![](https://images.aatbio.com/dataset/ic50/p2x-purinoceptor-4_1ae4cdbe15d8ef0ea45d00891c1f4348.svg) | CID 9841560 | IC50 | 350.0 [1], 500.0 [2] |
![](https://images.aatbio.com/dataset/ic50/p2x-purinoceptor-4_43cef558f354ca01d14a0c51699f6e63.svg) | Paroxetine | IC50 | 1870.0 [1], 4680.0 [2] |
![](https://images.aatbio.com/dataset/ic50/p2x-purinoceptor-4_d7281b90886e3a49d827e6cdc8f46d75.svg) | Benzyl 10H-phenoxazine-10-carboxylate | IC50 | 189.0 [1] |
![](https://images.aatbio.com/dataset/ic50/p2x-purinoceptor-4_2d46cd64b612bada34966bcfba251b25.svg) | Carbamazepine | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/p2x-purinoceptor-4_4dc438f6747ee1a2a43c99a9ab3957fc.svg) | Oxcarbazepine | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/p2x-purinoceptor-4_16271d46f50e105850b0ecf29bb95a95.svg) | Ppads | IC50 | 27500.0 [1] |
![](https://images.aatbio.com/dataset/ic50/p2x-purinoceptor-4_973cd7b6d3d5e13386c6a6d8612312ea.svg) | Carbamazepine-10,11-epoxide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/p2x-purinoceptor-4_bcc09aa3df38877182b37568a6fd2ba5.svg) | Eslicarbazepine acetate | IC50 | 20000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/p2x-purinoceptor-4_f0ff9790a19a35eb1c8503335ea13d90.svg) | Hexasodium;8-[[3-[[3-[(4,6,8-trisulfonatonaphthalen-1-yl)carbamoyl]phenyl]carbamoylamino]benzoyl]amino]naphthalene-1,3,5-trisulfonate | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/p2x-purinoceptor-4_a1f682f2081256f1284591a943726d63.svg) | Licarbazepine | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/p2x-purinoceptor-4_3331777d13482aa5d6492c6cf0e3da04.svg) | 10,11-Dihydrocarbamazepine | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/p2x-purinoceptor-4_06f194d2d695b5cd59ab980874cac1d6.svg) | 9-Chloroacridine | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/p2x-purinoceptor-4_88bfc2e097a3e213b8f59bafc8676784.svg) | 2,4-Pyrimidinediamine, 5-[5-iodo-4-methoxy-2-(1-methylethyl)phenoxy]- | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/p2x-purinoceptor-4_d87d7e5dc0814e129737012b15955463.svg) | CID 24883277 | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/p2x-purinoceptor-4_7bd1b405cadff6ff60cb960e8bae0479.svg) | 10-Tosyl-10H-phenoxazine | IC50 | 1380.0 [1] |
![](https://images.aatbio.com/dataset/ic50/p2x-purinoceptor-4_1d571a0dc41596f2a64a0005125a4e41.svg) | 5-Ethoxy-5,6-dihydrobenzo[b][1]benzazepine-11-carboxamide | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/p2x-purinoceptor-4_981fd24b9de41f5e02973f5e43fdd326.svg) | Dibenzo[b,f]azepine-5-carboxylic acid methyl ester | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/p2x-purinoceptor-4_562c414d77462662876af4bba7541aad.svg) | N,N-Diethyl-5H-dibenzo[b,f]azepine-5-carboxamide | IC50 | 11400.0 [1] |
![](https://images.aatbio.com/dataset/ic50/p2x-purinoceptor-4_3c9ff2901b1d7f5f7f660053058a9912.svg) | Dibenzo[b,f]azepine-5-carboxylic acid methylamide | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/p2x-purinoceptor-4_1c65f5e6b6854fc984382e9844b06c17.svg) | 2-Hydroxycarbamazepine | IC50 | 146000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/p2x-purinoceptor-4_eb0d80571fd57c47978b3096fa1e1177.svg) | 5-Acetyl-5H-dibenz[b,f]azepine | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/p2x-purinoceptor-4_2a37a604ccf18a307f0a6f4c9132c63b.svg) | CID 11636757 | IC50 | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/p2x-purinoceptor-4_8daf0e01e342c6e3674d49481e404abd.svg) | 3-Hydroxycarbamazepine | IC50 | 72800.0 [1] |
![](https://images.aatbio.com/dataset/ic50/p2x-purinoceptor-4_810e7c568288f85476c2bf9865cdcc2c.svg) | 9(10H)-Acridinone, 10-(phenylmethyl)- | IC50 | 5970.0 [1] |
![](https://images.aatbio.com/dataset/ic50/p2x-purinoceptor-4_eb015343fd527f43c41b3ba57379d5f8.svg) | N-(2-Hydroxyphenyl)benzamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/p2x-purinoceptor-4_000c82e836a931202963c197beffc45c.svg) | 2,3-Dihydro-1,4-benzoxazin-4-yl(phenyl)methanone | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/p2x-purinoceptor-4_e4609619e40bd74d8b9150587b19fd1d.svg) | [(3Ar,4R,6R,6aR)-4-(6-aminopurin-9-yl)-6-[[hydroxy-[hydroxy(phosphonooxy)phosphoryl]oxyphosphoryl]oxymethyl]-3',5'-dinitrospiro[3a,4,6,6a-tetrahydrofuro[3,4-d][1,3]dioxole-2,4'-cyclohexa-2,5-diene]-1'-ylidene]-dioxidoazanium | IC50 | 15200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/p2x-purinoceptor-4_c5f6df36d5e375f1e48a07bb9c35807b.svg) | Benzo[b][1]benzazepin-11-yl(piperidin-1-yl)methanone | IC50 | 13700.0 [1] |
![](https://images.aatbio.com/dataset/ic50/p2x-purinoceptor-4_8fbca1a150dd2d892a8460731419df33.svg) | Benzo[b][1]benzazepin-11-yl(pyrrolidin-1-yl)methanone | IC50 | 34100.0 [1] |
![](https://images.aatbio.com/dataset/ic50/p2x-purinoceptor-4_3357f63ede2132fc2bb683618bbb1488.svg) | 10-Methoxycarbamazepine | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/p2x-purinoceptor-4_c195338aa0210799997c5c38dea9b401.svg) | 11-Benzylbenzo[b][1]benzazepine | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/p2x-purinoceptor-4_3a2b4db3de070825e4f4627e32a0f5f2.svg) | N-Acetylphenoxazine | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/p2x-purinoceptor-4_41cdd47bbe7bb925f397208d2f33c10d.svg) | 10-[(4-Methoxyphenyl)methyl]acridin-9-one | IC50 | 10300.0 [1] |
![](https://images.aatbio.com/dataset/ic50/p2x-purinoceptor-4_07a511b94e1b4b77f999e2f4194b1a83.svg) | 2-Fluorocarbamazepine | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/p2x-purinoceptor-4_8f61aeef71418acd3381c81c504c8f78.svg) | 10-[(4-Nitrophenyl)methyl]acridin-9-one | IC50 | 2490.0 [1] |
![](https://images.aatbio.com/dataset/ic50/p2x-purinoceptor-4_0333825c9f51b3a92336abe41a5dfeb6.svg) | 10-Benzoylacridin-9-one | IC50 | 26900.0 [1] |
![](https://images.aatbio.com/dataset/ic50/p2x-purinoceptor-4_7f2bf924783f053a2d4ab104a6023c6d.svg) | N-(2-Hydroxyphenyl)morpholine-4-carboxamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/p2x-purinoceptor-4_6398775fcd07968ff44ac87050a7c033.svg) | Phenoxazine-10-carbonyl chloride | IC50 | 23200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/p2x-purinoceptor-4_2b7aaf3ef6dfc0df657ffdc76460249f.svg) | (4-Nitrophenyl)-phenoxazin-10-ylmethanone | IC50 | 4290.0 [1] |
![](https://images.aatbio.com/dataset/ic50/p2x-purinoceptor-4_b6816b6cd7846482a47b6ec9bde9060c.svg) | (4E)-5-Cyclohexyl-4-[hydroxy-(4-methoxyphenyl)methylidene]-1-[4-(1,2-oxazol-3-yl)phenyl]pyrrolidine-2,3-dione | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/p2x-purinoceptor-4_5e1e4811d4d129c3dc4ee88c1c10610c.svg) | Benzyl(2-Hydroxyphenyl)Carbamate | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/p2x-purinoceptor-4_d26f685844b9c2a2e00d263f4650237b.svg) | Phenoxazin-10-yl(phenyl)methanone | IC50 | 4110.0 [1] |
![](https://images.aatbio.com/dataset/ic50/p2x-purinoceptor-4_6b0595cada5960135d2368bcd448e17b.svg) | N-[3-(Dimethylamino)propyl]benzo[b][1]benzazepine-11-carboxamide | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/p2x-purinoceptor-4_81eb8bca7b605bcaa5729ce4b2238070.svg) | N-[2-[2-(2-Benzamidophenoxy)ethoxy]phenyl]benzamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/p2x-purinoceptor-4_6cc3ee311fcd1c0c80301f1d23a86537.svg) | N-Phenylbenzo[b][1]benzazepine-11-carboxamide | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/p2x-purinoceptor-4_8d5153547218722e97437323691d079c.svg) | N-[(2R)-1-(4-Acetylpiperazin-1-yl)propan-2-yl]-1-methyl-3-phenylthieno[2,3-c]pyrazole-5-carboxamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/p2x-purinoceptor-4_ee93da4c7f12f4bda69b9a0f4172aad5.svg) | 2-Phenyl-4-propyl-N-[1-(4-pyrimidin-2-ylpiperazin-1-yl)propan-2-yl]-1,3-oxazole-5-carboxamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/p2x-purinoceptor-4_fb4a7c26b436f86f266063d6072916bd.svg) | (4S)-N-[4-Chloro-5-(2-hydroxyethoxy)-2-methylphenyl]-4-(4-fluorophenyl)-2-oxo-3,4-dihydro-1H-pyridine-5-carboxamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/p2x-purinoceptor-4_4c8b105fb54f455b24d7130c499f952c.svg) | 5-Benzoyl-5H-dibenz[b,f]azepin | IC50 | 23300.0 [1] |
![](https://images.aatbio.com/dataset/ic50/p2x-purinoceptor-4_0404cdad8594db95e75722a397f393f9.svg) | 2-Methylbenzo[b][1]benzazepine-11-carboxamide | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/p2x-purinoceptor-4_5735588b93314c2f06862a4dc832fb8b.svg) | 5-Aminobenzo[b][1]benzazepine-11-carboxamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/p2x-purinoceptor-4_ed5c6806be966b451d93ce7029a26dd7.svg) | 2-Methoxybenzo[b][1]benzazepine-11-carboxamide | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/p2x-purinoceptor-4_f095876f759984e44ae2082bed74564c.svg) | 10-Benzyl-10H-phenoxazine | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/p2x-purinoceptor-4_87d335782e16414e376459dd8c65982c.svg) | (4-Methylphenyl)methyl phenoxazine-10-carboxylate | IC50 | 2280.0 [1] |
![](https://images.aatbio.com/dataset/ic50/p2x-purinoceptor-4_959a38c741440d165398d5f4ebf25354.svg) | (4-Methoxyphenyl)methyl phenoxazine-10-carboxylate | IC50 | 2640.0 [1] |
![](https://images.aatbio.com/dataset/ic50/p2x-purinoceptor-4_a2b906be5cd1b2e27bd5aba899d08141.svg) | N-Propan-2-ylphenoxazine-10-carboxamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/p2x-purinoceptor-4_30269edb77731a5d710bae8cf7d6a231.svg) | Phenoxazin-10-yl(piperidin-1-yl)methanone | IC50 | 10700.0 [1] |
![](https://images.aatbio.com/dataset/ic50/p2x-purinoceptor-4_7b8034f5895db0aa6addc982c88383a7.svg) | Methyl phenoxazine-10-carboxylate | IC50 | 52300.0 [1] |
![](https://images.aatbio.com/dataset/ic50/p2x-purinoceptor-4_4c97d2f77fe4eebbee64b5688acc7272.svg) | Benzyl 2H-benzo[b][1,4]oxazine-4(3H)-carboxylate | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/p2x-purinoceptor-4_7745b83513180560d8646225ab9b6316.svg) | 1-Phenoxazin-10-yl-2-phenylethanone | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/p2x-purinoceptor-4_40d8e1a1598c93569a835c5c72ee3f2f.svg) | N-[3-(Dimethylamino)propyl]phenoxazine-10-carboxamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/p2x-purinoceptor-4_d648500ee031c8c60c1dbedb850f8422.svg) | 10-Benzylsulfonylphenoxazine | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/p2x-purinoceptor-4_1f36ff44f441e3051137c4d72443cb0a.svg) | N-Methylphenoxazine-10-carboxamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/p2x-purinoceptor-4_b2e391278a4a002aa00c251b135ee228.svg) | N-Benzylphenoxazine-10-carboxamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/p2x-purinoceptor-4_80d9c9a034b2acab02ce10d5fbd191df.svg) | 2-Phenylethyl phenoxazine-10-carboxylate | IC50 | 3930.0 [1] |
![](https://images.aatbio.com/dataset/ic50/p2x-purinoceptor-4_3151596db571876b3f66f0f6f90f864b.svg) | S-(2-Phenylethyl) phenoxazine-10-carbothioate | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/p2x-purinoceptor-4_e7ad078098dc2b9ff0a9b3deb8c129a6.svg) | N,N-Diethyl-9-oxoacridine-10-carboxamide | IC50 | 39100.0 [1] |
![](https://images.aatbio.com/dataset/ic50/p2x-purinoceptor-4_cd60d3b52af16cd57d13c8e1369a9a9f.svg) | N-(2-Hydroxyphenyl)-2-[(1R,2S,5R)-5-methyl-2-propan-2-ylcyclohexyl]oxyacetamide | IC50 | 3390.0 [1] |
![](https://images.aatbio.com/dataset/ic50/p2x-purinoceptor-4_43041868883ba4432aaedfe51fd9c6d1.svg) | N-Cyclohexylphenoxazine-10-carboxamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/p2x-purinoceptor-4_89dc9aed7ab1f15498e55a3be664fb99.svg) | N,N-Diethylphenoxazine-10-carboxamide | IC50 | 17400.0 [1] |
![](https://images.aatbio.com/dataset/ic50/p2x-purinoceptor-4_7a05bbcf9decf492f1a701538e8138d8.svg) | (4-Nitrophenyl)methyl phenoxazine-10-carboxylate | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/p2x-purinoceptor-4_9b8dbfe22ac6d86653389bfd955d113e.svg) | N-[2-(2-Bromoethoxy)phenyl]-2-[(1R,2S,5R)-5-methyl-2-propan-2-ylcyclohexyl]oxyacetamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/p2x-purinoceptor-4_e31e801b74e0df946b67bf2a1e87b234.svg) | N-(2-Phenylethyl)phenoxazine-10-carboxamide | IC50 | 1780.0 [1] |
![](https://images.aatbio.com/dataset/ic50/p2x-purinoceptor-4_385924d069401cc10d9ab2f5e77a27e5.svg) | N,N-Di(propan-2-yl)phenoxazine-10-carboxamide | IC50 | 12400.0 [1] |
![](https://images.aatbio.com/dataset/ic50/p2x-purinoceptor-4_f9009b5c43d564b631cbbdbe606c0e94.svg) | (4-Chlorophenyl)-phenoxazin-10-ylmethanone | IC50 | 5290.0 [1] |
![](https://images.aatbio.com/dataset/ic50/p2x-purinoceptor-4_bf463d591ad832f0bb55528162d0fd29.svg) | 9-Phenyl-10-benzyl-9,10-dihydroacridine-9-ol | IC50 | 2440.0 [1] |
![](https://images.aatbio.com/dataset/ic50/p2x-purinoceptor-4_ae38c150371735975744ea020c17ffd6.svg) | 2,3-Dihydro-1,4-benzoxazin-4-yl(morpholin-4-yl)methanone | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/p2x-purinoceptor-4_be915d289ec60b4fa71ed1f27583e835.svg) | Phenoxazine-10-carboxamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/p2x-purinoceptor-4_f44bfaabe8b3369b8da402bc0afeae9b.svg) | N-(1-Methylpiperidin-4-yl)phenoxazine-10-carboxamide | IC50 | 45800.0 [1] |
![](https://images.aatbio.com/dataset/ic50/p2x-purinoceptor-4_e39f5b6103909d987fbfec7ca51de639.svg) | N,N-Dipropylphenoxazine-10-carboxamide | IC50 | 2690.0 [1] |
![](https://images.aatbio.com/dataset/ic50/p2x-purinoceptor-4_a63bf1c3fb6d1526ed8a1bedb16f6960.svg) | Morpholin-4-yl(phenoxazin-10-yl)methanone | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/p2x-purinoceptor-4_316f7b58866e22defd996b944f3b40ef.svg) | 10-[(4-Methylphenyl)methyl]acridin-9-one | IC50 | 11800.0 [1] |
![](https://images.aatbio.com/dataset/ic50/p2x-purinoceptor-4_5b909cefe484298704fc410b2a54c072.svg) | N-[(3,5-Dichlorophenyl)methyl]phenoxazine-10-carboxamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/p2x-purinoceptor-4_af326236bc607652b4f1ecdb50d05552.svg) | N,N-Dimethylphenoxazine-10-carboxamide | IC50 | 24600.0 [1] |
![](https://images.aatbio.com/dataset/ic50/p2x-purinoceptor-4_76533e42ffe2a883bdd6cdae1bd542c6.svg) | Propan-2-yl phenoxazine-10-carboxylate | IC50 | 2350.0 [1] |
![](https://images.aatbio.com/dataset/ic50/p2x-purinoceptor-4_502d4ce6866ebd75888f03b92121c6dd.svg) | (4-Chlorophenyl)methyl phenoxazine-10-carboxylate | IC50 | 1020.0 [1] |
![](https://images.aatbio.com/dataset/ic50/p2x-purinoceptor-4_a15b0dbcae027156522d0192dda4d88d.svg) | (4-Aminophenyl)-phenoxazin-10-ylmethanone | IC50 | 10800.0 [1] |
![](https://images.aatbio.com/dataset/ic50/p2x-purinoceptor-4_ca3e42e857bd7e40b2fff111528ec431.svg) | N-[(4-Chlorophenyl)methyl]phenoxazine-10-carboxamide | IC50 | 9540.0 [1] |
![](https://images.aatbio.com/dataset/ic50/p2x-purinoceptor-4_e814477a5345b441792a6d32199aadac.svg) | (4-Methylpiperazin-1-yl)-phenoxazin-10-ylmethanone | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/p2x-purinoceptor-4_25d35fa3ca70d0ee3eab124fa6cbbba1.svg) | N,N-Di(propan-2-yl)benzo[b][1]benzazepine-11-carboxamide | IC50 | 3440.0 [1] |
![](https://images.aatbio.com/dataset/ic50/p2x-purinoceptor-4_b0ab585de16f4c40d013c7c31ad3a27c.svg) | N-[2-(Dimethylamino)ethyl]-N-methylbenzo[b][1]benzazepine-11-carboxamide | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/p2x-purinoceptor-4_85c1926cf62f00c592482bbd260c96b0.svg) | N-(4-Aminocyclohexyl)benzo[b][1]benzazepine-11-carboxamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/p2x-purinoceptor-4_75dbecb1cdb2b1e3bf8bf662f347c0f0.svg) | Benzyl benzo[b][1]benzazepine-11-carboxylate | IC50 | 6020.0 [1] |
![](https://images.aatbio.com/dataset/ic50/p2x-purinoceptor-4_6080b948a7562dc3a75f1da3a1edccb3.svg) | 11-N,11-N-Diethyl-1-N,1-N-di(propan-2-yl)benzo[b][1]benzazepine-1,11-dicarboxamide | IC50 | 52500.0 [1] |
![](https://images.aatbio.com/dataset/ic50/p2x-purinoceptor-4_1af92317dcda952e17fbaf44ae181b4f.svg) | 2-Methylpropyl benzo[b][1]benzazepine-11-carboxylate | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/p2x-purinoceptor-4_ebdb138bf0ac02007ab8b1e76f4e4612.svg) | N-Tert-butylbenzo[b][1]benzazepine-11-carboxamide | IC50 | 13800.0 [1] |
![](https://images.aatbio.com/dataset/ic50/p2x-purinoceptor-4_98823bb1b0cea7779c30cbf8942b1c2b.svg) | N-(4-Hydroxycyclohexyl)benzo[b][1]benzazepine-11-carboxamide | IC50 | 20000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/p2x-purinoceptor-4_3958a4f92021753b1d5cc45619ebc39a.svg) | 2-(Dimethylamino)benzo[b][1]benzazepine-11-carboxamide | IC50 | 15300.0 [1] |
![](https://images.aatbio.com/dataset/ic50/p2x-purinoceptor-4_4967c7141ec5e11373e8aea611ce43b6.svg) | N-[2-(4-Methoxyphenyl)ethyl]benzo[b][1]benzazepine-11-carboxamide | IC50 | 27400.0 [1] |
![](https://images.aatbio.com/dataset/ic50/p2x-purinoceptor-4_955cb1f279c60eb3f33bb591a2108b07.svg) | N-Butylbenzo[b][1]benzazepine-11-carboxamide | IC50 | 100000.0 [1] |