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Oligosaccharyl transferase 48 kDa subunit Inhibitors (IC50, Ki)

Structure
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Compound Name
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Standard Type
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Standard Values (in nM)
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(3R,6S)-6-(2-Aminoethyl)-N-[(2S,3R)-1-[[(2S)-1-[[(2S,3R)-1-amino-3-hydroxy-1-oxobutan-2-yl]amino]-3-methyl-1-oxobutan-2-yl]amino]-3-hydroxy-1-oxobutan-2-yl]-5,8-dioxo-1-thia-4,7-diazacyclotridecane-3-carboxamideKi82.0 [1]
(3R,6S)-N-[(2S,3R)-1-[[(2S)-1-[[(2S,3R)-1-[[(2S)-1-Amino-3-(4-nitrophenyl)-1-oxopropan-2-yl]amino]-3-hydroxy-1-oxobutan-2-yl]amino]-3-methyl-1-oxobutan-2-yl]amino]-3-hydroxy-1-oxobutan-2-yl]-6-[2-(decylamino)ethyl]-5,8-dioxo-1-thia-4,7-diazacyclotridecane-3-carboxamideKi61.0 [1]
(3R,6S)-N-[(2S,3R)-1-[[(2S)-1-[[(2S,3R)-1-[[(2S)-1-Amino-3-(4-nitrophenyl)-1-oxopropan-2-yl]amino]-3-hydroxy-1-oxobutan-2-yl]amino]-3-methyl-1-oxobutan-2-yl]amino]-3-hydroxy-1-oxobutan-2-yl]-6-[2-(naphthalen-2-ylamino)ethyl]-5,8-dioxo-1-thia-4,7-diazacyclotridecane-3-carboxamideKi40.0 [1]
(3R,6S)-6-(2-Aminoethyl)-N-[(2S,3R)-1-[[(2S)-1-[[(2S,3R)-1-[[(2S)-1-amino-3-(4-nitrophenyl)-1-oxopropan-2-yl]amino]-3-hydroxy-1-oxobutan-2-yl]amino]-3-methyl-1-oxobutan-2-yl]amino]-3-hydroxy-1-oxobutan-2-yl]-5,8-dioxo-1-thia-4,7-diazacyclotridecane-3-carboxamideKi37.0 [1]
(3R,6S)-N-[(2S,3R)-3-Hydroxy-1-[[(2S)-1-[[(2S,3R)-3-hydroxy-1-[2-(4-nitrophenyl)ethylamino]-1-oxobutan-2-yl]amino]-3-methyl-1-oxobutan-2-yl]amino]-1-oxobutan-2-yl]-6-[2-(naphthalen-2-ylamino)ethyl]-5,8-dioxo-1-thia-4,7-diazacyclotridecane-3-carboxamideKi10.0 [1]
(3R,6S)-6-(2-Aminoethyl)-N-[(2S,3R)-3-hydroxy-1-[[(2S)-1-[[(2S,3R)-3-hydroxy-1-[2-(4-nitrophenyl)ethylamino]-1-oxobutan-2-yl]amino]-3-methyl-1-oxobutan-2-yl]amino]-1-oxobutan-2-yl]-5,8-dioxo-1-thia-4,7-diazacyclotridecane-3-carboxamideKi20.0 [1]
(3R,6S)-6-(2-Aminoethyl)-N-[(2S,3R)-3-hydroxy-1-[[(2S)-1-[[(2S,3R)-3-hydroxy-1-oxo-1-(4-phenylbutylamino)butan-2-yl]amino]-3-methyl-1-oxobutan-2-yl]amino]-1-oxobutan-2-yl]-5,8-dioxo-1-thia-4,7-diazacyclotridecane-3-carboxamideKi50.0 [1]
(3R,6S)-N-[(2S,3R)-3-Hydroxy-1-[[(2S)-1-[[(2S,3R)-3-hydroxy-1-oxo-1-(2-phenylethylamino)butan-2-yl]amino]-3-methyl-1-oxobutan-2-yl]amino]-1-oxobutan-2-yl]-6-[2-(naphthalen-2-ylamino)ethyl]-5,8-dioxo-1-thia-4,7-diazacyclotridecane-3-carboxamideKi18.0 [1]
(3R,6S)-6-(2-Aminoethyl)-N-[(2S,3R)-3-hydroxy-1-[[(2S)-1-[[(2S,3R)-3-hydroxy-1-oxo-1-(2-phenylethylamino)butan-2-yl]amino]-3-methyl-1-oxobutan-2-yl]amino]-1-oxobutan-2-yl]-5,8-dioxo-1-thia-4,7-diazacyclotridecane-3-carboxamideKi44.0 [1]
(3R,6S)-N-[(2S,3R)-1-[[(2S)-1-[[(2S,3R)-1-[[(2S)-1-Amino-3-(4-nitrophenyl)-1-oxopropan-2-yl]amino]-3-hydroxy-1-oxobutan-2-yl]amino]-3-methyl-1-oxobutan-2-yl]amino]-3-hydroxy-1-oxobutan-2-yl]-6-[2-(naphthalen-1-ylamino)ethyl]-5,8-dioxo-1-thia-4,7-diazacyclotridecane-3-carboxamideKi98.0 [1]
(2S)-N-[2-[[(2S,3R)-1-[[(2S)-1-[[(2S,3R)-1-Amino-3-hydroxy-1-oxobutan-2-yl]amino]-3-methyl-1-oxobutan-2-yl]amino]-3-hydroxy-1-oxobutan-2-yl]amino]-2-oxoethyl]-2-(benzylamino)-5-[(4-nitrophenyl)methylamino]pentanamideKi154.0 [1]
(2S)-N-[2-[[(2S,3R)-1-[[(2S)-1-[[(2S,3S)-1-Amino-3-hydroxy-1-oxobutan-2-yl]amino]-3-methyl-1-oxobutan-2-yl]amino]-3-hydroxy-1-oxobutan-2-yl]amino]-2-oxoethyl]-2,5-bis(benzylamino)pentanamideKi5000.0 [1]
(2S)-N-[2-[[(2S,3R)-1-[[(2S)-1-[[(2S,3R)-1-Amino-3-hydroxy-1-oxobutan-2-yl]amino]-3-methyl-1-oxobutan-2-yl]amino]-3-hydroxy-1-oxobutan-2-yl]amino]-2-oxoethyl]-2-(benzylamino)-5-[(4-methoxyphenyl)methylamino]pentanamideKi305.0 [1]
Items per page: 1 - 10 of 13
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References

This online tool may be cited as follows

MLA

"Quest Database™ Oligosaccharyl transferase 48 kDa subunit Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 21 Nov. 2024, https://www.aatbio.com/data-sets/oligosaccharyl-transferase-48-kda-subunit-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, November 21). Quest Database™ Oligosaccharyl transferase 48 kDa subunit Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/oligosaccharyl-transferase-48-kda-subunit-inhibitors-ic50-ki.
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