![](https://images.aatbio.com/dataset/ic50/oligopeptide-transporter-small-intestine-isoform_f4f025c62f2c5350c6593657708b1070.svg) | Valacyclovir | IC50 | 400000.0 [1], 431000.0 [2], 1100000.0 [3], 1420000.0 [4], 3400000.0 [5] |
![](https://images.aatbio.com/dataset/ic50/oligopeptide-transporter-small-intestine-isoform_f4f025c62f2c5350c6593657708b1070.svg) | Valacyclovir | Ki | 490000.0 [1], 740000.0 [2], 4080000.0 [3] |
![](https://images.aatbio.com/dataset/ic50/oligopeptide-transporter-small-intestine-isoform_9e85f1be5d21e3e9ed59594d3ae43ee0.svg) | Cefadroxil | IC50 | 870000.0 [1], 5400000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/oligopeptide-transporter-small-intestine-isoform_9e85f1be5d21e3e9ed59594d3ae43ee0.svg) | Cefadroxil | Ki | 1450000.0 [1], 7200000.0 [2], 9100000.0 [3] |
![](https://images.aatbio.com/dataset/ic50/oligopeptide-transporter-small-intestine-isoform_ee2a2a7889c5a7f23c360411dbafdadc.svg) | Phe-ala | IC50 | 180.0 [1], 70000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/oligopeptide-transporter-small-intestine-isoform_ee2a2a7889c5a7f23c360411dbafdadc.svg) | Phe-ala | Ki | 180.0 [1], 110000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/oligopeptide-transporter-small-intestine-isoform_2c408dfb7afe6b52eacdcd2181b2a45f.svg) | Cephalexin | IC50 | 5200000.0 [1], 13700000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/oligopeptide-transporter-small-intestine-isoform_2c408dfb7afe6b52eacdcd2181b2a45f.svg) | Cephalexin | Ki | 14000000.0 [1], 14400000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/oligopeptide-transporter-small-intestine-isoform_e09a7fe94aa6dc4a5b1d0f381b6f4f00.svg) | Cefixime | IC50 | 10000000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/oligopeptide-transporter-small-intestine-isoform_e09a7fe94aa6dc4a5b1d0f381b6f4f00.svg) | Cefixime | Ki | 1310000.0 [1], 12000000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/oligopeptide-transporter-small-intestine-isoform_f3a84782e93ba33584eead2640a4fa1d.svg) | Cephradine | IC50 | 15000000.0 [1], 15300000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/oligopeptide-transporter-small-intestine-isoform_f3a84782e93ba33584eead2640a4fa1d.svg) | Cephradine | Ki | 9800.0 [1], 9800000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/oligopeptide-transporter-small-intestine-isoform_1def19f9cd50998381d74df24a1b8967.svg) | L-Alanyl-L-alanine | IC50 | 63000.0 [1], 250000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/oligopeptide-transporter-small-intestine-isoform_1def19f9cd50998381d74df24a1b8967.svg) | L-Alanyl-L-alanine | Ki | 78000.0 [1], 140000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/oligopeptide-transporter-small-intestine-isoform_d5d57efdc5d415231812009b408cf2d9.svg) | Ceftibuten | Ki | 340000.0 [1], 710000.0 [2], 870000.0 [3] |
![](https://images.aatbio.com/dataset/ic50/oligopeptide-transporter-small-intestine-isoform_9b4952434b1a1879f3e78c42939caed9.svg) | Cyclacillin | IC50 | 350000.0 [1], 600000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/oligopeptide-transporter-small-intestine-isoform_9b4952434b1a1879f3e78c42939caed9.svg) | Cyclacillin | Ki | 500000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/oligopeptide-transporter-small-intestine-isoform_5b9940280eb50971a5b7493ada8712ad.svg) | Ampicillin | IC50 | 10000000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/oligopeptide-transporter-small-intestine-isoform_5b9940280eb50971a5b7493ada8712ad.svg) | Ampicillin | Ki | 14500000.0 [1], 15000000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/oligopeptide-transporter-small-intestine-isoform_abe754d59f1e9e9e7badbc5f50617dad.svg) | Cefaclor | IC50 | 8200000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/oligopeptide-transporter-small-intestine-isoform_abe754d59f1e9e9e7badbc5f50617dad.svg) | Cefaclor | Ki | 10000000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/oligopeptide-transporter-small-intestine-isoform_25382ff031f2a04ed0bbdf1f66e763a9.svg) | Glycylglycine | IC50 | 820000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/oligopeptide-transporter-small-intestine-isoform_25382ff031f2a04ed0bbdf1f66e763a9.svg) | Glycylglycine | Ki | 1000000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/oligopeptide-transporter-small-intestine-isoform_6c38bc51cf4974218a216b006d7bbfa1.svg) | Glycylsarcosine | IC50 | 1160000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/oligopeptide-transporter-small-intestine-isoform_6c38bc51cf4974218a216b006d7bbfa1.svg) | Glycylsarcosine | Ki | 830000.0 [1], 12800000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/oligopeptide-transporter-small-intestine-isoform_ab627db436627cd770977e492344013b.svg) | Glycyl-L-proline | IC50 | 330000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/oligopeptide-transporter-small-intestine-isoform_ab627db436627cd770977e492344013b.svg) | Glycyl-L-proline | Ki | 300000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/oligopeptide-transporter-small-intestine-isoform_ca1626d7295624d995bcdd9b7bbd8274.svg) | Phe-gly | IC50 | 200.0 [1], 170000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/oligopeptide-transporter-small-intestine-isoform_ca1626d7295624d995bcdd9b7bbd8274.svg) | Phe-gly | Ki | 200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/oligopeptide-transporter-small-intestine-isoform_82e795cad0453391f305a4eea4dab161.svg) | Glycyl-L-histidine | IC50 | 810000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/oligopeptide-transporter-small-intestine-isoform_82e795cad0453391f305a4eea4dab161.svg) | Glycyl-L-histidine | Ki | 1000000.0 [1], 4100000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/oligopeptide-transporter-small-intestine-isoform_e3c309d0812c33841cb983c7a4df1d0c.svg) | Asp-Asp | IC50 | 630000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/oligopeptide-transporter-small-intestine-isoform_e3c309d0812c33841cb983c7a4df1d0c.svg) | Asp-Asp | Ki | 410000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/oligopeptide-transporter-small-intestine-isoform_088d619370b7a1158a7205526cd2f81f.svg) | Ala-asp | IC50 | 450000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/oligopeptide-transporter-small-intestine-isoform_088d619370b7a1158a7205526cd2f81f.svg) | Ala-asp | Ki | 78000.0 [1], 260000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/oligopeptide-transporter-small-intestine-isoform_1f8742af9f3ff48ab105d27bf6d6248c.svg) | Pro-glu | IC50 | 12300000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/oligopeptide-transporter-small-intestine-isoform_1f8742af9f3ff48ab105d27bf6d6248c.svg) | Pro-glu | Ki | 20000000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/oligopeptide-transporter-small-intestine-isoform_f027fe601214bf89be887d416118a4b9.svg) | Tyr-Ala | IC50 | 110000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/oligopeptide-transporter-small-intestine-isoform_f027fe601214bf89be887d416118a4b9.svg) | Tyr-Ala | Ki | 90000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/oligopeptide-transporter-small-intestine-isoform_417493ec904781ce7f246e48336d69cd.svg) | Trp-Ala | IC50 | 260000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/oligopeptide-transporter-small-intestine-isoform_417493ec904781ce7f246e48336d69cd.svg) | Trp-Ala | Ki | 160000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/oligopeptide-transporter-small-intestine-isoform_490ef4d9e618dfcc70b6a41f8affbfc0.svg) | Ala-Lys | IC50 | 280000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/oligopeptide-transporter-small-intestine-isoform_490ef4d9e618dfcc70b6a41f8affbfc0.svg) | Ala-Lys | Ki | 117000.0 [1], 210000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/oligopeptide-transporter-small-intestine-isoform_f4992be17174bfa54bfa5b4a5b055ddd.svg) | Penicillin g | Ki | 30000000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/oligopeptide-transporter-small-intestine-isoform_f6083e307fb5b0c7b62d62e2f8808336.svg) | Enalapril | IC50 | 4500000.0 [1], 15000000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/oligopeptide-transporter-small-intestine-isoform_a01f0545e37e044d3063e3004c1d976c.svg) | Ceftriaxone | Ki | 30000000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/oligopeptide-transporter-small-intestine-isoform_cf9e99cc0ec161936ae5f39aadf2c4dc.svg) | Cefotaxime | Ki | 30000000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/oligopeptide-transporter-small-intestine-isoform_e1760d62cd8cd44e822d02efdcffaa3e.svg) | Oxacillin | Ki | 12000000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/oligopeptide-transporter-small-intestine-isoform_c77009e93d3f4908c62d842dd93a87cb.svg) | Cephalothin | Ki | 10000000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/oligopeptide-transporter-small-intestine-isoform_1f659e20e6919e67a589983b3ad2f40e.svg) | Cefuroxime | Ki | 26000000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/oligopeptide-transporter-small-intestine-isoform_ddce11da5e2e16912a45a18ad7a5cb38.svg) | Cloxacillin | Ki | 2500000.0 [1], 3000000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/oligopeptide-transporter-small-intestine-isoform_5d300885ae1748b0e63151e6b738a321.svg) | Cefamandole | Ki | 8100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/oligopeptide-transporter-small-intestine-isoform_c30a9fc6d9c28f7b3568b348f7656956.svg) | Latamoxef | Ki | 12000000.0 [1], 12300000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/oligopeptide-transporter-small-intestine-isoform_e92b9426ec3ed0b62b36d44608851ece.svg) | Dicloxacillin | Ki | 7200000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/oligopeptide-transporter-small-intestine-isoform_52803b0030aad77f118c9b91e61ba91e.svg) | Cysteinylglycine | Ki | 200000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/oligopeptide-transporter-small-intestine-isoform_d2076417c43167844e15f0c4408a6ce9.svg) | Cephapirin | Ki | 10000000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/oligopeptide-transporter-small-intestine-isoform_e15582b8e36c0d21cace0e48a392d2f4.svg) | Cefmetazole | Ki | 28000000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/oligopeptide-transporter-small-intestine-isoform_bcaaa31f39fefac153ddedffe39c7f10.svg) | (6R,7R)-7-[[(2Z)-2-(2-Amino-1,3-thiazol-4-yl)-2-methoxyiminoacetyl]amino]-3-(6,7-dihydro-5H-cyclopenta[b]pyridin-1-ium-1-ylmethyl)-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid | Ki | 30000000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/oligopeptide-transporter-small-intestine-isoform_114241d4bfeb027a1bffecfb81599f70.svg) | D-Alanyl-D-alanine | Ki | 30000000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/oligopeptide-transporter-small-intestine-isoform_4f6fed2871165ce47ff922230d7a56d6.svg) | Cefodizime | Ki | 22000000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/oligopeptide-transporter-small-intestine-isoform_7c00d6a8afd8f379c23f8bfaabdb054a.svg) | Alanyl-D-alanine | Ki | 4200000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/oligopeptide-transporter-small-intestine-isoform_eb0f9094e69d343f8e0083c4a3eed977.svg) | Glycylglycylglycine | IC50 | 1070000.0 [1], 1400000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/oligopeptide-transporter-small-intestine-isoform_65754cb5cdce590022c288feaeb8e647.svg) | Prolylglycine | IC50 | 16000000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/oligopeptide-transporter-small-intestine-isoform_65754cb5cdce590022c288feaeb8e647.svg) | Prolylglycine | Ki | 22000000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/oligopeptide-transporter-small-intestine-isoform_bb398aa6e29543647a4d9ea269b4e97c.svg) | Lysylglutamic acid | IC50 | 820000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/oligopeptide-transporter-small-intestine-isoform_bb398aa6e29543647a4d9ea269b4e97c.svg) | Lysylglutamic acid | Ki | 1300000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/oligopeptide-transporter-small-intestine-isoform_66070919fed532f6f69e782ca4b0624b.svg) | Glycyl-L-leucine | IC50 | 70000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/oligopeptide-transporter-small-intestine-isoform_66070919fed532f6f69e782ca4b0624b.svg) | Glycyl-L-leucine | Ki | 160000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/oligopeptide-transporter-small-intestine-isoform_5f26da99a33846171c0c8a4373561983.svg) | Ala-Gly | Ki | 140000.0 [1], 7300000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/oligopeptide-transporter-small-intestine-isoform_22c51d61b150efc4c5978cf59fbedae7.svg) | Pro-Pro | IC50 | 800000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/oligopeptide-transporter-small-intestine-isoform_22c51d61b150efc4c5978cf59fbedae7.svg) | Pro-Pro | Ki | 1200000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/oligopeptide-transporter-small-intestine-isoform_6b4b914380fb4dbded1b12bbda2608b2.svg) | H-Phe-phe-OH | Ki | 110000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/oligopeptide-transporter-small-intestine-isoform_1e6b6c7f1d043a75d64dfb3d39a08e13.svg) | Ala-Tyr | IC50 | 170000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/oligopeptide-transporter-small-intestine-isoform_1e6b6c7f1d043a75d64dfb3d39a08e13.svg) | Ala-Tyr | Ki | 150000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/oligopeptide-transporter-small-intestine-isoform_5a3e8ca6ec56a8cf0c2f943446b0de77.svg) | Val-Tyr | Ki | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/oligopeptide-transporter-small-intestine-isoform_59839b0019b2bf9da37f873c78f5131b.svg) | Pro-leu | IC50 | 620000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/oligopeptide-transporter-small-intestine-isoform_59839b0019b2bf9da37f873c78f5131b.svg) | Pro-leu | Ki | 470000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/oligopeptide-transporter-small-intestine-isoform_63aaf70011783ab6cabef5c54a8d020f.svg) | Leucylproline | Ki | 110000.0 [1], 180000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/oligopeptide-transporter-small-intestine-isoform_123cd421e275d4a2faaa976a7842a9ef.svg) | Metampicillin | Ki | 12700000.0 [1], 13000000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/oligopeptide-transporter-small-intestine-isoform_3f7a912ccf2e9cf9847e91a8008f0d93.svg) | Glycyl-L-aspartic acid | IC50 | 380000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/oligopeptide-transporter-small-intestine-isoform_3f7a912ccf2e9cf9847e91a8008f0d93.svg) | Glycyl-L-aspartic acid | Ki | 350000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/oligopeptide-transporter-small-intestine-isoform_60121d503706f71426ca7c8613a5cca1.svg) | Glutamylalanine | Ki | 250000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/oligopeptide-transporter-small-intestine-isoform_3901cbd950a25d295629da83633680c2.svg) | Aspartyllysine | Ki | 108000.0 [1], 860000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/oligopeptide-transporter-small-intestine-isoform_1bf1f7accb93005d180cc0ca9719d1c2.svg) | (2R)-1-[(2S)-2,6-Diaminohexanoyl]pyrrolidine-2-carboxylic acid | IC50 | 390000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/oligopeptide-transporter-small-intestine-isoform_1bf1f7accb93005d180cc0ca9719d1c2.svg) | (2R)-1-[(2S)-2,6-Diaminohexanoyl]pyrrolidine-2-carboxylic acid | Ki | 350000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/oligopeptide-transporter-small-intestine-isoform_80360b6ba12273846380f1f40b8459ac.svg) | Aspartylalanine | Ki | 320000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/oligopeptide-transporter-small-intestine-isoform_8487c45653b5c8d73d8a55843f100f69.svg) | Val-phe | Ki | 50000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/oligopeptide-transporter-small-intestine-isoform_bc53321d8879b7b5a96f4a4de2658e29.svg) | L-Lysyl-L-alanine | Ki | 340000.0 [1], 419000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/oligopeptide-transporter-small-intestine-isoform_2a32ad54ebf0a30ae43fab269948cc62.svg) | Pro-Ser | IC50 | 16000000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/oligopeptide-transporter-small-intestine-isoform_2a32ad54ebf0a30ae43fab269948cc62.svg) | Pro-Ser | Ki | 14000000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/oligopeptide-transporter-small-intestine-isoform_b8d683d6fd876b2b6cb6622bbd9c43c1.svg) | Tyrosylphenylalanine | Ki | 90000.0 [1], 140000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/oligopeptide-transporter-small-intestine-isoform_59fe48af2fdf97c0dc1cb59711b54f8a.svg) | Ala-Ser | Ki | 140000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/oligopeptide-transporter-small-intestine-isoform_1cf9b4c84c92140f4cbd70694fc7c61f.svg) | H-D-Phe-Ala-OH | Ki | 7000000.0 [1], 7100000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/oligopeptide-transporter-small-intestine-isoform_4d76b6a385e5c793f8b3f2bca4e87fda.svg) | Ser-Ala | Ki | 140000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/oligopeptide-transporter-small-intestine-isoform_4bc76d48890c94878801a60589e1a67c.svg) | Glu-lys | IC50 | 720000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/oligopeptide-transporter-small-intestine-isoform_4bc76d48890c94878801a60589e1a67c.svg) | Glu-lys | Ki | 510000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/oligopeptide-transporter-small-intestine-isoform_1d2775f0f3f5e8fecdd7558afa6c40eb.svg) | Pro-Asp | IC50 | 9160000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/oligopeptide-transporter-small-intestine-isoform_1d2775f0f3f5e8fecdd7558afa6c40eb.svg) | Pro-Asp | Ki | 9800000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/oligopeptide-transporter-small-intestine-isoform_c5f9790b613639f0118a37319ed134a5.svg) | Alanyl ornithine | Ki | 970000.0 [1], 980000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/oligopeptide-transporter-small-intestine-isoform_dcac1165cadb8f4c8628077d23a0576a.svg) | 1-(2-Aminopropanethioyl)pyrrolidine-2-carboxylic acid | Ki | 300000.0 [1], 330000.0 [2] |