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Opioid receptors; mu & kappa Inhibitors (IC50, Ki)

Structure
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Compound Name
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Standard Type
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▼
Standard Values (in nM)
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▼
NaloxoneIC509.0 [1], 127.0 [2]
NaltrexoneIC502.6 [1], 12.0 [2]
trans-3,4-Dichloro-N-methyl-N-[2-(1-pyrrolidinyl)cyclohexyl]-benzeneacetamideIC505.0 [1], 3100.0 [2]
LevallorphanIC500.67 [1], 2.6 [2]
CyprodimeIC50170.0 [1], 628.0 [2]
N-[(4R,4As,7S,7aR,12bS)-4a,9-dihydroxy-3-methyl-1,2,4,5,6,7,7a,13-octahydro-4,12-methanobenzofuro[3,2-e]isoquinolin-7-yl]acetamideIC5066.8 [1]
N,N'-Bis[(4R,4aS,7S,7aR,12bS)-4a,9-dihydroxy-3-methyl-1,2,4,5,6,7,7a,13-octahydro-4,12-methanobenzofuro[3,2-e]isoquinolin-7-yl]butanediamideIC5030.2 [1]
N,N'-Bis[2-[[2-[[2-[[(4R,4aS,7S,7aR,12bS)-4a,9-dihydroxy-3-methyl-1,2,4,5,6,7,7a,13-octahydro-4,12-methanobenzofuro[3,2-e]isoquinolin-7-yl]amino]-2-oxoethyl]amino]-2-oxoethyl]amino]-2-oxoethyl]butanediamideIC5025.1 [1]
N,N'-Bis[2-[[2-[[(4R,4aS,7S,7aR,12bS)-4a,9-dihydroxy-3-methyl-1,2,4,5,6,7,7a,13-octahydro-4,12-methanobenzofuro[3,2-e]isoquinolin-7-yl]amino]-2-oxoethyl]amino]-2-oxoethyl]butanediamideIC503.9 [1]
N,N'-Bis[2-[[(4R,4aS,7S,7aR,12bS)-4a,9-dihydroxy-3-methyl-1,2,4,5,6,7,7a,13-octahydro-4,12-methanobenzofuro[3,2-e]isoquinolin-7-yl]amino]-2-oxoethyl]butanediamideIC5022.0 [1]
N,N'-Bis[(4R,4aR,7R,7aS,12bS)-4a,9-dihydroxy-3-methyl-1,2,4,5,6,7,7a,13-octahydro-4,12-methanobenzofuro[3,2-e]isoquinolin-7-yl]butanediamideIC5015.7 [1]
N,N'-Bis[2-[[(4R,4aR,7R,7aS,12bS)-4a,9-dihydroxy-3-methyl-1,2,4,5,6,7,7a,13-octahydro-4,12-methanobenzofuro[3,2-e]isoquinolin-7-yl]amino]-2-oxoethyl]butanediamideIC5019.2 [1]
N,N'-Bis[2-[[2-[[(4R,4aR,7R,7aS,12bS)-4a,9-dihydroxy-3-methyl-1,2,4,5,6,7,7a,13-octahydro-4,12-methanobenzofuro[3,2-e]isoquinolin-7-yl]amino]-2-oxoethyl]amino]-2-oxoethyl]butanediamideIC506.3 [1]
N-[(4R,4As,7R,7aR,12bS)-4a,9-dihydroxy-3-methyl-1,2,4,5,6,7,7a,13-octahydro-4,12-methanobenzofuro[3,2-e]isoquinolin-7-yl]acetamideIC5045.9 [1]
N,N'-Bis[2-[[2-[[2-[[(4R,4aR,7R,7aS,12bS)-4a,9-dihydroxy-3-methyl-1,2,4,5,6,7,7a,13-octahydro-4,12-methanobenzofuro[3,2-e]isoquinolin-7-yl]amino]-2-oxoethyl]amino]-2-oxoethyl]amino]-2-oxoethyl]butanediamideIC5012.6 [1]
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References

This online tool may be cited as follows

MLA

"Quest Database™ Opioid receptors; mu & kappa Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 20 Feb. 2025, https://www.aatbio.com/data-sets/opioid-receptors-mu-kappa-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2025, February 20). Quest Database™ Opioid receptors; mu & kappa Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/opioid-receptors-mu-kappa-inhibitors-ic50-ki.
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