![](https://images.aatbio.com/dataset/ic50/platelet-derived-growth-factor-receptor_b2d54f313fd6fae3559ad99a1d264705.svg) | Imatinib | IC50 | 50.0 [1], 400.0 [2] |
![](https://images.aatbio.com/dataset/ic50/platelet-derived-growth-factor-receptor_814ad9e264ab2b2e27706d05bd4c2f07.svg) | 4-(6,7-Dimethoxy-quinoxalin-2-ylamino)-cyclohexanol | IC50 | 68.0 [1], 76.0 [2] |
![](https://images.aatbio.com/dataset/ic50/platelet-derived-growth-factor-receptor_0777dc765086e0fe44c81bec0cc1dba3.svg) | 4-Methyl-N-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | IC50 | 10.0 [1] |
![](https://images.aatbio.com/dataset/ic50/platelet-derived-growth-factor-receptor_ba62e48f8b5dfdb7ab85063c90b10bee.svg) | 3-(3-Thienyl)-6,7-dimethoxyquinoline | IC50 | 20.0 [1], 461.0 [2] |
![](https://images.aatbio.com/dataset/ic50/platelet-derived-growth-factor-receptor_1ab933be3af068e2d39845a83560bd49.svg) | N-[3-(4-Pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | IC50 | 5000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/platelet-derived-growth-factor-receptor_373d0e788d177eebf741620cf2b0bdf0.svg) | 4-(6,7-Dimethoxyquinoxaline-2-ylamino)cyclohexanecarboxylic acid methyl ester | IC50 | 28.0 [1], 49.0 [2], 345.0 [3] |
![](https://images.aatbio.com/dataset/ic50/platelet-derived-growth-factor-receptor_0e7b73ababb2246a51be20848a7a9b76.svg) | 6-(2,6-Dichlorophenyl)-2-{[3-(hydroxymethyl)phenyl]amino}-8-methylpyrido[2,3-D]pyrimidin-7(8H)-one | IC50 | 45.0 [1], 139.0 [2] |
![](https://images.aatbio.com/dataset/ic50/platelet-derived-growth-factor-receptor_8b41edc658ff384bedf4ec89c5c66dfb.svg) | N-[4-Methyl-3-[(4-pyridin-3-ylpyrimidin-2-yl)amino]phenyl]benzamide | IC50 | 100.0 [1] |
![](https://images.aatbio.com/dataset/ic50/platelet-derived-growth-factor-receptor_6db682cb0ba0382bb8605ed11f70bce3.svg) | Pyrido(2,3-d)pyrimidin-7(8H)-one, 6-(2,6-dichlorophenyl)-2-((4-fluorophenyl)amino)-8-methyl- | IC50 | 47.0 [1], 1250.0 [2] |
![](https://images.aatbio.com/dataset/ic50/platelet-derived-growth-factor-receptor_1c3f448dcdf6985f3b83c6259ce95880.svg) | N-(5-Amino-2-methylphenyl)-4-(3-pyridyl)-2-pyrimidineamine | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/platelet-derived-growth-factor-receptor_f1ad2b0ad65cacce5e9c9e9cbd966efd.svg) | 2-(3-Methylcyclohexylamino)-6,7-dimethoxyquinoxaline | IC50 | 41.0 [1] |
![](https://images.aatbio.com/dataset/ic50/platelet-derived-growth-factor-receptor_6b570d98b870cd72e04c3ed7a581167e.svg) | 2-Cyclohexylamino-6,7-dimethoxyquinoxaline | IC50 | 124.0 [1] |
![](https://images.aatbio.com/dataset/ic50/platelet-derived-growth-factor-receptor_84471a7719c085f985196d7ed8a14937.svg) | 5,7-Dimethoxy-3-(4-pyridinyl)quinoline | IC50 | 80.0 [1] |
![](https://images.aatbio.com/dataset/ic50/platelet-derived-growth-factor-receptor_84471a7719c085f985196d7ed8a14937.svg) | 5,7-Dimethoxy-3-(4-pyridinyl)quinoline | Ki | 14.0 [1] |
![](https://images.aatbio.com/dataset/ic50/platelet-derived-growth-factor-receptor_1ccd3b2521eb51116027a74a09cb2b7c.svg) | N-[4-Methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-acetamide | IC50 | 50000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/platelet-derived-growth-factor-receptor_69655e17af756ced10a634d48ae5f4ab.svg) | 2-(Phenylamino)-6,7-dimethoxyquinoxaline | IC50 | 6.0 [1] |
![](https://images.aatbio.com/dataset/ic50/platelet-derived-growth-factor-receptor_935fd4575ca3ba0db7bb0be07cad1d52.svg) | 2-Methoxy-N-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | IC50 | 300.0 [1] |
![](https://images.aatbio.com/dataset/ic50/platelet-derived-growth-factor-receptor_e940243148096a0894dd0157ec3910e0.svg) | N-[4-Methyl-3-[(4-pyridin-3-ylpyrimidin-2-yl)amino]phenyl]naphthalene-2-carboxamide | IC50 | 50.0 [1] |
![](https://images.aatbio.com/dataset/ic50/platelet-derived-growth-factor-receptor_84cc0e17a8d178e1438ce3abd0efd420.svg) | 4-Chloro-N-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | IC50 | 10.0 [1] |
![](https://images.aatbio.com/dataset/ic50/platelet-derived-growth-factor-receptor_1d5eba4b4bb57896dda18b1604bab021.svg) | Staurosporine | IC50 | 2.0 [1] |
![](https://images.aatbio.com/dataset/ic50/platelet-derived-growth-factor-receptor_7de5848be93196a6906eba944a298431.svg) | Sunitinib | IC50 | 80.0 [1] |
![](https://images.aatbio.com/dataset/ic50/platelet-derived-growth-factor-receptor_a7afc429fb2d8ce8facb9c0cc833f028.svg) | N-(3-Chlorophenyl)-6,7-dimethoxyquinazolin-4-amine | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/platelet-derived-growth-factor-receptor_ad465c21dbd002c135a4fe93dc9f7695.svg) | N-(3-Bromophenyl)-6,7-dimethoxyquinazolin-4-amine | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/platelet-derived-growth-factor-receptor_291fdc26c251ab1eb139e1406ed05831.svg) | Canertinib | IC50 | 50000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/platelet-derived-growth-factor-receptor_ddc31cb72a8aa21440e26147cfc64b1b.svg) | Lfm-a13 | IC50 | 500000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/platelet-derived-growth-factor-receptor_e98e38f8f3edf8be20fec1223eba919f.svg) | 6,7-Dimethyl-2-phenylquinoxaline | IC50 | 0.0 [1] |
![](https://images.aatbio.com/dataset/ic50/platelet-derived-growth-factor-receptor_94feb385cecaa610e1d68d9fb9d55ef3.svg) | Pyridone 6 | IC50 | 1490.0 [1] |
![](https://images.aatbio.com/dataset/ic50/platelet-derived-growth-factor-receptor_33bc0283962e2a0c3729440054f4f20b.svg) | 6-(2,6-Dichlorophenyl)-8-methyl-2-((3-(methylthio)phenyl)amino)pyrido[2,3-d]pyrimidin-7(8H)-one | IC50 | 1660.0 [1] |
![](https://images.aatbio.com/dataset/ic50/platelet-derived-growth-factor-receptor_5f0648764433a139fcbde34dddb456ff.svg) | 6-(2,6-Dichlorophenyl)-2-[(4-Fluoro-3-Methylphenyl)amino]-8-Methylpyrido[2,3-D]pyrimidin-7(8h)-One | IC50 | 1430.0 [1] |
![](https://images.aatbio.com/dataset/ic50/platelet-derived-growth-factor-receptor_eecff12231f5f450d936f7633fcd7db0.svg) | Unii-NA856793UT | IC50 | 50000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/platelet-derived-growth-factor-receptor_3d9c4e87ec0a775c8d3f9ae4ae00a310.svg) | 7-[cis-4-(4-Methylpiperazin-1-Yl)cyclohexyl]-5-(4-Phenoxyphenyl)-7h-Pyrrolo[2,3-D]pyrimidin-4-Amine | IC50 | 20000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/platelet-derived-growth-factor-receptor_ab2268bff60761ec9560ebfb5b03f869.svg) | CID 6918852 | Ki | 5000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/platelet-derived-growth-factor-receptor_e963c3aa05ad7127bcceb46efc475941.svg) | 6-(2,6-Dichlorophenyl)-8-methyl-2-(4-morpholin-4-ylanilino)pyrido[2,3-d]pyrimidin-7-one | IC50 | 636.0 [1] |
![](https://images.aatbio.com/dataset/ic50/platelet-derived-growth-factor-receptor_5c898ffa00cf3f2b994bb59aea767af1.svg) | 9-Hydroxy-4-phenyl-6H-pyrrolo[3,4-C]carbazole-1,3-dione | IC50 | 50000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/platelet-derived-growth-factor-receptor_cc4ece185f9b4c4aae0cb0a1535db1b0.svg) | (Z)-3-(3,4-Dimethoxy-phenyl)-2-pyridin-3-yl-acrylonitrile | IC50 | 3000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/platelet-derived-growth-factor-receptor_229be97168f5a1e19a21ea31c162ddf6.svg) | 3-(4-{4-Aminofuro[2,3-d]pyrimidin-5-yl}phenyl)-1-[2-fluoro-5-(trifluoromethyl)phenyl]urea | IC50 | 27.54 [1] |
![](https://images.aatbio.com/dataset/ic50/platelet-derived-growth-factor-receptor_b2e0374192c14780687bb9ed1d5a397b.svg) | PDGF Receptor Tyrosine Kinase Inhibitor III | IC50 | 80.0 [1] |
![](https://images.aatbio.com/dataset/ic50/platelet-derived-growth-factor-receptor_eafb0e81bf1ead1a6d779e2f6e43f30b.svg) | PDGF Receptor Tyrosine Kinase Inhibitor II | IC50 | 1100.0 [1] |
![](https://images.aatbio.com/dataset/ic50/platelet-derived-growth-factor-receptor_3d027434bed540e43919919e9f91203b.svg) | VEGF Receptor 2 Kinase Inhibitor I | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/platelet-derived-growth-factor-receptor_bbb936490cb2d36df2f50d54114bf2ad.svg) | 1-[4-(4-Aminothieno[2,3-d]pyrimidin-5-yl)phenyl]-3-(3-methylphenyl)urea | IC50 | 48.0 [1] |
![](https://images.aatbio.com/dataset/ic50/platelet-derived-growth-factor-receptor_5f02b655eda2ba8c931019b391ac0d51.svg) | 2-[2-[4-[4-(4-Tert-butylanilino)phenoxy]-6-methoxyquinolin-7-yl]oxyethylamino]ethanol | IC50 | 480.0 [1] |
![](https://images.aatbio.com/dataset/ic50/platelet-derived-growth-factor-receptor_10b979513d2e855fbc4454fcc705914e.svg) | 1-[2-Amino-6-(2,6-dichlorophenyl)pyrido[2,3-d]pyrimidin-7-yl]-3-tert-butylurea | IC50 | 1250.0 [1] |
![](https://images.aatbio.com/dataset/ic50/platelet-derived-growth-factor-receptor_8dd9e09809fda3f168eb4b9ad40384a9.svg) | N-(3-Cyclopropyl-1H-pyrazol-5-YL)-2-(2-naphthyl)acetamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/platelet-derived-growth-factor-receptor_58c90006fc0e17833fa580fd32d26841.svg) | 3-(3-Chlorophenyl)-5,7-dimethoxychromen-4-one | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/platelet-derived-growth-factor-receptor_c7ea91415258cf701a653bfc92e395ff.svg) | (5-Hydroxy-1H-indol-2-yl)-(1H-indol-2-yl)methanone | IC50 | 200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/platelet-derived-growth-factor-receptor_fa164f67dd00f6d2e9f05348b548a4dc.svg) | 4-(6,7-Dimethoxy-4-quinazolinyl)-N-(4-nitrophenyl)-1-piperazinecarboxamide | IC50 | 700.0 [1] |
![](https://images.aatbio.com/dataset/ic50/platelet-derived-growth-factor-receptor_017ea60e9b689094fe878e36635d2d23.svg) | N-(4-Chlorophenyl)-4-(6,7-dimethoxyquinazolin-4-yl)piperazine-1-carboxamide | IC50 | 1100.0 [1] |
![](https://images.aatbio.com/dataset/ic50/platelet-derived-growth-factor-receptor_c7c31ad92e1b0b77d0138e3a513f200e.svg) | N-Benzyl-4-(6,7-dimethoxyquinazolin-4-yl)piperazine-1-carbothioamide | IC50 | 550.0 [1] |
![](https://images.aatbio.com/dataset/ic50/platelet-derived-growth-factor-receptor_6238525de36d6e163d562db0dd8c6cad.svg) | 4-[(4-Methyl-1-piperazinyl)methyl]-N-[3-[[4-(3-pyridinyl)-2-pyrimidinyl]amino]phenyl]-benzamide | IC50 | 200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/platelet-derived-growth-factor-receptor_a790cac18f0dd5a580111474d0503b4d.svg) | 1,3-Diphenyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/platelet-derived-growth-factor-receptor_ce6920acc50917e483b92e9ba93d1188.svg) | 6-Acetyl-8-cyclopentyl-5-methyl-2-(4-piperazin-1-yl-phenylamino)-8H-pyrido[2,3-d]pyrimidin-7-one | IC50 | 2460.0 [1] |
![](https://images.aatbio.com/dataset/ic50/platelet-derived-growth-factor-receptor_5b10441bbfcd2a7880fba7127c6144c0.svg) | 3-[[5-[6-[(3-Chlorophenyl)amino]pyrazinyl]-3-pyridinyl]amino]-1-propanol | IC50 | 360.0 [1] |
![](https://images.aatbio.com/dataset/ic50/platelet-derived-growth-factor-receptor_9dabcb9dd97dc98e9c2238fea0fb3696.svg) | Glycine, N,N-dimethyl-, 2-(1H-indol-2-ylcarbonyl)-1H-indol-5-yl ester | IC50 | 100.0 [1] |
![](https://images.aatbio.com/dataset/ic50/platelet-derived-growth-factor-receptor_1c2f21fb84105173318aedd7aa2c5bfc.svg) | Thienopyrimidine deriv. 28 | IC50 | 60.0 [1] |
![](https://images.aatbio.com/dataset/ic50/platelet-derived-growth-factor-receptor_fd951065be8c84c1b332e18593d47262.svg) | N-(1,3-Benzodioxol-5-ylmethyl)-4-(6,7-dimethoxyquinazolin-4-yl)piperazine-1-carbothioamide | IC50 | 140.0 [1] |
![](https://images.aatbio.com/dataset/ic50/platelet-derived-growth-factor-receptor_bfc068b0de37e23c3c1f9268b88d562f.svg) | [4-[(2S)-2-Acetamido-3-[[(2S)-1-[[(2S)-1-(dibutylamino)-1-oxopropan-2-yl]amino]-3-methyl-1-oxobutan-2-yl]amino]-3-oxopropyl]phenyl] dihydrogen phosphate | IC50 | 77.0 [1] |
![](https://images.aatbio.com/dataset/ic50/platelet-derived-growth-factor-receptor_eccca8e1619e296862aaaa9d609c2860.svg) | 20-Ethyl-17,23-dioxa-4,14,20,26-tetrazahexacyclo[24.6.1.17,14.02,6.08,13.027,32]tetratriaconta-1(33),2(6),7(34),8,10,12,27,29,31-nonaene-3,5-dione | IC50 | 4400.0 [1] |
![](https://images.aatbio.com/dataset/ic50/platelet-derived-growth-factor-receptor_2f0440ad99a8f224adf7a929c6c5c12f.svg) | 3-(1H-Indol-3-yl)quinoline | IC50 | 8000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/platelet-derived-growth-factor-receptor_220d42a418e0b76bdf8e695de7abd6b8.svg) | 2-(3-Aminophenylamino)-6-(2,6-dichlorophenyl)-8-methylpyrido[2,3-d]pyrimidin-7(8H)-one | IC50 | 24.0 [1] |
![](https://images.aatbio.com/dataset/ic50/platelet-derived-growth-factor-receptor_ff9c97ae965f3c38b1a326d77574c930.svg) | N-(4-Bromophenyl)-4-(6,7-dimethoxyquinazolin-4-yl)piperazine-1-carboxamide | IC50 | 530.0 [1] |
![](https://images.aatbio.com/dataset/ic50/platelet-derived-growth-factor-receptor_a92ac6270ebde090c81e2e9c7c6cf7bc.svg) | N-(4-Tert-butylphenyl)-4-(6,7-dimethoxyquinazolin-4-yl)piperazine-1-carboxamide | IC50 | 30.0 [1] |
![](https://images.aatbio.com/dataset/ic50/platelet-derived-growth-factor-receptor_95493f8d18603aa8ebb85025d281548b.svg) | 4-(6,7-Dimethoxyquinazolin-4-yl)-N-(4-propan-2-ylphenyl)piperazine-1-carboxamide | IC50 | 80.0 [1] |
![](https://images.aatbio.com/dataset/ic50/platelet-derived-growth-factor-receptor_f438e3c7bf9e45199e79c5809088cdbb.svg) | N-(4-Chlorophenyl)-4-(6,7-dimethoxyquinazolin-4-yl)piperazine-1-carbothioamide | IC50 | 790.0 [1] |
![](https://images.aatbio.com/dataset/ic50/platelet-derived-growth-factor-receptor_fa5e07784488382cd6f4b6c8e05eed3d.svg) | [3-(2-Imidazol-1-yl-ethoxy)-phenyl]-(4-pyridin-3-yl-pyrimidin-2-yl)-amine | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/platelet-derived-growth-factor-receptor_c96eb92a27fb9bb63cf7e9d2ca4db08d.svg) | 3-[5-[3-(2-Methoxyethoxy)prop-1-ynyl]thiophen-3-yl]-7-(1,2,4-triazol-1-ylmethyl)-1,4-dihydroindeno[1,2-c]pyrazole | IC50 | 84.0 [1] |
![](https://images.aatbio.com/dataset/ic50/platelet-derived-growth-factor-receptor_1c0672b167275420873e93bbcbc80ed2.svg) | (3-Imidazol-1-yl-phenyl)-(4-pyridin-3-yl-pyrimidin-2-yl)-amine | IC50 | 18000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/platelet-derived-growth-factor-receptor_a48938f0bcc140c4b47f4c8bb103a1f3.svg) | (3-Chloro-phenyl)-(4-pyridin-3-yl-pyrimidin-2-yl)-amine | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/platelet-derived-growth-factor-receptor_3c0f6a73cbc4459571db355cf32beaf5.svg) | 2-(Phenylamino)quinoxaline | IC50 | 5100.0 [1] |
![](https://images.aatbio.com/dataset/ic50/platelet-derived-growth-factor-receptor_6873ea49735d36649ab7181056d0b14f.svg) | 4-(Benzothiazol-6-ylamino)-6-(benzyl-isopropyl-amino)-[1,3,5]triazin-2-ol | IC50 | 12500.0 [1] |
![](https://images.aatbio.com/dataset/ic50/platelet-derived-growth-factor-receptor_428de67b623f9bcea05ecbbdd5883d96.svg) | 6-[(4-Methylpiperazin-1-yl)methyl]-3-[5-(3-phenoxyprop-1-ynyl)thiophen-3-yl]-1,4-dihydroindeno[1,2-c]pyrazole | IC50 | 58.0 [1] |
![](https://images.aatbio.com/dataset/ic50/platelet-derived-growth-factor-receptor_482caccce5577424472b4f30ef45663d.svg) | [6-Chloro-4-methyl-3-[[3-(methylsulfamoylamino)phenyl]methyl]-2-oxochromen-7-yl] N,N-dimethylcarbamate | IC50 | 50000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/platelet-derived-growth-factor-receptor_27026f966ba91a62c343a6cb4f61c185.svg) | 7-((1H-Imidazol-1-yl)methyl)-3-(thiophen-3-yl)-1,4-dihydroindeno[1,2-c]pyrazole | IC50 | 50000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/platelet-derived-growth-factor-receptor_03a355acde03979fd5dbde19609eb8e0.svg) | 7-[(4-Methylpiperazin-1-yl)methyl]-3-thiophen-3-yl-1,4-dihydroindeno[1,2-c]pyrazole | IC50 | 50000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/platelet-derived-growth-factor-receptor_460f9101e7943d38d0b2ef84527ff304.svg) | 2-Aminopyrido[2,3-d]pyrimidin-7(8H)-one 46 | IC50 | 500.0 [1] |
![](https://images.aatbio.com/dataset/ic50/platelet-derived-growth-factor-receptor_8232754fecc261b7459667e77731da57.svg) | 2-Aminopyrido[2,3-d]pyrimidin-7(8H)-one 50 | IC50 | 76.0 [1] |
![](https://images.aatbio.com/dataset/ic50/platelet-derived-growth-factor-receptor_a5e2edf16746073d4f4a1ab199c697f7.svg) | 2-Aminopyrido[2,3-d]pyrimidin-7(8H)-one 51 | IC50 | 82.0 [1] |
![](https://images.aatbio.com/dataset/ic50/platelet-derived-growth-factor-receptor_08200d339f414120a8135a9db47a1f10.svg) | 1-[2-Amino-6-(2,6-dimethylphenyl)pyrido[2,3-d]pyrimidin-7-yl]-3-tert-butylurea | IC50 | 340.0 [1] |
![](https://images.aatbio.com/dataset/ic50/platelet-derived-growth-factor-receptor_d40fcb2be0a9cddaf2d96063b00d9a24.svg) | 1-[2-Amino-6-(2,3,5,6-tetramethylphenyl)pyrido[2,3-d]pyrimidin-7-yl]-3-tert-butylurea | IC50 | 50000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/platelet-derived-growth-factor-receptor_15f1422e39010bb4b4ec1df07625e658.svg) | 1-(2-Amino-6-phenylpyrido[2,3-d]pyrimidin-7-yl)-3-tert-butylurea | IC50 | 13240.0 [1] |
![](https://images.aatbio.com/dataset/ic50/platelet-derived-growth-factor-receptor_1d4695468dde2d60ae8b28d9b9ad4e73.svg) | PD089828 analog 12 | IC50 | 50000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/platelet-derived-growth-factor-receptor_6cf7886a5b82a2bf609f0a60248cf8d4.svg) | 1-[2-Amino-6-(3,5-diethoxyphenyl)pyrido[2,3-d]pyrimidin-7-yl]-3-tert-butylurea | IC50 | 50000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/platelet-derived-growth-factor-receptor_98ddcb182ba99dbe35bc1cff3e6008b6.svg) | PD089828 analog 31 | IC50 | 50000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/platelet-derived-growth-factor-receptor_63e4642dfc493032f304638d6c920ebc.svg) | Bis(1H-2-indolyl)methanone 11 | IC50 | 300.0 [1] |
![](https://images.aatbio.com/dataset/ic50/platelet-derived-growth-factor-receptor_fc8e0ee4e89abe2e1f2bae64b674ecd0.svg) | Bis(1H-2-indolyl)methanone 12 | IC50 | 300.0 [1] |
![](https://images.aatbio.com/dataset/ic50/platelet-derived-growth-factor-receptor_be130926288e95a2e738065fb0b2790a.svg) | Acetic acid, methoxy-, 2-(1H-indol-2-ylcarbonyl)-1H-indol-5-yl ester | IC50 | 200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/platelet-derived-growth-factor-receptor_dfa25059701399b6aea342e563393987.svg) | 3-[[4-[4-[(3-Chlorophenyl)amino]-1,3,5-triazin-2-yl]-2-pyridinyl]amino]-1-Propanol | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/platelet-derived-growth-factor-receptor_0e57dd1eb58b575cc332fec3561866e1.svg) | N-(4-Pyridin-4-yl-pyrimidin-2-yl)-benzene-1,3-diamine | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/platelet-derived-growth-factor-receptor_392fa124e10264240b17243651a4f4e0.svg) | N-(4-Pyridin-3-yl-pyrimidin-2-yl)-benzene-1,3-diamine | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/platelet-derived-growth-factor-receptor_d37189895be31a0566a9ac4c34fce103.svg) | 2-Chloro-N-[4-(4,5-dichloro-2-fluoro-phenylamino)-quinazolin-6-yl]-acetamide | IC50 | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/platelet-derived-growth-factor-receptor_74f40f0841354156dfe0679af418412b.svg) | 6-(2,6-Dichlorophenyl)-8-methyl-2-[4-(4-methylpiperazine-1-carbonyl)anilino]pyrido[2,3-d]pyrimidin-7-one | IC50 | 14.0 [1] |
![](https://images.aatbio.com/dataset/ic50/platelet-derived-growth-factor-receptor_6991f3374d93faff474372a5e671f4e9.svg) | 6,7-Dimethoxy-3-((E)-styryl)-quinoline | IC50 | 5.0 [1] |
![](https://images.aatbio.com/dataset/ic50/platelet-derived-growth-factor-receptor_53e7a7486c5bedc031e625a35c1abf10.svg) | 6,7-Dimethoxy-3-(4-methoxy-3-methyl-phenyl)-quinoline | IC50 | 400.0 [1] |
![](https://images.aatbio.com/dataset/ic50/platelet-derived-growth-factor-receptor_40cb9fb3058875da4f2a5b0a0235e254.svg) | 6-(2,6-Dichlorophenyl)-2-(4-iodophenylamino)-8-methylpyrido[2,3-d]pyrimidin-7(8H)-one | IC50 | 203.0 [1] |
![](https://images.aatbio.com/dataset/ic50/platelet-derived-growth-factor-receptor_fae93bb232969759d34c3ee50fd93daf.svg) | 3-(4-Fluoro-phenyl)-6,7-dimethoxy-quinoline | IC50 | 60.0 [1] |
![](https://images.aatbio.com/dataset/ic50/platelet-derived-growth-factor-receptor_c4b2ab60a253bfa905828e72348b7733.svg) | 3-[[4-(3-Pyridinyl)-2-pyrimidinyl]amino]benzoic acid | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/platelet-derived-growth-factor-receptor_e585aecd77d4d0082e60a38a1a577928.svg) | 3-(2-Cyclohexyl-ethyl)-6,7-dimethoxy-quinoline | IC50 | 500.0 [1] |
![](https://images.aatbio.com/dataset/ic50/platelet-derived-growth-factor-receptor_285974c5411aa98e6af3d8fc51150102.svg) | 3-(1H-Indol-3-yl)-7,8-dimethoxy-quinoline | IC50 | 50000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/platelet-derived-growth-factor-receptor_516729703440656f0da95fd0e05265ee.svg) | 3-(2,4-Dimethoxy-phenyl)-6,7-dimethoxy-quinoline | IC50 | 50000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/platelet-derived-growth-factor-receptor_9956f5332ef1d08478f3c6bff358a946.svg) | 4-(6,7-Dimethoxy-quinolin-3-yl)-benzoic acid ethyl ester | IC50 | 200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/platelet-derived-growth-factor-receptor_d5b019986aa49dc386aa234b795fb6dc.svg) | 3-Hydroxy-6,7-dimethoxyquinoline | IC50 | 20000.0 [1] |