloro-5-[(2,4-dioxoquinazolin-1-yl)methyl]pyridin-3-yl]carbamoyl]pyrrolidine-1-carboxylate | IC50 | 12.2 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-2_68efb4305bf0130f8de33b3c9971ef10.svg) | Tert-butyl (3S)-3-[[5-[(2,4-dioxoquinazolin-1-yl)methyl]pyridin-3-yl]carbamoyl]pyrrolidine-1-carboxylate | IC50 | 100.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-2_57e0db592b134e40c00dc2e10e96fbaf.svg) | (3S)-1-(Cyclopropylmethyl)-N-[5-[(2,4-dioxoquinazolin-1-yl)methyl]-2-fluoropyridin-3-yl]pyrrolidine-3-carboxamide | IC50 | 3.6 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-2_67c970df5e1784e20b52399af9473258.svg) | (3S)-N-[2-Chloro-5-[(2,4-dioxoquinazolin-1-yl)methyl]phenyl]pyrrolidine-3-carboxamide;2,2,2-trifluoroacetic acid | IC50 | 100.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-2_b3da336ed2cd3a4541ddadb7ecd75e57.svg) | 2-[4-(Trifluoromethyl)phenyl]-7,8-dihydro-3H-thiopyrano[4,3-d]pyrimidine-4,5-dione | IC50 | 141.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-2_8e56ecf98beb12180cb5d4f9f2363019.svg) | 2-[3-(Propylamino)pyrrolidine-1-carbonyl]-1H-benzimidazole-4-carboxamide | IC50 | 75.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-2_9a4f0247e7e9cd7bc0a052adec7c0dad.svg) | (3S)-1-(Cyclopropanecarbonyl)-N-[5-[(2,4-dioxoquinazolin-1-yl)methyl]-2-fluoropyridin-3-yl]pyrrolidine-3-carboxamide | IC50 | 4.5 [1] |