Phospholipase A-2-activating protein Inhibitors (IC50, Ki)

Structure ▲ ▼	Compound Name ▲ ▼	Standard Type ▲ ▼	Standard Values (in nM) ▲ ▼
	Tryptophan	IC50	5000.0 [1]
	Leucine	IC50	5000.0 [1]
	Phenylalanine	IC50	5000.0 [1]
	Theophylline	IC50	5000.0 [1]
	Levamisole	IC50	5000.0 [1]
	L-Homoarginine	IC50	5000.0 [1]
	(S)-2-Amino-4-methylpentanamide	IC50	5000.0 [1]
	5Z-7-Oxozeaenol	IC50	11.0 [1]
	2,5-Dimethoxy-N-(3-quinolinyl)benzenesulfonamide	IC50	100000.0 [1]
	1-(3,4-Dihydroxyphenyl)-2-{[1-(4-methoxyphenyl)-1H-tetrazol-5-yl]thio}ethanone	IC50	2000.0 [1]
	2-{[2-(3,4-Dihydroxyphenyl)-2-oxoethyl]thio}-4-(methoxymethyl)-6-methylnicotinonitrile	IC50	2200.0 [1]
	1-(3,4-Dihydroxyphenyl)-2-(1-imidazolyl)ethanone	IC50	2100.0 [1]
	1-(3,4-Dihydroxy-phenyl)-2-(5-phenyl-4H-[1,2,4]triazol-3-ylsulfanyl)-ethanone	IC50	100000.0 [1]
	1-(3,4-Dihydroxyphenyl)-2-[(4,6-dimethyl-2-pyrimidinyl)thio]ethanone	IC50	2500.0 [1]
	2-(5-(3-Aminophenyl)-4-methyl-4H-1,2,4-triazol-3-ylthio)-1-phenylethanone	IC50	100000.0 [1]
	3-[2-(3,4-Dihydroxyphenyl)-2-oxoethyl]-6,7-dimethoxy-2-benzofuran-1(3H)-one	IC50	3000.0 [1]
	1-(3,4-Dihydroxyphenyl)-2-(4-methyl-5-phenyl-4H-1,2,4-triazol-3-ylthio)ethanone	IC50	6700.0 [1]
	2-(4,6-Dimethylpyrimidin-2-ylthio)-1-(4-methoxyphenyl)ethanone	IC50	100000.0 [1]
	(4S,6Z,9S,10S,12E)-9,10,18-Trihydroxy-16-methoxy-4,7-dimethyl-3-oxabicyclo[12.4.0]octadeca-1(14),6,12,15,17-pentaene-2,8-dione	IC50	10000.0 [1]
	(4S,6Z,9S,10S,12E)-9,10,18-Trihydroxy-16-methoxy-4,6-dimethyl-3-oxabicyclo[12.4.0]octadeca-1(14),6,12,15,17-pentaene-2,8-dione	IC50	10000.0 [1]
	2-(4,6-Dimethylpyrimidin-2-ylthio)-1-(4-hydroxyphenyl)ethanone	IC50	100000.0 [1]
	1-(1,3-Benzodioxol-5-yl)-2-(4,6-dimethylpyrimidin-2-yl)sulfanylethanone	IC50	100000.0 [1]
	2-(4,6-Dimethylpyrimidin-2-yl)sulfanyl-1-(4-hydroxy-3-methoxyphenyl)ethanone	IC50	100000.0 [1]
	2-(4-Bromo-2-methylimidazol-1-yl)-1-(3,4-dihydroxyphenyl)ethanone	IC50	4900.0 [1]
	2-(4-Bromoimidazol-1-yl)-1-(3,4-dihydroxyphenyl)ethanone	IC50	15800.0 [1]
	1-(3,4-Dihydroxyphenyl)-2-(2-phenylimidazol-1-yl)ethanone	IC50	17200.0 [1]
	1-(3,4-Dihydroxyphenyl)-2-(2-ethyl-1-imidazolyl)ethanone	IC50	800.0 [1]
	2-(1H-Benzimidazol-2-ylamino)-1-(3,4-dihydroxyphenyl)ethanone	IC50	9100.0 [1]
	1-(3,4-Dihydroxyphenyl)-2-(1,2,4-triazol-4-yl)ethanone	IC50	13400.0 [1]
	1-(3,4-Dihydroxyphenyl)-2-(5,6-dimethylbenzimidazol-1-yl)ethanone	IC50	5800.0 [1]
	1-(3,4-Dihydroxyphenyl)-2-(2-methyl-1-imidazolyl)ethanone	IC50	14300.0 [1]
	2-(Benzimidazol-1-yl)-1-(3,4-dihydroxyphenyl)ethanone	IC50	800.0 [1]
	1-(3,4-Dihydroxyphenyl)-2-(2-methyl-1-benzimidazolyl)ethanone	IC50	6600.0 [1]
	1-(3,4-Dihydroxyphenyl)-2-(4-methylimidazol-1-yl)ethanone	IC50	5800.0 [1]
	4-((4,6-Dimethylpyrimidin-2-ylamino)methyl)benzene-1,2-diol	IC50	51200.0 [1]
	1-(3,4-Dihydroxyphenyl)-2-(4-methyl-1-pyrazolyl)ethanone	IC50	2700.0 [1]
	2-(4,6-Dimethylpyrimidin-2-ylthio)-1-(3-hydroxyphenyl)ethanone	IC50	100000.0 [1]
	N-(3,4-Dihydroxybenzyl)-4,5-dimethylfuran-2-carboxamide	IC50	100000.0 [1]
	N-(3,4-Dihydroxyphenethyl)-4,5-dimethylfuran-2-carboxamide	IC50	100000.0 [1]
	(4S,6E,9S,10S,12E)-7-Fluoro-9,10,18-trihydroxy-16-methoxy-4-methyl-3-oxabicyclo[12.4.0]octadeca-1(14),6,12,15,17-pentaene-2,8-dione	IC50	36.0 [1]
	Isoproterenone	IC50	39300.0 [1]

Entire TableStructureCompound NameStandard TypeStandard Values (in nM)

Items per page: 510All1 - 10 of 41 ⟨⟩

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References

This online tool may be cited as follows

MLA	"Quest Database™ Phospholipase A-2-activating protein Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 20 Feb. 2025, https://www.aatbio.com/data-sets/phospholipase-a-2-activating-protein-inhibitors-ic50-ki.
APA	AAT Bioquest, Inc. (2025, February 20). Quest Database™ Phospholipase A-2-activating protein Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/phospholipase-a-2-activating-protein-inhibitors-ic50-ki.
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