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Peregrin Inhibitors (IC50, Ki)

Structure
▲
▼
Compound Name
▲
▼
Standard Type
▲
▼
Standard Values (in nM)
▲
▼
CID 40642506IC5040.0 [1], 50.12 [2]
CID 122705990IC502280.0 [1], 3150.0 [2], 10000.0 [3]
CID 91827373IC503.1 [1], 70.0 [2], 114.0 [3]
4-Cyano-N-(1,3-dimethyl-2-oxoquinolin-6-yl)benzenesulfonamideIC507.9 [1], 140.0 [2]
N-[1,3-Dimethyl-6-[(2R)-2-methylpiperazin-1-yl]-2-oxobenzimidazol-5-yl]-2-methoxybenzamideIC502.51 [1], 7.94 [2], 19.95 [3]
4-Cyano-N-(1,3-diethyl-2-oxoquinolin-6-yl)benzenesulfonamideIC5020000.0 [1], 100000.0 [2]
6-(3-Hydroxypropyl)-2-(1-methyl-2-oxo-3H-benzimidazol-5-yl)benzo[de]isoquinoline-1,3-dioneIC5010000.0 [1], 20000.0 [2]
CID 15990224IC5079.43 [1], 1000.0 [2]
4-Cyano-N-(3-ethyl-1-methyl-2-oxoquinolin-6-yl)benzenesulfonamideIC50180.0 [1]
4-Cyano-N-(1-methyl-2-oxoquinolin-6-yl)benzenesulfonamideIC5043.0 [1]
3-Cyano-N-(1-methyl-2-oxoquinolin-6-yl)benzenesulfonamideIC5056.0 [1]
2-Cyano-N-(1-methyl-2-oxoquinolin-6-yl)benzenesulfonamideIC50430.0 [1]
N-[1,3-Dimethyl-6-[(2R)-2-methylpiperazin-1-yl]-2-oxobenzimidazol-5-yl]-N-ethyl-2-methoxybenzamideIC501000.0 [1], 3981.07 [2]
N-(1-Methyl-2-oxoquinolin-6-yl)benzenesulfonamideIC5065.0 [1]
2-Methoxy-N-(1,3,6-trimethyl-2-oxobenzimidazol-5-yl)benzamideIC501584.89 [1]
2-Methoxy-N-(6-methoxy-1,3-dimethyl-2-oxobenzimidazol-5-yl)benzamideIC50125.89 [1]
N-(1,3-Dimethyl-2-oxoquinolin-6-yl)-2-methoxybenzenesulfonamideIC509.0 [1]
2-(1,3,6-Trimethyl-2-Oxidanylidene-Benzimidazol-5-Yl)benzo[de]isoquinoline-1,3-DioneIC501550.0 [1], 10000.0 [2]
2-(6-Methoxy-1,3-dimethyl-2-oxobenzimidazol-5-yl)benzo[de]isoquinoline-1,3-dioneIC501150.0 [1], 10000.0 [2]
1-Methyl-2-quinoloneIC504800.0 [1]
4-[(2s,4r)-1-Acetyl-4-[(4-Chlorophenyl)amino]-2-Methyl-1,2,3,4-Tetrahydroquinolin-6-Yl]benzoic AcidIC503.98 [1]
N-(1,3-Dimethyl-2-oxo-2,3-dihydro-1H-benzimidazol-5-yl)-2,4-dimethylbenzenesulfonamideIC50199.53 [1]
1,3-Dimethyl-2-oxo-2,3-dihydro-1H-benzimidazole-5-carboxamideIC5010000.0 [1]
N-(1,3-Dimethyl-2-oxo-2,3-dihydro-1H-benzoimidazol-5-yl)-3-methoxy-benzamideIC503162.28 [1]
N-(1,3-Dimethyl-6-morpholin-4-yl-2-oxobenzimidazol-5-yl)-3-methoxybenzamideIC50630.96 [1]
N-(1,3-Dimethyl-2-oxo-6-pyrrolidin-1-ylbenzimidazol-5-yl)-3-methoxybenzamideIC50316.23 [1]
N-(1,3-Dimethyl-2-oxo-6-piperidin-1-ylbenzimidazol-5-yl)benzamideIC50100.0 [1]
N-(1,3-Dimethyl-2-oxo-2,3-dihydro-1H-benzimidazol-5-yl)-5,6,7,8-tetrahydro-2-naphthalenesulfonamideIC50330.0 [1]
N-(1,3-Dimethyl-2-oxo-2,3-dihydro-1H-benzoimidazol-5-yl)-2-methoxy-benzamideIC502511.89 [1]
3-[7-(Difluoromethyl)-6-(1-methylpyrazol-4-yl)-3,4-dihydro-2H-quinolin-1-yl]-N-methyl-1-(oxan-4-yl)-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-5-carboxamideIC504600.0 [1]
CID 35397514IC50270.0 [1]
N-(1,3-Dimethyl-2-oxo-6-piperidin-1-ylbenzimidazol-5-yl)-2,2-dimethylpropanamideIC50630.96 [1]
N-(1,3-Dimethyl-2-oxo-6-piperidin-1-ylbenzimidazol-5-yl)-2-methylbenzamideIC50316.23 [1]
N-(1,3-Dimethyl-6-morpholin-4-yl-2-oxobenzimidazol-5-yl)-2-methoxybenzamideIC50125.89 [1]
N-(1,4-Dimethyl-7-morpholin-4-yl-2,3-dioxoquinoxalin-6-yl)-4-(2-methylpropyl)benzenesulfonamideIC501900.0 [1]
N-[4-[(1,4-Dimethyl-7-morpholin-4-yl-2,3-dioxoquinoxalin-6-yl)sulfamoyl]phenyl]-3-methylbutanamideIC502000.0 [1]
N-(1,4-Dimethyl-2,3-dioxo-7-pyrrolidin-1-ylquinoxalin-6-yl)-2-methoxybenzamideIC5027000.0 [1]
N-[6-(4-Methoxyphenoxy)-1,3-Dimethyl-2-Oxo-2,3-Dihydro-1h-Benzimidazol-5-Yl]benzenesulfonamideIC50660.0 [1]
3,4-Dimethoxy-N-[6-(4-methoxyphenoxy)-1,3-dimethyl-2-oxobenzimidazol-5-yl]benzenesulfonamideIC50340.0 [1]
1-(3-Phenylazanyl-1,4,6,7-Tetrahydropyrazolo[4,3-C]pyridin-5-Yl)ethanoneIC5020000.0 [1]
6-Amino-1-Methylquinolin-2(1h)-OneIC502100.0 [1]
2-Methoxy-N-(1-methyl-2-oxo-6-piperidin-1-yl-3H-benzimidazol-5-yl)benzamideIC50630.96 [1]
2-Methoxy-N-(3-methyl-2-oxo-6-piperidin-1-yl-1H-benzimidazol-5-yl)benzamideIC5019952.62 [1]
4-Cyano-N-(3-ethyl-1-methyl-2-oxoquinolin-6-yl)-2-methoxybenzenesulfonamideIC5093.0 [1]
4-Cyano-N-methyl-N-(1-methyl-2-oxoquinolin-6-yl)benzenesulfonamideIC50910.0 [1]
N-(1-Methyl-2-oxoquinolin-6-yl)ethanesulfonamideIC501200.0 [1]
4-Cyano-2-methoxy-N-(7-methoxy-1,3-dimethyl-2-oxoquinolin-6-yl)benzenesulfonamideIC5012.0 [1]
N-(1-Methyl-2-oxoquinolin-6-yl)methanesulfonamideIC502200.0 [1]
N-(1-Methyl-2-oxoquinolin-6-yl)cyclopropanesulfonamideIC50520.0 [1]
4-Cyano-N-(7-methoxy-1-methyl-2-oxoquinolin-6-yl)-N-methylbenzenesulfonamideIC501000.0 [1]
N-(1-Methyl-2-oxoquinolin-6-yl)cyclohexanesulfonamideIC50380.0 [1]
3-Chloro-4-cyano-N-(1-methyl-2-oxoquinolin-6-yl)benzenesulfonamideIC5062.0 [1]
4-Cyano-N-(1-ethyl-3-methyl-2-oxoquinolin-6-yl)benzenesulfonamideIC5015.0 [1]
N-(1-Methyl-2-oxoquinolin-6-yl)propane-2-sulfonamideIC501100.0 [1]
4-Cyano-N-(8-fluoro-1,3-dimethyl-2-oxoquinolin-6-yl)-2-methoxybenzenesulfonamideIC5012.0 [1]
4-Cyano-N-(1-methyl-2-oxo-7-propan-2-yloxyquinolin-6-yl)benzenesulfonamideIC5039.0 [1]
4-Cyano-N-(7-ethoxy-1-methyl-2-oxoquinolin-6-yl)benzenesulfonamideIC5055.0 [1]
4-Cyano-N-(1,3-dimethyl-2-oxoquinolin-6-yl)-2-methoxy-N-methylbenzenesulfonamideIC5052.0 [1]
3,4-Dichloro-N-(1-methyl-2-oxoquinolin-6-yl)benzenesulfonamideIC5044.0 [1]
4-Cyano-N-(7-methoxy-1-methyl-2-oxoquinolin-6-yl)benzenesulfonamideIC5053.0 [1]
N-(7-Methoxy-1-methyl-2-oxoquinolin-6-yl)benzenesulfonamideIC5029.0 [1]
N-(4-Cyanophenyl)-1-methyl-2-oxoquinoline-6-sulfonamideIC50100.0 [1]
4-Cyano-N-(7-methoxy-1,3-dimethyl-2-oxoquinolin-6-yl)benzenesulfonamideIC5015.0 [1]
N-(7-Methoxy-1,3-dimethyl-2-oxoquinolin-6-yl)benzenesulfonamideIC5017.0 [1]
4-Cyano-N-(7-Methoxy-1,4-Dimethyl-2-Oxo-1,2-Dihydroquinolin-6-Yl)benzene-1-SulfonamideIC5060.0 [1]
4-Cyano-N-(1,4-dimethyl-2-oxoquinolin-6-yl)benzenesulfonamideIC5024.0 [1]
1-[3-[7-(Difluoromethyl)-6-(1-methylpyrazol-4-yl)-3,4-dihydro-2H-quinolin-1-yl]-1-(oxan-4-yl)-6,7-dihydro-4H-pyrazolo[4,3-c]pyridin-5-yl]ethanoneIC5020000.0 [1]
1-[3-[2-Fluoro-4-(1-methylpyrazol-4-yl)anilino]-1-[(3R)-oxolan-3-yl]-6,7-dihydro-4H-pyrazolo[4,3-c]pyridin-5-yl]ethanoneIC5020000.0 [1]
3-Ethyl-N-[4-(piperidin-1-ylmethyl)-1,3-thiazol-2-yl]pyridine-4-carboxamideIC50515000.0 [1]
7-Oxo-N-[4-(piperidin-1-ylmethyl)-1,3-thiazol-2-yl]azepane-2-carboxamideIC50293000.0 [1]
8-[[(3R,4R)-3-[(1,1-Dioxothian-4-yl)methoxy]-1-methylpiperidin-4-yl]amino]-3-methyl-5-(5-methylpyridin-3-yl)-1H-1,7-naphthyridin-2-oneKi5011.87 [1]
N-(1,3-Dimethyl-2-oxobenzimidazol-5-yl)-2,2-dimethyl-3,4-dihydrochromene-6-sulfonamideIC50310.0 [1]
(2S)-N-(1,3-Dimethyl-2-oxobenzimidazol-5-yl)-2,3-dimethoxy-2,3-dimethyl-1,4-benzodioxine-6-sulfonamideIC501400.0 [1]
N-(1,3-Dimethyl-2-oxobenzimidazol-5-yl)-3,4-dihydro-2H-chromene-6-sulfonamideIC50270.0 [1]
N-(1,3-Dimethyl-2-oxo-6-phenoxybenzimidazol-5-yl)-2-methylbenzenesulfonamideIC50430.0 [1]
N-(1,3-Dimethyl-2-oxo-6-phenoxybenzimidazol-5-yl)-3-methoxybenzenesulfonamideIC50430.0 [1]
N-(1,3-Dimethyl-2-oxo-6-phenoxybenzimidazol-5-yl)-5,6,7,8-tetrahydronaphthalene-2-sulfonamideIC502680.0 [1]
N-(1,3-Dimethyl-2-oxo-6-propan-2-yloxybenzimidazol-5-yl)pyridine-4-carboxamideIC50794.33 [1]
N-[1,3-Dimethyl-6-[(3S)-3-methylpiperazin-1-yl]-2-oxobenzimidazol-5-yl]-2-methoxybenzamideIC5079.43 [1]
2-[2-(Dimethylamino)ethoxy]-N-(1,3-dimethyl-2-oxo-6-propan-2-yloxybenzimidazol-5-yl)benzamideIC50316.23 [1]
N-(1,3-Dimethyl-2-oxo-6-propan-2-yloxybenzimidazol-5-yl)pyridine-2-carboxamideIC5063.1 [1]
N-(1,3-Dimethyl-2-oxo-6-propan-2-yloxybenzimidazol-5-yl)pyridine-3-carboxamideIC501258.93 [1]
N-(1,3-Dimethyl-2-oxo-6-propan-2-yloxybenzimidazol-5-yl)pyrimidine-4-carboxamideIC50125.89 [1]
N-(1,3-Dimethyl-2-oxo-6-propan-2-yloxybenzimidazol-5-yl)-2-methoxypyridine-3-carboxamideIC5031.62 [1]
N-(1,3-Dimethyl-2-oxo-6-piperidin-4-ylbenzimidazol-5-yl)-2-methoxybenzamideIC503162.28 [1]
N-[1,3-Dimethyl-2-oxo-6-(1,2,3,6-tetrahydropyridin-4-yl)benzimidazol-5-yl]-2-methoxybenzamideIC501258.93 [1]
N-[1,3-Dimethyl-6-[(2R)-2-methylpyrrolidin-1-yl]-2-oxobenzimidazol-5-yl]-2-methoxybenzamideIC505.01 [1]
N-[1,3-Dimethyl-6-[(2S)-2-methylpyrrolidin-1-yl]-2-oxobenzimidazol-5-yl]-2-methoxybenzamideIC5015.85 [1]
N-[1,3-Dimethyl-6-[(2S)-2-methylpiperazin-1-yl]-2-oxobenzimidazol-5-yl]-2-methoxybenzamideIC50125.89 [1]
N-[1,3-Dimethyl-6-[(3R)-3-methylpiperazin-1-yl]-2-oxobenzimidazol-5-yl]-2-methoxybenzamideIC50125.89 [1]
N-(1,3-Dimethyl-2-oxo-6-propan-2-yloxybenzimidazol-5-yl)-3-methoxypyridine-2-carboxamideIC50100.0 [1]
N-(1,3-Dimethyl-2-oxo-6-propan-2-yloxybenzimidazol-5-yl)-2,6-dimethoxybenzamideIC501995.26 [1]
N-[3-(2-Hydroxyethyl)-1-methyl-2-oxo-6-propan-2-yloxybenzimidazol-5-yl]-2-methoxybenzamideIC501258.93 [1]
N-(1,3-Dimethyl-2-oxo-6-piperazin-1-ylbenzimidazol-5-yl)-2-methoxybenzamideIC5079.43 [1]
2-[2-(Dimethylamino)-2-oxoethoxy]-N-(1,3-dimethyl-2-oxo-6-propan-2-yloxybenzimidazol-5-yl)benzamideIC50100.0 [1]
N-(1,3-Dimethyl-2-oxo-6-propan-2-yloxybenzimidazol-5-yl)-2-(1-methylpyrrolidin-3-yl)oxybenzamideIC50316.23 [1]
N-(1,3-Dimethyl-2-oxo-6-propan-2-yloxybenzimidazol-5-yl)acetamideIC501000.0 [1]
N-(1,3-Dimethyl-2-oxo-6-propan-2-yloxybenzimidazol-5-yl)butanamideIC501258.93 [1]
N-(1,3-Dimethyl-2-oxo-6-propan-2-yloxybenzimidazol-5-yl)pyrrolidine-3-carboxamideIC50794.33 [1]
N-(1,3-Dimethyl-2-oxo-6-propan-2-yloxybenzimidazol-5-yl)oxane-4-carboxamideIC501584.89 [1]
Items per page: 1 - 10 of 100
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References

This online tool may be cited as follows

MLA

"Quest Database™ Peregrin Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 22 Feb. 2025, https://www.aatbio.com/data-sets/peregrin-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2025, February 22). Quest Database™ Peregrin Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/peregrin-inhibitors-ic50-ki.
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