| m-Xylylenediphosphonic Acid | IC50 | 200000.0 [1] |
| m-Xylylenediphosphonic Acid | Ki | 120000.0 [1] |
| [Fluoro-[6-[fluoro(phosphono)methyl]pyridin-2-yl]methyl]phosphonic acid | IC50 | 87000.0 [1] |
| [Fluoro-[6-[fluoro(phosphono)methyl]pyridin-2-yl]methyl]phosphonic acid | Ki | 61000.0 [1] |
| [6-(Phosphonomethyl)pyridin-2-yl]methylphosphonic acid | IC50 | 182000.0 [1] |
| [6-(Phosphonomethyl)pyridin-2-yl]methylphosphonic acid | Ki | 80000.0 [1] |
| [Hydroxy-[3-[hydroxy(phosphono)methyl]phenyl]methyl]phosphonic acid | IC50 | 150000.0 [1] |
| [Hydroxy-[3-[hydroxy(phosphono)methyl]phenyl]methyl]phosphonic acid | Ki | 75000.0 [1] |
| 2-(Phosphonomethyl)prop-2-enylphosphonic acid | IC50 | 87000.0 [1] |
| 2-(Phosphonomethyl)prop-2-enylphosphonic acid | Ki | 61000.0 [1] |
| [Hydroxy-[6-[hydroxy(phosphono)methyl]pyridin-2-yl]methyl]phosphonic acid | IC50 | 163000.0 [1] |
| [Hydroxy-[6-[hydroxy(phosphono)methyl]pyridin-2-yl]methyl]phosphonic acid | Ki | 156000.0 [1] |
| [Chloro-[6-[chloro(phosphono)methyl]pyridin-2-yl]methyl]phosphonic acid | IC50 | 1340.0 [1] |
| [Chloro-[6-[chloro(phosphono)methyl]pyridin-2-yl]methyl]phosphonic acid | Ki | 330.0 [1] |
| [Fluoro-[3-[fluoro(phosphono)methyl]phenyl]methyl]phosphonic acid | IC50 | 1300.0 [1] |
| [Fluoro-[3-[fluoro(phosphono)methyl]phenyl]methyl]phosphonic acid | Ki | 690.0 [1] |
| Adenosine | IC50 | 3000000.0 [1] |
| N6-Cyclopentyladenosine | IC50 | 3900000.0 [1] |
| N6-Benzyladenosine | IC50 | 1000000.0 [1] |
| 2-Aminoadenosine | IC50 | 3500000.0 [1] |
| (2R,3R,4S,5R)-2-[6-(Cycloheptylamino)purin-9-yl]-5-(hydroxymethyl)oxolane-3,4-diol | IC50 | 3900000.0 [1] |
| (2R,3S,4R,5R)-2-(Hydroxymethyl)-5-[6-(pentylamino)purin-9-yl]oxolane-3,4-diol | IC50 | 3000000.0 [1] |
| 2-[6-Amino-2-(2-phenyl-propylamino)-purin-9-yl]-5-hydroxymethyl-tetrahydro-furan-3,4-diol | IC50 | 700000.0 [1] |
| (3R,4S,5R)-2-[2-Amino-6-(cyclopentylamino)purin-9-yl]-5-(hydroxymethyl)oxolane-3,4-diol | IC50 | 1500000.0 [1] |
| (2R,3R,4S,5R)-2-[6-Amino-2-(cyclohexylamino)purin-9-yl]-5-(hydroxymethyl)oxolane-3,4-diol | IC50 | 1500000.0 [1] |
| (2R,3R,4S,5R)-2-(6-Amino-2-cyclopentylamino-purin-9-yl)-5-hydroxymethyl-tetrahydro-furan-3,4-diol | IC50 | 1500000.0 [1] |
| [4-(Phosphonomethyl)phenyl]methylphosphonic Acid | IC50 | 193000.0 [1] |
| (3R,4S,5R)-2-[6-Amino-2-(3-phenylpropylamino)purin-9-yl]-5-(hydroxymethyl)oxolane-3,4-diol | IC50 | 1800000.0 [1] |
| (3R,4S,5R)-2-[6-Amino-2-(benzylamino)purin-9-yl]-5-(hydroxymethyl)oxolane-3,4-diol | IC50 | 3500000.0 [1] |
| (3R,4S,5R)-2-[6-(2-Aminoethylamino)purin-9-yl]-5-(hydroxymethyl)oxolane-3,4-diol | IC50 | 2500000.0 [1] |
| (3R,4S,5R)-2-[2,6-Bis(2-phenylethylamino)purin-9-yl]-5-(hydroxymethyl)oxolane-3,4-diol | IC50 | 30000.0 [1] |
| (2R,3R,4S,5R)-2-[6-Amino-2-(propylamino)purin-9-yl]-5-(hydroxymethyl)oxolane-3,4-diol | IC50 | 1500000.0 [1] |
| [(3-Phosphonophenyl)hydroxymethyl]phosphonic acid | IC50 | 102000.0 [1] |
| [[4-(Phosphonomethyl)phenyl]fluoromethyl]phosphonic acid | IC50 | 10700.0 [1] |
| [[3-(Phosphonodifluoromethyl)phenyl]difluoromethyl]phosphonic acid | IC50 | 960.0 [1] |
| [[4-(Phosphonomethyl)phenyl]chloromethyl]phosphonic acid | IC50 | 9400.0 [1] |
| [Fluoro-[4-[fluoro(phosphono)methyl]phenyl]methyl]phosphonic acid | IC50 | 1150.0 [1] |
| [4-[Hydroxy(phosphono)methyl]phenyl]methylphosphonic acid | IC50 | 89000.0 [1] |
| [[3-(Phosphonomethyl)phenyl]fluoromethyl]phosphonic acid | IC50 | 8350.0 [1] |
| [2,4-Dimethyl-5-(phosphonomethyl)phenyl]methylphosphonic acid | IC50 | 73000.0 [1] |
| [Hydroxy-[4-[hydroxy(phosphono)methyl]phenyl]methyl]phosphonic acid | IC50 | 181000.0 [1] |
| [(3-Phosphonophenyl)methyl]phosphonic acid | IC50 | 138000.0 [1] |
| [(3-Phosphonophenyl)difluoromethyl]phosphonic acid | IC50 | 1000.0 [1] |
| [Chloro-[3-[chloro(phosphono)methyl]phenyl]methyl]phosphonic acid | IC50 | 1000.0 [1] |
| [(3-Phosphonophenyl)fluoromethyl]phosphonic acid | IC50 | 16000.0 [1] |
| [3-Methyl-5-(phosphonomethyl)phenyl]methylphosphonic acid | IC50 | 99000.0 [1] |
| [[3-(Phosphonomethyl)phenyl]difluoromethyl]phosphonic acid | IC50 | 1800.0 [1] |
| [[4-(Phosphonodifluoromethyl)phenyl]difluoromethyl]phosphonic acid | IC50 | 980.0 [1] |
| [[6-(Phosphonodifluoromethyl)-2-pyridinyl]difluoromethyl]phosphonic acid | IC50 | 1170.0 [1] |
| [3-[Hydroxy(phosphono)methyl]phenyl]methylphosphonic acid | IC50 | 68800.0 [1] |
| [2-Fluoro-3-(phosphonomethyl)phenyl]methylphosphonic acid | IC50 | 147000.0 [1] |
| [Chloro-[4-[chloro(phosphono)methyl]phenyl]methyl]phosphonic acid | IC50 | 1080.0 [1] |
| [[3-[Difluoro(phosphono)methyl]-5-methylphenyl]-difluoromethyl]phosphonic acid | IC50 | 880.0 [1] |
| [[3-(Phosphonomethyl)phenyl]chloromethyl]phosphonic acid | IC50 | 8000.0 [1] |
| [(3-Phosphonophenyl)chloromethyl]phosphonic acid | IC50 | 17000.0 [1] |
| [[4-(Phosphonomethyl)phenyl]difluoromethyl]phosphonic acid | IC50 | 1980.0 [1] |
| [2,4,6-Trimethyl-3-(phosphonomethyl)phenyl]methylphosphonic acid | IC50 | 78000.0 [1] |
| o-Xylylenediphosphonic Acid | IC50 | 107000.0 [1] |
| (2R,3R,4S,5R)-2-[6-Amino-2-[(2-hydroxy-2-phenylethyl)amino]purin-9-yl]-5-(hydroxymethyl)oxolane-3,4-diol | IC50 | 1400000.0 [1] |
| [Dichloro-[3-[dichloro(phosphono)methyl]phenyl]methyl]phosphonic acid | IC50 | 3600.0 [1] |
| (3R,4S,5R)-2-[2-Amino-6-[2-(4-hydroxy-3-methoxyphenyl)ethylamino]purin-9-yl]-5-(hydroxymethyl)oxolane-3,4-diol | IC50 | 1500000.0 [1] |
| (3R,4S,5R)-2-[2-Amino-6-[2-(3-methoxyphenyl)ethylamino]purin-9-yl]-5-(hydroxymethyl)oxolane-3,4-diol | IC50 | 1900000.0 [1] |
| (3R,4S,5R)-2-[6-Amino-2-[(2-chlorophenyl)methylamino]purin-9-yl]-5-(hydroxymethyl)oxolane-3,4-diol | IC50 | 2000000.0 [1] |
| (3R,4S,5R)-2-[2-Amino-6-(cycloheptylamino)purin-9-yl]-5-(hydroxymethyl)oxolane-3,4-diol | IC50 | 2500000.0 [1] |
| (3R,4S,5R)-2-[2-Amino-6-(3-aminopropylamino)purin-9-yl]-5-(hydroxymethyl)oxolane-3,4-diol | IC50 | 4000000.0 [1] |
| (3R,4S,5R)-2-[2-Amino-6-[2-(2-methoxyphenyl)ethylamino]purin-9-yl]-5-(hydroxymethyl)oxolane-3,4-diol | IC50 | 1800000.0 [1] |
| (3R,4S,5R)-2-[2-Amino-6-(benzylamino)purin-9-yl]-5-(hydroxymethyl)oxolane-3,4-diol | IC50 | 600000.0 [1] |
| (3R,4S,5R)-2-[2-Amino-6-[5-[[2-amino-9-[(3S,4R,5S)-3,4-dihydroxy-5-(hydroxymethyl)oxolan-2-yl]purin-6-yl]amino]pentylamino]purin-9-yl]-5-(hydroxymethyl)oxolane-3,4-diol | IC50 | 1000000.0 [1] |
| (3R,4S,5R)-2-[6-Amino-2-(butylamino)purin-9-yl]-5-(hydroxymethyl)oxolane-3,4-diol | IC50 | 1500000.0 [1] |
| (3R,4S,5R)-2-[2-Amino-6-(cyclohexylmethylamino)purin-9-yl]-5-(hydroxymethyl)oxolane-3,4-diol | IC50 | 2500000.0 [1] |
| (3R,4S,5R)-2-[6-Amino-2-[(4-methoxyphenyl)methylamino]purin-9-yl]-5-(hydroxymethyl)oxolane-3,4-diol | IC50 | 1000000.0 [1] |
| (3R,4S,5R)-2-[2-Amino-6-(3-phenylpropylamino)purin-9-yl]-5-(hydroxymethyl)oxolane-3,4-diol | IC50 | 4000000.0 [1] |
| (3R,4S,5R)-2-[2-Amino-6-[2-(4-hydroxyphenyl)ethylamino]purin-9-yl]-5-(hydroxymethyl)oxolane-3,4-diol | IC50 | 130000.0 [1] |
| (3R,4S,5R)-2-[2-Amino-6-(pentylamino)purin-9-yl]-5-(hydroxymethyl)oxolane-3,4-diol | IC50 | 2000000.0 [1] |
| (3R,4S,5R)-2-[2-Amino-6-[2-(3-chlorophenyl)ethylamino]purin-9-yl]-5-(hydroxymethyl)oxolane-3,4-diol | IC50 | 1200000.0 [1] |
| (3R,4S,5R)-2-[2-Amino-6-(2-phenylpropylamino)purin-9-yl]-5-(hydroxymethyl)oxolane-3,4-diol | IC50 | 2900000.0 [1] |
| (3R,4S,5R)-2-[2-Amino-6-(ethylamino)purin-9-yl]-5-(hydroxymethyl)oxolane-3,4-diol | IC50 | 3500000.0 [1] |
| (3R,4S,5R)-2-[2-Amino-6-(1-phenylethylamino)purin-9-yl]-5-(hydroxymethyl)oxolane-3,4-diol | IC50 | 2900000.0 [1] |
| (3R,4S,5R)-2-[2-Amino-6-[2-(2-chlorophenyl)ethylamino]purin-9-yl]-5-(hydroxymethyl)oxolane-3,4-diol | IC50 | 1900000.0 [1] |
| (3R,4S,5R)-2-[6-Amino-2-[(3-methylphenyl)methylamino]purin-9-yl]-5-(hydroxymethyl)oxolane-3,4-diol | IC50 | 1500000.0 [1] |
| (3R,4S,5R)-2-[2-Amino-6-(furan-2-ylmethylamino)purin-9-yl]-5-(hydroxymethyl)oxolane-3,4-diol | IC50 | 1500000.0 [1] |
| (3R,4S,5R)-2-[6-Amino-2-[2-(2,4-dichlorophenyl)ethylamino]purin-9-yl]-5-(hydroxymethyl)oxolane-3,4-diol | IC50 | 600000.0 [1] |
| (3R,4S,5R)-2-[2-Amino-6-[2-(4-methylphenyl)ethylamino]purin-9-yl]-5-(hydroxymethyl)oxolane-3,4-diol | IC50 | 200000.0 [1] |
| (3R,4S,5R)-2-[6-Amino-2-(cycloheptylamino)purin-9-yl]-5-(hydroxymethyl)oxolane-3,4-diol | IC50 | 3000000.0 [1] |
| (3R,4S,5R)-2-[6-Amino-2-[(2-methoxyphenyl)methylamino]purin-9-yl]-5-(hydroxymethyl)oxolane-3,4-diol | IC50 | 1400000.0 [1] |
| (3R,4S,5R)-2-[2-Amino-6-[2-(4-methoxyphenyl)ethylamino]purin-9-yl]-5-(hydroxymethyl)oxolane-3,4-diol | IC50 | 1500000.0 [1] |
| (3R,4S,5R)-2-[2-Amino-6-(prop-2-ynylamino)purin-9-yl]-5-(hydroxymethyl)oxolane-3,4-diol | IC50 | 1500000.0 [1] |
| (3R,4S,5R)-2-[2-Amino-6-[2-(3-hydroxyphenyl)ethylamino]purin-9-yl]-5-(hydroxymethyl)oxolane-3,4-diol | IC50 | 250000.0 [1] |
| (3R,4S,5R)-2-[2-Amino-6-[2-(4-aminophenyl)ethylamino]purin-9-yl]-5-(hydroxymethyl)oxolane-3,4-diol | IC50 | 250000.0 [1] |
| (3R,4S,5R)-2-[6-Amino-2-[(3-chlorophenyl)methylamino]purin-9-yl]-5-(hydroxymethyl)oxolane-3,4-diol | IC50 | 800000.0 [1] |
| (3R,4S,5R)-2-[2-Amino-6-[2-(3,4-dihydroxyphenyl)ethylamino]purin-9-yl]-5-(hydroxymethyl)oxolane-3,4-diol | IC50 | 250000.0 [1] |
| (3R,4S,5R)-2-[6-Amino-2-[2-(4-hydroxyphenyl)ethylamino]purin-9-yl]-5-(hydroxymethyl)oxolane-3,4-diol | IC50 | 500000.0 [1] |
| (3R,4S,5R)-2-[2-Amino-6-(2-phenylethylamino)purin-9-yl]-5-(hydroxymethyl)oxolane-3,4-diol | IC50 | 200000.0 [1] |
| (3R,4S,5R)-2-[2-Amino-6-(naphthalen-1-ylmethylamino)purin-9-yl]-5-(hydroxymethyl)oxolane-3,4-diol | IC50 | 1900000.0 [1] |
| (3R,4S,5R)-2-[6-Amino-2-(2-phenylpropylamino)purin-9-yl]-5-(hydroxymethyl)oxolane-3,4-diol | IC50 | 3500000.0 [1] |
| (3R,4S,5R)-2-[6-Amino-2-(oxolan-2-ylmethylamino)purin-9-yl]-5-(hydroxymethyl)oxolane-3,4-diol | IC50 | 800000.0 [1] |
| (3R,4S,5R)-2-[6-Amino-2-[2-(4-aminophenyl)ethylamino]purin-9-yl]-5-(hydroxymethyl)oxolane-3,4-diol | IC50 | 500000.0 [1] |
| (3R,4S,5R)-2-[2-Amino-6-[4-[[2-amino-9-[(3S,4R,5S)-3,4-dihydroxy-5-(hydroxymethyl)oxolan-2-yl]purin-6-yl]amino]butylamino]purin-9-yl]-5-(hydroxymethyl)oxolane-3,4-diol | IC50 | 750000.0 [1] |
| (3R,4S,5R)-2-[2-Amino-6-(butylamino)purin-9-yl]-5-(hydroxymethyl)oxolane-3,4-diol | IC50 | 900000.0 [1] |
| (3R,4S,5R)-2-[6-Amino-2-[2-(2-chlorophenyl)ethylamino]purin-9-yl]-5-(hydroxymethyl)oxolane-3,4-diol | IC50 | 2200000.0 [1] |