| 3-(2,4-Dimethylpyrido[2',3':3,4]pyrazolo[1,5-a]pyrimidin-3-yl)-N-(3-(methylthio)phenyl)propanamide | IC50 | 25.0 [1], 360.0 [2] |
| 3-(4,6-Dimethyl-3,7,8,10-tetrazatricyclo[7.4.0.02,7]trideca-1,3,5,8,10,12-hexaen-5-yl)-N-(3-methoxyphenyl)propanamide | IC50 | 1640.0 [1] |
| 3-(4,6-Dimethyl-3,7,8,10-tetrazatricyclo[7.4.0.02,7]trideca-1,3,5,8,10,12-hexaen-5-yl)-N-[(4-methoxyphenyl)methyl]propanamide | IC50 | 25840.0 [1] |
| 2-(2,3-Dichlorophenyl)-N-(3-methylbutyl)-1,3-thiazole-4-carboxamide | IC50 | 2450.0 [1] |
| 3-(4,6-Dimethyl-3,7,8,10-tetrazatricyclo[7.4.0.02,7]trideca-1,3,5,8,10,12-hexaen-5-yl)-N-(4-methylsulfanylphenyl)propanamide | IC50 | 10510.0 [1] |
| 3-(4,6-Dimethyl-3,7,8,10-tetrazatricyclo[7.4.0.02,7]trideca-1,3,5,8,10,12-hexaen-5-yl)-N-phenylpropanamide | IC50 | 24500.0 [1] |
| 3-(4,6-Dimethyl-3,7,8,10-tetrazatricyclo[7.4.0.02,7]trideca-1,3,5,8,10,12-hexaen-5-yl)-N-methyl-N-phenylpropanamide | IC50 | 56000.0 [1] |
| N-(Cyclohexylmethyl)-3-(4,6-dimethyl-3,7,8,10-tetrazatricyclo[7.4.0.02,7]trideca-1,3,5,8,10,12-hexaen-5-yl)propanamide | IC50 | 40890.0 [1] |
| 3-(4,6-Dimethyl-3,7,8,10-tetrazatricyclo[7.4.0.02,7]trideca-1,3,5,8,10,12-hexaen-5-yl)-N-(4-methylphenyl)propanamide | IC50 | 25560.0 [1] |
| 3-(4,6-Dimethyl-3,7,8,10-tetrazatricyclo[7.4.0.02,7]trideca-1,3,5,8,10,12-hexaen-5-yl)-N-(2-fluorophenyl)propanamide | IC50 | 13640.0 [1] |
| 3-(4,6-Dimethyl-3,7,8,10-tetrazatricyclo[7.4.0.02,7]trideca-1,3,5,8,10,12-hexaen-5-yl)-N-[(4-fluorophenyl)methyl]propanamide | IC50 | 56000.0 [1] |
| 3-(4,6-Dimethyl-3,7,8,10-tetrazatricyclo[7.4.0.02,7]trideca-1,3,5,8,10,12-hexaen-5-yl)-N-[(3-fluorophenyl)methyl]propanamide | IC50 | 10050.0 [1] |
| 3-(4,6-Dimethyl-3,7,8,10-tetrazatricyclo[7.4.0.02,7]trideca-1,3,5,8,10,12-hexaen-5-yl)-N-[(3-methoxyphenyl)methyl]propanamide | IC50 | 56000.0 [1] |
| 3-(4,6-Dimethyl-3,7,8,10-tetrazatricyclo[7.4.0.02,7]trideca-1,3,5,8,10,12-hexaen-5-yl)-N-[3-(trifluoromethyl)phenyl]propanamide | IC50 | 830.0 [1] |
| Methyl 3-[3-(4,6-dimethyl-3,7,8,10-tetrazatricyclo[7.4.0.02,7]trideca-1,3,5,8,10,12-hexaen-5-yl)propanoylamino]benzoate | IC50 | 56000.0 [1] |
| N-Cyclohexyl-3-(4,6-dimethyl-3,7,8,10-tetrazatricyclo[7.4.0.02,7]trideca-1,3,5,8,10,12-hexaen-5-yl)propanamide | IC50 | 56000.0 [1] |
| 3-(4,6-Dimethyl-3,7,8,10-tetrazatricyclo[7.4.0.02,7]trideca-1,3,5,8,10,12-hexaen-5-yl)-N-(2-methoxyphenyl)propanamide | IC50 | 56000.0 [1] |
| 3-(4,6-Dimethyl-3,7,8,10-tetrazatricyclo[7.4.0.02,7]trideca-1,3,5,8,10,12-hexaen-5-yl)-N-(3-methylphenyl)propanamide | IC50 | 3840.0 [1] |
| 3-(4,6-Dimethyl-3,7,8,10-tetrazatricyclo[7.4.0.02,7]trideca-1,3,5,8,10,12-hexaen-5-yl)-N-(4-fluorophenyl)propanamide | IC50 | 56000.0 [1] |
| 3-(4,6-Dimethyl-3,7,8,10-tetrazatricyclo[7.4.0.02,7]trideca-1,3,5,8,10,12-hexaen-5-yl)-N-(4-methoxyphenyl)propanamide | IC50 | 11290.0 [1] |
| 3-(4,6-Dimethyl-3,7,8,10-tetrazatricyclo[7.4.0.02,7]trideca-1,3,5,8,10,12-hexaen-5-yl)-N-(3-fluorophenyl)propanamide | IC50 | 620.0 [1] |
| 3-(12-Oxo-7-thia-9,11-diazatricyclo[6.4.0.02,6]dodeca-1(8),2(6),9-trien-10-yl)-N-(4-propan-2-ylphenyl)propanamide | IC50 | 120.0 [1] |
| N-(Bicyclo[2.2.1]hept-2-yl)-4-[(ethylsulfonyl)amino]benzamide | IC50 | 180.0 [1] |
| N-(4-Acetamidophenyl)-3-(4,6-dimethyl-3,7,8,10-tetrazatricyclo[7.4.0.02,7]trideca-1,3,5,8,10,12-hexaen-5-yl)propanamide | IC50 | 350.0 [1] |