 | (2R)-5-(Diaminomethylideneamino)-2-[(2,2-diphenylacetyl)amino]-N-[(4-hydroxyphenyl)methyl]pentanamide | IC50 | 3.98 [1], 8.8 [2], 10.23 [3], 11.75 [4], 16.22 [5] |
| (2R)-5-(Diaminomethylideneamino)-2-[(2,2-diphenylacetyl)amino]-N-[(4-hydroxyphenyl)methyl]pentanamide | Ki | 14.9 [1] |
 | Ethyl 2-[[N'-[(4R)-4-[(2,2-diphenylacetyl)amino]-5-[(4-hydroxyphenyl)methylamino]-5-oxopentyl]carbamimidoyl]carbamoylamino]acetate | IC50 | 0.13 [1] |
 | (2R)-5-[[Amino-[2-(propanoylamino)ethylcarbamoylamino]methylidene]amino]-2-[(2,2-diphenylacetyl)amino]-N-[(4-hydroxyphenyl)methyl]pentanamide;2,2,2-trifluoroacetic acid | IC50 | 0.17 [1] |
| (2R)-5-[[Amino-[2-(propanoylamino)ethylcarbamoylamino]methylidene]amino]-2-[(2,2-diphenylacetyl)amino]-N-[(4-hydroxyphenyl)methyl]pentanamide;2,2,2-trifluoroacetic acid | Ki | 0.08 [1], 0.1 [2], 0.23 [3], 0.31 [4] |
 | (2R)-5-[[Amino-(ethylcarbamoylamino)methylidene]amino]-2-[(2,2-diphenylacetyl)amino]-N-[(4-hydroxyphenyl)methyl]pentanamide | IC50 | 0.1 [1], 0.12 [2], 0.24 [3], 0.48 [4], 1.23 [5] |
 | Ethyl 3-[[N'-[(4R)-4-[(2,2-diphenylacetyl)amino]-5-[(4-hydroxyphenyl)methylamino]-5-oxopentyl]carbamimidoyl]carbamoylamino]propanoate | IC50 | 0.16 [1] |
| Ethyl 3-[[N'-[(4R)-4-[(2,2-diphenylacetyl)amino]-5-[(4-hydroxyphenyl)methylamino]-5-oxopentyl]carbamimidoyl]carbamoylamino]propanoate | Ki | 0.3 [1], 0.49 [2] |
 | (2R)-5-[[Amino-[(1-methyltriazol-4-yl)methylcarbamoylamino]methylidene]amino]-2-[(2,2-diphenylacetyl)amino]-N-[(4-hydroxyphenyl)methyl]pentanamide;2,2,2-trifluoroacetic acid | IC50 | 0.35 [1] |
| (2R)-5-[[Amino-[(1-methyltriazol-4-yl)methylcarbamoylamino]methylidene]amino]-2-[(2,2-diphenylacetyl)amino]-N-[(4-hydroxyphenyl)methyl]pentanamide;2,2,2-trifluoroacetic acid | Ki | 0.34 [1], 0.56 [2] |
 | Human Neuropeptide Y | IC50 | 1.2 [1] |
| Human Neuropeptide Y | Ki | 0.5 [1] |
 | CID 16132350 | IC50 | 3.07 [1] |
| CID 16132350 | Ki | 0.12 [1], 0.5 [2], 2.0 [3] |
 | CID 145948574 | IC50 | 1.78 [1] |
| CID 145948574 | Ki | 0.41 [1], 0.6 [2], 0.7 [3] |
 | 4-(3-Piperidinopropoxy)-2-(4-chlorophenoxymethyl)-1-[3-(3-piperidinyl)propyl]-1H-benzimidazole | Ki | 1.7 [1], 2.0 [2] |
 | 2-Diphenylacetylamino-5-guanidino-pentanoic acid 4-hydroxy-benzylamide | IC50 | 5.9 [1], 17.0 [2] |
| 2-Diphenylacetylamino-5-guanidino-pentanoic acid 4-hydroxy-benzylamide | Ki | 4.6 [1] |
 | 1-[2-[(4-Chlorophenoxy)methyl]-1-[3-[(3S)-piperidin-3-yl]propyl]indol-3-yl]-2-(4-piperidin-1-ylpiperidin-1-yl)ethanone | Ki | 0.75 [1], 1.8 [2] |
 | Bms-193885 | IC50 | 4.2 [1] |
| Bms-193885 | Ki | 3.3 [1] |
 | Neuropeptide Y (24-36) amide, N-acetyl-(leu(28,31))- | Ki | 210.0 [1] |
 | FR-226928 free base | IC50 | 9500.0 [1], 9600.0 [2] |
 | 1-Methyl-2-(4-chlorophenoxymethyl)-3-(piperidinomethyl)-1H-indole | Ki | 2310.0 [1], 2315.0 [2] |
 | Dimethyl 4-[3-[3-[4-(2-methoxyphenyl)piperazin-1-yl]propylcarbamoylamino]phenyl]-2,6-dimethyl-1,4-dihydropyridine-3,5-dicarboxylate | IC50 | 12.0 [1] |
| Dimethyl 4-[3-[3-[4-(2-methoxyphenyl)piperazin-1-yl]propylcarbamoylamino]phenyl]-2,6-dimethyl-1,4-dihydropyridine-3,5-dicarboxylate | Ki | 12.0 [1] |
 | (2S)-2-[[(2S)-2-[[(2S,3R)-2-[[(2S)-2-[[(2S)-2-[[(2S)-4-Amino-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[(2-aminobenzoyl)amino]-5-carbamimidamidopentanoyl]amino]-3-(1H-imidazol-5-yl)propanoyl]amino]-3-(4-hydroxyphenyl)propanoyl]amino]-4-methylpentanoyl]amino]-4-oxobutanoyl]amino]-4-methylpentanoyl]amino]-3-methylbutanoyl]amino]-3-hydroxybutanoyl]amino]-5-carbamimidamidopentanoyl]amino]-N-[(2S)-1-[[(2S)-1-amino-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]amino]-5-carbamimidamido-1-oxopentan-2-yl]pentanediamide | Ki | 1000.0 [1] |
 | N-[[4-[(1,2,3,4-Tetrahydronaphthalen-2-ylmethylamino)methyl]cyclohexyl]methyl]naphthalene-1-sulfonamide | IC50 | 1300.0 [1] |
| N-[[4-[(1,2,3,4-Tetrahydronaphthalen-2-ylmethylamino)methyl]cyclohexyl]methyl]naphthalene-1-sulfonamide | Ki | 3548.0 [1] |
 | (2R)-5-[[Amino-(propanoylamino)methylidene]amino]-2-[(2,2-diphenylacetyl)amino]-N-[(4-hydroxyphenyl)methyl]pentanamide | Ki | 1.0 [1], 1.2 [2] |
 | (2S)-2-[[(2S)-2-[[(2S,3R)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-Acetamidopropanoyl]amino]-3-hydroxypropanoyl]amino]-4-methylpentanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]-3-(1H-imidazol-4-yl)propanoyl]amino]-3-(4-hydroxyphenyl)propanoyl]amino]-4-methylpentanoyl]amino]-4-amino-4-oxobutanoyl]amino]-4-methylpentanoyl]amino]-3-methylbutanoyl]amino]-3-hydroxybutanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]-N-[(2S)-1-[[(2S)-1-amino-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]amino]-5-(diaminomethylideneamino)-1-oxopentan-2-yl]pentanediamide | IC50 | 1000.0 [1] |
| (2S)-2-[[(2S)-2-[[(2S,3R)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-Acetamidopropanoyl]amino]-3-hydroxypropanoyl]amino]-4-methylpentanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]-3-(1H-imidazol-4-yl)propanoyl]amino]-3-(4-hydroxyphenyl)propanoyl]amino]-4-methylpentanoyl]amino]-4-amino-4-oxobutanoyl]amino]-4-methylpentanoyl]amino]-3-methylbutanoyl]amino]-3-hydroxybutanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]-N-[(2S)-1-[[(2S)-1-amino-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]amino]-5-(diaminomethylideneamino)-1-oxopentan-2-yl]pentanediamide | Ki | 118.0 [1] |
 | (2S)-2-[[(2S)-2-[[(2S)-5-Amino-2-[[(2S)-2-[[(2S,3R)-2-[[(2S,3S)-2-[[(2S)-2-[[(2S)-4-amino-2-[[(2S,3S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[6-[[(2S)-6-amino-2-[[(2S)-2-[[(2S)-1-[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]pyrrolidine-2-carbonyl]amino]-3-hydroxypropanoyl]amino]hexanoyl]amino]hexanoylamino]-5-(diaminomethylideneamino)pentanoyl]amino]-3-(1H-imidazol-4-yl)propanoyl]amino]-3-(4-hydroxyphenyl)propanoyl]amino]-3-methylpentanoyl]amino]-4-oxobutanoyl]amino]-4-methylpentanoyl]amino]-3-methylpentanoyl]amino]-3-hydroxybutanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]-5-oxopentanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]-3-(4-hydroxyphenyl)propanoic acid | Ki | 261.0 [1], 398.11 [2] |
 | 2-[(4-Chlorophenoxy)methyl]-4-methyl-1-[3-[1-(3-piperidin-1-ylpropyl)piperidin-4-yl]propyl]benzimidazole | Ki | 4.5 [1] |
 | (2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2R)-2-Amino-3-[[(2R)-2-amino-3-[[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-amino-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]amino]-5-(diaminomethylideneamino)-1-oxopentan-2-yl]amino]-1-oxopentan-2-yl]amino]-5-(diaminomethylideneamino)-1-oxopentan-2-yl]amino]-3-(1H-indol-3-yl)-1-oxopropan-2-yl]amino]-3-oxopropyl]disulfanyl]propanoyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]pentanoyl]amino]-N-[(2S)-1-amino-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]-5-(diaminomethylideneamino)pentanamide | Ki | 46.0 [1], 340.0 [2] |
 | Unii-glz1WA47Q8 | IC50 | 7.0 [1] |
| Unii-glz1WA47Q8 | Ki | 1.0 [1] |
 | [5-Bromo-2-[[3-[2-[4-(dimethylamino)piperidin-1-yl]ethyl]-1-benzothiophen-2-yl]methoxy]phenyl]methanol | Ki | 15.0 [1], 1200.0 [2] |
 | Dimethyl 4-[3-[[N-cyano-N'-[2-[[1-(2-methoxyphenyl)piperidin-4-yl]amino]ethyl]carbamimidoyl]amino]phenyl]-2,6-dimethyl-1,4-dihydropyridine-3,5-dicarboxylate | IC50 | 4.0 [1] |
| Dimethyl 4-[3-[[N-cyano-N'-[2-[[1-(2-methoxyphenyl)piperidin-4-yl]amino]ethyl]carbamimidoyl]amino]phenyl]-2,6-dimethyl-1,4-dihydropyridine-3,5-dicarboxylate | Ki | 3.6 [1] |
 | Dimethyl 4-[3-[2-[[1-(2-methoxyphenyl)piperidin-4-yl]amino]ethylcarbamoylamino]phenyl]-2,6-dimethyl-1,4-dihydropyridine-3,5-dicarboxylate | IC50 | 2.0 [1] |
| Dimethyl 4-[3-[2-[[1-(2-methoxyphenyl)piperidin-4-yl]amino]ethylcarbamoylamino]phenyl]-2,6-dimethyl-1,4-dihydropyridine-3,5-dicarboxylate | Ki | 1.9 [1] |
 | N-[1-(7-Hydroxy-1,3,4,5-tetrahydro-2-benzazepin-2-yl)-1-oxo-5-[[N'-(3-phenylpropyl)carbamimidoyl]amino]pentan-2-yl]-2-(4-phenylphenyl)acetamide | IC50 | 11900.0 [1], 22000.0 [2] |
 | 5-(Diaminomethylideneamino)-2-[(2,2-diphenylacetyl)amino]-N-[(1S)-2-hydroxy-1-phenylethyl]pentanamide | IC50 | 184.0 [1], 900.0 [2] |
 | N-[(1R)-2-Amino-2-oxo-1-phenylethyl]-5-(diaminomethylideneamino)-2-[(2,2-diphenylacetyl)amino]pentanamide | IC50 | 2400.0 [1], 4600.0 [2] |
 | 5-(Diaminomethylideneamino)-2-[(2,2-diphenylacetyl)amino]-N-[(1R)-1-phenylethyl]pentanamide | IC50 | 150.0 [1], 200.0 [2] |
 | N-[5-(Diaminomethylideneamino)-1-(7-hydroxy-1,3,4,5-tetrahydro-2-benzazepin-2-yl)-1-oxopentan-2-yl]-2,2-diphenylacetamide | IC50 | 280.0 [1], 670.0 [2] |
 | 5-(Diaminomethylideneamino)-2-[(2,2-diphenylacetyl)amino]-N-[1-(4-hydroxyphenyl)ethyl]pentanamide | IC50 | 19.0 [1], 60.0 [2] |
 | N-Benzyl-2-[[2-(4-chlorophenyl)-2-phenylacetyl]amino]-5-(diaminomethylideneamino)pentanamide | IC50 | 81.0 [1], 170.0 [2] |
 | 2-[[2-(4-Chlorophenyl)-2-phenylacetyl]amino]-5-(diaminomethylideneamino)-N-[(1S)-2,3-dihydro-1H-inden-1-yl]pentanamide | IC50 | 3000.0 [1], 5300.0 [2] |
 | 1-[2-[2-[(2,4-Dichlorophenoxy)methyl]-1-benzothiophen-3-yl]ethyl]-N,N-dimethylpiperidin-4-amine | Ki | 140.0 [1], 4700.0 [2] |
 | [(1R,4R)-4-[[(1S)-2,2-Difluoro-1-(4-methoxyphenyl)ethyl]amino]-2,2-dimethylcyclohexyl]-[4-phenyl-4-(pyrrolidine-1-carbonyl)piperidin-1-yl]methanone | IC50 | 280.0 [1] |
| [(1R,4R)-4-[[(1S)-2,2-Difluoro-1-(4-methoxyphenyl)ethyl]amino]-2,2-dimethylcyclohexyl]-[4-phenyl-4-(pyrrolidine-1-carbonyl)piperidin-1-yl]methanone | Ki | 22.0 [1] |
 | CID 71566722 | IC50 | 74.0 [1], 80.0 [2] |
 | 4-N-[2-[2-[2-[[(Z)-[Amino-[[(4R)-4-[(2,2-diphenylacetyl)amino]-5-[(4-hydroxyphenyl)methylamino]-5-oxopentyl]amino]methylidene]carbamoyl]amino]ethoxy]ethoxy]ethyl]-1-N-[2-[2-[[4-[2-[2-[2-[[(Z)-[amino-[[(4R)-4-[(2,2-diphenylacetyl)amino]-5-[(4-hydroxyphenyl)methylamino]-5-oxopentyl]amino]methylidene]carbamoyl]amino]ethoxy]ethoxy]ethylcarbamoyl]benzoyl]amino]ethyl-[2-(propanoylamino)ethyl]amino]ethyl]benzene-1,4-dicarboxamide;2,2,2-trifluoroacetic acid | Ki | 64.0 [1], 110.0 [2] |
 | N'-[2-[2-[2-[[(Z)-[Amino-[[(4R)-4-[(2,2-diphenylacetyl)amino]-5-[(4-hydroxyphenyl)methylamino]-5-oxopentyl]amino]methylidene]carbamoyl]amino]ethoxy]ethoxy]ethyl]-N-[2-[2-[[4-[2-[2-[2-[[(Z)-[amino-[[(4R)-4-[(2,2-diphenylacetyl)amino]-5-[(4-hydroxyphenyl)methylamino]-5-oxopentyl]amino]methylidene]carbamoyl]amino]ethoxy]ethoxy]ethylamino]-4-oxobutanoyl]amino]ethyl-(2-aminoethyl)amino]ethyl]butanediamide;2,2,2-trifluoroacetic acid | Ki | 25.0 [1], 37.0 [2] |
 | 4-N-[2-[2-[2-[[(Z)-[Amino-[[(4R)-4-[(2,2-diphenylacetyl)amino]-5-[(4-hydroxyphenyl)methylamino]-5-oxopentyl]amino]methylidene]carbamoyl]amino]ethoxy]ethoxy]ethyl]-1-N-[2-[2-[[4-[2-[2-[2-[[(Z)-[amino-[[(4R)-4-[(2,2-diphenylacetyl)amino]-5-[(4-hydroxyphenyl)methylamino]-5-oxopentyl]amino]methylidene]carbamoyl]amino]ethoxy]ethoxy]ethylcarbamoyl]benzoyl]amino]ethyl-(2-aminoethyl)amino]ethyl]benzene-1,4-dicarboxamide;2,2,2-trifluoroacetic acid | Ki | 24.0 [1], 48.0 [2] |
 | N'-[2-[2-Aminoethyl-[2-[[5-[4-[[4-[[[(2R)-5-carbamimidamido-2-[(2,2-diphenylacetyl)amino]pentanoyl]amino]methyl]phenyl]methylcarbamoylamino]butylamino]-5-oxopentanoyl]amino]ethyl]amino]ethyl]-N-[4-[[4-[[[(2R)-5-carbamimidamido-2-[(2,2-diphenylacetyl)amino]pentanoyl]amino]methyl]phenyl]methylcarbamoylamino]butyl]pentanediamide;2,2,2-trifluoroacetic acid | Ki | 330.0 [1], 430.0 [2] |
 | N'-[2-[2-[2-[[(Z)-[Amino-[[(4R)-5-[[4-[(carbamoylamino)methyl]phenyl]methylamino]-4-[(2,2-diphenylacetyl)amino]-5-oxopentyl]amino]methylidene]carbamoyl]amino]ethoxy]ethoxy]ethyl]-N-[2-[2-[[4-[2-[2-[2-[[(Z)-[amino-[[(4R)-5-[[4-[(carbamoylamino)methyl]phenyl]methylamino]-4-[(2,2-diphenylacetyl)amino]-5-oxopentyl]amino]methylidene]carbamoyl]amino]ethoxy]ethoxy]ethylamino]-4-oxobutanoyl]amino]ethyl-(2-aminoethyl)amino]ethyl]butanediamide;2,2,2-trifluoroacetic acid | Ki | 210.0 [1], 230.0 [2] |
 | N'-[2-[2-[2-[[(Z)-[Amino-[[(4R)-4-[(2,2-diphenylacetyl)amino]-5-[(4-hydroxyphenyl)methylamino]-5-oxopentyl]amino]methylidene]carbamoyl]amino]ethoxy]ethoxy]ethyl]-N-[2-[2-[[5-[2-[2-[2-[[(Z)-[amino-[[(4R)-4-[(2,2-diphenylacetyl)amino]-5-[(4-hydroxyphenyl)methylamino]-5-oxopentyl]amino]methylidene]carbamoyl]amino]ethoxy]ethoxy]ethylamino]-5-oxopentanoyl]amino]ethyl-(2-aminoethyl)amino]ethyl]pentanediamide;2,2,2-trifluoroacetic acid | Ki | 29.0 [1], 50.0 [2] |
 | N'-[3-(2,6-Dichloro-4-propoxyphenyl)-2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl]-N-(oxan-4-yl)ethane-1,2-diamine | IC50 | 207.0 [1] |
| N'-[3-(2,6-Dichloro-4-propoxyphenyl)-2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl]-N-(oxan-4-yl)ethane-1,2-diamine | Ki | 8.0 [1] |
 | N'-[3-(2,6-Dichloro-4-ethoxyphenyl)-2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl]-N-(oxan-4-yl)ethane-1,2-diamine | IC50 | 15.0 [1] |
| N'-[3-(2,6-Dichloro-4-ethoxyphenyl)-2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl]-N-(oxan-4-yl)ethane-1,2-diamine | Ki | 3.0 [1] |
 | N-[2-[4-[(E)-2-(1-Azatricyclo[7.3.1.05,13]trideca-5,7,9(13)-trien-7-yl)ethenyl]-2,6-dimethylpyridin-1-ium-1-yl]ethyl]-N'-[N'-[(4R)-4-[(2,2-diphenylacetyl)amino]-5-[(4-hydroxyphenyl)methylamino]-5-oxopentyl]carbamimidoyl]pentanediamide | Ki | 22.0 [1] |
 | (2R)-5-[[Amino-[4-[4-[2-[(1E,3E)-4-[4-(dimethylamino)phenyl]buta-1,3-dienyl]-1,3-benzothiazol-3-ium-3-yl]butanoylamino]butylcarbamoylamino]methylidene]amino]-2-[(2,2-diphenylacetyl)amino]-N-[(4-hydroxyphenyl)methyl]pentanamide | Ki | 26.0 [1] |
 | N-[6-[[(E)-[Amino-[[(4S)-5-[2-(3,5-dioxo-1,2-diphenyl-1,2,4-triazolidin-4-yl)ethylamino]-5-oxo-4-[[2-[1-[2-oxo-2-[4-(6-oxo-5,11-dihydrobenzo[c][1]benzazepin-11-yl)piperazin-1-yl]ethyl]cyclopentyl]acetyl]amino]pentyl]amino]methylidene]carbamoyl]amino]hexyl]-N'-[2-[2-[[4-[6-[[(E)-[amino-[[(4R)-4-[(2,2-diphenylacetyl)amino]-5-[(4-hydroxyphenyl)methylamino]-5-oxopentyl]amino]methylidene]carbamoyl]amino]hexylamino]-4-oxobutanoyl]amino]ethyl-(2-aminoethyl)amino]ethyl]butanediamide | Ki | 230.0 [1], 260.0 [2] |
 | Unii-PX9azu7qpk | IC50 | 4.7 [1] |
 | Peptide YY | Ki | 0.13 [1] |
 | (2S)-5-(Diaminomethylideneamino)-2-[(2,2-diphenylacetyl)amino]-N-[(4-hydroxyphenyl)methyl]pentanamide | Ki | 10000.0 [1] |
 | Benextramine | Ki | 1800.0 [1] |
 | BIBO-3304 free base | Ki | 0.25 [1] |
 | Cipargamin | IC50 | 10000.0 [1] |
 | N-[[4-[[(4-Aminoquinazolin-2-yl)amino]methyl]cyclohexyl]methyl]naphthalene-1-sulfonamide | IC50 | 8370.0 [1] |
 | 4-(4-Butylpiperidin-1-yl)-1-o-tolylbutan-1-one | Ki | 1000.0 [1] |
 | N-[[4-(4,5-Dihydro-[1]benzothiepino[5,4-d][1,3]thiazol-2-ylamino)cyclohexyl]methyl]methanesulfonamide | IC50 | 1000.0 [1] |
 | 9-(2-Hydroxy-4,4-dimethyl-6-oxo-1-cyclohexen-1-yl)-3,3-dimethyl-2,3,4,9-tetrahydro-1H-xanthen-1-one | IC50 | 10000.0 [1] |
 | 3-Amino-2-[4-(4-quinolin-2-ylpiperazin-1-yl)butyl]-5,6,7,8-tetrahydroquinazolin-4-one | IC50 | 1000.0 [1] |
 | Propan-2-yl N-[3-chloro-5-[1-[[6-[2-(5-ethyl-4-methyl-1,3-thiazol-2-yl)ethyl]-4-morpholin-4-ylpyridin-2-yl]amino]ethyl]phenyl]carbamate | IC50 | 1.4 [1] |
 | (2S)-1-[(2S)-4-Amino-2-[[(2S,3S)-2-amino-3-methylpentanoyl]amino]-4-oxobutanoyl]-N-[(2S,3S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-amino-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]amino]-5-(diaminomethylideneamino)-1-oxopentan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]amino]-5-(diaminomethylideneamino)-1-oxopentan-2-yl]amino]-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]amino]-3-methyl-1-oxopentan-2-yl]pyrrolidine-2-carboxamide | Ki | 5.0 [1] |
 | CID 16200926 | Ki | 21.0 [1] |
 | N-[1-[3-(3-Oxo-1,4-benzoxazin-4-yl)propyl]piperidin-4-yl]-2-phenylacetamide | Ki | 1000.0 [1] |
 | 4-(Pyridin-2-yl)-N-[4-(trifluoromethyl)phenyl]-1,3-thiazol-2-amine | Ki | 31622.78 [1] |
 | 3-Oxo-N-(5-phenylpyrazin-2-yl)spiro[2-benzofuran-1,4'-piperidine]-1'-carboxamide | IC50 | 10000.0 [1] |
 | N-{3-Chloro-4-[4-(phenylcarbonyl)piperazin-1-yl]phenyl}-2,2-dimethylpropanamide | Ki | 6309.57 [1] |
 | CID 44351001 | Ki | 460.0 [1] |
 | CID 44351041 | Ki | 2.0 [1] |
 | (2R)-5-(Diaminomethylideneamino)-N-[2-(3,5-dioxo-1,2-diphenyl-1,2,4-triazolidin-4-yl)ethyl]-2-[[2-[1-[2-oxo-2-[4-(6-oxo-5,11-dihydrobenzo[c][1]benzazepin-11-yl)piperazin-1-yl]ethyl]cyclopentyl]acetyl]amino]pentanamide | Ki | 5000.0 [1] |
 | 3-[2-[6-[2-[(2-Methylpropan-2-yl)oxy]ethoxy]pyridin-3-yl]-1H-imidazol-5-yl]benzonitrile | IC50 | 1000.0 [1] |
 | N-[[4-[(Naphthalen-2-ylmethylamino)methyl]cyclohexyl]methyl]naphthalene-2-sulfonamide | IC50 | 10000.0 [1] |
 | 1-(Difluoromethyl)-5-[(4S,5S)-5-(4-fluorophenyl)-5-(6-fluoropyridin-3-yl)-4-methyl-1,4-dihydroimidazol-2-yl]pyridin-2-one | IC50 | 10000.0 [1] |
 | 4-Bromo-N-[[4-[(thiophene-2-carbonylamino)carbamoyl]cyclohexyl]methyl]benzenesulfonamide | IC50 | 10000.0 [1] |
 | CID 118718116 | Ki | 1000.0 [1] |
 | CID 118718124 | Ki | 14.0 [1] |
 | CID 118718320 | Ki | 260.0 [1] |
 | 2-[(4S,5S)-5-(4-Fluorophenyl)-5-(6-fluoropyridin-3-yl)-4-methyl-1,4-dihydroimidazol-2-yl]pyridine-4-carbonitrile | IC50 | 10000.0 [1] |
 | CID 44349418 | Ki | 2.9 [1] |
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