 | Juglone | IC50 | 5900.0 [1], 10030.0 [2], 10120.0 [3], 10810.0 [4] |
 | Cyclic crypeveic | IC50 | 500.0 [1] |
 | Cyclic crypeveic | Ki | 200.0 [1], 520.0 [2] |
 | [(2R)-2-(1-Benzothiophene-2-carbonylamino)-3-(3-fluorophenyl)propyl] dihydrogen phosphate | IC50 | 6.0 [1], 50.0 [2] |
 | [(2R)-2-(1-Benzothiophene-2-carbonylamino)-3-(3-fluorophenyl)propyl] dihydrogen phosphate | Ki | 6.0 [1] |
 | Acetyl-11-keto-beta-boswellic acid | IC50 | 50360.0 [1], 52990.0 [2] |
 | Procodazole | IC50 | 10000.0 [1], 740000.0 [2] |
 | 1,7-Diphenylheptan-4-yl (2S)-1-[[(2R)-1-phenyl-3-phosphonooxypropan-2-yl]carbamoyl]piperidine-2-carboxylate | IC50 | 800.0 [1] |
 | 1,7-Diphenylheptan-4-yl (2S)-1-[[(2R)-1-phenyl-3-phosphonooxypropan-2-yl]carbamoyl]piperidine-2-carboxylate | Ki | 800.0 [1] |
 | [(2R)-2-(1-Benzothiophene-2-carbonylamino)-3-phenylpropyl] dihydrogen phosphate | IC50 | 180.0 [1] |
 | [(2R)-2-(1-Benzothiophene-2-carbonylamino)-3-phenylpropyl] dihydrogen phosphate | Ki | 179.0 [1] |
 | (2R)-3-(6-Fluoro-1H-indol-2-yl)-2-(naphthalene-2-carbonylamino)propanoic acid | IC50 | 2960.0 [1] |
 | (2R)-3-(6-Fluoro-1H-indol-2-yl)-2-(naphthalene-2-carbonylamino)propanoic acid | Ki | 138.0 [1] |
 | 3-Fluoro-N-(naphthalen-2-ylcarbonyl)-D-phenylalanine | IC50 | 12000.0 [1] |
 | 3-Fluoro-N-(naphthalen-2-ylcarbonyl)-D-phenylalanine | Ki | 12000.0 [1] |
 | Piperidine-1-dithiocarboxylic acid, anhydrosulphide | IC50 | 4000.0 [1] |
 | Piperidine-1-dithiocarboxylic acid, anhydrosulphide | Ki | 50.0 [1] |
 | (2R,4E)-2-[(Naphthalen-2-ylcarbonyl)amino]-5-phenylpent-4-enoic acid | IC50 | 50000.0 [1] |
 | (2R,4E)-2-[(Naphthalen-2-ylcarbonyl)amino]-5-phenylpent-4-enoic acid | Ki | 1800.0 [1] |
 | (3R)-4-(3-Fluorophenyl)-3-(naphthalene-2-carbonylamino)butanoic acid | IC50 | 50000.0 [1] |
 | (3R)-4-(3-Fluorophenyl)-3-(naphthalene-2-carbonylamino)butanoic acid | Ki | 5700.0 [1] |
 | (2R)-3-(3-Methylphenyl)-2-(naphthalene-2-carbonylamino)propanoic acid | IC50 | 50000.0 [1] |
 | (2R)-3-(3-Methylphenyl)-2-(naphthalene-2-carbonylamino)propanoic acid | Ki | 2800.0 [1] |
 | (3R)-4-(3-Methylphenyl)-3-(naphthalene-2-carbonylamino)butanoic acid | IC50 | 50000.0 [1] |
 | (3R)-4-(3-Methylphenyl)-3-(naphthalene-2-carbonylamino)butanoic acid | Ki | 9700.0 [1] |
 | (2R)-3-(3-Cyanophenyl)-2-(naphthalene-2-carbonylamino)propanoic acid | IC50 | 50000.0 [1] |
 | (2R)-3-(3-Cyanophenyl)-2-(naphthalene-2-carbonylamino)propanoic acid | Ki | 3200.0 [1] |
 | (3R)-4-(3-Cyanophenyl)-3-(naphthalene-2-carbonylamino)butanoic acid | IC50 | 50000.0 [1] |
 | (3R)-4-(3-Cyanophenyl)-3-(naphthalene-2-carbonylamino)butanoic acid | Ki | 2300.0 [1] |
 | (2R)-2-(Naphthalene-2-carbonylamino)-3-[3-(trifluoromethyl)phenyl]propanoic acid | IC50 | 50000.0 [1] |
 | (2R)-2-(Naphthalene-2-carbonylamino)-3-[3-(trifluoromethyl)phenyl]propanoic acid | Ki | 1800.0 [1] |
 | (3R)-3-(Naphthalene-2-carbonylamino)-4-[3-(trifluoromethyl)phenyl]butanoic acid | IC50 | 50000.0 [1] |
 | (3R)-3-(Naphthalene-2-carbonylamino)-4-[3-(trifluoromethyl)phenyl]butanoic acid | Ki | 13000.0 [1] |
 | (2R)-3-(3-Chlorophenyl)-2-(naphthalene-2-carbonylamino)propanoic acid | IC50 | 50000.0 [1] |
 | (2R)-3-(3-Chlorophenyl)-2-(naphthalene-2-carbonylamino)propanoic acid | Ki | 3400.0 [1] |
 | (3R)-4-(3-Chlorophenyl)-3-(naphthalene-2-carbonylamino)butanoic acid | IC50 | 50000.0 [1] |
 | (3R)-4-(3-Chlorophenyl)-3-(naphthalene-2-carbonylamino)butanoic acid | Ki | 2000.0 [1] |
 | (2R)-3-(3,4-Difluorophenyl)-2-(naphthalene-2-carbonylamino)propanoic acid | IC50 | 50000.0 [1] |
 | (2R)-3-(3,4-Difluorophenyl)-2-(naphthalene-2-carbonylamino)propanoic acid | Ki | 23000.0 [1] |
 | (3R)-4-(3,4-Difluorophenyl)-3-(naphthalene-2-carbonylamino)butanoic acid | IC50 | 50000.0 [1] |
 | (3R)-4-(3,4-Difluorophenyl)-3-(naphthalene-2-carbonylamino)butanoic acid | Ki | 82000.0 [1] |
 | (2R)-3-(3,4-Dichlorophenyl)-2-(naphthalene-2-carbonylamino)propanoic acid | IC50 | 50000.0 [1] |
 | (2R)-3-(3,4-Dichlorophenyl)-2-(naphthalene-2-carbonylamino)propanoic acid | Ki | 2200.0 [1] |
 | (2R)-2-(Naphthalene-2-carbonylamino)-3-(3,4,5-trifluorophenyl)propanoic acid | IC50 | 50000.0 [1] |
 | (2R)-2-(Naphthalene-2-carbonylamino)-3-(3,4,5-trifluorophenyl)propanoic acid | Ki | 9000.0 [1] |
 | (2R)-3-(4-Cyanophenyl)-2-(naphthalene-2-carbonylamino)propanoic acid | IC50 | 50000.0 [1] |
 | (2R)-3-(4-Cyanophenyl)-2-(naphthalene-2-carbonylamino)propanoic acid | Ki | 3000.0 [1] |
 | (R)-N-(2-(4-Fluorophenyl)-1-(1H-tetrazol-5-yl)ethyl)-2-naphthamide | IC50 | 50000.0 [1] |
 | (R)-N-(2-(4-Fluorophenyl)-1-(1H-tetrazol-5-yl)ethyl)-2-naphthamide | Ki | 4000.0 [1] |
 | N-[(1R)-1-(2H-Tetrazol-5-yl)-2-[4-(trifluoromethyl)phenyl]ethyl]naphthalene-2-carboxamide | IC50 | 50000.0 [1] |
 | N-[(1R)-1-(2H-Tetrazol-5-yl)-2-[4-(trifluoromethyl)phenyl]ethyl]naphthalene-2-carboxamide | Ki | 8500.0 [1] |
 | (2R)-2-(Naphthalene-2-carbonylamino)-5-phenylpent-4-ynoic acid | IC50 | 50000.0 [1] |
 | (2R)-2-(Naphthalene-2-carbonylamino)-5-phenylpent-4-ynoic acid | Ki | 12800.0 [1] |
 | (2R)-5-(3-Fluorophenyl)-2-(naphthalene-2-carbonylamino)pent-4-ynoic acid | IC50 | 50000.0 [1] |
 | (2R)-5-(3-Fluorophenyl)-2-(naphthalene-2-carbonylamino)pent-4-ynoic acid | Ki | 1870.0 [1] |
 | (2R)-5-(2-Hydroxyphenyl)-2-(naphthalene-2-carbonylamino)pent-4-ynoic acid | IC50 | 50000.0 [1] |
 | (2R)-5-(2-Hydroxyphenyl)-2-(naphthalene-2-carbonylamino)pent-4-ynoic acid | Ki | 4430.0 [1] |
 | (2R)-2-(Naphthalene-2-carbonylamino)-5-thiophen-2-ylpent-4-ynoic acid | IC50 | 50000.0 [1] |
 | (2R)-2-(Naphthalene-2-carbonylamino)-5-thiophen-2-ylpent-4-ynoic acid | Ki | 7000.0 [1] |
 | (E,2R)-5-(3-Fluorophenyl)-2-(naphthalene-2-carbonylamino)pent-4-enoic acid | IC50 | 50000.0 [1] |
 | (E,2R)-5-(3-Fluorophenyl)-2-(naphthalene-2-carbonylamino)pent-4-enoic acid | Ki | 890.0 [1] |
 | (R)-2-(Benzo[b]thiophene-2-carboxamido)-5-phenylpent-4-enoic acid | IC50 | 50000.0 [1] |
 | (R)-2-(Benzo[b]thiophene-2-carboxamido)-5-phenylpent-4-enoic acid | Ki | 3700.0 [1] |
 | (E,2R)-5-(Cyclohexen-1-yl)-2-(naphthalene-2-carbonylamino)pent-4-enoic acid | IC50 | 50000.0 [1] |
 | (E,2R)-5-(Cyclohexen-1-yl)-2-(naphthalene-2-carbonylamino)pent-4-enoic acid | Ki | 2000.0 [1] |
 | Cycloheximide | Ki | 200000.0 [1] |
 | Tretinoin | IC50 | 820.0 [1] |
 | (-)-Epigallocatechin gallate | IC50 | 20000.0 [1] |
 | Enoxolone | IC50 | 10000.0 [1] |
 | 5-Pyridin-2-yl-1H-pyrazole-3-carboxylic acid | IC50 | 720000.0 [1] |
 | 5-(2-Methoxyphenyl)-2-furoic acid | IC50 | 1000000.0 [1] |
 | 5-Methyl-1H-indole-2-carboxylic acid | IC50 | 16000.0 [1] |
 | PPIase-Parvulin Inhibitor | IC50 | 1500.0 [1] |
 | 6-Methyl-1H-indole-2-carboxylic acid | IC50 | 630000.0 [1] |
 | 2-Phenyl-1H-imidazole-4-carboxylic acid | IC50 | 180000.0 [1] |
 | 2-(3-Chloro-4-fluorophenyl)-3(2H)-isothiazolone | IC50 | 6100.0 [1] |
 | 2-Chloro-N-cyclopentyl-5-nitropyrimidin-4-amine | IC50 | 100000.0 [1] |
 | Elemonic acid | IC50 | 13160.0 [1] |
 | 2-Phenyl-1H-imidazole-4,5-dicarboxylic acid | IC50 | 1460.0 [1] |
 | [(2R)-2-[[(2S)-2-[[(2S)-2-Acetamidopropanoyl]amino]propanoyl]amino]-3-[(2S)-2-[[(2S)-5-(diaminomethylideneamino)-1-(4-nitroanilino)-1-oxopentan-2-yl]carbamoyl]pyrrolidin-1-yl]-3-oxopropyl] dihydrogen phosphate | IC50 | 1000.0 [1] |
 | 2-Chloro-4-cyclohexyloxy-5-nitropyrimidine | IC50 | 100000.0 [1] |
 | 2-Chloro-4-cyclopentyloxy-5-nitropyrimidine | IC50 | 100000.0 [1] |
 | 2-(2-Chloro-5-nitropyrimidin-4-yl)oxybenzonitrile | IC50 | 9050.0 [1] |
 | 2-Chloro-4-naphthalen-1-yloxy-5-nitropyrimidine | IC50 | 22600.0 [1] |
 | 2-Chloro-4-naphthalen-2-yloxy-5-nitropyrimidine | IC50 | 16550.0 [1] |
 | [(2R,3Z)-2-[[(2S)-2-[[(2S)-2-Acetamido-3-phenylpropanoyl]amino]-3-phenylpropanoyl]amino]-3-[(2R)-2-[[(2S)-1-amino-5-(diaminomethylideneamino)-1-oxopentan-2-yl]carbamoyl]cyclopentylidene]propyl] dihydrogen phosphate | IC50 | 1500.0 [1] |
 | 2-Chloro-4-(3-methoxyphenoxy)-5-nitropyrimidine | IC50 | 5040.0 [1] |
 | 2-Chloro-4-(2-fluorophenoxy)-5-nitropyrimidine | IC50 | 2520.0 [1] |
 | 2-Chloro-4-(2-methoxyphenoxy)-5-nitropyrimidine | IC50 | 4030.0 [1] |
 | (2R)-2-[[2-(9H-Fluoren-9-yl)acetyl]amino]-3-(6-fluoro-1H-indol-2-yl)propanoic acid | Ki | 12.0 [1] |
 | 2-[2-(2,6-Dichlorophenyl)ethyl]-4-[(6-fluoro-1H-indol-2-yl)methyl]-5H-1,3-thiazole-4-carboxylic acid | Ki | 196.0 [1] |
 | [(2R,3S)-3-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-6-[5-[(3As,4S,6aR)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]pentanoylamino]-2-acetamidohexanoyl]amino]propanoyl]amino]propanoyl]amino]-3-thiophen-2-ylpropanoyl]amino]-4-[(2S)-2-[[(2S)-1-[[(2S)-1,5-diamino-1,5-dioxopentan-2-yl]amino]-1-oxo-3-(4-phenylphenyl)propan-2-yl]carbamoyl]pyrrolidin-1-yl]-4-oxobutan-2-yl] dihydrogen phosphate | IC50 | 22000.0 [1] |
 | (2R)-2-(1-Benzothiophene-2-carbonylamino)-3-(6-fluoro-1H-benzimidazol-2-yl)propanoic acid | Ki | 76.0 [1] |
 | 2-[(E)-2-(2,6-Dichlorophenyl)ethenyl]-4-[(6-fluoro-1H-indol-2-yl)methyl]-5H-1,3-thiazole-4-carboxylic acid | Ki | 580.0 [1] |
 | [(2R,3R)-3-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-6-[5-[(3As,4S,6aR)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]pentanoylamino]-2-acetamidohexanoyl]amino]propanoyl]amino]propanoyl]amino]-3-(1-benzothiophen-3-yl)propanoyl]amino]-4-[(2S)-2-[[(2S)-1-[[(2S)-1,5-diamino-1,5-dioxopentan-2-yl]amino]-3-naphthalen-2-yl-1-oxopropan-2-yl]carbamoyl]piperidin-1-yl]-4-oxobutan-2-yl] dihydrogen phosphate | Ki | 1.2 [1] |
 | 2-(9H-Fluoren-9-ylmethyl)-4-[(6-fluoro-1H-indol-2-yl)methyl]-5H-1,3-thiazole-4-carboxylic acid | Ki | 320.0 [1] |
 | 3-(6-Fluoro-1h-Benzimidazol-2-Yl)-N-(Naphthalen-2-Ylcarbonyl)-D-Alanine | Ki | 80.0 [1] |
 | 4-[(6-Fluoro-1H-indol-2-yl)methyl]-2-naphthalen-2-yl-5H-1,3-thiazole-4-carboxylic acid | Ki | 1360.0 [1] |
 | (2R)-2-[3-(2,6-Dichlorophenyl)propanoylamino]-3-(6-fluoro-1H-indol-2-yl)propanoic acid | Ki | 75.0 [1] |
 | [(2R)-3-(3-Methylphenyl)-2-(naphthalene-2-carbonylamino)propyl] dihydrogen phosphate | Ki | 32.0 [1] |