 | 4,4'-Oxydibenzamide | IC50 | 10000.0 [1], 23000.0 [2], 23400.0 [3] |
 | 3,5,7,8-Tetrahydro-2-[4-(trifluoromethyl)phenyl]-4H-thiopyrano[4,3-d]pyrimidin-4-one | IC50 | 5011.87 [1], 5888.44 [2] |
 | 3-[[(Z)-4-[4-(4-Chlorophenyl)piperazin-1-yl]-4-oxobut-2-enoyl]amino]benzamide | IC50 | 160.0 [1], 616.6 [2] |
 | 3-[[(Z)-4-[4-(4-Fluorophenyl)piperazin-1-yl]-4-oxobut-2-enoyl]amino]benzamide | IC50 | 700.0 [1], 707.95 [2] |
 | N~2~,N~2~-Dimethyl-N~1~-(6-oxo-5,6-dihydrophenanthridin-2-YL)glycinamide | IC50 | 4168.69 [1] |
 | Veliparib | IC50 | 89125.09 [1] |
 | Rucaparib | IC50 | 8912.51 [1] |
 | Niraparib | IC50 | 1737.8 [1] |
 | Bmn-673 8R,9S | IC50 | 25118.86 [1] |
 | 4-Methoxybenzamide | IC50 | 10000.0 [1] |
 | 5-(2-Oxo-2-phenylethoxy)isoquinolin-1(2H)-one | IC50 | 5754.4 [1] |
 | Morpholin-4-Yl[4-(Tetrazolo[1,5-A]quinoxalin-4-Ylamino)phenyl]methanone | IC50 | 5011.87 [1] |
 | 2-[4-[6-[(3R,5S)-3,5-Dimethylpiperazin-1-yl]-4-methylpyridin-3-yl]phenyl]-7-methyl-3H-pyrrolo[2,3-d]pyrimidin-4-one | IC50 | 2691.53 [1] |
 | (2z)-4-[(3-Carbamoylphenyl)amino]-4-Oxobut-2-Enoic Acid | IC50 | 20000.0 [1] |
 | 4-(4-Carbamoylphenoxy)benzoic acid | IC50 | 10000.0 [1] |
 | (2E)-4-[(3-Carbamoylphenyl)amino]-4-oxobut-2-enoic acid | IC50 | 20000.0 [1] |
 | 4-[(2-Fluorophenyl)methoxy]benzamide | IC50 | 10000.0 [1] |
 | N-{4-[(2-Chlorophenyl)(Pyrimidin-4-Yl)carbamoyl]phenyl}-4-Methoxybenzamide | IC50 | 10000.0 [1] |
 | (Z)-4-(3-Carbamoylanilino)-3-methyl-4-oxobut-2-enoic acid | IC50 | 20000.0 [1] |
 | (Z)-4-(3-Carbamoylanilino)-2-methyl-4-oxobut-2-enoic acid | IC50 | 20000.0 [1] |
 | 2-[(3-Carbamoylphenyl)carbamoyl]cyclopentene-1-carboxylic acid | IC50 | 20000.0 [1] |
 | 3-(3,4-Dimethyl-2,5-dioxopyrrol-1-yl)benzamide | IC50 | 20000.0 [1] |
 | (Z)-N'-(3-Carbamoylphenyl)-N-methylbut-2-enediamide | IC50 | 20000.0 [1] |
 | (E)-N'-(3-Carbamoylphenyl)-N-methylbut-2-enediamide | IC50 | 18620.87 [1] |
 | 3-[[(Z)-4-Oxo-4-pyrrolidin-1-ylbut-2-enoyl]amino]benzamide | IC50 | 20000.0 [1] |
 | (Z)-N-(3-Carbamoylphenyl)-N',N'-diethylbut-2-enediamide | IC50 | 20000.0 [1] |
 | Methyl (Z)-4-(3-carbamoylanilino)-4-oxobut-2-enoate | IC50 | 1659.59 [1] |
 | N-[2-(9H-Carbazol-1-yl)phenyl]methanesulfonamide | IC50 | 900.0 [1] |
 | 1-[3-[4-(2-Chlorophenyl)-5-pyrimidin-4-yl-1,2,4-triazol-3-yl]cyclobutyl]-2-oxo-3H-benzimidazole-5-carbonitrile | IC50 | 10000.0 [1] |
 | 4-[3-[4-(4-Fluorophenyl)piperidine-1-carbonyl]phenoxy]benzamide | IC50 | 5200.0 [1] |
 | N-[2-(9H-Carbazol-1-yl)phenyl]acetamide | IC50 | 720.0 [1] |
 | 4-[3-(4-Oxo-3H-quinazolin-2-yl)propanoylamino]-N-quinolin-8-ylbenzamide | IC50 | 100000.0 [1] |
 | 4-[3-(8-Methyl-4-oxo-3H-quinazolin-2-yl)propanoylamino]-N-quinolin-8-ylbenzamide | IC50 | 100000.0 [1] |
 | 3-[3-[4-(2-Fluorophenyl)piperazin-1-yl]-2,5-dioxopyrrolidin-1-yl]benzamide | IC50 | 20000.0 [1] |
 | 3-[[(Z)-4-Oxo-4-(4-pyrimidin-2-ylpiperazin-1-yl)but-2-enoyl]amino]benzamide | IC50 | 2818.38 [1] |
 | 3-[[(Z)-4-[4-(4-Fluorophenyl)piperidin-1-yl]-4-oxobut-2-enoyl]amino]benzamide | IC50 | 275.42 [1] |
 | 3-[[(Z)-4-Oxo-4-(4-phenylpiperazin-1-yl)but-2-enoyl]amino]benzamide | IC50 | 891.25 [1] |
 | 3-[[(Z)-4-[4-(4-Methoxyphenyl)piperazin-1-yl]-4-oxobut-2-enoyl]amino]benzamide | IC50 | 3388.44 [1] |
 | 3-[[(Z)-4-Oxo-4-(3-phenylpiperidin-1-yl)but-2-enoyl]amino]benzamide | IC50 | 690.0 [1] |
 | Ethyl 2-[1-[(Z)-4-(3-carbamoylanilino)-4-oxobut-2-enoyl]piperidin-4-yl]acetate | IC50 | 407.38 [1] |
 | 3-[[(Z)-4-Oxo-4-[4-(2-phenylethyl)piperidin-1-yl]but-2-enoyl]amino]benzamide | IC50 | 676.08 [1] |
 | 3-[[(Z)-4-[4-(2-Fluorophenyl)piperazin-1-yl]-4-oxobut-2-enoyl]amino]benzamide | IC50 | 407.38 [1] |
 | 3-[[(Z)-4-(2-Benzylpiperidin-1-yl)-4-oxobut-2-enoyl]amino]benzamide | IC50 | 3500.0 [1] |
 | 3-[[(Z)-4-Oxo-4-(3-phenoxypiperidin-1-yl)but-2-enoyl]amino]benzamide | IC50 | 1400.0 [1] |
 | 3-[[(Z)-4-(4-Benzylpiperidin-1-yl)-4-oxobut-2-enoyl]amino]benzamide | IC50 | 446.68 [1] |
 | Tert-butyl 4-[(Z)-4-(3-carbamoylanilino)-4-oxobut-2-enoyl]piperazine-1-carboxylate | IC50 | 371.54 [1] |
 | 3-[[(Z)-4-Oxo-4-(2-phenylpiperidin-1-yl)but-2-enoyl]amino]benzamide | IC50 | 1100.0 [1] |
 | 3-[[(Z)-4-Oxo-4-(4-phenylpiperidin-1-yl)but-2-enoyl]amino]benzamide | IC50 | 2238.72 [1] |
 | 3-[[(Z)-4-Oxo-4-[4-(4-phenylphenyl)piperazin-1-yl]but-2-enoyl]amino]benzamide | IC50 | 4168.69 [1] |
 | 4-[3-(3-Phenylpiperidine-1-carbonyl)phenoxy]benzamide | IC50 | 3600.0 [1] |
 | 4-[3-[4-(3-Fluorophenyl)piperidine-1-carbonyl]phenoxy]benzamide | IC50 | 1500.0 [1] |
 | 4-[3-[4-(3-Fluorophenyl)piperazine-1-carbonyl]phenoxy]benzamide | IC50 | 4786.3 [1] |
 | 4-[3-[4-(4-Chlorophenyl)piperazine-1-carbonyl]phenoxy]benzamide | IC50 | 4677.35 [1] |
 | 4-[3-(2-Phenylpiperidine-1-carbonyl)phenoxy]benzamide | IC50 | 4265.8 [1] |
 | 4-[3-(4-Phenylpiperazine-1-carbonyl)phenoxy]benzamide | IC50 | 1047.13 [1] |
 | 4-[3-[4-(4-Fluorophenyl)-4-hydroxypiperidine-1-carbonyl]phenoxy]benzamide | IC50 | 1288.25 [1] |
 | 4-[3-[4-(2-Fluorophenyl)piperazine-1-carbonyl]phenoxy]benzamide | IC50 | 1071.52 [1] |
 | 4-[3-[4-(3,4-Difluorophenyl)piperazine-1-carbonyl]phenoxy]benzamide | IC50 | 691.83 [1] |
 | 4-[3-[4-(4-Methoxyphenyl)piperazine-1-carbonyl]phenoxy]benzamide | IC50 | 5754.4 [1] |
 | 4-[3-(4-Phenylpiperidine-1-carbonyl)phenoxy]benzamide | IC50 | 2430.0 [1] |
 | 4-[3-[4-(4-Fluorophenyl)piperazine-1-carbonyl]phenoxy]benzamide | IC50 | 776.25 [1] |
 | 4-[3-(3-Phenylpyrrolidine-1-carbonyl)phenoxy]benzamide | IC50 | 3235.94 [1] |
 | 2-(9H-Carbazol-1-yl)-4-(trifluoromethyl)aniline | IC50 | 50000.0 [1] |
 | N-[2-(9H-Carbazol-1-yl)phenyl]-2-(2,5-dimethylphenyl)acetamide | IC50 | 44600.0 [1] |
 | N-[3-(9H-Carbazol-1-yl)pyridin-4-yl]acetamide | IC50 | 50000.0 [1] |
 | N-[2-(9H-Carbazol-1-yl)phenyl]benzamide | IC50 | 1900.0 [1] |
 | 2-(9H-Carbazol-1-yl)-3-methylaniline | IC50 | 50000.0 [1] |
 | N-[2-(9-Hydroxy-9H-fluoren-1-yl)phenyl]acetamide | IC50 | 50000.0 [1] |
 | N-[2-(9H-Carbazol-1-yl)phenyl]-2-(4-fluorophenyl)acetamide | IC50 | 50000.0 [1] |
 | N-[2-(9H-Carbazol-1-yl)phenyl]pentanamide | IC50 | 50000.0 [1] |
 | N-[2-(9H-Carbazol-1-yl)phenyl]-2-[3-(trifluoromethyl)phenyl]acetamide | IC50 | 7100.0 [1] |
 | N-[2-(9H-Carbazol-1-yl)pyridin-3-yl]acetamide | IC50 | 50000.0 [1] |
 | N-[2-(6,7,8,9-Tetrahydro-5H-carbazol-1-yl)phenyl]acetamide | IC50 | 1100.0 [1] |
 | N-[2-(9H-Carbazol-1-yl)phenyl]cyclohexanecarboxamide | IC50 | 50000.0 [1] |
 | N-[2-(9H-Carbazol-1-yl)phenyl]-2-(6-cyanopyridin-3-yl)acetamide | IC50 | 3500.0 [1] |
 | 2-(1,3-Benzodioxol-5-yl)-N-[2-(9H-carbazol-1-yl)phenyl]acetamide | IC50 | 6900.0 [1] |
 | N-[2-(9H-Carbazol-1-yl)phenyl]-2-(3,4-dichlorophenyl)acetamide | IC50 | 6300.0 [1] |
 | N-[2-(9H-Carbazol-1-yl)phenyl]-1-(3-cyanophenyl)methanesulfonamide | IC50 | 660.0 [1] |
 | N-[2-(2,3,4,5-Tetrahydro-1H-pyrido[4,3-b]indol-6-yl)phenyl]acetamide | IC50 | 50000.0 [1] |
 | 1-[2-(Dimethylsulfamoylamino)phenyl]-9H-carbazole | IC50 | 2500.0 [1] |
 | N-[2-(9H-Carbazol-1-yl)phenyl]-2-pyrazin-2-ylacetamide | IC50 | 2100.0 [1] |
 | N-[2-(9-Oxofluoren-1-yl)phenyl]acetamide | IC50 | 50000.0 [1] |
 | N-[2-(9H-Carbazol-1-yl)-3-methylphenyl]acetamide | IC50 | 1700.0 [1] |
 | N-[2-(9H-Carbazol-1-yl)-5-methylphenyl]methanesulfonamide | IC50 | 1100.0 [1] |
 | N-[2-(9H-Carbazol-1-yl)phenyl]-2-(3-fluorophenyl)acetamide | IC50 | 4200.0 [1] |
 | N-[2-(9H-Carbazol-1-yl)phenyl]propane-1-sulfonamide | IC50 | 2900.0 [1] |
 | N-[2-(9H-Carbazol-1-yl)phenyl]-1-(5-cyano-2-fluorophenyl)methanesulfonamide | IC50 | 1200.0 [1] |
 | N-[2-(9H-Carbazol-1-yl)phenyl]-2-(2-cyanopyridin-4-yl)acetamide | IC50 | 2400.0 [1] |
 | N-[2-(7,8-Dichloro-9H-carbazol-1-yl)phenyl]acetamide | IC50 | 1400.0 [1] |
 | N-[2-(9H-Carbazol-1-yl)phenyl]-2-pyridin-3-ylacetamide | IC50 | 1100.0 [1] |
 | N-[2-(9-Benzylcarbazol-1-yl)phenyl]acetamide | IC50 | 50000.0 [1] |
 | N-[2-(4-Oxo-1,6-diazatetracyclo[7.6.1.05,16.010,15]hexadeca-2,5,7,9(16),10,12,14-heptaen-3-yl)phenyl]acetamide | IC50 | 50000.0 [1] |
 | N-[2-(9H-Carbazol-1-yl)phenyl]-2-(dimethylamino)acetamide | IC50 | 5500.0 [1] |
 | N-[2-(6-Methoxy-9H-carbazol-1-yl)phenyl]acetamide | IC50 | 50000.0 [1] |
 | N-[2-(9H-Carbazol-1-yl)phenyl]-2-(4-chlorophenyl)acetamide | IC50 | 6200.0 [1] |
 | N-(2-Dibenzofuran-4-ylphenyl)acetamide | IC50 | 50000.0 [1] |
 | N-[2-(9H-Carbazol-1-yl)phenyl]propanamide | IC50 | 1000.0 [1] |
 | 2-(9H-Carbazol-1-yl)-5-methylaniline | IC50 | 50000.0 [1] |
 | N-[2-(9-Methylcarbazol-1-yl)phenyl]acetamide | IC50 | 50000.0 [1] |
 | N-[2-(9H-Carbazol-1-yl)phenyl]butane-1-sulfonamide | IC50 | 3300.0 [1] |