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Norepinephrine transporter Inhibitors (IC50, Ki)

Structure
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▼
Compound Name
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▼
Standard Type
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▼
Standard Values (in nM)
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▼
CocaineIC50378.0 [1]
CocaineKi264.0 [1]
DesipramineIC503.4 [1]
DesipramineKi0.6 [1], 2.1 [2], 3.4 [3], 5.11 [4]
DuloxetineIC505.0 [1]
DuloxetineKi7.94 [1]
FluoxetineIC502000.0 [1]
FluoxetineKi440.0 [1], 1292.0 [2], 1560.0 [3], 2000.0 [4]
AtomoxetineIC505.0 [1]
VenlafaxineIC50535.0 [1]
VenlafaxineKi210.0 [1], 385.0 [2], 553.0 [3], 2685.0 [4]
ProtriptylineIC501.1 [1], 7.1 [2], 17.0 [3]
ProtriptylineKi2.0 [1], 2.1 [2], 2.3 [3], 6.8 [4]
2-[(2-Ethoxyphenoxy)-phenylmethyl]morpholineIC503.2 [1]
2-[(2-Ethoxyphenoxy)-phenylmethyl]morpholineKi1.1 [1], 5.0 [2]
NisoxetineIC508.3 [1]
NisoxetineKi1.6 [1], 6.0 [2]
BupropionIC501850.0 [1]
BupropionKi6970.0 [1]
Venlafaxine hydrochlorideIC502550.0 [1]
MazindolIC500.92 [1], 4.9 [2]
MazindolKi11.3 [1], 13.5 [2], 18.0 [3]
MidalcipranIC500.79 [1], 77.0 [2], 5500.0 [3]
MidalcipranKi85.0 [1]
1-(3,4-Dichlorophenyl)-3-azabicyclo[3.1.0]hexaneIC5020.0 [1], 20.3 [2], 72.4 [3], 143.0 [4]
1-(3,4-Dichlorophenyl)-3-azabicyclo[3.1.0]hexaneKi63.0 [1]
Rel-1-(3,4-dichlorophenyl)-6-(methoxymethyl)-3-azabicyclo[4.1.0]heptaneIC502.0 [1], 8.1 [2]
Rel-1-(3,4-dichlorophenyl)-6-(methoxymethyl)-3-azabicyclo[4.1.0]heptaneKi7.94 [1], 12.02 [2], 12.59 [3]
ReboxetineIC502.0 [1], 3.0 [2], 3.1 [3]
ReboxetineKi0.3 [1], 1.04 [2]
NomifensineIC50630.96 [1]
NomifensineKi3.8 [1], 5.0 [2], 23.0 [3]
MadamIC50100.0 [1]
MadamKi61.0 [1], 320.4 [2], 325.0 [3]
AmitifadineIC5022.8 [1], 71.4 [2]
AmitifadineKi63.1 [1], 147.91 [2]
3-(4-Iodo-phenyl)-8-methyl-8-aza-bicyclo[3.2.1]octane-2-carboxylic acid methyl esterKi1.4 [1], 11.2 [2], 22.0 [3], 36.0 [4]
(R)-Sila-VenlafaxineIC50200.0 [1], 251.0 [2]
4-(3,4-Dimethoxy-phenyl)-4a,5,8,8a-tetrahydro-2H-phthalazin-1-oneIC50100000.0 [1]
4-(3,4-Dimethoxy-phenyl)-4a,5,8,8a-tetrahydro-2H-phthalazin-1-oneKi100000.0 [1]
(S)-N-(2,3-Dimethylbenzyl)-N-(tetrahydro-2H-pyran-4-yl)pyrrolidin-3-amineIC507.0 [1]
(1S,5S,6S)-1-(3,4-Dichlorophenyl)-6-(ethoxymethyl)-3-azabicyclo[3.1.0]hexaneIC500.16 [1]
(1S,5S,6S)-1-(3,4-Dichlorophenyl)-6-(ethoxymethyl)-3-azabicyclo[3.1.0]hexaneKi0.5 [1], 1.58 [2]
2-[5-[3-(5-Fluoro-2-methoxyphenyl)propyl]oxolan-2-yl]ethanamineIC501930.0 [1], 5133.0 [2]
2-[5-[3-(5-Fluoro-2-methoxyphenyl)propyl]oxolan-2-yl]ethanamineKi10600.0 [1], 30430.0 [2]
Dimethyl-((2S,3S)-3-naphthalen-2-yl-bicyclo[2.2.1]hept-2-ylmethyl)-amineIC5025.0 [1]
Dimethyl-((2S,3S)-3-naphthalen-2-yl-bicyclo[2.2.1]hept-2-ylmethyl)-amineKi152.0 [1]
(1S,2R)-1-(1H-Indol-1-yl)-3-(methylamino)-1-phenylpropan-2-olIC5023.0 [1], 28.0 [2]
(cis)-2-(5-Bromopentyl)-4-(3,4-dimethoxyphenyl)-4a,5,8,8a-tetrahydrophthalazin-1(2H)-oneIC50100000.0 [1]
(cis)-2-(5-Bromopentyl)-4-(3,4-dimethoxyphenyl)-4a,5,8,8a-tetrahydrophthalazin-1(2H)-oneKi39119.0 [1]
(2S)-4-[3-(2-Fluorophenyl)-2,2-dioxo-2lambda6,1,3-benzothiadiazol-1-yl]-1-(methylamino)butan-2-olIC501.0 [1], 2.0 [2], 4.0 [3], 6.0 [4]
(2R)-4-[3-(2-Fluorophenyl)-2,2-dioxo-2lambda6,1,3-benzothiadiazol-1-yl]-1-(methylamino)butan-2-olIC503.0 [1], 4.0 [2], 9.0 [3]
MethylphenidateIC5061.0 [1]
MethylphenidateKi340.0 [1], 660.0 [2]
CitalopramKi2178.0 [1], 6190.0 [2], 1000000.0 [3]
ParoxetineIC50100.0 [1]
ParoxetineKi86.0 [1], 90.0 [2]
3,4-MethylenedioxymethamphetamineIC50405.0 [1], 1995.26 [2]
SertralineIC50825.0 [1]
SertralineKi976.6 [1]
TenamfetamineIC50266.0 [1], 3162.28 [2]
VanoxerineIC5079.0 [1], 110.0 [2]
Methyl (1R,2S,3S,5R)-3-(4-fluorophenyl)-8-methyl-8-azabicyclo[3.2.1]octane-2-carboxylateIC50834.0 [1]
Methyl (1R,2S,3S,5R)-3-(4-fluorophenyl)-8-methyl-8-azabicyclo[3.2.1]octane-2-carboxylateKi503.0 [1], 635.0 [2]
1-[2-(Diphenylmethoxy)ethyl]-4-(3-phenylpropyl)piperazineIC50165.0 [1], 1261.0 [2]
1-[2-(Diphenylmethoxy)ethyl]-4-(3-phenylpropyl)piperazineKi630.0 [1]
2-((2-((Dimethylamino)methyl)phenyl)thio)-5-iodophenylamineKi699.0 [1], 1352.0 [2]
Benzonitrile, 3-amino-4-((2-((dimethylamino)methyl)phenyl)thio)-Ki1000.0 [1], 1350.0 [2], 5127.0 [3]
N,N-Diallyl-5-methoxytryptamineIC5042657.95 [1]
N,N-Diallyl-5-methoxytryptamineKi10000.0 [1]
(S)-VenlafaxineIC50149.0 [1], 754.0 [2]
3-Amino-4-[[2-[(dimethylamino)methyl]phenyl]thio]benzenemethanolKi303.0 [1], 787.4 [2]
BMS-505130 free baseIC509200.0 [1]
BMS-505130 free baseKi4600.0 [1]
Morpholine, 2-((S)-(2-methoxyphenoxy)phenylmethyl)-, (2S)-Ki0.95 [1], 7.93 [2]
6-(4-Chloro-phenyl)-2,3,4,6-tetrahydro-pyrimido[2,1-a]isoindol-6-olIC504.9 [1]
6-(4-Chloro-phenyl)-2,3,4,6-tetrahydro-pyrimido[2,1-a]isoindol-6-olKi18.0 [1], 18.2 [2]
2-Methyl-N-[(2-phenylphenyl)methyl]-N-[(3S)-pyrrolidin-3-yl]propanamideIC5014.0 [1]
2-Methyl-N-[(2-phenylphenyl)methyl]-N-[(3S)-pyrrolidin-3-yl]propanamideKi6.0 [1]
(1S,5R)-1-(3,4-Dichlorophenyl)-3-azabicyclo(3.1.0)hexaneIC50103.0 [1]
(1S,5R)-1-(3,4-Dichlorophenyl)-3-azabicyclo(3.1.0)hexaneKi58.88 [1], 794.33 [2]
(S)-N-(2,3-Dichlorobenzyl)-N-(pyrrolidin-3-yl)isobutyramideIC5023.0 [1]
(S)-N-(2,3-Dichlorobenzyl)-N-(pyrrolidin-3-yl)isobutyramideKi52.0 [1]
1-[(1R)-2-(2-Ethoxyphenyl)-1-phenylethyl]piperazineIC5016.0 [1], 18.0 [2]
1-[(1R)-2-(2-Ethoxyphenyl)-1-phenylethyl]piperazineKi12.0 [1]
Methyl 2-(3,4-dichlorophenyl)cyclopent-1-enecarboxylateKi11000.0 [1], 28000.0 [2]
(R)-3-(4-(Dimethylamino)cyclohex-1-enyl)-1H-indole-5-carbonitrileIC50390.0 [1]
Silacyclohexan-1-ol, 1-[2-(dimethylamino)-1-(4-methoxyphenyl)ethyl]-IC50109.0 [1]
[(2S,3S)-3-(3-Chloro-phenyl)-bicyclo[2.2.2]oct-2-ylmethyl]-dimethyl-amineIC5044.0 [1]
[(2S,3S)-3-(3-Chloro-phenyl)-bicyclo[2.2.2]oct-2-ylmethyl]-dimethyl-amineKi51.0 [1]
2-(Tert-butylamino)-1-(3-chlorophenyl)butan-1-oneIC50607.0 [1], 969.0 [2]
2-(Tert-butylamino)-1-(3-chlorophenyl)butan-1-oneKi3195.0 [1]
2-(Tert-butylamino)-1-(3-chlorophenyl)pentan-1-oneIC50370.0 [1], 472.0 [2]
2-(Tert-butylamino)-1-(3-chlorophenyl)pentan-1-oneKi1171.0 [1]
1-(3-Bromophenyl)-2-(tert-butylamino)propan-1-oneIC505600.0 [1], 6500.0 [2]
1-(3-Bromophenyl)-2-(tert-butylamino)propan-1-oneKi7140.0 [1]
1-(3-Chlorophenyl)-2-(piperidin-1-yl)propan-1-oneIC502520.0 [1], 4798.0 [2]
1-(3-Chlorophenyl)-2-(piperidin-1-yl)propan-1-oneKi4760.0 [1]
1-(3-Chlorophenyl)-2-(dimethylamino)propan-1-oneIC501260.0 [1], 1520.0 [2]
1-(3-Chlorophenyl)-2-(dimethylamino)propan-1-oneKi3090.0 [1]
Items per page: 1 - 10 of 100
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References

This online tool may be cited as follows

MLA

"Quest Database™ Norepinephrine transporter Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 20 Feb. 2025, https://www.aatbio.com/data-sets/norepinephrine-transporter-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2025, February 20). Quest Database™ Norepinephrine transporter Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/norepinephrine-transporter-inhibitors-ic50-ki.
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