![](https://images.aatbio.com/dataset/ic50/peroxisome-proliferator-activated-receptor-alpha_75de8bb67a0e2555d13e845be859468c.svg) | Rosiglitazone | IC50 | 10000.0 [1], 15000.0 [2], 50000.0 [3], 100000.0 [4] |
![](https://images.aatbio.com/dataset/ic50/peroxisome-proliferator-activated-receptor-alpha_75de8bb67a0e2555d13e845be859468c.svg) | Rosiglitazone | Ki | 33300.0 [1] |
![](https://images.aatbio.com/dataset/ic50/peroxisome-proliferator-activated-receptor-alpha_2deff51ca7df7c17041b5f1bdaa9bce1.svg) | Fenofibric acid | IC50 | 10000.0 [1], 24000.0 [2], 35000.0 [3] |
![](https://images.aatbio.com/dataset/ic50/peroxisome-proliferator-activated-receptor-alpha_2deff51ca7df7c17041b5f1bdaa9bce1.svg) | Fenofibric acid | Ki | 35000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/peroxisome-proliferator-activated-receptor-alpha_b5a2498ba76e0a74b43478962185f1cc.svg) | Endurobol | IC50 | 463.0 [1], 1995.26 [2] |
![](https://images.aatbio.com/dataset/ic50/peroxisome-proliferator-activated-receptor-alpha_aed333a52366f4f302bf087e5c103f48.svg) | 2-Methyl-3-{4-[2-(5-methyl-2-phenyl-oxazol-4-yl)-ethoxy]-phenyl}-2-phenoxy-propionic acid | IC50 | 42.0 [1] |
![](https://images.aatbio.com/dataset/ic50/peroxisome-proliferator-activated-receptor-alpha_8c1068f2a127c296cb0d1e6a0c1bdea0.svg) | Farglitazar | IC50 | 2870.0 [1] |
![](https://images.aatbio.com/dataset/ic50/peroxisome-proliferator-activated-receptor-alpha_8c1068f2a127c296cb0d1e6a0c1bdea0.svg) | Farglitazar | Ki | 489.78 [1], 490.0 [2] |
![](https://images.aatbio.com/dataset/ic50/peroxisome-proliferator-activated-receptor-alpha_3f535485f4136475bd96fea9d1049700.svg) | 5-[3-[3-(4-Phenoxy-2-propylphenoxy)propoxy]phenyl]-1,3-thiazolidine-2,4-dione | IC50 | 28.0 [1] |
![](https://images.aatbio.com/dataset/ic50/peroxisome-proliferator-activated-receptor-alpha_3f535485f4136475bd96fea9d1049700.svg) | 5-[3-[3-(4-Phenoxy-2-propylphenoxy)propoxy]phenyl]-1,3-thiazolidine-2,4-dione | Ki | 30.0 [1] |
![](https://images.aatbio.com/dataset/ic50/peroxisome-proliferator-activated-receptor-alpha_03f092899b0bd9c810c7a4e0e83e60b6.svg) | F3MethylAA | IC50 | 280.0 [1], 310.0 [2] |
![](https://images.aatbio.com/dataset/ic50/peroxisome-proliferator-activated-receptor-alpha_f31ed59aacf7f1a64de01fe0d16adc5d.svg) | (2S)-2-(4-[2-(3-[2,4-Difluorophenyl]-1-heptylureido)ethyl]phenoxy)-2-methylbutyric acid | IC50 | 348.0 [1], 538.0 [2], 740.0 [3] |
![](https://images.aatbio.com/dataset/ic50/peroxisome-proliferator-activated-receptor-alpha_8fa4bab24a63d98653dcfb9859ac5704.svg) | (2S)-2-Methyl-3-[4-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl]-2-phenoxypropanoic acid | IC50 | 21.0 [1] |
![](https://images.aatbio.com/dataset/ic50/peroxisome-proliferator-activated-receptor-alpha_154415637c0e204eb7978910d28e9430.svg) | 2-Methyl-2-{4-[2-(5-methyl-2-phenyl-oxazol-4-yl)-ethoxy]-phenoxy}-3-phenyl-propionic acid | IC50 | 678.0 [1], 680.0 [2] |
![](https://images.aatbio.com/dataset/ic50/peroxisome-proliferator-activated-receptor-alpha_466025246c4c2d204e96b6678df0c533.svg) | (2R)-2-Methyl-3-[4-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl]-2-phenoxypropanoic acid | IC50 | 1545.25 [1], 1546.0 [2] |
![](https://images.aatbio.com/dataset/ic50/peroxisome-proliferator-activated-receptor-alpha_c7401f0cad421127f6a699f1316fe28e.svg) | (R)-3-(4-(3-(2-Benzoyl-4-ethylphenoxy)butoxy)-2-methylphenyl)propanoic acid | IC50 | 4257.0 [1] |
![](https://images.aatbio.com/dataset/ic50/peroxisome-proliferator-activated-receptor-alpha_6741916ec0ffbe7b9094a90fb9dbbf57.svg) | (S)-3-{4-[2-(5-Methyl-2-phenyl-oxazol-4-yl)-ethoxy]-phenyl}-2-pyrrol-1-yl-propionic acid | IC50 | 697.0 [1] |
![](https://images.aatbio.com/dataset/ic50/peroxisome-proliferator-activated-receptor-alpha_6741916ec0ffbe7b9094a90fb9dbbf57.svg) | (S)-3-{4-[2-(5-Methyl-2-phenyl-oxazol-4-yl)-ethoxy]-phenyl}-2-pyrrol-1-yl-propionic acid | Ki | 560.0 [1] |
![](https://images.aatbio.com/dataset/ic50/peroxisome-proliferator-activated-receptor-alpha_d8855eab1fc786a760a2efa7c6c16311.svg) | 2-[3-[2-[[Cyclopropanecarbonyl(ethyl)amino]methyl]-4-(6-ethoxypyridin-3-yl)phenyl]-4-methoxyphenyl]acetic acid | IC50 | 250000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/peroxisome-proliferator-activated-receptor-alpha_a16d649a1f71d4918aafff4db968f9dd.svg) | Arachidonic acid | IC50 | 1200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/peroxisome-proliferator-activated-receptor-alpha_edbdf21aebcb7609b93378bfd38b4072.svg) | Oleic acid | IC50 | 600.0 [1] |
![](https://images.aatbio.com/dataset/ic50/peroxisome-proliferator-activated-receptor-alpha_fb032a9524e407c27b6318fb40a37503.svg) | Linoleic acid | IC50 | 1100.0 [1] |
![](https://images.aatbio.com/dataset/ic50/peroxisome-proliferator-activated-receptor-alpha_fcb134416d1d6bfbb104b783c370b009.svg) | Eicosapentaenoic acid | IC50 | 1100.0 [1] |
![](https://images.aatbio.com/dataset/ic50/peroxisome-proliferator-activated-receptor-alpha_637c0cd22ea54919094e88b6070c5665.svg) | Linolenic acid | IC50 | 1200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/peroxisome-proliferator-activated-receptor-alpha_59247e969f873dd9bb0acfdb506a2d9c.svg) | Dihomo-gamma-linolenic acid | IC50 | 1400.0 [1] |
![](https://images.aatbio.com/dataset/ic50/peroxisome-proliferator-activated-receptor-alpha_ba70d60ff21c7329a3800eef4aa21a00.svg) | Pirinixic acid | IC50 | 10110.0 [1], 36300.0 [2] |
![](https://images.aatbio.com/dataset/ic50/peroxisome-proliferator-activated-receptor-alpha_b8e655e36944d4874d04dc97fc7b1b55.svg) | gamma-Linolenic acid | IC50 | 270.0 [1] |
![](https://images.aatbio.com/dataset/ic50/peroxisome-proliferator-activated-receptor-alpha_946ab26ca5195a11909dd213deedcf09.svg) | Palmitoleic acid | IC50 | 1700.0 [1] |
![](https://images.aatbio.com/dataset/ic50/peroxisome-proliferator-activated-receptor-alpha_6761c94e1af0b9bcc1a2008bf25c1fd5.svg) | Muraglitazar | IC50 | 190.0 [1], 250.0 [2] |
![](https://images.aatbio.com/dataset/ic50/peroxisome-proliferator-activated-receptor-alpha_b62696cb8f1e3dee221a92314df5a62b.svg) | Erucic acid | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/peroxisome-proliferator-activated-receptor-alpha_85eae0074a1e33ccdf892e730891b099.svg) | GW7647 | IC50 | 0.46 [1] |
![](https://images.aatbio.com/dataset/ic50/peroxisome-proliferator-activated-receptor-alpha_85eae0074a1e33ccdf892e730891b099.svg) | GW7647 | Ki | 0.05 [1] |
![](https://images.aatbio.com/dataset/ic50/peroxisome-proliferator-activated-receptor-alpha_ef7a72d98f4717d81d508690e85597cd.svg) | Tesaglitazar | IC50 | 3800.0 [1] |
![](https://images.aatbio.com/dataset/ic50/peroxisome-proliferator-activated-receptor-alpha_ef7a72d98f4717d81d508690e85597cd.svg) | Tesaglitazar | Ki | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/peroxisome-proliferator-activated-receptor-alpha_141e0d0cc895ed114cd0a27b7f852066.svg) | Ragaglitazar | IC50 | 980.0 [1] |
![](https://images.aatbio.com/dataset/ic50/peroxisome-proliferator-activated-receptor-alpha_141e0d0cc895ed114cd0a27b7f852066.svg) | Ragaglitazar | Ki | 980.0 [1] |
![](https://images.aatbio.com/dataset/ic50/peroxisome-proliferator-activated-receptor-alpha_ba977d4dcd8ecefee03f9e57f2048777.svg) | 5-((2,4-Dioxo-5-thiazolidinyl)methyl)-2-methoxy-N-((4-(trifluoromethyl)phenyl)methyl)benzamide | IC50 | 914.0 [1] |
![](https://images.aatbio.com/dataset/ic50/peroxisome-proliferator-activated-receptor-alpha_ba977d4dcd8ecefee03f9e57f2048777.svg) | 5-((2,4-Dioxo-5-thiazolidinyl)methyl)-2-methoxy-N-((4-(trifluoromethyl)phenyl)methyl)benzamide | Ki | 230.0 [1] |
![](https://images.aatbio.com/dataset/ic50/peroxisome-proliferator-activated-receptor-alpha_de71a3aa6943bcc015c5c2225b309ed9.svg) | LY-518674 | IC50 | 23.99 [1], 24.0 [2] |
![](https://images.aatbio.com/dataset/ic50/peroxisome-proliferator-activated-receptor-alpha_44ab4f38c19ea27223223e749e193c65.svg) | Naveglitazar | IC50 | 2710.19 [1], 2711.0 [2] |
![](https://images.aatbio.com/dataset/ic50/peroxisome-proliferator-activated-receptor-alpha_080138ed28375f2f72ae1e8524bbfbf7.svg) | Benzeneacetic acid, 3-chloro-4-((3-((3-phenyl-7-propyl-6-benzofuranyl)oxy)propyl)thio)- | IC50 | 53.95 [1], 54.0 [2] |
![](https://images.aatbio.com/dataset/ic50/peroxisome-proliferator-activated-receptor-alpha_4e46db8f9f161f75023b6297fbae4165.svg) | CID 9890319 | IC50 | 174.0 [1] |
![](https://images.aatbio.com/dataset/ic50/peroxisome-proliferator-activated-receptor-alpha_4e46db8f9f161f75023b6297fbae4165.svg) | CID 9890319 | Ki | 170.0 [1] |
![](https://images.aatbio.com/dataset/ic50/peroxisome-proliferator-activated-receptor-alpha_5b3d8dcb3afe298fdfab33dec2702b3f.svg) | (2S)-2-Methyl-3-[4-[2-(5-methyl-2-thiophen-2-yl-1,3-oxazol-4-yl)ethoxy]phenyl]-2-phenoxypropanoic acid | IC50 | 28.0 [1] |
![](https://images.aatbio.com/dataset/ic50/peroxisome-proliferator-activated-receptor-alpha_64678f8de19632509f726c56457de37d.svg) | CID 9889841 | IC50 | 570.0 [1], 570.16 [2] |
![](https://images.aatbio.com/dataset/ic50/peroxisome-proliferator-activated-receptor-alpha_82c598d3b2db149ab88ed4435573cc90.svg) | 2-Methyl-3-[4-[2-(5-methyl-2-thiophen-2-yl-1,3-oxazol-4-yl)ethoxy]phenyl]-2-phenoxypropanoic acid | IC50 | 45.0 [1] |
![](https://images.aatbio.com/dataset/ic50/peroxisome-proliferator-activated-receptor-alpha_82c598d3b2db149ab88ed4435573cc90.svg) | 2-Methyl-3-[4-[2-(5-methyl-2-thiophen-2-yl-1,3-oxazol-4-yl)ethoxy]phenyl]-2-phenoxypropanoic acid | Ki | 4.0 [1] |
![](https://images.aatbio.com/dataset/ic50/peroxisome-proliferator-activated-receptor-alpha_230830782ac7043954839dd225426ca6.svg) | 2-{5-[3-(6-Benzoyl-1-propylnaphthalen-2-yloxy)propoxy]indol-1-YL}ethanoic acid | IC50 | 112.98 [1], 113.0 [2] |
![](https://images.aatbio.com/dataset/ic50/peroxisome-proliferator-activated-receptor-alpha_9e0411d99b7e1fca741170518542c99e.svg) | 4-Methoxy-N-(2,4,6-trimethylphenyl)benzenesulfonamide | IC50 | 25118.86 [1] |
![](https://images.aatbio.com/dataset/ic50/peroxisome-proliferator-activated-receptor-alpha_b45f89156f53d631f2d7ba0d19a25b50.svg) | (2R)-7-(3-(2-Chloro-4-(4-fluorophenoxy)phenoxy)propoxy)-2-ethylchromane-2-carboxylic acid | IC50 | 60.0 [1] |
![](https://images.aatbio.com/dataset/ic50/peroxisome-proliferator-activated-receptor-alpha_e943ef3e09ebceb09db527cf097980ba.svg) | 2-Methyl-2-{4-[2-(5-methyl-2-phenyloxazol-4-yl)ethoxy]phenoxy}propionic Acid | IC50 | 1445.0 [1], 1736.0 [2] |
![](https://images.aatbio.com/dataset/ic50/peroxisome-proliferator-activated-receptor-alpha_e108a3b315f11f394679f4afb3557524.svg) | {3-Chloro-4-[3-(3-hydroxy-4-propionyl-2-propyl-phenoxy)-propylsulfanyl]-phenyl}-acetic acid | IC50 | 599.79 [1], 600.0 [2] |
![](https://images.aatbio.com/dataset/ic50/peroxisome-proliferator-activated-receptor-alpha_8c5687ad78b9e8e8477870d681dd5a05.svg) | 3-[4-[3-[(1R)-1-[(5-Chloro-1,3-dimethylindole-2-carbonyl)amino]ethyl]-5-fluorophenoxy]-2-ethylphenyl]propanoic acid | IC50 | 10256.52 [1], 10257.0 [2] |
![](https://images.aatbio.com/dataset/ic50/peroxisome-proliferator-activated-receptor-alpha_f10c3b86acd5ef4906728f936e43f1cc.svg) | 2-[4-[3-[2-Chloro-4-(4-fluorophenoxy)phenoxy]propoxy]phenoxy]-2-methylpropanoic acid | IC50 | 30.0 [1] |
![](https://images.aatbio.com/dataset/ic50/peroxisome-proliferator-activated-receptor-alpha_2263515c8509463dbef0b10dbed2f0a0.svg) | {4-[3-(4-Acetyl-3-hydroxy-2-propyl-phenoxy)-propylsulfanyl]-3-chloro-phenyl}-acetic acid | IC50 | 7396.05 [1], 7400.0 [2] |
![](https://images.aatbio.com/dataset/ic50/peroxisome-proliferator-activated-receptor-alpha_e83dd943a64f093c68242bfd53cd47d5.svg) | {3-Chloro-4-[3-(3-ethyl-7-propyl-benzofuran-6-yloxy)-propylsulfanyl]-phenyl}-acetic acid | IC50 | 1730.0 [1] |
![](https://images.aatbio.com/dataset/ic50/peroxisome-proliferator-activated-receptor-alpha_1a5e81e4d50f3bc3a245ee176e97a9cf.svg) | 2-{5-[3-(7-Propyl-3-trifluoromethylbenzo[D]isoxazol-6-yloxy)propoxy]indol-1-YL}ethanoic acid | IC50 | 495.45 [1], 496.0 [2] |
![](https://images.aatbio.com/dataset/ic50/peroxisome-proliferator-activated-receptor-alpha_bb56ae6b93156121c41aff0e7e34b439.svg) | (2S)-2-Methoxy-3-{4-[5-(4-phenoxy-phenoxy)-pent-1-ynyl]-phenyl}-propionic acid | IC50 | 769.13 [1], 770.0 [2] |
![](https://images.aatbio.com/dataset/ic50/peroxisome-proliferator-activated-receptor-alpha_214e1e9a45799dfbefa357cc929cd50c.svg) | 2-[4-[3-[1-[(3,4-Dimethylphenyl)methyl]-4-methyl-5-oxo-1,2,4-triazol-3-yl]propyl]phenoxy]-2-methylpropanoic acid | IC50 | 11.99 [1], 12.0 [2] |
![](https://images.aatbio.com/dataset/ic50/peroxisome-proliferator-activated-receptor-alpha_e477ba284cc5f1ee9677c928085ea8d9.svg) | (2R)-7-(3-(2-Chloro-4-cyclopentylphenoxy)propoxy)-2-methylchromane-2-carboxylic Acid | IC50 | 39.99 [1], 40.0 [2] |
![](https://images.aatbio.com/dataset/ic50/peroxisome-proliferator-activated-receptor-alpha_ba2d3ca32b20ccc073646bfcbadb447d.svg) | (S)-2-Ethoxy-3-{4-[3-(4-phenoxy-phenoxy)-propoxy]-phenyl}-propionic acid | IC50 | 1686.0 [1], 1686.55 [2] |
![](https://images.aatbio.com/dataset/ic50/peroxisome-proliferator-activated-receptor-alpha_046976101718a8f77089981314bf5ef7.svg) | 3-{4-[2-(2-Biphenyl-4-yl-5-methyl-oxazol-4-yl)ethoxy]-phenyl}-2-methyl-2-phenoxypropionic acid | IC50 | 503.0 [1] |
![](https://images.aatbio.com/dataset/ic50/peroxisome-proliferator-activated-receptor-alpha_964d21e48bbb8c35a463d423aa5f0ebf.svg) | 3-{4-[2-(2-Biphenyl-3-yl-5-methyl-oxazol-4-yl)ethoxy]-phenyl}-2-methyl-2-phenoxypropionic acid | IC50 | 167.0 [1] |
![](https://images.aatbio.com/dataset/ic50/peroxisome-proliferator-activated-receptor-alpha_5d662ab03dd2d3a5e37b85ab72147344.svg) | (S)-2-Methoxy-3-{4-[4-(4-phenoxy-phenoxy)-but-1-ynyl]-phenyl}-propionic acid | IC50 | 1153.45 [1], 1154.0 [2] |
![](https://images.aatbio.com/dataset/ic50/peroxisome-proliferator-activated-receptor-alpha_de2ac2cab437141b45c9346acce81814.svg) | (R)-7-[3-(2-Chloro-4-isobutyl-phenoxy)-propoxy]-2-methyl-chroman-2-carboxylic acid | IC50 | 16.0 [1] |
![](https://images.aatbio.com/dataset/ic50/peroxisome-proliferator-activated-receptor-alpha_55a815b159f098e3597df2a03b4ea720.svg) | 2-[4-[3-[1-[(4-Tert-butylphenyl)methyl]-4-methyl-5-oxo-1,2,4-triazol-3-yl]propyl]phenoxy]-2-methylpropanoic acid | IC50 | 15.0 [1] |
![](https://images.aatbio.com/dataset/ic50/peroxisome-proliferator-activated-receptor-alpha_c4ad20a6169379c8f4032ae1f9007c23.svg) | 2-(4-(4-(4-(Trifluoromethyl)benzyloxy)benzylthio)-5-methoxy-2-methylphenoxy)acetic acid | IC50 | 4.7 [1] |
![](https://images.aatbio.com/dataset/ic50/peroxisome-proliferator-activated-receptor-alpha_47ce909c2326f4765c60cba9a390d549.svg) | 2-[4-[3-[1-[(3-Methoxyphenyl)methyl]-5-oxo-4-propyl-1,2,4-triazol-3-yl]propyl]phenoxy]-2-methylpropanoic acid | IC50 | 19.0 [1], 19.01 [2] |
![](https://images.aatbio.com/dataset/ic50/peroxisome-proliferator-activated-receptor-alpha_373613e6ed91c22c3bfcd721b8db92a5.svg) | (R)-7-[3-(2-Chloro-4-trifluoromethyl-phenoxy)-propoxy]-2-ethyl-chroman-2-carboxylic acid | IC50 | 89.95 [1], 90.0 [2] |
![](https://images.aatbio.com/dataset/ic50/peroxisome-proliferator-activated-receptor-alpha_5eb88a4d9d8f538c540f222b2cd6de13.svg) | (S)-3-{4-[3-(Biphenyl-4-yloxy)-propoxy]-phenyl}-2-methoxy-propionic acid | IC50 | 567.54 [1], 568.0 [2] |
![](https://images.aatbio.com/dataset/ic50/peroxisome-proliferator-activated-receptor-alpha_3b5f77cab79541a7375a5d5993e685cc.svg) | (S)-3-{4-[3-(4-Benzoyl-phenoxy)-propoxy]-phenyl}-2-methoxy-propionic acid | IC50 | 469.89 [1], 470.0 [2] |
![](https://images.aatbio.com/dataset/ic50/peroxisome-proliferator-activated-receptor-alpha_2fa743d0c852be55efc70f2c9abe45da.svg) | (S)-2-Methoxy-3-{3-methoxy-4-[3-(4-phenoxy-phenoxy)-propoxy]-phenyl}-propionic acid | IC50 | 1349.0 [1] |
![](https://images.aatbio.com/dataset/ic50/peroxisome-proliferator-activated-receptor-alpha_93fa17ea759b6c248420f3988fccdc65.svg) | 3-[2-Ethyl-4-[(3R)-3-(4-ethyl-2-pyridin-2-ylphenoxy)butoxy]phenyl]propanoic acid | IC50 | 7345.14 [1], 7350.0 [2] |
![](https://images.aatbio.com/dataset/ic50/peroxisome-proliferator-activated-receptor-alpha_b4d47ccbf607a2a2c58fdb37f874f198.svg) | 3-[4-[(3R)-3-(4-Ethyl-2-pyridin-2-ylphenoxy)butoxy]-2-methylphenyl]propanoic acid | IC50 | 8290.0 [1], 8298.51 [2] |
![](https://images.aatbio.com/dataset/ic50/peroxisome-proliferator-activated-receptor-alpha_dca1d12844cbe906c38d15fa28fd6ce2.svg) | (2S)-3-[4-[2-(2-Cyclohexyl-5-methyl-1,3-oxazol-4-yl)ethoxy]phenyl]-2-methyl-2-phenoxypropanoic acid | IC50 | 17.99 [1], 18.0 [2] |
![](https://images.aatbio.com/dataset/ic50/peroxisome-proliferator-activated-receptor-alpha_121f20ca19eb3180b3b402ff5b79bfbf.svg) | 3-[4-[(3R)-3-[4-Ethyl-2-(1,3-oxazol-2-yl)phenoxy]butoxy]-2-methylphenyl]propanoic acid | IC50 | 10399.2 [1], 10400.0 [2] |
![](https://images.aatbio.com/dataset/ic50/peroxisome-proliferator-activated-receptor-alpha_030c5bbffed02a0a0810c7f4bc052892.svg) | 2-[5-[3-(6-Benzoylnaphthalen-2-yl)oxypropoxy]indol-1-yl]acetic acid | IC50 | 484.0 [1], 484.17 [2] |
![](https://images.aatbio.com/dataset/ic50/peroxisome-proliferator-activated-receptor-alpha_604d45f19cdc13229196b130f4ffd427.svg) | 2-[4-[3-[[[2-Fluoro-4-(trifluoromethyl)benzoyl]amino]methyl]-5-methylphenoxy]-2-methylphenoxy]-2-methylpropanoic acid | IC50 | 313.0 [1], 313.33 [2] |
![](https://images.aatbio.com/dataset/ic50/peroxisome-proliferator-activated-receptor-alpha_7b9938185fed2cf63fe05a1a3d945ba1.svg) | 2-(6-(3-(4-(4-Fluorobenzoyl)-2-propylphenoxy)propoxy)-1H-indol-1-yl)acetic acid | IC50 | 1047.0 [1], 1047.13 [2] |
![](https://images.aatbio.com/dataset/ic50/peroxisome-proliferator-activated-receptor-alpha_99407355fee4f6a2e82bcbbc57d28e0f.svg) | 2-[4-[3-[4-(2-Hydroxyethyl)-1-[(4-methylphenyl)methyl]-5-oxo-1,2,4-triazol-3-yl]propyl]phenoxy]-2-methylpropanoic acid | IC50 | 26.98 [1], 27.0 [2] |
![](https://images.aatbio.com/dataset/ic50/peroxisome-proliferator-activated-receptor-alpha_2cb9d4d2eedab9d9e304825fec433c70.svg) | 2-Methyl-2-[2-methyl-4-[3-[[[2-methyl-4-(trifluoromethyl)benzoyl]amino]methyl]phenoxy]phenoxy]propanoic acid | IC50 | 1761.98 [1], 1763.0 [2] |
![](https://images.aatbio.com/dataset/ic50/peroxisome-proliferator-activated-receptor-alpha_c204d546e7514a9d07add72ba86fc27c.svg) | 2-[4-[3-[1-(Cyclohexylmethyl)-5-oxo-4-propyl-1,2,4-triazol-3-yl]propyl]phenoxy]-2-methylpropanoic acid | IC50 | 250.0 [1], 250.03 [2] |
![](https://images.aatbio.com/dataset/ic50/peroxisome-proliferator-activated-receptor-alpha_e5c0ef830c001552f2cb0f029f54fd71.svg) | 3-[2-Ethyl-4-[(3R)-3-[2-pyridin-2-yl-4-(trifluoromethyl)phenoxy]butoxy]phenyl]propanoic acid | IC50 | 6090.0 [1], 6095.37 [2] |
![](https://images.aatbio.com/dataset/ic50/peroxisome-proliferator-activated-receptor-alpha_9d5a14fa7a7a8a39457fc59afd3d5e15.svg) | (2R)-2-Methyl-3-[4-[2-(5-methyl-2-thiophen-2-yl-1,3-oxazol-4-yl)ethoxy]phenyl]-2-phenoxypropanoic acid | IC50 | 618.0 [1], 618.02 [2] |
![](https://images.aatbio.com/dataset/ic50/peroxisome-proliferator-activated-receptor-alpha_2f9ca5fda6f65db4ee25815fe6c1d4ab.svg) | 3-(1-(3-(7-Propyl-3-(trifluoromethyl)benzo[d]isoxazol-6-yloxy)propyl)-1H-indol-5-yl)propanoic acid | IC50 | 449.78 [1], 450.0 [2] |
![](https://images.aatbio.com/dataset/ic50/peroxisome-proliferator-activated-receptor-alpha_1a3875fc6561b1fdeb93e80f169fea37.svg) | 2-(4-(3-(6-Benzoyl-1-propylnaphthalen-2-yloxy)propoxy)-1H-indol-1-yl)acetic acid | IC50 | 578.0 [1], 578.1 [2] |
![](https://images.aatbio.com/dataset/ic50/peroxisome-proliferator-activated-receptor-alpha_6e3d3e4ed17bbdd05689e75776d00c89.svg) | 2-(6-(3-(6-Benzoylnaphthalen-2-yloxy)propoxy)-1H-indol-1-yl)acetic acid | IC50 | 4486.0 [1], 4487.45 [2] |
![](https://images.aatbio.com/dataset/ic50/peroxisome-proliferator-activated-receptor-alpha_59c182515bd94155974ee6fc19892283.svg) | 2-(5-(3-(4-(4-Fluorobenzoyl)-2-propylphenoxy)propoxy)-1H-indol-1-yl)acetic acid | IC50 | 469.89 [1], 470.0 [2] |
![](https://images.aatbio.com/dataset/ic50/peroxisome-proliferator-activated-receptor-alpha_ec17412f339dfa3b1c8f30cc09afaaf1.svg) | 2-(6-(3-(4-(4-Fluorobenzoyl)phenoxy)propoxy)-1H-indol-1-yl)acetic acid | IC50 | 115.88 [1], 116.0 [2] |
![](https://images.aatbio.com/dataset/ic50/peroxisome-proliferator-activated-receptor-alpha_2f9ff7233fee13b2a6dad4f60a503676.svg) | 2-(1-(3-(7-Propyl-3-(trifluoromethyl)benzo[d]isoxazol-6-yloxy)propyl)-1H-indol-5-yl)acetic acid | IC50 | 400.0 [1] |
![](https://images.aatbio.com/dataset/ic50/peroxisome-proliferator-activated-receptor-alpha_508cf86550f54e08e753cf94d6008f94.svg) | 2-(6-(3-(6-Benzoyl-1-propylnaphthalen-2-yloxy)propoxy)-1H-indol-1-yl)acetic acid | IC50 | 4486.0 [1], 4487.45 [2] |
![](https://images.aatbio.com/dataset/ic50/peroxisome-proliferator-activated-receptor-alpha_ea2ee1f3ece051f370081f3ca1c0c020.svg) | 2-(4-(3-(4-(4-Fluorobenzoyl)-2-propylphenoxy)propoxy)-1H-indol-1-yl)acetic acid | IC50 | 414.0 [1] |
![](https://images.aatbio.com/dataset/ic50/peroxisome-proliferator-activated-receptor-alpha_128b1a5625a2ebd341ee5926de09182f.svg) | 3-[4-[(3R)-3-[4-Ethyl-2-(1,3-thiazol-4-yl)phenoxy]butoxy]-2-methylphenyl]propanoic acid | IC50 | 4100.0 [1], 4102.04 [2] |
![](https://images.aatbio.com/dataset/ic50/peroxisome-proliferator-activated-receptor-alpha_44a9bfe78d1b4cdacbfef6172d7562b9.svg) | 4-[({1-[(E)-{[4-(Morpholin-4-yl)phenyl]imino}methyl]naphthalen-2-yl}oxy)methyl]benzoic acid | IC50 | 42953.64 [1], 43000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/peroxisome-proliferator-activated-receptor-alpha_a433e14bf1588fa8e8a2118ee4b5b113.svg) | (R)-3-{4-[3-(4-Ethyl-2-phenoxy-phenoxy)-butoxy]-2-methyl-phenyl}-propionic acid | IC50 | 3758.0 [1], 3758.37 [2] |
![](https://images.aatbio.com/dataset/ic50/peroxisome-proliferator-activated-receptor-alpha_134f5c7890b0de64a76af987d1542871.svg) | (R)-3-{2-Methyl-4-[3-(2-phenoxy-4-trifluoromethoxy-phenoxy)-butoxy]-phenyl}-propionic acid | IC50 | 897.0 [1], 897.43 [2] |
![](https://images.aatbio.com/dataset/ic50/peroxisome-proliferator-activated-receptor-alpha_f4a82b09cdf34f849d21cfd09a8ee681.svg) | (R)-3-{4-[3-(4-Chloro-2-phenoxy-phenoxy)-butoxy]-2-trifluoromethyl-phenyl}-propionic acid | IC50 | 4385.31 [1], 4386.0 [2] |
![](https://images.aatbio.com/dataset/ic50/peroxisome-proliferator-activated-receptor-alpha_68cbd9bf90c68dea5e743e9f9858f82d.svg) | 2-(4-(3-(2-Benzoyl-4-ethylphenoxy)propoxy)phenoxy)-2-methylpropanoic acid | IC50 | 1398.0 [1], 1399.59 [2] |
![](https://images.aatbio.com/dataset/ic50/peroxisome-proliferator-activated-receptor-alpha_ab780977de368d75d3bcafed08810242.svg) | (R)-3-{4-[3-(4-Chloro-2-phenoxy-phenoxy)-butoxy]-2-methyl-phenyl}-propionic acid | IC50 | 5303.0 [1], 5308.84 [2] |
![](https://images.aatbio.com/dataset/ic50/peroxisome-proliferator-activated-receptor-alpha_54a676751d973fe4f4f8103b94adc6f0.svg) | (R)-3-{2-Methyl-4-[3-(2-phenoxy-4-trifluoromethyl-phenoxy)-butoxy]-phenyl}-propionic acid | IC50 | 1037.0 [1], 1037.53 [2] |