 | 4-[(1R,5S)-9-(3-Bicyclo[3.3.1]nonanyl)-9-azabicyclo[3.3.1]nonan-3-yl]-3-oxoquinoxaline-2-carboxylic acid | Ki | 2.4 [1], 178.0 [2] |
 | 4-[(1R,5S)-8-Cycloundecyl-8-azabicyclo[3.2.1]octan-3-yl]-3-oxoquinoxaline-2-carboxylic acid | Ki | 9.0 [1] |
 | 4-[(1R,5S)-8-Cyclododecyl-8-azabicyclo[3.2.1]octan-3-yl]-3-oxoquinoxaline-2-carboxylic acid | Ki | 43.1 [1] |
 | 4-[(1R,5S)-8-(3-Bicyclo[3.3.1]nonanyl)-8-azabicyclo[3.2.1]octan-3-yl]-3-oxoquinoxaline-2-carboxylic acid | Ki | 5.7 [1] |
 | (1S,2S,6R,14R,15R,16R)-5-(Cyclopropylmethyl)-11,15-dimethoxy-16-(phenylmethoxymethyl)-13-oxa-5-azahexacyclo[13.2.2.12,8.01,6.02,14.012,20]icosa-8(20),9,11-triene | Ki | 532.0 [1], 859.27 [2] |
 | 4-[(1R,5S)-8-Cyclooctyl-8-azabicyclo[3.2.1]octan-3-yl]-3-oxoquinoxaline-2-carboxylic acid | Ki | 12.6 [1], 299.0 [2] |
 | (2S)-2-[[4-[(1R,5S)-8-Cyclooctyl-8-azabicyclo[3.2.1]octan-3-yl]-3-oxoquinoxalin-2-yl]amino]-3-hydroxypropanoic acid | Ki | 8.2 [1], 285.0 [2] |
 | 2-[[4-[(1R,5S)-8-Cyclooctyl-8-azabicyclo[3.2.1]octan-3-yl]-3-oxoquinoxalin-2-yl]amino]acetic acid | Ki | 61.4 [1], 1716.0 [2] |
 | 2-[[4-[(1R,5S)-8-Cyclooctyl-8-azabicyclo[3.2.1]octan-3-yl]-3-oxoquinoxalin-2-yl]amino]acetamide | Ki | 6.42 [1], 233.7 [2] |
 | 4-[(1R,5S)-8-Cyclooctyl-8-azabicyclo[3.2.1]octan-3-yl]-3-oxo-N-(6-oxo-1H-pyridin-3-yl)quinoxaline-2-carboxamide | Ki | 7.5 [1], 103.0 [2] |
 | 3-Oxo-4-[(1R,5S)-8-(3-tricyclo[3.3.1.03,7]nonanyl)-8-azabicyclo[3.2.1]octan-3-yl]quinoxaline-2-carboxylic acid | Ki | 15.4 [1], 364.0 [2] |
 | 1-[(1R,5S)-8-Cyclooctyl-8-azabicyclo[3.2.1]octan-3-yl]-3-[[(2R)-2,3-dihydroxypropyl]amino]quinoxalin-2-one | Ki | 6.5 [1], 288.0 [2] |
 | 4-[(1R,5S)-8-(1-Adamantyl)-8-azabicyclo[3.2.1]octan-3-yl]-3-oxoquinoxaline-2-carboxylic acid | Ki | 89.9 [1], 275.0 [2] |
 | Cebranopadol | Ki | 22.0 [1] |
 | N-[(E)-(2,3-Dihydroxyphenyl)methylideneamino]-4-[(4,6-dimethylpyrimidin-2-yl)sulfanylmethyl]benzamide | Ki | 836.0 [1] |
 | N,N-Dimethyl-1'-phenylspiro[4,9-dihydro-3H-pyrano[3,4-b]indole-1,4'-cyclohexane]-1'-amine | Ki | 0.6 [1] |
 | (1S,2S,6R,14R,15R,16R)-5-(Cyclopropylmethyl)-16-[(3,4-dichlorophenyl)methoxymethyl]-11,15-dimethoxy-5-methyl-13-oxa-5-azoniahexacyclo[13.2.2.12,8.01,6.02,14.012,20]icosa-8(20),9,11-triene | Ki | 20000.0 [1] |
 | (1S,2S,6R,14R,15R,16R)-5-(Cyclopropylmethyl)-11,15-dimethoxy-5-methyl-16-[(4-methylphenyl)methoxymethyl]-13-oxa-5-azoniahexacyclo[13.2.2.12,8.01,6.02,14.012,20]icosa-8(20),9,11-triene | Ki | 20000.0 [1] |
 | 3-Amino-1-[4-[(1R,5S)-9-[(1S,6R)-8-bicyclo[4.3.1]decanyl]-9-azabicyclo[3.3.1]nonan-3-yl]-3-oxoquinoxalin-2-yl]azetidine-3-carboxylic acid | Ki | 0.22 [1] |
 | (2S)-1-[4-[(1R,5S)-9-[(1S,5R)-3-Bicyclo[3.3.1]nonanyl]-9-azabicyclo[3.3.1]nonan-3-yl]-3-oxoquinoxalin-2-yl]azetidine-2-carboxylic acid | Ki | 27.1 [1] |
 | 1-[4-[(1R,5S)-9-[(1S,6R)-8-Bicyclo[4.3.1]decanyl]-9-azabicyclo[3.3.1]nonan-3-yl]-3-oxoquinoxalin-2-yl]-3-(dimethylamino)azetidine-3-carboxylic acid | Ki | 0.34 [1] |
 | (2S,3R)-1-[4-[(1R,5S)-9-[(1S,6R)-8-Bicyclo[4.3.1]decanyl]-9-azabicyclo[3.3.1]nonan-3-yl]-3-oxoquinoxalin-2-yl]-3-(methylamino)azetidine-2-carboxylic acid | Ki | 1.98 [1] |
 | (2R)-1-[4-[(1R,5S)-8-[(1S,5R)-7-Methyl-3-bicyclo[3.3.1]nonanyl]-8-azabicyclo[3.2.1]octan-3-yl]-3-oxoquinoxalin-2-yl]azetidine-2-carboxylic acid | Ki | 43.0 [1] |
 | 2-[1-[4-[(1R,5S)-9-[(1S,5R)-7-Methyl-3-bicyclo[3.3.1]nonanyl]-9-azabicyclo[3.3.1]nonan-3-yl]-3-oxoquinoxalin-2-yl]azetidin-3-yl]acetic acid | Ki | 1.03 [1] |
 | (2R)-1-[4-[(1R,5S)-9-[(1S,5R)-7-Methyl-3-bicyclo[3.3.1]nonanyl]-9-azabicyclo[3.3.1]nonan-3-yl]-3-oxoquinoxalin-2-yl]azetidine-2-carboxylic acid | Ki | 9.8 [1] |
 | (2S)-1-[4-[(1S,5R)-9-[(1S,5R)-3-Bicyclo[3.3.1]nonanyl]-3-oxa-9-azabicyclo[3.3.1]nonan-7-yl]-3-oxoquinoxalin-2-yl]azetidine-2-carboxylic acid | Ki | 294.0 [1] |
 | (2S,3R)-1-[4-[(1R,5S)-9-[(1S,5R)-3-Bicyclo[3.3.1]nonanyl]-9-azabicyclo[3.3.1]nonan-3-yl]-3-oxoquinoxalin-2-yl]-3-(dimethylamino)azetidine-2-carboxylic acid | Ki | 23.0 [1] |
 | (2R)-1-[4-[(1R,5S)-9-[(1S,3S,5R,7S)-9-Methyl-5-tricyclo[5.2.1.03,9]decanyl]-9-azabicyclo[3.3.1]nonan-3-yl]-3-oxoquinoxalin-2-yl]azetidine-2-carboxylic acid | Ki | 0.89 [1] |
 | (2S)-1-[4-[(1R,5S)-8-[(1S,5R)-7-Methyl-3-bicyclo[3.3.1]nonanyl]-8-azabicyclo[3.2.1]octan-3-yl]-3-oxoquinoxalin-2-yl]azetidine-2-carboxylic acid | Ki | 19.2 [1] |
 | (2S)-1-[4-[(1R,5S)-9-[(1S,3S,5R,7S)-9-Methyl-5-tricyclo[5.2.1.03,9]decanyl]-9-azabicyclo[3.3.1]nonan-3-yl]-3-oxoquinoxalin-2-yl]azetidine-2-carboxylic acid | Ki | 7.44 [1] |
 | 1-[4-[(1R,5S)-9-[(1S,3S,5R,7S)-9-Methyl-5-tricyclo[5.2.1.03,9]decanyl]-3-oxa-9-azabicyclo[3.3.1]nonan-7-yl]-3-oxoquinoxalin-2-yl]azetidine-3-carboxylic acid | Ki | 381.0 [1] |
 | (2S,3S)-1-[4-[(1R,5S)-9-[(1S,5R)-3-Bicyclo[3.3.1]nonanyl]-9-azabicyclo[3.3.1]nonan-3-yl]-3-oxoquinoxalin-2-yl]-3-methoxyazetidine-2-carboxylic acid | Ki | 11.9 [1] |
 | (2S)-1-[4-[(1R,5S)-9-[(1S,3S,5R,7S)-9-Methyl-5-tricyclo[5.2.1.03,9]decanyl]-3-oxa-9-azabicyclo[3.3.1]nonan-7-yl]-3-oxoquinoxalin-2-yl]azetidine-2-carboxylic acid | Ki | 55.5 [1] |
 | (2S)-1-[4-[(1S,5R)-9-[2-[(1S,2S,5S)-6,6-Dimethyl-2-bicyclo[3.1.1]heptanyl]ethyl]-9-azabicyclo[3.3.1]nonan-3-yl]-3-oxoquinoxalin-2-yl]azetidine-2-carboxylic acid | Ki | 23.6 [1] |
 | (2S,3R)-3-Amino-1-[4-[(1R,5S)-9-[(1S,6R)-8-bicyclo[4.3.1]decanyl]-9-azabicyclo[3.3.1]nonan-3-yl]-3-oxoquinoxalin-2-yl]azetidine-2-carboxylic acid | Ki | 1.98 [1] |
 | (2S,3R)-1-[4-[(1R,5S)-9-[(1S,6R)-8-Bicyclo[4.3.1]decanyl]-9-azabicyclo[3.3.1]nonan-3-yl]-3-oxoquinoxalin-2-yl]-3-(dimethylamino)azetidine-2-carboxylic acid | Ki | 1.97 [1] |
 | (2S)-1-[4-[(1R,5S)-9-[(1S,5R)-3-Bicyclo[3.3.1]nonanyl]-9-azabicyclo[3.3.1]nonan-3-yl]-3-oxoquinoxalin-2-yl]pyrrolidine-2-carboxylic acid | Ki | 98.0 [1] |
 | (2S)-1-[4-[(1R,5S)-9-[(1S,3S,5R,7S)-9-Methyl-5-tricyclo[5.2.1.03,9]decanyl]-9-azabicyclo[3.3.1]nonan-3-yl]-3-oxoquinoxalin-2-yl]pyrrolidine-2-carboxylic acid | Ki | 15.0 [1] |
 | 2-[1-[4-[(1R,5S)-9-[(1S,3S,5R,7S)-9-Methyl-5-tricyclo[5.2.1.03,9]decanyl]-3-oxa-9-azabicyclo[3.3.1]nonan-7-yl]-3-oxoquinoxalin-2-yl]azetidin-3-yl]acetic acid | Ki | 264.0 [1] |
 | (2S)-1-[4-[(1S,5R)-9-[(1R,5S)-3-Bicyclo[3.3.2]decanyl]-3-oxa-9-azabicyclo[3.3.1]nonan-7-yl]-3-oxoquinoxalin-2-yl]pyrrolidine-2-carboxylic acid | Ki | 511.0 [1] |
 | 2-[1-[4-[(1R,5S)-9-[(1S,6R)-8-Bicyclo[4.3.1]decanyl]-9-azabicyclo[3.3.1]nonan-3-yl]-3-oxoquinoxalin-2-yl]azetidin-3-yl]acetic acid | Ki | 1.32 [1] |
 | (2S)-1-[4-[(1R,5S)-9-[(1S,3S,5R,7S)-9-Methyl-5-tricyclo[5.2.1.03,9]decanyl]-3-oxa-9-azabicyclo[3.3.1]nonan-7-yl]-3-oxoquinoxalin-2-yl]pyrrolidine-2-carboxylic acid | Ki | 272.0 [1] |
 | (2R)-1-[4-[(1S,5R)-9-[2-[(1S,2S,5S)-6,6-Dimethyl-2-bicyclo[3.1.1]heptanyl]ethyl]-9-azabicyclo[3.3.1]nonan-3-yl]-3-oxoquinoxalin-2-yl]azetidine-2-carboxylic acid | Ki | 80.0 [1] |
 | (2S,3R)-3-Acetamido-1-[4-[(1R,5S)-9-[(1S,5R)-3-bicyclo[3.3.1]nonanyl]-9-azabicyclo[3.3.1]nonan-3-yl]-3-oxoquinoxalin-2-yl]azetidine-2-carboxylic acid | Ki | 39.9 [1] |
 | (2S,3R)-3-Acetamido-1-[4-[(1R,5S)-9-[(1S,6R)-8-bicyclo[4.3.1]decanyl]-9-azabicyclo[3.3.1]nonan-3-yl]-3-oxoquinoxalin-2-yl]azetidine-2-carboxylic acid | Ki | 3.14 [1] |
 | (1S,2S,6R,14R,15R,16R)-5-(Cyclopropylmethyl)-16-[[4-(1,1-difluoroethyl)phenyl]methoxymethyl]-11,15-dimethoxy-5-methyl-13-oxa-5-azoniahexacyclo[13.2.2.12,8.01,6.02,14.012,20]icosa-8(20),9,11-triene | Ki | 20000.0 [1] |
 | N,N,3,6-Tetramethyl-1'-phenylspiro[4,9-dihydro-3H-pyrano[3,4-b]indole-1,4'-cyclohexane]-1'-amine | Ki | 4.4 [1] |
 | 1'-(4-Fluorophenyl)-N,N-dimethylspiro[4,9-dihydro-3H-pyrano[3,4-b]indole-1,4'-cyclohexane]-1'-amine | Ki | 3.2 [1] |
 | 7-Fluoro-N,N-dimethyl-1'-phenylspiro[2,3,4,9-tetrahydropyrido[3,4-b]indole-1,4'-cyclohexane]-1'-amine | Ki | 6.9 [1] |
 | 1-[1'-(Dimethylamino)-1'-phenylspiro[4,9-dihydro-3H-pyrido[3,4-b]indole-1,4'-cyclohexane]-2-yl]ethanone | Ki | 2.4 [1] |
 | 1'-(3-Fluorophenyl)-N,N-dimethylspiro[4,9-dihydro-3H-pyrano[3,4-b]indole-1,4'-cyclohexane]-1'-amine | Ki | 1.2 [1] |
 | N,N-Dimethyl-1'-phenylspiro[2,3,4,9-tetrahydropyrido[3,4-b]indole-1,4'-cyclohexane]-1'-amine | Ki | 3.4 [1] |
 | N,N,3-Trimethyl-1'-phenylspiro[4,9-dihydro-3H-pyrano[3,4-b]indole-1,4'-cyclohexane]-1'-amine | Ki | 42.0 [1] |
 | N,N-Dimethyl-1'-phenylspiro[4,9-dihydro-3H-thiopyrano[3,4-b]indole-1,4'-cyclohexane]-1'-amine | Ki | 3.7 [1] |
 | N,N,3-Trimethyl-6-nitro-1'-phenylspiro[4,9-dihydro-3H-pyrano[3,4-b]indole-1,4'-cyclohexane]-1'-amine | Ki | 29.0 [1] |
 | N,N,3-Trimethyl-1'-phenylspiro[2,3,4,9-tetrahydropyrido[3,4-b]indole-1,4'-cyclohexane]-1'-amine | Ki | 0.5 [1] |
 | 6-Fluoro-N,N,3-trimethyl-1'-phenylspiro[4,9-dihydro-3H-pyrano[3,4-b]indole-1,4'-cyclohexane]-1'-amine | Ki | 83.0 [1] |
 | 1'-(Dimethylamino)-1'-phenylspiro[4,9-dihydro-3H-pyrano[3,4-b]indole-1,4'-cyclohexane]-6-ol | Ki | 1.6 [1] |
 | 1'-Benzyl-N,N-dimethylspiro[2,3,4,9-tetrahydropyrido[3,4-b]indole-1,4'-cyclohexane]-1'-amine | Ki | 1.1 [1] |
 | 6-Fluoro-N,N-dimethyl-1'-phenylspiro[2,3,4,9-tetrahydropyrido[3,4-b]indole-1,4'-cyclohexane]-1'-amine | Ki | 1.4 [1] |
 | N,N,6-Trimethyl-1'-phenylspiro[2,3,4,9-tetrahydropyrido[3,4-b]indole-1,4'-cyclohexane]-1'-amine | Ki | 32.0 [1] |
 | 6-Bromo-N,N,3-trimethyl-1'-phenylspiro[4,9-dihydro-3H-pyrano[3,4-b]indole-1,4'-cyclohexane]-1'-amine | Ki | 23.0 [1] |
 | 6-Bromo-N,N-dimethyl-1'-phenylspiro[4,9-dihydro-3H-pyrano[3,4-b]indole-1,4'-cyclohexane]-1'-amine | Ki | 52.0 [1] |
 | 6-Methoxy-N,N-dimethyl-1'-phenylspiro[4,9-dihydro-3H-pyrano[3,4-b]indole-1,4'-cyclohexane]-1'-amine | Ki | 5.8 [1] |
 | Lexanopadol | Ki | 10.0 [1] |
 | N-Methyl-1'-phenylspiro[4,9-dihydro-3H-pyrano[3,4-b]indole-1,4'-cyclohexane]-1'-amine | Ki | 1.4 [1] |
 | 2-[[(3S)-1-[4-(1-Cyclooctylpiperidin-4-yl)-3-oxoquinoxalin-2-yl]pyrrolidin-3-yl]amino]acetic acid | Ki | 500.0 [1] |
 | 3-(2,3,3a,4,6,6a-Hexahydro-1H-pyrrolo[3,4-c]pyrrole-5-carbonyl)-1-(1-cyclooctylpiperidin-4-yl)quinoxalin-2-one | Ki | 52.8 [1] |
 | 1-[4-[3-(2,3,3a,4,6,6a-Hexahydro-1H-pyrrolo[3,4-c]pyrrol-5-yl)-2-oxoquinoxalin-1-yl]piperidin-1-yl]cyclooctane-1-carboxamide | Ki | 44.6 [1] |
 | N,N,6-Trimethyl-1'-phenylspiro[4,9-dihydro-3H-pyrano[3,4-b]indole-1,4'-cyclohexane]-1'-amine | Ki | 4.5 [1] |
 | 1'-(4-Fluorophenyl)-N,N-dimethyl-2-oxospiro[3,4-dihydrothiopyrano[3,4-b][1]benzothiole-1,4'-cyclohexane]-1'-amine | Ki | 62.0 [1] |
 | Methyl 1'-(dimethylamino)-1'-phenylspiro[2,3,4,9-tetrahydropyrido[3,4-b]indole-1,4'-cyclohexane]-3-carboxylate | Ki | 0.9 [1] |
 | (1S,2S,6R,14R,15R,16R)-5-(Cyclopropylmethyl)-11,15-dimethoxy-16-[[4-(trifluoromethyl)phenyl]methoxymethyl]-13-oxa-5-azahexacyclo[13.2.2.12,8.01,6.02,14.012,20]icosa-8(20),9,11-triene | Ki | 3957.55 [1] |
 | (1S,2S,6R,14R,15R,16R)-16-(Cyclohexylmethoxymethyl)-11,15-dimethoxy-5-methyl-13-oxa-5-azahexacyclo[13.2.2.12,8.01,6.02,14.012,20]icosa-8(20),9,11-triene | Ki | 1034.67 [1] |
 | (1S,2S,6R,14R,15R,16R)-11,15-Dimethoxy-5-methyl-16-[[4-(trifluoromethyl)phenyl]methoxymethyl]-13-oxa-5-azahexacyclo[13.2.2.12,8.01,6.02,14.012,20]icosa-8(20),9,11-triene | Ki | 13803.96 [1] |
 | (1S,2S,6R,14R,15R,16R)-5-(Cyclopropylmethyl)-16-[(3,4-dichlorophenyl)methoxymethyl]-11,15-dimethoxy-13-oxa-5-azahexacyclo[13.2.2.12,8.01,6.02,14.012,20]icosa-8(20),9,11-triene | Ki | 823.29 [1] |
 | (2S,6R)-11,15-Dimethoxy-5-methyl-16-(phenylmethoxymethyl)-13-oxa-5-azahexacyclo[13.2.2.12,8.01,6.02,14.012,20]icosa-8(20),9,11-triene | Ki | 569.0 [1] |
 | (2S,6R)-11,15-Dimethoxy-5-methyl-16-(prop-2-enoxymethyl)-13-oxa-5-azahexacyclo[13.2.2.12,8.01,6.02,14.012,20]icosa-8(20),9,11-triene | Ki | 1295.55 [1] |
 | (1S,2S,6R,14R,15R,16R)-16-[(4-Tert-butylphenyl)methoxymethyl]-11,15-dimethoxy-5-methyl-13-oxa-5-azahexacyclo[13.2.2.12,8.01,6.02,14.012,20]icosa-8(20),9,11-triene | Ki | 4555.05 [1] |
 | (1S,2S,6R,14R,15R,16R)-11,15-Dimethoxy-5-methyl-16-(phenoxymethyl)-13-oxa-5-azahexacyclo[13.2.2.12,8.01,6.02,14.012,20]icosa-8(20),9,11-triene | Ki | 2571.83 [1] |
 | (1S,2S,6R,14R,15R,16R)-16-(Cyclohexylmethoxymethyl)-5-(cyclopropylmethyl)-11,15-dimethoxy-13-oxa-5-azahexacyclo[13.2.2.12,8.01,6.02,14.012,20]icosa-8(20),9,11-triene | Ki | 1165.91 [1] |
 | (1S,2S,6R,14R,15R,16R)-11,15-Dimethoxy-5-methyl-16-[(3-methylphenyl)methoxymethyl]-13-oxa-5-azahexacyclo[13.2.2.12,8.01,6.02,14.012,20]icosa-8(20),9,11-triene | Ki | 1602.42 [1] |
 | (1S,2S,6R,14R,15R,16R)-5-(Cyclopropylmethyl)-11,15-dimethoxy-16-[(4-phenylphenyl)methoxymethyl]-13-oxa-5-azahexacyclo[13.2.2.12,8.01,6.02,14.012,20]icosa-8(20),9,11-triene | Ki | 20000.0 [1] |
 | (1S,2S,6R,14R,15R,16R)-16-[(4-Chlorophenyl)methoxymethyl]-11,15-dimethoxy-5-methyl-13-oxa-5-azahexacyclo[13.2.2.12,8.01,6.02,14.012,20]icosa-8(20),9,11-triene | Ki | 1116.98 [1] |
 | (1S,2S,6R,14R,15R,16R)-5-(Cyclopropylmethyl)-11,15-dimethoxy-16-(phenoxymethyl)-13-oxa-5-azahexacyclo[13.2.2.12,8.01,6.02,14.012,20]icosa-8(20),9,11-triene | Ki | 9605.7 [1] |
 | (1S,2S,6R,14R,15R,16R)-11,15-Dimethoxy-5-methyl-16-(naphthalen-2-ylmethoxymethyl)-13-oxa-5-azahexacyclo[13.2.2.12,8.01,6.02,14.012,20]icosa-8(20),9,11-triene | Ki | 20000.0 [1] |
 | 4-[(1R,5S)-9-Cyclodecyl-9-azabicyclo[3.3.1]nonan-3-yl]-3-oxoquinoxaline-2-carboxylic acid | Ki | 1.8 [1] |
 | 4-[(1R,5S)-9-[(1S,5R)-7-Methyl-3-bicyclo[3.3.1]nonanyl]-9-azabicyclo[3.3.1]nonan-3-yl]-3-oxoquinoxaline-2-carboxylic acid | Ki | 1.1 [1] |
 | 4-[(1R,5S)-8-(9-Bicyclo[3.3.1]nonanyl)-8-azabicyclo[3.2.1]octan-3-yl]-3-oxoquinoxaline-2-carboxylic acid | Ki | 4.8 [1] |
 | 4-[(1R,5S)-8-Cyclononyl-8-azabicyclo[3.2.1]octan-3-yl]-3-oxoquinoxaline-2-carboxylic acid | Ki | 2.0 [1] |
 | 4-[(1R,5S)-9-Cyclononyl-9-azabicyclo[3.3.1]nonan-3-yl]-3-oxoquinoxaline-2-carboxylic acid | Ki | 1.4 [1] |
 | 4-[(1R,5S)-8-Cyclodecyl-8-azabicyclo[3.2.1]octan-3-yl]-3-oxoquinoxaline-2-carboxylic acid | Ki | 2.5 [1] |
 | 4-[(1R,5S)-9-(1-Bicyclo[3.3.1]nonanyl)-9-azabicyclo[3.3.1]nonan-3-yl]-3-oxoquinoxaline-2-carboxylic acid | Ki | 30.2 [1] |
 | 4-[(1R,5S)-8-Cyclooctyl-8-azabicyclo[3.2.1]octan-3-yl]-3-oxo-N-(2H-tetrazol-5-ylmethyl)quinoxaline-2-carboxamide | Ki | 157.0 [1] |
 | 4-[(1R,5S)-8-Cyclooctyl-8-azabicyclo[3.2.1]octan-3-yl]-N-hydroxy-3-oxoquinoxaline-2-carboxamide | Ki | 2.7 [1] |
 | 2-[2-[4-(1-Cyclooctylpiperidin-4-yl)-3-oxoquinoxalin-2-yl]-1,3,3a,4,6,6a-hexahydropyrrolo[3,4-c]pyrrol-5-yl]-2-oxoacetic acid | Ki | 71.4 [1] |
 | 3-(5-Acetyl-1,3,3a,4,6,6a-hexahydropyrrolo[3,4-c]pyrrol-2-yl)-1-(1-cyclooctylpiperidin-4-yl)quinoxalin-2-one | Ki | 96.5 [1] |
 | (1S,3R)-3-[[4-(1-Cyclooctylpiperidin-4-yl)-3-oxoquinoxalin-2-yl]amino]cyclopentane-1-carboxylic acid | Ki | 607.4 [1] |
 | 4-[[[4-[(1R,5S)-8-Cyclooctyl-8-azabicyclo[3.2.1]octan-3-yl]-3-oxoquinoxalin-2-yl]amino]methyl]benzoic acid | Ki | 456.0 [1] |
 | 3-[(3S)-3-Aminopyrrolidin-1-yl]-1-(1-cyclooctylpiperidin-4-yl)quinoxalin-2-one | Ki | 4.0 [1] |
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