 | Tacrolimus | Ki | 79.0 [1], 80.0 [2] |
 | 2-[3-[(1R)-3-(3,4-Dimethoxyphenyl)-1-[(2S)-1-(3,3-dimethyl-2-oxopentanoyl)piperidine-2-carbonyl]oxypropyl]phenoxy]acetic acid | IC50 | 6300.0 [1], 8360.0 [2] |
 | SAFit1 | Ki | 4.0 [1] |
 | SAFit2 | Ki | 6.0 [1] |
 | Sirolimus | Ki | 3.0 [1] |
 | (S)-3-(Pyridin-3-yl)propyl 1-(3,3-dimethyl-2-oxopentanoyl)pyrrolidine-2-carboxylate | IC50 | 100000.0 [1] |
 | Biricodar | IC50 | 8520.0 [1] |
 | Timcodar | IC50 | 100000.0 [1] |
 | (S)-1-(3,3-Dimethyl-2-oxo-pentanoyl)-piperidine-2-carboxylic acid 3-pyridin-3-yl-propyl ester | IC50 | 150000.0 [1] |
 | 2-[3-[(1R)-1-[(2S)-1-[(2S)-2-Cyclohexyl-2-phenylacetyl]piperidine-2-carbonyl]oxy-3-(3,4-dimethoxyphenyl)propyl]phenoxy]acetic acid | Ki | 600.0 [1] |
 | Methyl (2S)-1-(3,3-dimethyl-2-oxopentanoyl)piperidine-2-carboxylate | IC50 | 100000.0 [1] |
 | (2S)-N-(1-Carbamoylcyclobutyl)-1-[(2S)-2-cyclohexyl-2-(3,4,5-trimethoxyphenyl)acetyl]piperidine-2-carboxamide | Ki | 4900.0 [1] |
 | (2S)-N-[1-[(2-Amino-2-oxoethyl)carbamoyl]cyclopentyl]-1-[(2S)-2-cyclohexyl-2-(3,4,5-trimethoxyphenyl)acetyl]piperidine-2-carboxamide | Ki | 800.0 [1] |
 | (2S)-N-[(1R)-2-Amino-2-oxo-1-phenylethyl]-1-[(2S)-2-cyclohexyl-2-(3,4,5-trimethoxyphenyl)acetyl]piperidine-2-carboxamide | Ki | 1500.0 [1] |
 | CID 117967787 | Ki | 140.0 [1] |
 | (2S)-N-[(2S,3S)-1-Amino-3-methyl-1-oxopentan-2-yl]-1-[(2S)-2-cyclohexyl-2-(3,4,5-trimethoxyphenyl)acetyl]piperidine-2-carboxamide | Ki | 7100.0 [1] |
 | (2R)-2-[[(2S)-1-[(2S)-2-Cyclohexyl-2-(3,4,5-trimethoxyphenyl)acetyl]piperidine-2-carbonyl]amino]pentanediamide | Ki | 3400.0 [1] |
 | 2-[3-[(1R)-1-[(2S)-1-[(2R)-2-Cyclohexylpent-4-enoyl]piperidine-2-carbonyl]oxy-3-(3,4-dimethoxyphenyl)propyl]phenoxy]acetic acid | Ki | 3400.0 [1] |
 | (2S)-N-[(2S)-1-Amino-1-oxobutan-2-yl]-1-[(2S)-2-cyclohexyl-2-(3,4,5-trimethoxyphenyl)acetyl]piperidine-2-carboxamide | Ki | 3600.0 [1] |
 | (2S)-N-[(2S)-1-Amino-3-hydroxy-1-oxopropan-2-yl]-1-[(2S)-2-cyclohexyl-2-(3,4,5-trimethoxyphenyl)acetyl]piperidine-2-carboxamide | Ki | 62900.0 [1] |
 | (2S)-N-[(2S)-1-Amino-1-oxopropan-2-yl]-1-[(2S)-2-cyclohexyl-2-(3,4,5-trimethoxyphenyl)acetyl]piperidine-2-carboxamide | Ki | 17100.0 [1] |
 | 2-[3-[(1R)-1-[[(2S)-1-[(2S)-2-Cyclohexyl-2-(3,4,5-trimethoxyphenyl)acetyl]piperidine-2-carbonyl]amino]-3-(3,4-dimethoxyphenyl)propyl]phenoxy]acetic acid | Ki | 43.0 [1] |
 | (2S)-N-(4-Amino-2-methyl-4-oxobutan-2-yl)-1-[(2S)-2-cyclohexyl-2-(3,4,5-trimethoxyphenyl)acetyl]piperidine-2-carboxamide | Ki | 3800.0 [1] |
 | (2S)-N-[(2R)-1-Amino-3-(1H-imidazol-5-yl)-1-oxopropan-2-yl]-1-[(2S)-2-cyclohexyl-2-(3,4,5-trimethoxyphenyl)acetyl]piperidine-2-carboxamide | Ki | 3800.0 [1] |
 | (2S)-N-[(2R)-1-Amino-1-oxopropan-2-yl]-1-[(2S)-2-cyclohexyl-2-(3,4,5-trimethoxyphenyl)acetyl]piperidine-2-carboxamide | Ki | 10000.0 [1] |
 | (2S)-N-(1-Carbamoylcyclopropyl)-1-[(2S)-2-cyclohexyl-2-(3,4,5-trimethoxyphenyl)acetyl]piperidine-2-carboxamide | Ki | 19500.0 [1] |
 | (2S)-N-[(2S)-1-Amino-3-(1H-imidazol-5-yl)-1-oxopropan-2-yl]-1-[(2S)-2-cyclohexyl-2-(3,4,5-trimethoxyphenyl)acetyl]piperidine-2-carboxamide | Ki | 13400.0 [1] |
 | (2S)-N-[(2R)-1-Amino-1-oxobutan-2-yl]-1-[(2S)-2-cyclohexyl-2-(3,4,5-trimethoxyphenyl)acetyl]piperidine-2-carboxamide | Ki | 4500.0 [1] |
 | (2S)-N-[(2S)-1-Amino-1-oxo-3-phenylpropan-2-yl]-1-[(2S)-2-cyclohexyl-2-(3,4,5-trimethoxyphenyl)acetyl]piperidine-2-carboxamide | Ki | 6500.0 [1] |
 | (2S)-N-[(2S)-1-Amino-3-methyl-1-oxobutan-2-yl]-1-[(2S)-2-cyclohexyl-2-(3,4,5-trimethoxyphenyl)acetyl]piperidine-2-carboxamide | Ki | 12600.0 [1] |
 | (2S)-N-[(2R)-1-Amino-1-oxo-3-phenylpropan-2-yl]-1-[(2S)-2-cyclohexyl-2-(3,4,5-trimethoxyphenyl)acetyl]piperidine-2-carboxamide | Ki | 1400.0 [1] |
 | (2S)-N-[(2R)-1-Amino-4-hydroxy-1-oxobutan-2-yl]-1-[(2S)-2-cyclohexyl-2-(3,4,5-trimethoxyphenyl)acetyl]piperidine-2-carboxamide | Ki | 4200.0 [1] |
 | (2S)-N-[(2S)-1-Amino-4-hydroxy-1-oxobutan-2-yl]-1-[(2S)-2-cyclohexyl-2-(3,4,5-trimethoxyphenyl)acetyl]piperidine-2-carboxamide | Ki | 13000.0 [1] |
 | (2S)-N-[(2S)-1-Amino-4-methyl-1-oxopentan-2-yl]-1-[(2S)-2-cyclohexyl-2-(3,4,5-trimethoxyphenyl)acetyl]piperidine-2-carboxamide | Ki | 8700.0 [1] |
 | (2S)-N-[(2S)-1-Amino-4-cyclohexyl-1-oxobutan-2-yl]-1-[(2S)-2-cyclohexyl-2-(3,4,5-trimethoxyphenyl)acetyl]piperidine-2-carboxamide | Ki | 12000.0 [1] |
 | (2S)-N-[(2S)-1-Amino-3-cyclohexyl-1-oxopropan-2-yl]-1-[(2S)-2-cyclohexyl-2-(3,4,5-trimethoxyphenyl)acetyl]piperidine-2-carboxamide | Ki | 17800.0 [1] |
 | 2-[3-[(1R)-1-[(2S)-1-[(2R)-2-Cyclohexylpropanoyl]piperidine-2-carbonyl]oxy-3-(3,4-dimethoxyphenyl)propyl]phenoxy]acetic acid | Ki | 1200.0 [1] |
 | (2S)-N-(1-Carbamoylcyclohexyl)-1-[(2S)-2-cyclohexyl-2-(3,4,5-trimethoxyphenyl)acetyl]piperidine-2-carboxamide | Ki | 1900.0 [1] |
 | (2S)-1-[(2S)-2-Cyclohexyl-2-(3,4,5-trimethoxyphenyl)acetyl]-N-ethylpiperidine-2-carboxamide | Ki | 55000.0 [1] |
 | (2S)-N-[(2R,3R)-1-Amino-3-methyl-1-oxopentan-2-yl]-1-[(2S)-2-cyclohexyl-2-(3,4,5-trimethoxyphenyl)acetyl]piperidine-2-carboxamide | Ki | 3200.0 [1] |
 | (2S)-N-[(2S)-1-Amino-1-oxo-4-phenylbutan-2-yl]-1-[(2S)-2-cyclohexyl-2-(3,4,5-trimethoxyphenyl)acetyl]piperidine-2-carboxamide | Ki | 9100.0 [1] |
 | (2S)-N-(2-Amino-2-oxoethyl)-1-[(2S)-2-cyclohexyl-2-(3,4,5-trimethoxyphenyl)acetyl]piperidine-2-carboxamide | Ki | 36700.0 [1] |
 | (2S)-N-[(1S)-2-Amino-2-oxo-1-phenylethyl]-1-[(2S)-2-cyclohexyl-2-(3,4,5-trimethoxyphenyl)acetyl]piperidine-2-carboxamide | Ki | 3100.0 [1] |
 | (2S)-N-[(2R)-1-Amino-3-hydroxy-1-oxopropan-2-yl]-1-[(2S)-2-cyclohexyl-2-(3,4,5-trimethoxyphenyl)acetyl]piperidine-2-carboxamide | Ki | 2800.0 [1] |
 | (2S)-N-[(1S)-2-Amino-1-cyclohexyl-2-oxoethyl]-1-[(2S)-2-cyclohexyl-2-(3,4,5-trimethoxyphenyl)acetyl]piperidine-2-carboxamide | Ki | 4300.0 [1] |
 | (2S)-2-[[(2S)-1-[(2S)-2-Cyclohexyl-2-(3,4,5-trimethoxyphenyl)acetyl]piperidine-2-carbonyl]amino]pentanediamide | Ki | 345000.0 [1] |
 | (2S)-N-(1-Amino-2-methyl-1-oxopropan-2-yl)-1-[(2S)-2-cyclohexyl-2-(3,4,5-trimethoxyphenyl)acetyl]piperidine-2-carboxamide | Ki | 2200.0 [1] |
 | (2S)-N-[(2R)-1-Amino-3-methyl-1-oxobutan-2-yl]-1-[(2S)-2-cyclohexyl-2-(3,4,5-trimethoxyphenyl)acetyl]piperidine-2-carboxamide | Ki | 5000.0 [1] |
 | (2S)-N-(3-Amino-3-oxopropyl)-1-[(2S)-2-cyclohexyl-2-(3,4,5-trimethoxyphenyl)acetyl]piperidine-2-carboxamide | Ki | 7900.0 [1] |
 | (2S)-N-(4-Carbamoyloxan-4-yl)-1-[(2S)-2-cyclohexyl-2-(3,4,5-trimethoxyphenyl)acetyl]piperidine-2-carboxamide | Ki | 1800.0 [1] |
 | 2-[3-[(1R)-1-[(2S)-1-[(2S)-2-Cyclohexyl-2-(3,5-dimethoxyphenyl)acetyl]piperidine-2-carbonyl]oxy-3-(3,4-dimethoxyphenyl)propyl]phenoxy]acetic acid | Ki | 110.0 [1] |
 | 2-[3-[(1R)-1-[(2S)-1-[(2S)-2-Cyclohexyl-2-(3-methoxyphenyl)acetyl]piperidine-2-carbonyl]oxy-3-(3,4-dimethoxyphenyl)propyl]phenoxy]acetic acid | Ki | 160.0 [1] |
 | 2-[3-[(1R)-1-[(2S)-1-(2-Cyclohexylacetyl)piperidine-2-carbonyl]oxy-3-(3,4-dimethoxyphenyl)propyl]phenoxy]acetic acid | Ki | 4200.0 [1] |
 | [(1R)-3-(3,4-Dimethoxyphenyl)-1-[3-(2-morpholin-4-ylethoxy)phenyl]propyl] (2S)-1-[(2S)-2-cyclohexyl-3-(methoxymethoxy)propanoyl]piperidine-2-carboxylate | Ki | 4100.0 [1] |
 | [(1R)-3-(3,4-Dimethoxyphenyl)-1-[3-(2-morpholin-4-ylethoxy)phenyl]propyl] (2S)-1-[(2S)-2-cyclohexyl-3-hydroxypropanoyl]piperidine-2-carboxylate | Ki | 2000.0 [1] |
 | [(1R)-3-(3,4-Dimethoxyphenyl)-1-[3-(2-morpholin-4-ylethoxy)phenyl]propyl] (2S)-1-[(2S)-3-acetyloxy-2-cyclohexylpropanoyl]piperidine-2-carboxylate | Ki | 2100.0 [1] |
 | [(1R)-3-(3,4-Dimethoxyphenyl)-1-[3-(2-morpholin-4-ylethoxy)phenyl]propyl] (2S)-1-[(2S,3R)-2-cyclohexyl-3-(methoxymethoxy)butanoyl]piperidine-2-carboxylate | Ki | 2000.0 [1] |
 | [(1R)-3-(3,4-Dimethoxyphenyl)-1-[3-(2-morpholin-4-ylethoxy)phenyl]propyl] (2S)-1-[(2S)-2-cyclohexyl-3-oxobutanoyl]piperidine-2-carboxylate | Ki | 2500.0 [1] |
 | [(1R)-3-(3,4-Dimethoxyphenyl)-1-[3-(2-morpholin-4-ylethoxy)phenyl]propyl] (2S)-1-[(E,2S,3R)-2-cyclohexyl-3-hydroxyhex-4-enoyl]piperidine-2-carboxylate | Ki | 1100.0 [1] |
 | [(1R)-3-(3,4-Dimethoxyphenyl)-1-[3-(2-morpholin-4-ylethoxy)phenyl]propyl] (2S)-1-[(2R,3R)-2-cyclohexyl-3-hydroxy-4-methylpentanoyl]piperidine-2-carboxylate | Ki | 13000.0 [1] |
 | [(1R)-3-(3,4-Dimethoxyphenyl)-1-[3-(2-morpholin-4-ylethoxy)phenyl]propyl] (2S)-1-[(2S,3R)-2-cyclohexyl-3-(methoxymethoxy)-5-methylhexanoyl]piperidine-2-carboxylate | Ki | 17000.0 [1] |
 | [(1R)-3-(3,4-Dimethoxyphenyl)-1-[3-(2-morpholin-4-ylethoxy)phenyl]propyl] (2S)-1-[(2S,3R)-2-cyclohexyl-3-hydroxy-5-methylhexanoyl]piperidine-2-carboxylate | Ki | 9000.0 [1] |
 | [(1R)-3-(3,4-Dimethoxyphenyl)-1-[3-(2-morpholin-4-ylethoxy)phenyl]propyl] (2S)-1-[(2R,3S)-2-cyclohexyl-3-hydroxy-3-phenylpropanoyl]piperidine-2-carboxylate | Ki | 100000.0 [1] |
 | (2S)-N-(4-Amino-4-oxobutyl)-1-[(2S)-2-cyclohexyl-2-(3,4,5-trimethoxyphenyl)acetyl]piperidine-2-carboxamide | Ki | 5700.0 [1] |
 | (2S)-N-(5-Amino-5-oxopentyl)-1-[(2S)-2-cyclohexyl-2-(3,4,5-trimethoxyphenyl)acetyl]piperidine-2-carboxamide | Ki | 3900.0 [1] |
 | (1S,5S,6R)-10-(3,5-Dichlorophenyl)sulfonyl-5-(methoxymethyl)-3-(pyridin-2-ylmethyl)-3,10-diazabicyclo[4.3.1]decan-2-one | Ki | 24.5 [1] |
 | [(1R)-1-(3-Aminophenyl)-3-(3,4-dimethoxyphenyl)propyl] (2S)-1-(3,3-dimethyl-2-oxopentanoyl)piperidine-2-carboxylate | IC50 | 3800.0 [1] |
 | 2-[3-[(1R)-3-(3,4-Dimethoxyphenyl)-1-[(2S)-1-[2-[(1S,2R)-2-ethyl-1-hydroxycyclohexyl]-2-oxoacetyl]piperidine-2-carbonyl]oxypropyl]phenoxy]acetic acid | IC50 | 5800.0 [1] |
 | 2-[3-[(1R)-3-(3,4-Dimethoxyphenyl)-1-[(2S)-1-[2-[(1R,2S)-2-ethyl-1-hydroxycyclohexyl]-2-oxoacetyl]piperidine-2-carbonyl]oxypropyl]phenoxy]acetic acid | IC50 | 3900.0 [1] |
 | 2-[3-[(1R)-3-(3,4-Dimethoxyphenyl)-1-[(2S)-1-[2-[(1S,2S)-1-hydroxy-2-(hydroxymethyl)cyclohexyl]-2-oxoacetyl]piperidine-2-carbonyl]oxypropyl]phenoxy]acetic acid | IC50 | 8500.0 [1] |
 | 2-(3,4-Dimethoxyphenoxy)ethyl (2S)-1-(3,3-dimethyl-2-oxopentanoyl)piperidine-2-carboxylate | IC50 | 100000.0 [1] |
 | [(1R)-3-(3,4-Dimethoxyphenyl)-1-[3-(2-morpholin-4-ylethoxy)phenyl]propyl] (2S)-1-(3,3-dimethyl-2-oxopentanoyl)piperidine-2-carboxylate | IC50 | 4150.0 [1] |
 | [(1R)-3-(3,4-Dimethoxyphenyl)-1-[3-(2-morpholin-4-ylethoxy)phenyl]propyl] (2S)-1-(3,3-dimethyl-2-oxopentanoyl)pyrrolidine-2-carboxylate | IC50 | 15340.0 [1] |
 | 2-[3-[(1R)-3-(3,4-Dimethoxyphenyl)-1-[(2S)-1-[2-oxo-2-(3,4,5-trimethoxyphenyl)acetyl]piperidine-2-carbonyl]oxypropyl]phenoxy]acetic acid | IC50 | 19300.0 [1] |
 | 2-[3-[(1R)-3-(3,4-Dimethoxyphenyl)-1-[(2S)-1-[2-[(1S,2R)-1-hydroxy-2-methylcyclohexyl]-2-oxoacetyl]piperidine-2-carbonyl]oxypropyl]phenoxy]acetic acid | IC50 | 4270.0 [1] |
 | 2-[3-[(1R)-3-(3,4-Dimethoxyphenyl)-1-[(2S)-1-[2-[(1R,2S)-1-hydroxy-2-methylcyclohexyl]-2-oxoacetyl]piperidine-2-carbonyl]oxypropyl]phenoxy]acetic acid | IC50 | 4540.0 [1] |
 | 2-[3-[(1R)-3-(3,4-Dimethoxyphenyl)-1-[(2S)-1-[2-[(1S,2S)-1-hydroxy-2-methylcyclohexyl]-2-oxoacetyl]piperidine-2-carbonyl]oxypropyl]phenoxy]acetic acid | IC50 | 4180.0 [1] |
 | 2-[3-[(1R)-3-(3,4-Dimethoxyphenyl)-1-[(2S)-1-[2-[(1R,2R)-1-hydroxy-2-methylcyclohexyl]-2-oxoacetyl]piperidine-2-carbonyl]oxypropyl]phenoxy]acetic acid | IC50 | 4960.0 [1] |
 | 2-[3-[(1R)-3-(3,4-Dimethoxyphenyl)-1-[(2S)-1-(4-pyrimidin-2-ylphenyl)sulfonylpiperidine-2-carbonyl]oxypropyl]phenoxy]acetic acid | IC50 | 62800.0 [1] |
 | 2-[3-[(1R)-1-[(2S)-1-(3-Chlorophenyl)sulfonylpiperidine-2-carbonyl]oxy-3-(3,4-dimethoxyphenyl)propyl]phenoxy]acetic acid | IC50 | 30700.0 [1] |
 | 2-[3-[(1R)-1-[(2S)-1-(1,3-Benzothiazol-6-ylsulfonyl)piperidine-2-carbonyl]oxy-3-(3,4-dimethoxyphenyl)propyl]phenoxy]acetic acid | IC50 | 11600.0 [1] |
 | 2-[3-[(1R)-3-(3,4-Dimethoxyphenyl)-1-[(2S)-1-(furan-3-ylsulfonyl)piperidine-2-carbonyl]oxypropyl]phenoxy]acetic acid | IC50 | 100000.0 [1] |
 | 2-[3-[(1R)-1-[(2S)-1-(1-Benzothiophen-2-ylsulfonyl)piperidine-2-carbonyl]oxy-3-(3,4-dimethoxyphenyl)propyl]phenoxy]acetic acid | IC50 | 67100.0 [1] |
 | 2-[3-[(1R)-1-[(2S)-1-(3-Cyanophenyl)sulfonylpiperidine-2-carbonyl]oxy-3-(3,4-dimethoxyphenyl)propyl]phenoxy]acetic acid | IC50 | 28500.0 [1] |
 | 2-[3-[(1R)-3-(3,4-Dimethoxyphenyl)-1-[(2S)-1-(3-nitrophenyl)sulfonylpiperidine-2-carbonyl]oxypropyl]phenoxy]acetic acid | IC50 | 47200.0 [1] |
 | 2-[3-[(1R)-1-[(2S)-1-(3-Aminophenyl)sulfonylpiperidine-2-carbonyl]oxy-3-(3,4-dimethoxyphenyl)propyl]phenoxy]acetic acid | IC50 | 45400.0 [1] |
 | 2-[3-[(1R)-3-(3,4-Dimethoxyphenyl)-1-[(2S)-1-(3-fluorophenyl)sulfonylpiperidine-2-carbonyl]oxypropyl]phenoxy]acetic acid | IC50 | 54050.0 [1] |
 | 2-[3-[(1R)-1-[(2S)-1-(3-Bromophenyl)sulfonylpiperidine-2-carbonyl]oxy-3-(3,4-dimethoxyphenyl)propyl]phenoxy]acetic acid | IC50 | 15780.0 [1] |
 | 2-[3-[(1R)-1-[(2S)-1-(3,5-Dichlorophenyl)sulfonylpiperidine-2-carbonyl]oxy-3-(3,4-dimethoxyphenyl)propyl]phenoxy]acetic acid | IC50 | 22600.0 [1] |
 | 2-[3-[(1R)-1-[(2S)-1-(3,4-Dichlorophenyl)sulfonylpiperidine-2-carbonyl]oxy-3-(3,4-dimethoxyphenyl)propyl]phenoxy]acetic acid | IC50 | 100000.0 [1] |
 | 2-[3-[(1R)-3-(3,4-Dimethoxyphenyl)-1-[(2S)-1-(3,4-dimethoxyphenyl)sulfonylpiperidine-2-carbonyl]oxypropyl]phenoxy]acetic acid | IC50 | 100000.0 [1] |
 | 2-[3-[(1R)-1-[(2S)-1-(3-Chloro-4-methoxyphenyl)sulfonylpiperidine-2-carbonyl]oxy-3-(3,4-dimethoxyphenyl)propyl]phenoxy]acetic acid | IC50 | 29600.0 [1] |
 | 2-[3-[(1R)-1-[(2S)-1-(3,5-Difluorophenyl)sulfonylpiperidine-2-carbonyl]oxy-3-(3,4-dimethoxyphenyl)propyl]phenoxy]acetic acid | IC50 | 88200.0 [1] |
 | 2-[3-[(1R)-1-[(2S)-1-[3,5-Bis(trifluoromethyl)phenyl]sulfonylpiperidine-2-carbonyl]oxy-3-(3,4-dimethoxyphenyl)propyl]phenoxy]acetic acid | IC50 | 100000.0 [1] |
 | 2-[3-[(1R)-1-[(2S)-1-[3-Bromo-5-(trifluoromethyl)phenyl]sulfonylpiperidine-2-carbonyl]oxy-3-(3,4-dimethoxyphenyl)propyl]phenoxy]acetic acid | IC50 | 100000.0 [1] |
 | 2-[3-[(1R)-1-[(2S)-1-[3,5-Bis(methoxycarbonyl)phenyl]sulfonylpiperidine-2-carbonyl]oxy-3-(3,4-dimethoxyphenyl)propyl]phenoxy]acetic acid | IC50 | 100000.0 [1] |
 | 2-[3-[(1R)-1-[(2S)-1-(3,5-Dichloro-4-hydroxyphenyl)sulfonylpiperidine-2-carbonyl]oxy-3-(3,4-dimethoxyphenyl)propyl]phenoxy]acetic acid | IC50 | 6200.0 [1] |
 | 2-[3-[(1R)-1-[(2S)-1-(3,5-Dichloro-4-methoxyphenyl)sulfonylpiperidine-2-carbonyl]oxy-3-(3,4-dimethoxyphenyl)propyl]phenoxy]acetic acid | IC50 | 16400.0 [1] |
 | 2-[3-[(1R)-1-[(2S)-1-(4-Acetamido-3,5-dichlorophenyl)sulfonylpiperidine-2-carbonyl]oxy-3-(3,4-dimethoxyphenyl)propyl]phenoxy]acetic acid | IC50 | 16100.0 [1] |
 | 2-[3-[(1R)-3-(3,4-Dimethoxyphenyl)-1-[(2S)-1-[(7-nitro-2,3-dihydro-1-benzofuran-5-yl)sulfonyl]piperidine-2-carbonyl]oxypropyl]phenoxy]acetic acid | IC50 | 27200.0 [1] |