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Neurotensin receptor 3 Inhibitors (IC50, Ki)

Structure
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Compound Name
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Standard Type
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Standard Values (in nM)
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2-[(6-Methylpyridin-2-Yl)carbamoyl]-5-(Trifluoromethyl)benzoic AcidIC50316.23 [1], 330.0 [2]
NeurotensinIC50360.0 [1]
MeclinertantIC50238.0 [1]
(2S)-2-[[(2S,3R)-2-[[(2S)-2-[[(2S)-1-[(2S)-2-[[(2S)-2-Amino-5-(diaminomethylideneamino)pentanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]pyrrolidine-2-carbonyl]amino]-3-(4-hydroxyphenyl)propanoyl]amino]-3-methylpentanoyl]amino]-4-methylpentanoic acidIC50640.0 [1]
5-Phenyl-1,3,4-oxadiazol-2-olIC50125892.54 [1]
5(4H)-Isoxazolone, 3-phenyl-IC50158489.32 [1]
N-[(7-Hydroxy-4-Methyl-2-Oxo-2h-Chromen-8-Yl)methyl]-L-LeucineIC504000.0 [1]
(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-1-[(2S)-2-Amino-5-[[amino-[[(2S)-2,7-diaminoheptanoyl]amino]methylidene]amino]pentanoyl]pyrrolidine-2-carbonyl]amino]-3-(4-hydroxyphenyl)propanoyl]amino]-3,3-dimethylbutanoyl]amino]-4-methylpentanoic acidIC504000.0 [1]
3-(3-Methylbutyl)-4H-1,2,4-oxadiazol-5-oneIC50125892.54 [1]
3-(3-Methylbutyl)-4H-triazol-5-oneIC5063095.73 [1]
N-Methyl-3-(3-methylbutyl)-5-oxo-4H-triazole-4-carboxamideIC5039810.72 [1]
N-[3-(3-Methylbutyl)-5-oxo-4H-triazol-4-yl]pyridine-3-carboxamideIC5012589.25 [1]
3-(3-Methylbutyl)-5-oxo-N-pyridin-3-yl-4H-triazole-4-carboxamideIC503981.07 [1]
3-(3-Methylbutyl)-4H-1,2-oxazol-5-oneIC5012589.25 [1]
3-(3-Methylbutyl)-5-oxo-N-pyridin-4-yl-4H-triazole-4-carboxamideIC5063095.73 [1]
6-Methyl-N-[3-(3-methylbutyl)-5-oxo-4H-triazol-4-yl]pyridine-2-carboxamideIC5039810.72 [1]
4-Methyl-3-(3-methylbutyl)-4H-triazol-5-oneIC5079432.82 [1]
3-(3-Methylbutyl)-N-(6-methylpyridin-2-yl)-5-oxo-4H-triazole-4-carboxamideIC5012589.25 [1]
3-(3-Methylbutyl)-5-oxo-4H-triazole-4-carboxamideIC5050118.72 [1]
N-[3-(3-Methylbutyl)-5-oxo-4H-triazol-4-yl]acetamideIC5031622.78 [1]
N-[3-(3-Methylbutyl)-5-oxo-4H-triazol-4-yl]pyridine-4-carboxamideIC5019952.62 [1]
3-Benzyl-5(4H)-isoxazoloneIC5079432.82 [1]
(2S)-2-[[(2S,3S)-2-[[(2S)-2-[[(2S)-1-[(2S)-2-Amino-5-[[amino-[[(2S)-2,7-diaminoheptanoyl]amino]methylidene]amino]pentanoyl]pyrrolidine-2-carbonyl]amino]-3-(4-hydroxyphenyl)propanoyl]amino]-3-methylpentanoyl]amino]-4-methylpentanoic acidIC501200.0 [1]
(2S)-2-[[(2S,3S)-2-[[(2S)-2-[[(2S)-1-[(2S)-2-Amino-5-[[amino-[[(2S)-2-amino-6-(dimethylamino)hexanoyl]amino]methylidene]amino]pentanoyl]pyrrolidine-2-carbonyl]amino]-3-(4-hydroxyphenyl)propanoyl]amino]-3-methylpentanoyl]amino]-4-methylpentanoic acidIC501620.0 [1]
(2S)-2-[[(2S,3S)-2-[[(2S)-2-[[(2S)-1-[(2S)-2-Amino-5-[[amino-[[(2S)-2-amino-5-(2-amino-4,5-dihydroimidazol-1-yl)pentanoyl]amino]methylidene]amino]pentanoyl]pyrrolidine-2-carbonyl]amino]-3-(4-hydroxyphenyl)propanoyl]amino]-3-methylpentanoyl]amino]-4-methylpentanoic acidIC50590.0 [1]
(2S)-2-[[(2S,3S)-2-[[(2S)-2-[[(2S)-1-[(2S)-2-Amino-5-[[amino-[[(2S)-2-amino-5-(imidazolidin-2-ylamino)pentanoyl]amino]methylidene]amino]pentanoyl]pyrrolidine-2-carbonyl]amino]-3-(4-hydroxyphenyl)propanoyl]amino]-3-methylpentanoyl]amino]-4-methylpentanoic acidIC50510.0 [1]
(2S)-2-[[(2S,3S)-2-[[(2S)-2-[[(2S)-1-[(2S)-2-Amino-5-[[amino-[[(2S)-2-amino-5-[[amino(ethylamino)methylidene]amino]pentanoyl]amino]methylidene]amino]pentanoyl]pyrrolidine-2-carbonyl]amino]-3-(4-hydroxyphenyl)propanoyl]amino]-3-methylpentanoyl]amino]-4-methylpentanoic acidIC50480.0 [1]
(2S,3S)-2-[[(2S)-2-[[(2S)-1-[(2S)-2-[[(2S)-2-[[(2S)-1-[(2S)-6-Amino-2-[[(2S)-4-amino-2-[[2-[[(2S)-2-[[(2S)-2-[[(2S)-2-amino-4-carboxybutanoyl]amino]-4-methylpentanoyl]amino]-3-(4-hydroxyphenyl)propanoyl]amino]acetyl]amino]-4-oxobutanoyl]amino]hexanoyl]pyrrolidine-2-carbonyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]pyrrolidine-2-carbonyl]amino]-3-(4-hydroxyphenyl)propanoyl]amino]-3-methylpentanoic acidIC50440.0 [1]
(2S)-2-[[(2S,3S)-2-[[(2S)-2-[[(2S)-1-[(2S)-2-Amino-5-[[amino-[[(2S)-2-amino-7-(methylamino)heptanoyl]amino]methylidene]amino]pentanoyl]pyrrolidine-2-carbonyl]amino]-3-(4-hydroxyphenyl)propanoyl]amino]-3-methylpentanoyl]amino]-4-methylpentanoic acidIC50400.0 [1]
(2S)-2-[[(2S,3S)-2-[[(2S)-2-[[(2S)-1-[(2S)-2-Amino-5-[[amino-[[(2S)-2-amino-7-(dimethylamino)heptanoyl]amino]methylidene]amino]pentanoyl]pyrrolidine-2-carbonyl]amino]-3-(4-hydroxyphenyl)propanoyl]amino]-3-methylpentanoyl]amino]-4-methylpentanoic acidIC50700.0 [1]
(2S)-2-[[(2S,3S)-2-[[(2S)-2-[[(2S)-1-[(2S)-2-Amino-5-[[amino-[[(2S)-2-amino-5-(diaminomethylideneamino)pentanoyl]amino]methylidene]amino]pentanoyl]pyrrolidine-2-carbonyl]amino]-3-(4-hydroxyphenyl)propanoyl]amino]-3-methylpentanoyl]amino]-4-methylpentanoic acidIC501740.0 [1]
(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-1-[(2S)-2-Amino-5-[[amino-[[(2S)-2,7-diaminoheptanoyl]amino]methylidene]amino]pentanoyl]pyrrolidine-2-carbonyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]-3,3-dimethylbutanoyl]amino]-4-methylpentanoic acidIC5053700.0 [1]
[(4S)-4-Amino-5-[[N'-[(4S)-4-amino-5-[(2S)-2-[[(2S)-1-[[(2S,3S)-1-[[(1S)-1-carboxy-3-methylbutyl]amino]-3-methyl-1-oxopentan-2-yl]amino]-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]carbamoyl]pyrrolidin-1-yl]-5-oxopentyl]carbamimidoyl]amino]-5-oxopentyl]-trimethylazaniumIC502000.0 [1]
[(6S)-6-Amino-7-[[N'-[(4S)-4-amino-5-[(2S)-2-[[(2S)-1-[[(2S,3S)-1-[[(1S)-1-carboxy-3-methylbutyl]amino]-3-methyl-1-oxopentan-2-yl]amino]-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]carbamoyl]pyrrolidin-1-yl]-5-oxopentyl]carbamimidoyl]amino]-7-oxoheptyl]-trimethylazaniumIC50550.0 [1]
(2S)-2-[[(2S,3S)-2-[[(2S)-2-[[(2S)-1-[(2S)-2-Amino-5-[[amino-[[(2S)-2-amino-6-(methylamino)hexanoyl]amino]methylidene]amino]pentanoyl]pyrrolidine-2-carbonyl]amino]-3-(4-hydroxyphenyl)propanoyl]amino]-3-methylpentanoyl]amino]-4-methylpentanoic acidIC501150.0 [1]
(2S)-2-[[(2S,3S)-2-[[(2S)-2-[[(2S)-1-[(2S)-2-Amino-5-[[amino-[[(2S)-2-amino-5-[(N'-methylcarbamimidoyl)amino]pentanoyl]amino]methylidene]amino]pentanoyl]pyrrolidine-2-carbonyl]amino]-3-(4-hydroxyphenyl)propanoyl]amino]-3-methylpentanoyl]amino]-4-methylpentanoic acidIC50720.0 [1]
(2S)-2-[[(2S,3S)-2-[[(2S)-2-[[(2S)-1-[(2S)-2-Amino-5-[[amino-[[(2S)-2,6-diaminohexanoyl]amino]methylidene]amino]pentanoyl]pyrrolidine-2-carbonyl]amino]-3-(4-hydroxyphenyl)propanoyl]amino]-3-methylpentanoyl]amino]-4-methylpentanoic acidIC50512.0 [1]
(2S)-2-[[(2S,3S)-2-[[(2S)-2-[[(2S)-1-[(2S)-2-Amino-5-[[amino-[[(2S)-2-amino-5-(dimethylamino)pentanoyl]amino]methylidene]amino]pentanoyl]pyrrolidine-2-carbonyl]amino]-3-(4-hydroxyphenyl)propanoyl]amino]-3-methylpentanoyl]amino]-4-methylpentanoic acidIC50480.0 [1]
(2S)-2-[[(2S,3S)-2-[[(2S)-2-[[(2S)-1-[(2S)-2-Amino-5-[[amino-[[(2S)-2-amino-5-(methylamino)pentanoyl]amino]methylidene]amino]pentanoyl]pyrrolidine-2-carbonyl]amino]-3-(4-hydroxyphenyl)propanoyl]amino]-3-methylpentanoyl]amino]-4-methylpentanoic acidIC50640.0 [1]
(2S)-2-[[(2S,3S)-2-[[(2S)-2-[[(2S)-1-[(2S)-2-Amino-5-[[amino-[[(2S)-2,5-diaminopentanoyl]amino]methylidene]amino]pentanoyl]pyrrolidine-2-carbonyl]amino]-3-(4-hydroxyphenyl)propanoyl]amino]-3-methylpentanoyl]amino]-4-methylpentanoic acidIC501400.0 [1]
[(5S)-5-Amino-6-[[N'-[(4S)-4-amino-5-[(2S)-2-[[(2S)-1-[[(2S,3S)-1-[[(1S)-1-carboxy-3-methylbutyl]amino]-3-methyl-1-oxopentan-2-yl]amino]-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]carbamoyl]pyrrolidin-1-yl]-5-oxopentyl]carbamimidoyl]amino]-6-oxohexyl]-trimethylazaniumIC503500.0 [1]
3-(2-Methylpropyl)-4H-1,2-oxazol-5-oneIC5031622.78 [1]
5-(3-Methylbutyl)-3H-1,3,4-oxadiazol-2-oneIC5063095.73 [1]
3-Benzyl-4H-triazol-5-oneIC50125892.54 [1]
5-Bromo-2-[(6-methylpyridin-2-yl)carbamoyl]benzoic acidIC50710.0 [1]
4-Bromo-2-[(6-methylpyridin-2-yl)carbamoyl]benzoic acidIC5012000.0 [1]
5-Chloro-2-[(6-methylpyridin-2-yl)carbamoyl]benzoic acidIC501400.0 [1]
5-Methyl-2-[(6-methylpyridin-2-yl)carbamoyl]benzoic acidIC506400.0 [1]
2-[(6-Methylpyridin-2-yl)carbamoyl]-5-propan-2-ylbenzoic acidIC501100.0 [1]
2-[(6-Methylpyridin-2-yl)carbamoyl]-5-nitrobenzoic acidIC501700.0 [1]
2-[(6-Methylpyridin-2-yl)carbamoyl]-4-(trifluoromethyl)benzoic acidIC509100.0 [1]
4,5-Dichloro-2-[(6-methylpyridin-2-yl)carbamoyl]benzoic acidIC50830.0 [1]
4,5-Dimethyl-2-[(6-methylpyridin-2-yl)carbamoyl]benzoic acidIC503400.0 [1]
5-Bromo-2-[(3-methylphenyl)carbamoyl]benzoic acidIC505200.0 [1]
5-Bromo-2-(pyridin-2-ylcarbamoyl)benzoic acidIC503600.0 [1]
5-Bromo-2-[(6-chloropyridin-2-yl)carbamoyl]benzoic acidIC501600.0 [1]
5-Bromo-2-[(4-methylpyridin-2-yl)carbamoyl]benzoic acidIC502400.0 [1]
5-Bromo-2-[(2-methylpyridin-4-yl)carbamoyl]benzoic acidIC501800.0 [1]
5-Bromo-2-[(2-methylpyrimidin-4-yl)carbamoyl]benzoic acidIC50490.0 [1]
2-[(6-Methoxypyridin-2-yl)carbamoyl]-5-(trifluoromethyl)benzoic acidIC501300.0 [1]
2-[(5,6-Dimethylpyridin-2-yl)carbamoyl]-5-(trifluoromethyl)benzoic acidIC50170.0 [1]
2-(5,6,7,8-Tetrahydroquinolin-2-ylcarbamoyl)-5-(trifluoromethyl)benzoic acidIC50100.0 [1]
Items per page: 1 - 10 of 62
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References

This online tool may be cited as follows

MLA

"Quest Database™ Neurotensin receptor 3 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 21 Dec. 2024, https://www.aatbio.com/data-sets/neurotensin-receptor-3-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, December 21). Quest Database™ Neurotensin receptor 3 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/neurotensin-receptor-3-inhibitors-ic50-ki.
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