![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-1_bba0e8ca6afb314c59542be5b90d2370.svg) | Olaparib | IC50 | 6.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-1_5bde39defdeb9b3639f2a3e58f77f3b5.svg) | Veliparib | IC50 | 10.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-1_5bde39defdeb9b3639f2a3e58f77f3b5.svg) | Veliparib | Ki | 5.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-1_66f579be2776d27a7c1330d28453bb08.svg) | 3-Aminobenzamide | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-1_66f579be2776d27a7c1330d28453bb08.svg) | 3-Aminobenzamide | Ki | 3100.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-1_7de353ee3e6da7d439f1ec3aa8996b73.svg) | 3,5,7,8-Tetrahydro-2-[4-(trifluoromethyl)phenyl]-4H-thiopyrano[4,3-d]pyrimidin-4-one | IC50 | 1200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-1_9d37a00818f71911ddc7ae7fb3af75a7.svg) | N~2~,N~2~-Dimethyl-N~1~-(6-oxo-5,6-dihydrophenanthridin-2-YL)glycinamide | IC50 | 110.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-1_4ce1e392071f9a35d153ee0e21369703.svg) | Rucaparib | IC50 | 26.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-1_4ce1e392071f9a35d153ee0e21369703.svg) | Rucaparib | Ki | 1.4 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-1_67f6ced2b72cac0cc2b4d65f0d199019.svg) | Niraparib | IC50 | 16.7 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-1_60c3f20b0f42dbc4974f096cbfd3e3d0.svg) | 6(5H)-Phenanthridinone | IC50 | 350.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-1_12897fe178d0c23398901a95d6f53cba.svg) | Nicotinamide | IC50 | 210000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-1_7afbbb1be7620705fc093aef5825493f.svg) | 5-Aminoisoquinolin-1(2H)-one | IC50 | 300.0 [1], 1000.0 [2], 1600.0 [3], 1800.0 [4] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-1_72be741f94b9c3b04dde685cca0d2342.svg) | 9,19-Diazapentacyclo[10.7.0.02,6.07,11.013,18]nonadeca-1(12),2(6),7(11),13,15,17-hexaene-8,10-dione | IC50 | 36.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-1_5edd145e846f9a798df250757d78c01c.svg) | 1H-Benzimidazole-4-carboxamide | IC50 | 240.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-1_5edd145e846f9a798df250757d78c01c.svg) | 1H-Benzimidazole-4-carboxamide | Ki | 95.0 [1], 240.0 [2] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-1_c0f257298c463f6c4382a3cdcd9f78df.svg) | 2-Phenylbenzimidazole-4-carboxamide | Ki | 15.0 [1], 17.0 [2] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-1_895ffca54a4e36e44050383b60daf9be.svg) | 8-Chloro-2-{3-[4-(4-fluorophenyl)-1,2,3,6-tetrahydropyridin-1-yl]propyl}-3,4-dihydroquinazolin-4-one | IC50 | 13.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-1_6af3cea59a029aa517c87fa218d1e204.svg) | 4-{[3-(Piperazine-1-carbonyl)phenyl]methyl}phthalazin-1(2H)-one | IC50 | 2.0 [1], 16.0 [2], 30.5 [3] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-1_7bc0a4f737bf6501b6ea0a212bb8e0d9.svg) | Benzamide | IC50 | 5400.0 [1], 20000.0 [2], 22000.0 [3] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-1_e436b7d5bd8c4c655e3fc8afe19f99cc.svg) | Talazoparib | IC50 | 0.6 [1], 7.2 [2] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-1_e436b7d5bd8c4c655e3fc8afe19f99cc.svg) | Talazoparib | Ki | 1.2 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-1_704edee049941e8d558af355b26c109e.svg) | 4-[3-(1,4-Diazepan-1-ylcarbonyl)-4-fluorobenzyl]phthalazin-1(2H)-one | IC50 | 3.4 [1], 7.0 [2] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-1_59860067917e0bb7819e6fe2eadb593a.svg) | 4-Benzyl-1(2H)-phthalazinone | IC50 | 770.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-1_f2b198c2d504e236c39c9f094ca41530.svg) | IWR-1-endo | IC50 | 18700.0 [1], 85000.0 [2], 100000.0 [3] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-1_028a11317906182ba0740511a9b10018.svg) | 4,4'-Oxydibenzamide | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-1_df648076470b085e16ee16ea1a5664bd.svg) | 5-Chloro-2-(3-(4-phenyl-5,6-dihydropyridin-1(2H)-yl)propyl)quinazolin-4(3H)-one | IC50 | 65.0 [1], 682.0 [2] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-1_85e553e8c353d11a071114967cb3946f.svg) | 1H-Benzimidazole-7-carboxamide, 2-[4-(2-pyridinyl)phenyl]- | IC50 | 83.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-1_85e553e8c353d11a071114967cb3946f.svg) | 1H-Benzimidazole-7-carboxamide, 2-[4-(2-pyridinyl)phenyl]- | Ki | 1.9 [1], 2.0 [2] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-1_a5e7467a4570aa0bb36152e9c72f923a.svg) | 2-Methyl-1H-benzo[d]imidazole-4-carboxamide | IC50 | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-1_a5e7467a4570aa0bb36152e9c72f923a.svg) | 2-Methyl-1H-benzo[d]imidazole-4-carboxamide | Ki | 99.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-1_c33de74e4fe8d6450ab460f469e45bb2.svg) | 2-{3-[4-Phenyl-3,6-dihydro-1(2H)-pyridinyl]propyl}-4(3H)-quinazolinone | IC50 | 16.0 [1], 21.0 [2] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-1_84dca3ee6dbea8267b44f5b9436e0d0b.svg) | 2-(3-(4-(4-Fluorophenyl)-5,6-dihydropyridin-1(2H)-yl)propyl)quinazolin-4(3H)-one | IC50 | 8.9 [1], 16.0 [2], 304.0 [3] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-1_070f0674798fe256ba9d0661f2545b49.svg) | 2-(3-(4-Phenylpiperidin-1-yl)propyl)quinazolin-4(3H)-one | IC50 | 46.0 [1], 79.0 [2] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-1_7078a04fd185fba8163ceadd68c36bcb.svg) | 2-(3-(4-(4-Chlorophenyl)-5,6-dihydropyridin-1(2H)-yl)propyl)quinazolin-4(3H)-one | IC50 | 8.9 [1], 23.0 [2] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-1_ccc8e52354e88c0ce3ebc531b75d83dd.svg) | N-Ethyl-3-((4-oxo-3,4-dihydrophthalazin-1-yl)methyl)benzamide | IC50 | 50.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-1_2acd9dcee0535fa7c95f7c76cd5d7c13.svg) | N-{3-[(4-Oxo-3,4-dihydrophthalazin-1-yl)methyl]phenyl}propanamide | IC50 | 20.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-1_0c910e9df8f26d2b4069eb5d31297518.svg) | 2-(4-Pyridine-3-ylphenyl)-1H-benzimidazole-4-carboxamide | IC50 | 22.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-1_0c910e9df8f26d2b4069eb5d31297518.svg) | 2-(4-Pyridine-3-ylphenyl)-1H-benzimidazole-4-carboxamide | Ki | 0.95 [1], 1.0 [2] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-1_3637811477648833019c73caac7a9bce.svg) | 2-Phenyl-2H-indazole-7-carboxamide | IC50 | 24.0 [1], 25.0 [2] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-1_198dd39f5dc86f39e84ee4e05843c7cb.svg) | 2-(4-((Methylamino)methyl)phenyl)-2H-indazole-7-carboxamide | IC50 | 3.8 [1], 5.0 [2] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-1_01ddfa2f93ef4fbed7b620e6200068c1.svg) | INO-1001 free base | IC50 | 1.0 [1], 40.0 [2] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-1_577097e8dbf2f5fc0bd003a841988c48.svg) | 4-[[4-Fluoro-3-[4-(4-iodobenzoyl)piperazine-1-carbonyl]phenyl]methyl]-2H-phthalazin-1-one | IC50 | 3.3 [1], 7.0 [2], 7.4 [3] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-1_00c2124fb9869b276d7ecf21eda38440.svg) | 4-[[4-Fluoro-3-[5-methyl-3-(trifluoromethyl)-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine-7-carbonyl]phenyl]methyl]-2H-phthalazin-1-one | IC50 | 0.74 [1], 10.0 [2], 17.33 [3] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-1_f81376922910f392e0880cf71b9288fa.svg) | 4-Hydroxyquinazoline | IC50 | 9500.0 [1], 15800.0 [2] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-1_b9bdcc0e12b4d8e3b0c1852ee169f316.svg) | 4-Amino-1,8-naphthalimide | IC50 | 26.0 [1], 180.0 [2] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-1_979b4880256c881f24510e2d72655f5e.svg) | Bmn-673 8R,9S | IC50 | 1.1 [1], 144.0 [2] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-1_94370288943b612cc279769e7021ed78.svg) | 1-Hydroxyisoquinoline | IC50 | 9.0 [1], 7000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-1_c2f08ad48d1818dd1b0795d49552b5b8.svg) | 2-(4-(Piperidin-3-yl)phenyl)-2H-indazole-7-carboxamide | IC50 | 3.2 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-1_5ad90ee8773be00da7d6ab421243600d.svg) | 3,4-Dihydro-5-(4-(1-piperidinyl)butoxy)-1(2H)-isoquinolinone | IC50 | 53.2 [1], 10820.0 [2] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-1_3cfc1d6ec3f125845b9f5dbd0e5a71b2.svg) | 5-Methyl-3,4-dihydroisoquinolin-1(2H)-one | IC50 | 160.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-1_3cfc1d6ec3f125845b9f5dbd0e5a71b2.svg) | 5-Methyl-3,4-dihydroisoquinolin-1(2H)-one | Ki | 70.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-1_6f319471151e9109735392e9e66bb80c.svg) | 3-(4-Oxo-3,4-Dihydroquinazolin-2-Yl)-N-[(1s)-1-Phenylethyl]propanamide | IC50 | 3700.0 [1], 6300.0 [2] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-1_9702119f8d8353419fd0adaa755f86bb.svg) | Nvp-tnks656 | IC50 | 19000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-1_0d917f12b4f21e18825c944259cad2ab.svg) | 2-(4-Methylphenyl)-4H-chromen-4-one | IC50 | 7100.0 [1], 25000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-1_ac816ce46bba81cb1254651c45ab97a7.svg) | 1H-Benzimidazole-7-carboxamide, 2-(1-propyl-4-piperidinyl)- | Ki | 8.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-1_b393e15c95cdf6cdd512c250386cf789.svg) | 2-(4-Hydroxyphenyl)-1h-Benzimidazole-4-Carboxamide | Ki | 6.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-1_6be00cc7d58fb38bfe7acfa9e9cc2db4.svg) | 2-(4-Methoxyphenyl)-1H-benzimidazole-4-carboxamide | IC50 | 60.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-1_6be00cc7d58fb38bfe7acfa9e9cc2db4.svg) | 2-(4-Methoxyphenyl)-1H-benzimidazole-4-carboxamide | Ki | 6.8 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-1_87e974ca514eed4e7d0e90da0a332e10.svg) | 1-[2-Fluoro-5-[(4-oxo-3H-phthalazin-1-yl)methyl]phenyl]pyrrolidine-2,5-dione | IC50 | 5.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-1_40c44b437a6507265b20004ecc92eea1.svg) | (S)-8-Chloro-2-(3-(4-phenylpiperidin-1-yl)cyclopent-1-enyl)quinazolin-4(3H)-one | IC50 | 8.7 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-1_65634b7e9ea50ff848e287746bd9c2f0.svg) | 5-Chloro-2-methyl-3H-quinazolin-4-one | IC50 | 1200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-1_736cd1a1103a1e8463eac5db2b41e4a4.svg) | 3-(4-Cyanophenyl)quinoxaline-5-carboxamide | IC50 | 101.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-1_8a3051c79523bfd80f1d6b9a674b8b3d.svg) | 9,19-Diazapentacyclo[10.7.0.02,6.07,11.013,18]nonadeca-1(12),2(6),7(11),13,15,17-hexaen-10-one | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-1_a55ce8f2d41684da38ec3f1921b1dd60.svg) | 9,19-Diazapentacyclo[10.7.0.02,6.07,11.013,18]nonadeca-1(12),2(6),7(11),13,15,17-hexaen-8-one | IC50 | 56.0 [1], 90.0 [2] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-1_522a9cadef4cfe638ddab2b289b01817.svg) | 2-(4-((Methylamino)methyl)phenyl)-1H-benzo[d]imidazole-4-carboxamide | Ki | 3.2 [1], 4.0 [2] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-1_ed032b520dda741af97e9e708ab4238d.svg) | 2-(3-(4-Phenyl-5,6-dihydropyridin-1(2H)-yl)propyl)phenanthridin-6(5H)-one | IC50 | 46.0 [1], 119.0 [2] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-1_8e6cc101412cb7a7e203fb178a32f9fd.svg) | 2-Phenyl-3,10-diazatricyclo[6.4.1.04,13]trideca-1,4,6,8(13)-tetraen-9-one | Ki | 6.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-1_789e5aa0df0419c8075a3223503b0749.svg) | 4-(4-(4-Phenyl-5,6-dihydropyridin-1(2H)-yl)butyl)phthalazin-1(2H)-one | IC50 | 64.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-1_c82ad92823dc5296b0a23fdd3865289f.svg) | Benzo[c][1,7]naphthyridin-6(5H)-one | IC50 | 169.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-1_431f0349231e919b699f911b76631b92.svg) | Benzo[c][1,5]naphthyridin-6(5H)-one | IC50 | 116.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-1_b7c025d7297f57f7f9ef951d1f74a34d.svg) | 2-(4-Aminophenyl)-1H-benzo[d]imidazole-4-carboxamide | IC50 | 30.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-1_b7c025d7297f57f7f9ef951d1f74a34d.svg) | 2-(4-Aminophenyl)-1H-benzo[d]imidazole-4-carboxamide | Ki | 11.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-1_3409d1cc4d3d82503ec6adaccf9b3e22.svg) | 2-[4-[(Dimethylamino)methyl]phenyl]-3,10-diazatricyclo[6.4.1.04,13]trideca-1,4,6,8(13)-tetraen-9-one | IC50 | 5.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-1_3409d1cc4d3d82503ec6adaccf9b3e22.svg) | 2-[4-[(Dimethylamino)methyl]phenyl]-3,10-diazatricyclo[6.4.1.04,13]trideca-1,4,6,8(13)-tetraen-9-one | Ki | 5.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-1_14ff37b6f7c4ac62e1683a17ed14ad52.svg) | 3-[(E)-N-Hydroxy-C-methylcarbonimidoyl]-1,10-diazatricyclo[6.4.1.04,13]trideca-2,4(13),5,7-tetraen-9-one | Ki | 39.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-1_f53cf1fd8276a1c2e7b2838dc7ddf500.svg) | 3-[(E)-Methoxyiminomethyl]-1,10-diazatricyclo[6.4.1.04,13]trideca-2,4(13),5,7-tetraen-9-one | Ki | 809.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-1_606305f987fe2aaffe3a46465e1f4ff1.svg) | 2-(4-Fluorophenyl)-3-[(E)-hydroxyiminomethyl]-1,10-diazatricyclo[6.4.1.04,13]trideca-2,4(13),5,7-tetraen-9-one | Ki | 6.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-1_14ac60c757bff7d7f4f1ffa768310001.svg) | 3-[(E)-Hydroxyiminomethyl]-1,10-diazatricyclo[6.4.1.04,13]trideca-2,4(13),5,7-tetraen-9-one | Ki | 9.4 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-1_1095e0b22f8f09aff7af7d38827d3aeb.svg) | 3-(Hydroxymethyl)-1,10-diazatricyclo[6.4.1.04,13]trideca-2,4(13),5,7-tetraen-9-one | Ki | 79.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-1_5013323d5971f1d681d7f60b81617e0c.svg) | 3-[(Z)-Methoxyiminomethyl]-1,10-diazatricyclo[6.4.1.04,13]trideca-2,4(13),5,7-tetraen-9-one | Ki | 121.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-1_34e4e0c421fd47df8b0d5adb04ed1a89.svg) | 1-[2-Fluoro-5-(4-oxo-3,4-dihydrophthalazin-1-ylmethyl)phenyl]-3-phenylpyrrolidine-2,5-dione | IC50 | 6.8 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-1_53e5f8fdbf55a7d64c7dc6b2badf43a4.svg) | 1-(2-Fluoro-5-((4-oxo-3,4-dihydrophthalazin-1-yl)methyl)phenyl)piperidine-2,6-dione | IC50 | 4.1 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-1_b649dfd201eeb1da12d8744051d2656a.svg) | 4-(4-Fluoro-3-(piperazine-1-carbonyl)benzyl)phthalazin-1(2H)-one | IC50 | 5.0 [1], 6.9 [2] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-1_16961a3567b47bf893f2999d74df7db6.svg) | 2-(4-Chlorophenyl)-3-[(E)-hydroxyiminomethyl]-1,10-diazatricyclo[6.4.1.04,13]trideca-2,4(13),5,7-tetraen-9-one | Ki | 7.5 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-1_9b90495c8b245e69058c90ae4912ffc4.svg) | 2-{3-[4-(4-Fluorophenyl)-3,6-dihydro-1(2H)-pyridinyl]propyl}-8-methyl-4(3H)-quinazolinone | IC50 | 8.0 [1], 16.0 [2] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-1_99fa22299b26e7551a3971655afb8a06.svg) | 8-Chloro-2-[3-(4-phenyl-1,2,3,6-tetrahydropyridin-1-yl)propyl]-3,4-dihydroquinazolin-4-one | IC50 | 26.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-1_2320f07b06d1a98ce6485951a52cffb3.svg) | 3H-Pyridazino(3,4,5-de)quinazolin-3-one, 8-((1,3-dihydro-2H-isoindol-2-yl)methyl)-1,2-dihydro- | IC50 | 2.0 [1], 12.0 [2] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-1_96d119e49b6772f7bb8017ef6549cb22.svg) | 5H-Benzo[c][1,6]naphthyridin-6-one | IC50 | 128.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-1_7ece0f852839b2e56a8318780322c2ef.svg) | 2-Nitro-6(5H)-phenanthridinone | IC50 | 156.0 [1], 350.0 [2] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-1_7c6504384a999afc5c25de8cb4475178.svg) | 3-Aminobenzo[c][1,5]naphthyridin-6(5H)-one | IC50 | 180.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-1_96fbcb07fe3e4a7820fea16e5de6be1c.svg) | 2-[1-(Propan-2-yl)pyrrolidin-3-yl]-1H-1,3-benzodiazole-4-carboxamide | Ki | 9.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-1_933f304621a4aca89a21a397d46d3284.svg) | 2-(Pyrrolidin-3-yl)-1H-1,3-benzodiazole-4-carboxamide | Ki | 4.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-1_ab13811a814ecb49233409a6f3ffdd13.svg) | 1-[2-Fluoro-5-(4-oxo-3,4-dihydrophthalazin-1-ylmethyl)phenyl]-3-methylpyrrolidine-2,5-dione | IC50 | 3.8 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-1_088a0723e264dbd9e9dbfafcb7340d6a.svg) | 4-(3-(2-Oxopyrrolidin-1-yl)benzyl)phthalazin-1(2H)-one | IC50 | 120.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-1_bd1340b764a830d28be9377a528c2230.svg) | 3,4-Dihydropyrrolo(3,2,1-jk)(1,4)benzodiazepin-1(2H)-one | Ki | 105.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-1_6fa3713ffb56898ab55638443fa6a72a.svg) | (R)-2-(4-(Piperidin-3-yl)phenyl)-2H-indazole-7-carboxamide | IC50 | 2.4 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-1_4026fc6979250bfc1845fabc7c54a0f6.svg) | 2-(Azetidin-3-yl)-1H-benzimidazole-4-carboxamide | Ki | 6.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-1_cfdc2ba519ed929479f439321a4607bd.svg) | 2-[(2r)-Pyrrolidin-2-yl]-1h-benzimidazole-4-carboxamide | Ki | 7.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-1_26e539bb2c6c1e29592d1dacb0d92dd3.svg) | 2-[(2s)-Pyrrolidin-2-yl]-1h-benzimidazole-4-carboxamide | Ki | 30.0 [1] |