![](https://images.aatbio.com/dataset/ic50/nuclear-receptor-ror-alpha_bc29448afbd834082697eaaff0360ff1.svg) | N-[4-(1,1,1,3,3,3-Hexafluoro-2-hydroxypropan-2-yl)phenyl]-N-(2,2,2-trifluoroethyl)benzenesulfonamide | IC50 | 2000.0 [1], 5011.87 [2], 11000.0 [3], 20000.0 [4] |
![](https://images.aatbio.com/dataset/ic50/nuclear-receptor-ror-alpha_bc29448afbd834082697eaaff0360ff1.svg) | N-[4-(1,1,1,3,3,3-Hexafluoro-2-hydroxypropan-2-yl)phenyl]-N-(2,2,2-trifluoroethyl)benzenesulfonamide | Ki | 132.0 [1] |
![](https://images.aatbio.com/dataset/ic50/nuclear-receptor-ror-alpha_d9300b9c5db9172269a90918adf94378.svg) | CID 44241473 | Ki | 172.0 [1] |
![](https://images.aatbio.com/dataset/ic50/nuclear-receptor-ror-alpha_dbe5b206d2de640c83715b21a7cf1333.svg) | 5-Butyl-2-[2,2,2-trifluoro-1-hydroxy-1-(trifluoromethyl)ethyl]phenanthridin-6-one | IC50 | 7200.0 [1], 9800.0 [2] |
![](https://images.aatbio.com/dataset/ic50/nuclear-receptor-ror-alpha_f2b40b6cf121be41d799a2ea8d2c35be.svg) | N-[4-[Hydroxy(dimethyl)silyl]phenyl]-N-(2,2,2-trifluoroethyl)benzenesulfonamide | IC50 | 30000.0 [1], 53000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/nuclear-receptor-ror-alpha_573d5a9fda73183a4ba97fe0320ec6c2.svg) | 4-Cyano-N-[3-[1-(cyclopentanecarbonyl)piperidin-4-yl]-1-methylindol-5-yl]pyridine-2-carboxamide | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/nuclear-receptor-ror-alpha_8506ef7d768446be03fec18e29c088bf.svg) | 2-Acetamido-N-[4-(5-cyano-3-fluoro-2-methoxyphenyl)thiophen-2-yl]-2-(4-ethylsulfonylphenyl)acetamide | IC50 | 19000.0 [1], 33000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/nuclear-receptor-ror-alpha_0da64dfbf8a32948c2a5448ccb46c180.svg) | N-[4-[5-Cyano-2-(2,2,2-trifluoroethoxy)pyridin-3-yl]thiophen-2-yl]-2-(4-ethylsulfonylphenyl)acetamide | IC50 | 6200.0 [1], 33000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/nuclear-receptor-ror-alpha_d22da0e144a9acba0dd45aee3e787804.svg) | 2-(4-Ethylsulfonylphenyl)-N-[4-[2-[4-(trifluoromethoxy)phenoxy]pyridin-3-yl]thiophen-2-yl]acetamide | IC50 | 33000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/nuclear-receptor-ror-alpha_5aa906899674b30f85dc3138034661d2.svg) | 2-Acetamido-N-[4-[5-cyano-2-(2,2,2-trifluoroethoxy)pyridin-3-yl]thiophen-2-yl]-2-(4-ethylsulfonylphenyl)acetamide | IC50 | 600.0 [1], 33000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/nuclear-receptor-ror-alpha_0c33410dfaf1c9a70f92bed30b45464c.svg) | 2-(4-Ethylsulfonylphenyl)-N-[4-[2-[[4-(trifluoromethoxy)phenyl]methoxy]pyridin-3-yl]thiophen-2-yl]acetamide | IC50 | 33000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/nuclear-receptor-ror-alpha_665885a26b029a7e5fa22a0c789c9273.svg) | (2R)-2-Acetamido-2-(4-ethylsulfonylphenyl)-N-[4-[2-[[4-(trifluoromethoxy)phenyl]methoxy]pyridin-3-yl]thiophen-2-yl]acetamide | IC50 | 9400.0 [1], 33000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/nuclear-receptor-ror-alpha_5d7ecbbec2169d781b8354a42c26d542.svg) | 4-Cyano-N-[3-[1-(cyclohexanecarbonyl)piperidin-4-yl]-1-methylindol-5-yl]pyridine-2-carboxamide | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/nuclear-receptor-ror-alpha_44795c2b7270c479cc4992bd0491449f.svg) | 3-Cyano-N-[3-[1-(cyclopentanecarbonyl)piperidin-4-yl]-1-methylindol-5-yl]benzamide | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/nuclear-receptor-ror-alpha_7f3f9d6989773277a63dc264420a06f9.svg) | 3-Cyano-N-[3-[1-(cyclopentanecarbonyl)piperidin-4-yl]-1H-indol-5-yl]benzamide | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/nuclear-receptor-ror-alpha_4fb901083691944934f10a258499025f.svg) | 7-Ketocholesterol | Ki | 12.0 [1] |
![](https://images.aatbio.com/dataset/ic50/nuclear-receptor-ror-alpha_1a68bce23b6fed9b3e58d128e2e9a857.svg) | 7alpha-Hydroxycholesterol | Ki | 12.0 [1] |
![](https://images.aatbio.com/dataset/ic50/nuclear-receptor-ror-alpha_8429446b1fa4184406937276f77b21dc.svg) | 7beta-Hydroxycholesterol | Ki | 12.0 [1] |
![](https://images.aatbio.com/dataset/ic50/nuclear-receptor-ror-alpha_cf63a793eb10bfb7723bcbd258978fd7.svg) | Ethyl 2-[2-[2-(2,3-dihydro-1,4-benzodioxin-6-ylamino)-2-oxoethyl]-1-oxoisoquinolin-5-yl]oxypropanoate | IC50 | 33000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/nuclear-receptor-ror-alpha_a43650a12f8ab3610a408dcc4012106b.svg) | CID 118622692 | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/nuclear-receptor-ror-alpha_e4ff5819ff293f0a07e37ee23b528c96.svg) | N-[4-(1,1,1,3,3,3-Hexafluoro-2-hydroxypropan-2-yl)phenyl]-2-thiophenesulfonamide | Ki | 220.0 [1] |
![](https://images.aatbio.com/dataset/ic50/nuclear-receptor-ror-alpha_c4866a34c6d2ba92acd6d6f18f0c2b53.svg) | Ethyl 2-[(2-{[(furan-2-ylmethyl)carbamoyl]methyl}-1-oxo-1,2-dihydroisoquinolin-5-yl)oxy]propanoate | IC50 | 33000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/nuclear-receptor-ror-alpha_fd7c31015cf52caba14b20222d5127d4.svg) | Ethyl 2-[2-[2-(1,3-benzodioxol-5-ylmethylamino)-2-oxoethyl]-1-oxoisoquinolin-5-yl]oxypropanoate | IC50 | 33000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/nuclear-receptor-ror-alpha_e9d1c5f56bbb9cef6d2446db4d9788d8.svg) | N-[5-(2-Chlorobenzoyl)-4-(3-chlorophenyl)-1,3-thiazol-2-yl]-2-(4-ethylsulfonylphenyl)acetamide | IC50 | 5011.87 [1] |
![](https://images.aatbio.com/dataset/ic50/nuclear-receptor-ror-alpha_27d89dd128e332c8a7bac5a0b04b3c65.svg) | 5-Butylphenanthridin-6(5H)-one | IC50 | 10200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/nuclear-receptor-ror-alpha_194a7da93d1c1444cd9c12fe1a5763b6.svg) | Ethyl 2-((2-(2-((4-fluorobenzyl)amino)-2-oxoethyl)-1-oxo-1,2-dihydroisoquinolin-5-yl)oxy)propanoate | IC50 | 1680.0 [1] |
![](https://images.aatbio.com/dataset/ic50/nuclear-receptor-ror-alpha_3292844ebc81e3cf6007e79e41d2f49c.svg) | Ethyl 2-[(2-{[(4-ethoxyphenyl)carbamoyl]methyl}-1-oxo-1,2-dihydroisoquinolin-5-yl)oxy]propanoate | IC50 | 22600.0 [1] |
![](https://images.aatbio.com/dataset/ic50/nuclear-receptor-ror-alpha_12cc3df65284c89cd5aa47ebacf6c559.svg) | Ethyl 2-[(1-oxo-2-{[(2-phenylethyl)carbamoyl]methyl}-1,2-dihydroisoquinolin-5-yl)oxy]propanoate | IC50 | 33000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/nuclear-receptor-ror-alpha_9b01cb9f8c5c85128e78ed8a178861a2.svg) | 5-Butyl-2-methylphenanthridin-6(5H)-one | IC50 | 17600.0 [1] |
![](https://images.aatbio.com/dataset/ic50/nuclear-receptor-ror-alpha_d9b6abe0fec65ffa11978462c49f5cdb.svg) | 5-Butyl-2-ethylphenanthridin-6(5H)-one | IC50 | 9000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/nuclear-receptor-ror-alpha_102970d308613a3ecec247e679e266a9.svg) | 5-Butyl-2-hydroxymethylphenanthridin-6(5H)-one | IC50 | 20000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/nuclear-receptor-ror-alpha_2e80e094ae9e012cbc087e6a18cb2656.svg) | Ethyl 2-({2-[(benzylcarbamoyl)methyl]-1-oxo-1,2-dihydroisoquinolin-5-yl}oxy)propanoate | IC50 | 3220.0 [1] |
![](https://images.aatbio.com/dataset/ic50/nuclear-receptor-ror-alpha_9c5f9ea48d6a220f2c40b9f501b11c67.svg) | 2-(5-Butoxy-1-oxo-2-isoquinolinyl)-N-(2,3-dihydro-1,4-benzodioxin-6-yl)acetamide | IC50 | 21500.0 [1] |
![](https://images.aatbio.com/dataset/ic50/nuclear-receptor-ror-alpha_2d6433b9aa0328eda895caa18d7dcee1.svg) | N-(5-Benzoyl-4-phenyl-1,3-thiazol-2-yl)-2-(4-ethylsulfonylphenyl)acetamide | IC50 | 5011.87 [1] |
![](https://images.aatbio.com/dataset/ic50/nuclear-receptor-ror-alpha_57dcbe872b6036a0ace704560f50edb0.svg) | 5-Nonyl-2-[2,2,2-trifluoro-1-hydroxy-1-(trifluoromethyl)ethyl]phenanthridin-6-one | IC50 | 20000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/nuclear-receptor-ror-alpha_c54893148d2a43d79fdb22dbf8ab8d39.svg) | 5-Butyl-2-tert-butylphenanthridin-6(5H)-one | IC50 | 11800.0 [1] |
![](https://images.aatbio.com/dataset/ic50/nuclear-receptor-ror-alpha_409797e514cbac7af22e8345dd6ab7cf.svg) | 5-Ethyl-2-[2,2,2-trifluoro-1-hydroxy-1-(trifluoromethyl)ethyl]phenanthridin-6-one | IC50 | 20000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/nuclear-receptor-ror-alpha_f7c475ecc3762fc60431438293ded326.svg) | 5-Hexyl-2-[2,2,2-trifluoro-1-hydroxy-1-(trifluoromethyl)ethyl]phenanthridin-6-one | IC50 | 7600.0 [1] |
![](https://images.aatbio.com/dataset/ic50/nuclear-receptor-ror-alpha_488f55862d9faf810cde2f204f7fc221.svg) | 2-(1,1,1,3,3,3-Hexafluoro-2-hydroxypropan-2-yl)-5-methylphenanthridin-6-one | IC50 | 20000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/nuclear-receptor-ror-alpha_3ee828407c9d6eb408a0a1dc67e28e7d.svg) | 5-(2,2,2-Trifluoroethyl)-2-[2,2,2-trifluoro-1-hydroxy-1-(trifluoromethyl)ethyl]phenanthridin-6-one | IC50 | 9900.0 [1] |
![](https://images.aatbio.com/dataset/ic50/nuclear-receptor-ror-alpha_1c0fb028a093502375ba3b3c5685a2a9.svg) | 5-(Cyclohexylmethyl)-2-[2,2,2-trifluoro-1-hydroxy-1-(trifluoromethyl)ethyl]phenanthridin-6-one | IC50 | 10300.0 [1] |
![](https://images.aatbio.com/dataset/ic50/nuclear-receptor-ror-alpha_dcdfcb682f1ea89dc1b7d0d7d2587d2f.svg) | 5-Butyl-2-isopropyl-phenanthridin-6-one | IC50 | 16700.0 [1] |
![](https://images.aatbio.com/dataset/ic50/nuclear-receptor-ror-alpha_7b1459728db581d2db3704bd206e36eb.svg) | 5-Butyl-3-methoxy-2-[2,2,2-trifluoro-1-hydroxy-1-(trifluoromethyl)ethyl]phenanthridin-6-one | IC50 | 7800.0 [1] |
![](https://images.aatbio.com/dataset/ic50/nuclear-receptor-ror-alpha_b5743fc115bd04528ca9fc798d2bcc00.svg) | 5-Butyl-4-methoxy-2-[2,2,2-trifluoro-1-hydroxy-1-(trifluoromethyl)ethyl]phenanthridin-6-one | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/nuclear-receptor-ror-alpha_21e1b398820aa54fe1c3072c761ab606.svg) | 5-Butyl-9-methoxy-2-[2,2,2-trifluoro-1-hydroxy-1-(trifluoromethyl)ethyl]phenanthridin-6-one | IC50 | 5300.0 [1] |
![](https://images.aatbio.com/dataset/ic50/nuclear-receptor-ror-alpha_92b987745af785397ee145b4be3f9147.svg) | 5-Butyl-10-methoxy-2-[2,2,2-trifluoro-1-hydroxy-1-(trifluoromethyl)ethyl]phenanthridin-6-one | IC50 | 9100.0 [1] |
![](https://images.aatbio.com/dataset/ic50/nuclear-receptor-ror-alpha_7f2bb6819e66100e8e46538c627a8646.svg) | N-(2,4-Difluorophenyl)-2-[4-[[2-(4-ethylsulfonylphenyl)acetyl]amino]-2-fluorophenyl]-2-methylpropanamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/nuclear-receptor-ror-alpha_8a9ca8d22c3507ed27cf6d6fe67379c2.svg) | 2-(1,1,1,3,3,3-Hexafluoro-2-hydroxypropan-2-yl)-5H-phenanthridin-6-one | IC50 | 20000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/nuclear-receptor-ror-alpha_c44b6f7a9745ea84c40007969305d742.svg) | 2-(1,1,1,3,3,3-Hexafluoro-2-hydroxypropan-2-yl)-5-propylphenanthridin-6-one | IC50 | 10800.0 [1] |
![](https://images.aatbio.com/dataset/ic50/nuclear-receptor-ror-alpha_c9b57d127598ebf3162dc7502571f763.svg) | [4-[(3R)-4-[5-(Hydroxymethyl)-4-(trifluoromethyl)pyrimidin-2-yl]-3-propan-2-ylpiperazin-1-yl]-2-methylsulfonylphenyl]methanol | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/nuclear-receptor-ror-alpha_6ce88abd520d2b354097eec897fc7de4.svg) | 4-Cyano-N-[3-[1-(cyclopentanecarbonyl)piperidin-4-yl]-1-ethylindol-5-yl]pyridine-2-carboxamide | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/nuclear-receptor-ror-alpha_6c1300f87a1524b70d70a57d575f29f3.svg) | N-(4-Ethylphenyl)-N-(2-methylpropyl)-3-(methylsulfonimidoyl)-4-(oxan-4-ylmethoxy)benzenesulfonamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/nuclear-receptor-ror-alpha_9d20dfdf0c959713c0c2ed060157312c.svg) | N-(4-Ethylphenyl)-N-(2-methylpropyl)-3-(methylsulfonimidoyl)-4-(oxan-4-ylmethoxy)benzenesulfonamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/nuclear-receptor-ror-alpha_5709e47f37656f2faf65d85e31038d03.svg) | 2-(5,5-Dibutylbenzo[b][1]benzosilol-2-yl)-1,1,1,3,3,3-hexafluoropropan-2-ol | IC50 | 6200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/nuclear-receptor-ror-alpha_ec2d4349fec4ae8f412e678afaa4774d.svg) | 2-(5,5-Dimethylbenzo[b][1]benzosilol-2-yl)-1,1,1,3,3,3-hexafluoropropan-2-ol | IC50 | 9400.0 [1] |
![](https://images.aatbio.com/dataset/ic50/nuclear-receptor-ror-alpha_47bebac6319cac9afb2cf939b6afa6eb.svg) | 2-(5-Butyl-5-methylbenzo[b][1]benzosilol-2-yl)-1,1,1,3,3,3-hexafluoropropan-2-ol | IC50 | 7700.0 [1] |
![](https://images.aatbio.com/dataset/ic50/nuclear-receptor-ror-alpha_a4bc12a3f30141746a9862c22ee03d7e.svg) | 4-[3-[2-Chloranyl-6-(Trifluoromethyl)phenoxy]-5-(Dimethylcarbamoyl)indazol-1-Yl]benzoic Acid | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/nuclear-receptor-ror-alpha_1549ab8fd9a52ac89ef4e927ade1d9e3.svg) | 4-[3-(2-Chloro-6-methylphenoxy)-5-(dimethylcarbamoyl)indazol-1-yl]benzoic acid | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/nuclear-receptor-ror-alpha_4248e27d22167b90ba16631c05a4df68.svg) | Chembl4175305 | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/nuclear-receptor-ror-alpha_e19df83f3101d53806c1cc8757dee35a.svg) | (4S)-4-Benzyl-1-[4-[(5S)-2-(2-cyclopentylethyl)-4,5-dihydro-1H-imidazol-5-yl]butyl]-3-(2-phenylethyl)imidazolidine-2-thione | IC50 | 6000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/nuclear-receptor-ror-alpha_d3b01d1b559aac650933fa348062a75a.svg) | (4R)-4-Tert-butyl-3-(2-phenylethyl)-1-[4-[(5S)-2-propyl-4,5-dihydro-1H-imidazol-5-yl]butyl]imidazolidine-2-thione | IC50 | 30100.0 [1] |
![](https://images.aatbio.com/dataset/ic50/nuclear-receptor-ror-alpha_bbe157f246c32e1756246c50afc43f0b.svg) | (4S)-4-Benzyl-1-[4-[(5S)-2-[(3-fluorophenyl)methyl]-4,5-dihydro-1H-imidazol-5-yl]butyl]-3-(2-phenylethyl)imidazolidine-2-thione | IC50 | 6800.0 [1] |
![](https://images.aatbio.com/dataset/ic50/nuclear-receptor-ror-alpha_79c97e2ac47b88faed41cc3df4986bfc.svg) | (4S)-4-Benzyl-3-[2-(2-bicyclo[2.2.1]heptanyl)ethyl]-1-[4-[(5S)-2-propyl-4,5-dihydro-1H-imidazol-5-yl]butyl]imidazolidine-2-thione | IC50 | 13000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/nuclear-receptor-ror-alpha_3000d065bc918f26a6733c93a668a9ae.svg) | (4S)-4-Benzyl-1-[4-[(5S)-2-[(3-methoxyphenyl)methyl]-4,5-dihydro-1H-imidazol-5-yl]butyl]-3-(2-phenylethyl)imidazolidine-2-thione | IC50 | 8000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/nuclear-receptor-ror-alpha_f4363e0415a07a5f16ee8abbedb60323.svg) | (4S)-4-Benzyl-3-(2-phenylethyl)-1-[4-[(5S)-2-prop-2-enyl-4,5-dihydro-1H-imidazol-5-yl]butyl]imidazolidine-2-thione | IC50 | 15000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/nuclear-receptor-ror-alpha_b7fc06837f8847322b59a7b0bbae3316.svg) | (4S)-3-[2-(2-Adamantyl)ethyl]-4-benzyl-1-[4-[(5S)-2-propyl-4,5-dihydro-1H-imidazol-5-yl]butyl]imidazolidine-2-thione | IC50 | 8400.0 [1] |
![](https://images.aatbio.com/dataset/ic50/nuclear-receptor-ror-alpha_1fe67bd541f1b000e887f1181cfe1fb2.svg) | (4S)-4-Benzyl-1-[4-[(5S)-2-[(4-fluorophenyl)methyl]-4,5-dihydro-1H-imidazol-5-yl]butyl]-3-(2-phenylethyl)imidazolidine-2-thione | IC50 | 9900.0 [1] |
![](https://images.aatbio.com/dataset/ic50/nuclear-receptor-ror-alpha_4938067a7084992245232de25caf88ce.svg) | (4S)-4-Benzyl-3-(2-phenylethyl)-1-[4-[(5S)-2-[(E)-prop-1-enyl]-4,5-dihydro-1H-imidazol-5-yl]butyl]imidazolidine-2-thione | IC50 | 12500.0 [1] |
![](https://images.aatbio.com/dataset/ic50/nuclear-receptor-ror-alpha_7e48079d23351232773c1c733b3f6c87.svg) | (4S)-4-Benzyl-3-(2-phenylethyl)-1-[4-[(5S)-2-(2-phenylpropyl)-4,5-dihydro-1H-imidazol-5-yl]butyl]imidazolidine-2-thione | IC50 | 7500.0 [1] |
![](https://images.aatbio.com/dataset/ic50/nuclear-receptor-ror-alpha_522b3f4b11e1bec441b8fc846b20e450.svg) | (4S)-4-Benzyl-1-[4-[(5S)-2-[(3-methylphenyl)methyl]-4,5-dihydro-1H-imidazol-5-yl]butyl]-3-(2-phenylethyl)imidazolidine-2-thione | IC50 | 6800.0 [1] |
![](https://images.aatbio.com/dataset/ic50/nuclear-receptor-ror-alpha_1b2c86f641d08da0a442282268422e9d.svg) | (4S)-4-Benzyl-1-[4-[(5S)-2-(cyclohexylmethyl)-4,5-dihydro-1H-imidazol-5-yl]butyl]-3-(2-phenylethyl)imidazolidine-2-thione | IC50 | 6400.0 [1] |
![](https://images.aatbio.com/dataset/ic50/nuclear-receptor-ror-alpha_335b6735a4f30e2b1fdbf0c327fbd1cc.svg) | (4S)-4-Benzyl-3-[(4-methylcyclohexyl)methyl]-1-[4-[(5S)-2-propyl-4,5-dihydro-1H-imidazol-5-yl]butyl]imidazolidine-2-thione | IC50 | 26000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/nuclear-receptor-ror-alpha_2e7fa87dec5a70495d09b5142cdbd5e5.svg) | (4S)-4-Butyl-3-(2-phenylethyl)-1-[4-[(5S)-2-propyl-4,5-dihydro-1H-imidazol-5-yl]butyl]imidazolidine-2-thione | IC50 | 11900.0 [1] |
![](https://images.aatbio.com/dataset/ic50/nuclear-receptor-ror-alpha_7ae1d709aa4a66f3bce967ae1b428f18.svg) | (4S)-4-Benzyl-3-(3-cyclopentylpropyl)-1-[4-[(5S)-2-propyl-4,5-dihydro-1H-imidazol-5-yl]butyl]imidazolidine-2-thione | IC50 | 5800.0 [1] |
![](https://images.aatbio.com/dataset/ic50/nuclear-receptor-ror-alpha_cd8bcfe221f82f98830b12d5cfffb678.svg) | 2-[4-[[2-(4-Ethylsulfonylphenyl)acetyl]amino]phenyl]-N-(4-fluorophenyl)-2-methylpropanamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/nuclear-receptor-ror-alpha_27505d0de3c5626e0b569b7f1be56a2f.svg) | N-(4-Cyanopyridin-2-yl)-2-[4-[[2-(4-ethylsulfonylphenyl)acetyl]amino]-2-fluorophenyl]-2-methylpropanamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/nuclear-receptor-ror-alpha_ae0d06f989dc682f0b44a5349e6ce5d4.svg) | N-[3-[1-(Cyclopentanecarbonyl)piperidin-4-yl]-1-methylindol-5-yl]benzamide | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/nuclear-receptor-ror-alpha_e3a43874bfb4bef42bc3cc214c9b2754.svg) | N-Benzyl-N-[4-[hydroxy(dimethyl)silyl]phenyl]benzenesulfonamide | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/nuclear-receptor-ror-alpha_3b527a6feda592f3e8df58435fcd6bce.svg) | N-[4-[Hydroxy(dimethyl)silyl]phenyl]-N-(2-phenylethyl)benzenesulfonamide | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/nuclear-receptor-ror-alpha_325bf0c3a7b2bde257c928432ca7bf1f.svg) | N-Ethyl-N-[4-[hydroxy(dimethyl)silyl]phenyl]benzenesulfonamide | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/nuclear-receptor-ror-alpha_375d5376e5e98e1738cb0227079378fd.svg) | N-Butyl-N-[4-[hydroxy(dimethyl)silyl]phenyl]benzenesulfonamide | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/nuclear-receptor-ror-alpha_4a0d09b6e45a297bd9e1c3fd47001df6.svg) | 2-[4-[[2-(4-Ethylsulfonylphenyl)acetyl]amino]-2-fluorophenyl]-N-(4-fluorophenyl)-2-methylpropanamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/nuclear-receptor-ror-alpha_07fa57b26ee5383485617d57eb1fd7f6.svg) | 5,5,8,8-Tetramethyl-N-phenyl-6,7-dihydronaphthalene-2-carboxamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/nuclear-receptor-ror-alpha_99ba73d1f296e2cc9347e60ec6839759.svg) | Ethyl 2-[(2-{[(4-ethylphenyl)carbamoyl]methyl}-1-oxo-1,2-dihydroisoquinolin-5-yl)oxy]propanoate | IC50 | 25000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/nuclear-receptor-ror-alpha_4d35e25ebde3684aac2c596316ec7055.svg) | Ethyl 2-[(2-{[(4-butylphenyl)carbamoyl]methyl}-1-oxo-1,2-dihydroisoquinolin-5-yl)oxy]propanoate | IC50 | 30700.0 [1] |
![](https://images.aatbio.com/dataset/ic50/nuclear-receptor-ror-alpha_ec60674ef71fdcade7f9c27ec8e42171.svg) | Ethyl 2-[(2-{[(4-methylphenyl)carbamoyl]methyl}-1-oxo-1,2-dihydroisoquinolin-5-yl)oxy]propanoate | IC50 | 36500.0 [1] |
![](https://images.aatbio.com/dataset/ic50/nuclear-receptor-ror-alpha_5ce21687e7da54975aaebd852831a574.svg) | 5-Butyl-2-hexylphenanthridin-6(5H)-one | IC50 | 10300.0 [1] |
![](https://images.aatbio.com/dataset/ic50/nuclear-receptor-ror-alpha_c9de77d1f6d157dea58df857c3f4291c.svg) | 1,1,4,4-Tetramethyl-N-phenyl-2,3-dihydro-1,4-benzodisiline-6-carboxamide | IC50 | 1300.0 [1] |
![](https://images.aatbio.com/dataset/ic50/nuclear-receptor-ror-alpha_7aabf5a0686f3eb38d78676369acb5b2.svg) | 5-Butyl-9-chloro-2-(1,1,1,3,3,3-hexafluoro-2-hydroxypropan-2-yl)phenanthridin-6-one | IC50 | 5600.0 [1] |
![](https://images.aatbio.com/dataset/ic50/nuclear-receptor-ror-alpha_34ad93034b7962f0d1a4d8882585937d.svg) | N-[5-(2-Chlorobenzoyl)-4-(2-chlorophenyl)-1,3-thiazol-2-yl]-2-(4-ethylsulfonylphenyl)acetamide | IC50 | 110.0 [1] |
![](https://images.aatbio.com/dataset/ic50/nuclear-receptor-ror-alpha_9e0e7e65330fc2913b1b5fb9f27dfa6f.svg) | 5-(Cyclopropylmethyl)-2-(1,1,1,3,3,3-hexafluoro-2-hydroxypropan-2-yl)phenanthridin-6-one | IC50 | 13600.0 [1] |
![](https://images.aatbio.com/dataset/ic50/nuclear-receptor-ror-alpha_2a07f0951b2b052b817e4735722db7d0.svg) | 2-(1,1,1,3,3,3-Hexafluoro-2-hydroxypropan-2-yl)-5-propan-2-ylphenanthridin-6-one | IC50 | 12300.0 [1] |
![](https://images.aatbio.com/dataset/ic50/nuclear-receptor-ror-alpha_7d5540967ad1512efe4db89fb6391edd.svg) | 5-Butyl-2-(1,1,1,3,3,3-hexafluoro-2-hydroxypropan-2-yl)-9-methylphenanthridin-6-one | IC50 | 7600.0 [1] |
![](https://images.aatbio.com/dataset/ic50/nuclear-receptor-ror-alpha_1999b10574dd4fbbbdd63600def83a4e.svg) | 5-Butyl-2-(1,1,1,3,3,3-hexafluoro-2-hydroxypropan-2-yl)-9-(trifluoromethyl)phenanthridin-6-one | IC50 | 5500.0 [1] |
![](https://images.aatbio.com/dataset/ic50/nuclear-receptor-ror-alpha_339f3fe7165dc02b56cbaa0e8f0bef1c.svg) | 5-Butyl-2-(1,1,1,3,3,3-hexafluoro-2-hydroxypropan-2-yl)-9-hydroxyphenanthridin-6-one | IC50 | 6400.0 [1] |