![](https://images.aatbio.com/dataset/ic50/neuropeptide-s-receptor_63fdedf3aa86fea51a0637df1f4ca79c.svg) | N-[(4-Fluorophenyl)methyl]-3-oxo-1,1-diphenyl-5,6,8,8a-tetrahydro-[1,3]oxazolo[3,4-a]pyrazine-7-carboxamide | IC50 | 14.0 [1], 420.0 [2] |
![](https://images.aatbio.com/dataset/ic50/neuropeptide-s-receptor_56f545077ee186dccbfd8155d8f5393f.svg) | CID 44156964 | IC50 | 11.0 [1], 55.0 [2], 785.0 [3] |
![](https://images.aatbio.com/dataset/ic50/neuropeptide-s-receptor_3bcc29786e7383c05f287871ab50352d.svg) | (1,2-Dimethylimidazo[1,2-a]pyridin-4-ium-3-yl)-diphenyl-sulfanylidene-lambda5-phosphane;iodide | IC50 | 30.0 [1], 51.0 [2] |
![](https://images.aatbio.com/dataset/ic50/neuropeptide-s-receptor_0d4c7ccacd1d3012831193b3c2c5a67d.svg) | [2-Methyl-1-[(E)-3-phenylprop-2-enyl]imidazo[1,2-a]pyridin-4-ium-3-yl]-diphenyl-sulfanylidene-lambda5-phosphane;bromide | IC50 | 0.96 [1], 1.3 [2], 3.5 [3], 45.0 [4] |
![](https://images.aatbio.com/dataset/ic50/neuropeptide-s-receptor_92406b199d3fe8d09b1f08a9cdd5fe46.svg) | [2-Methyl-1-(2-phenylethyl)imidazo[1,2-a]pyridin-4-ium-3-yl]-diphenyl-sulfanylidene-lambda5-phosphane;bromide | IC50 | 16.0 [1], 73.0 [2], 2100.0 [3] |
![](https://images.aatbio.com/dataset/ic50/neuropeptide-s-receptor_82527c73afce604418ed136799a32987.svg) | (2-Methyl-3-imidazo[1,2-a]pyridinyl)-diphenyl-sulfanylidenephosphorane | IC50 | 9.1 [1], 1000.0 [2], 18000.0 [3] |
![](https://images.aatbio.com/dataset/ic50/neuropeptide-s-receptor_72a5cbaa4686790516c7be23f9a9db2d.svg) | [2-Methyl-1-(4-phenylbutyl)imidazo[1,2-a]pyridin-4-ium-3-yl]-diphenyl-sulfanylidene-lambda5-phosphane;bromide | IC50 | 0.5 [1], 15.0 [2], 940.0 [3] |
![](https://images.aatbio.com/dataset/ic50/neuropeptide-s-receptor_4c6bc42f993bc3d33f4021212a7a2883.svg) | [2-Methyl-1-(5-phenylpentyl)imidazo[1,2-a]pyridin-4-ium-3-yl]-diphenyl-sulfanylidene-lambda5-phosphane;2,2,2-trifluoroacetate | IC50 | 6.2 [1], 13.0 [2], 710.0 [3] |
![](https://images.aatbio.com/dataset/ic50/neuropeptide-s-receptor_91a217da862af2ba23664454ceeecc07.svg) | (1-Benzyl-2-methylimidazo[1,2-a]pyridin-4-ium-3-yl)-diphenyl-sulfanylidene-lambda5-phosphane;2,2,2-trifluoroacetate | IC50 | 16.0 [1], 32.0 [2], 1300.0 [3] |
![](https://images.aatbio.com/dataset/ic50/neuropeptide-s-receptor_dd5f281d6e129f439b66a2d7b3810214.svg) | [2-Methyl-1-(3-phenylpropyl)imidazo[1,2-a]pyridin-4-ium-3-yl]-diphenyl-sulfanylidene-lambda5-phosphane;2,2,2-trifluoroacetate | IC50 | 0.5 [1], 110.0 [2] |
![](https://images.aatbio.com/dataset/ic50/neuropeptide-s-receptor_890666432d13d596982f13820be36745.svg) | 18-(3,4-Dimethoxyphenyl)-15-(2-morpholin-4-ylethyl)-11-oxa-13,15-diazatetracyclo[8.8.0.02,7.012,17]octadeca-1(10),2,4,6,8,13-hexaen-16-imine | IC50 | 190.0 [1], 1400.0 [2], 4900.0 [3] |
![](https://images.aatbio.com/dataset/ic50/neuropeptide-s-receptor_2ca73c0e7cf92868027e3f8b8c5139f7.svg) | 1-(3-Diphenylphosphinothioyl-2-methylimidazo[1,2-a]pyridin-4-ium-1-yl)-2-phenylethanone | IC50 | 13.0 [1], 80.0 [2], 2100.0 [3] |
![](https://images.aatbio.com/dataset/ic50/neuropeptide-s-receptor_fa427d30c0ceb09318e34f30fb98a59c.svg) | N-Benzyl-3-oxo-1,1-diphenyl-5,6,8,8a-tetrahydro-[1,3]oxazolo[3,4-a]pyrazine-7-carboxamide | IC50 | 2.0 [1], 26.0 [2] |
![](https://images.aatbio.com/dataset/ic50/neuropeptide-s-receptor_164c8e3826774088abd575986e86a1d6.svg) | CID 46203026 | IC50 | 43.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuropeptide-s-receptor_e6eb1c8ce1c286f3c7900555d79c054a.svg) | 5-Phenyl-2-[2-(piperidine-1-carbonyl)phenyl]-3H-pyrrolo[1,2-c]imidazol-1-one | IC50 | 10.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuropeptide-s-receptor_77113fdcfeec04374c4b5f91b460cae9.svg) | 3-Imidazo[1,2-a]pyridinyl-diphenyl-sulfanylidenephosphorane | IC50 | 4030.0 [1], 63000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/neuropeptide-s-receptor_bc6d484a1db6c49459616850ae330e9a.svg) | (1-Methylimidazo[1,2-a]pyridin-1-ium-3-yl)-diphenyl-sulfanylidene-lambda5-phosphane;methyl sulfate | IC50 | 2500.0 [1], 39000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/neuropeptide-s-receptor_5fc2f813afd095557e62c6bdcac91de9.svg) | [1-[(E)-3-(3-Methoxyphenyl)prop-2-enyl]-2-methylimidazo[1,2-a]pyridin-4-ium-3-yl]-diphenyl-sulfanylidene-lambda5-phosphane;2,2,2-trifluoroacetate | IC50 | 3.2 [1], 110.0 [2] |
![](https://images.aatbio.com/dataset/ic50/neuropeptide-s-receptor_dda514c585186a7fbf35089ff5e57d7d.svg) | [1-[(E)-3-(2-Chlorophenyl)prop-2-enyl]-2-methylimidazo[1,2-a]pyridin-4-ium-3-yl]-diphenyl-sulfanylidene-lambda5-phosphane;2,2,2-trifluoroacetate | IC50 | 3.4 [1], 94.0 [2] |
![](https://images.aatbio.com/dataset/ic50/neuropeptide-s-receptor_53f95a4510968b29b38d5f14cc320d6c.svg) | [1-[(E)-3-(3-Chlorophenyl)prop-2-enyl]-2-methylimidazo[1,2-a]pyridin-4-ium-3-yl]-diphenyl-sulfanylidene-lambda5-phosphane;2,2,2-trifluoroacetate | IC50 | 9.2 [1], 220.0 [2] |
![](https://images.aatbio.com/dataset/ic50/neuropeptide-s-receptor_3139865ca37bdf39fcc91f6a26fd081e.svg) | [1-[(E)-3-(4-Chlorophenyl)prop-2-enyl]-2-methylimidazo[1,2-a]pyridin-4-ium-3-yl]-diphenyl-sulfanylidene-lambda5-phosphane;2,2,2-trifluoroacetate | IC50 | 2.2 [1], 120.0 [2] |
![](https://images.aatbio.com/dataset/ic50/neuropeptide-s-receptor_1168c60887fa341659753043d4575e1a.svg) | [2-Methyl-1-[(E)-3-[4-(trifluoromethyl)phenyl]prop-2-enyl]imidazo[1,2-a]pyridin-4-ium-3-yl]-diphenyl-sulfanylidene-lambda5-phosphane;2,2,2-trifluoroacetate | IC50 | 4.5 [1], 400.0 [2] |
![](https://images.aatbio.com/dataset/ic50/neuropeptide-s-receptor_d0d54547cca41e47546f867eb971a929.svg) | [1-[(E)-3-(4-Bromophenyl)prop-2-enyl]-2-methylimidazo[1,2-a]pyridin-4-ium-3-yl]-diphenyl-sulfanylidene-lambda5-phosphane;2,2,2-trifluoroacetate | IC50 | 5.7 [1], 170.0 [2] |
![](https://images.aatbio.com/dataset/ic50/neuropeptide-s-receptor_30ec7447baeed473ed69820e698ee712.svg) | [1-[(E)-3-(3-Bromophenyl)prop-2-enyl]-2-methylimidazo[1,2-a]pyridin-4-ium-3-yl]-diphenyl-sulfanylidene-lambda5-phosphane;2,2,2-trifluoroacetate | IC50 | 23.0 [1], 670.0 [2] |
![](https://images.aatbio.com/dataset/ic50/neuropeptide-s-receptor_0ccab1586e1e680672046c1a963d920b.svg) | [2-Methyl-1-[(E)-3-naphthalen-2-ylprop-2-enyl]imidazo[1,2-a]pyridin-4-ium-3-yl]-diphenyl-sulfanylidene-lambda5-phosphane;bromide | IC50 | 64.0 [1], 1300.0 [2] |
![](https://images.aatbio.com/dataset/ic50/neuropeptide-s-receptor_2708d1cb1ee6acd376dcae4c4f4386b9.svg) | [1-[(E)-3-(4-Fluorophenyl)prop-2-enyl]-2-methylimidazo[1,2-a]pyridin-4-ium-3-yl]-diphenyl-sulfanylidene-lambda5-phosphane;2,2,2-trifluoroacetate | IC50 | 3.4 [1], 71.0 [2] |
![](https://images.aatbio.com/dataset/ic50/neuropeptide-s-receptor_d71aca2d15524495521fbd22701221bf.svg) | [1-[(E)-3-(3-Bromo-4-fluorophenyl)prop-2-enyl]-2-methylimidazo[1,2-a]pyridin-4-ium-3-yl]-diphenyl-sulfanylidene-lambda5-phosphane | IC50 | 45.0 [1], 840.0 [2] |
![](https://images.aatbio.com/dataset/ic50/neuropeptide-s-receptor_ccc04e72887a32640471530eee8901e2.svg) | [2-Methyl-1-[(E)-3-(4-methylphenyl)prop-2-enyl]imidazo[1,2-a]pyridin-4-ium-3-yl]-diphenyl-sulfanylidene-lambda5-phosphane | IC50 | 9.0 [1], 330.0 [2] |
![](https://images.aatbio.com/dataset/ic50/neuropeptide-s-receptor_462b685b8561c1078c30b2ab23aa673c.svg) | 5-Phenyl-N-[2-(piperidine-1-carbonyl)phenyl]thiophene-2-carboxamide | IC50 | 794.33 [1] |
![](https://images.aatbio.com/dataset/ic50/neuropeptide-s-receptor_f5836c38368401fa7adcd8ec39d8b5a5.svg) | (1,2-Dimethyl-3-indolyl)-diphenyl-sulfanylidenephosphorane | IC50 | 2800.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuropeptide-s-receptor_92d39b76bd7b65dabd4fa63090407b9b.svg) | Imidazo[1,2-a]pyridin-3-yl(diphenyl)phosphane | IC50 | 35000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuropeptide-s-receptor_713801d8b659d1eb3b80832bdfad0e83.svg) | 3-Diphenylphosphoryl-2-methylimidazo[1,2-a]pyridine | IC50 | 27000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuropeptide-s-receptor_597a279118a7ef8e0a77d2865624b89b.svg) | (1-Methyl-3-indolyl)-diphenyl-sulfanylidenephosphorane | IC50 | 7300.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuropeptide-s-receptor_03923dad1a1e34b09fdf53923f8e3702.svg) | 4-(5-Benzylimidazo[1,2-b]isoindol-5-yl)benzonitrile | IC50 | 387.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuropeptide-s-receptor_e6be1e45c0fa0f6eb2ab600677ddcd7b.svg) | 4-[5-(Cyclohexylmethyl)imidazo[1,2-b]isoindol-5-yl]benzonitrile | IC50 | 114.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuropeptide-s-receptor_9dde4222ec9526fb7507020fa5285ea5.svg) | 4-[5-(Cyclopentylmethyl)imidazo[1,2-b]isoindol-5-yl]benzonitrile | IC50 | 145.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuropeptide-s-receptor_d803f94fd0735dd216c63e46bf322818.svg) | 5-(6-Bromopyridin-3-yl)-5-(cyclopentylmethyl)imidazo[2,1-a]isoindole | IC50 | 851.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuropeptide-s-receptor_f37f62335c6e095ca71b9acb65a4d49b.svg) | 5-Benzyl-5-(5-bromopyridin-2-yl)imidazo[2,1-a]isoindole | IC50 | 2179.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuropeptide-s-receptor_e66666db925251d130485f91ea629b83.svg) | 5-(4-Chlorophenyl)-7-methoxy-5-(oxan-4-ylmethyl)imidazo[2,1-a]isoindole | IC50 | 82.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuropeptide-s-receptor_a8ed1795e5017abe35105bebf3a745ee.svg) | 5-(4-Bromophenyl)-5-(cyclopentylmethyl)imidazo[2,1-a]isoindole | IC50 | 321.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuropeptide-s-receptor_71cc2ccae16001fbbe1494cd8941c825.svg) | 5-(4-Bromophenyl)-5-(cyclohexylmethyl)imidazo[2,1-a]isoindole | IC50 | 254.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuropeptide-s-receptor_d2582ece5090c3e6c41c11da3ac5b7fd.svg) | 5-(4-Chlorophenyl)-6-methoxy-5-(oxan-4-ylmethyl)imidazo[2,1-a]isoindole | IC50 | 46.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuropeptide-s-receptor_c644f851e5b2ade20ee6f37c9eeaf36b.svg) | 5-Benzyl-5-(4-bromophenyl)-5H-imidazo[2,1-a]isoindole | IC50 | 163.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuropeptide-s-receptor_adf03326ab77143148ffb332ae848fda.svg) | 2-[[5-(4-Bromophenyl)imidazo[1,2-b]isoindol-5-yl]methyl]benzonitrile | IC50 | 369.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuropeptide-s-receptor_adb46cb3199e30ff484a29de4170c9c1.svg) | 5-(4-Bromophenyl)-5-(pyridin-3-ylmethyl)imidazo[2,1-a]isoindole | IC50 | 351.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuropeptide-s-receptor_e0a81fb61a6e6df51c9bd701718877eb.svg) | 5-Benzyl-5-(4-methylphenyl)imidazo[2,1-a]isoindole | IC50 | 1325.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuropeptide-s-receptor_aced220a8987410a03df64399e168c9c.svg) | N-[(1-Methyl-2-oxoquinolin-3-yl)methyl]-N-[[1-(4-methylpiperazin-1-yl)cyclohexyl]methyl]cyclohexanecarboxamide | IC50 | 18.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuropeptide-s-receptor_69aea382ca772094913e07dae69e2461.svg) | N-[(1-Methyl-2-oxoquinolin-3-yl)methyl]-N-(4-pyrrolidin-1-ylbutan-2-yl)cyclohexanecarboxamide | IC50 | 1577.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuropeptide-s-receptor_40cb2e4ceeb43d87ae06ca0a91dbfd8a.svg) | N-[(1-Methyl-2-oxoquinolin-3-yl)methyl]-N-(4-morpholin-4-ylbutan-2-yl)cyclohexanecarboxamide | IC50 | 725.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuropeptide-s-receptor_718320494ad41d78c9cdff5be588414c.svg) | N-[(1-Methyl-2-oxoquinolin-3-yl)methyl]-N-(2-methyl-4-pyrrolidin-1-ylbutan-2-yl)cyclohexanecarboxamide | IC50 | 326.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuropeptide-s-receptor_718f0f8924e8734ec7c5a50d79d5f1d8.svg) | N-[(1-Methyl-2-oxoquinolin-3-yl)methyl]-N-(2-methyl-4-piperidin-1-ylbutan-2-yl)cyclohexanecarboxamide | IC50 | 31.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuropeptide-s-receptor_4642ff2f55d708d0f2878c7b11d4bd41.svg) | N-(2-Methyl-4-morpholin-4-ylbutan-2-yl)-N-[(1-methyl-2-oxoquinolin-3-yl)methyl]cyclohexanecarboxamide | IC50 | 144.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuropeptide-s-receptor_d0073197ebe0f80c4e4a91c72e122e7b.svg) | N-[(1-Methyl-2-oxoquinolin-3-yl)methyl]-N-(3-methyl-1-piperidin-1-ylpentan-3-yl)cyclohexanecarboxamide | IC50 | 7.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuropeptide-s-receptor_34e0eaea28c1ad965fee0f45965c9eab.svg) | N-[1-(4-Fluoropiperidin-1-yl)-3-methylpentan-3-yl]-N-[(1-methyl-2-oxoquinolin-3-yl)methyl]cyclohexanecarboxamide | IC50 | 14.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuropeptide-s-receptor_2f6322fcab9c5d7bdccaa507a797a525.svg) | N-[1-(4,4-Difluoropiperidin-1-yl)-3-methylpentan-3-yl]-N-[(1-methyl-2-oxoquinolin-3-yl)methyl]cyclohexanecarboxamide | IC50 | 22.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuropeptide-s-receptor_38faf9d793b52a28696b2c453f272604.svg) | N-(3-Ethyl-1-morpholin-4-ylpentan-3-yl)-N-[(1-methyl-2-oxoquinolin-3-yl)methyl]cyclohexanecarboxamide | IC50 | 103.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuropeptide-s-receptor_a7c2169d874ce40b271920ca00a2c526.svg) | N-[(1-Methyl-2-oxoquinolin-3-yl)methyl]-N-[1-(2-morpholin-4-ylethyl)cyclohexyl]cyclohexanecarboxamide | IC50 | 398.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuropeptide-s-receptor_5b7bd4b3f6cf0aed350cf0436805d525.svg) | 6-Phenyl-N-[2-(piperidine-1-carbonyl)phenyl]pyridine-2-carboxamide | IC50 | 19.95 [1] |
![](https://images.aatbio.com/dataset/ic50/neuropeptide-s-receptor_14e187306393c649edffc4f886577924.svg) | 6-Phenyl-2-[2-(piperidine-1-carbonyl)phenyl]-3,4-dihydropyrrolo[1,2-a]pyrazin-1-one | IC50 | 5011.87 [1] |
![](https://images.aatbio.com/dataset/ic50/neuropeptide-s-receptor_ec068b38659175ad4d7c03bf9f2fd41a.svg) | 5-Phenyl-N-[2-(piperidine-1-carbonyl)phenyl]furan-2-carboxamide | IC50 | 31.62 [1] |
![](https://images.aatbio.com/dataset/ic50/neuropeptide-s-receptor_4931b3270d0bce49fa3c9cd0d88b5c99.svg) | 3-Phenyl-N-[2-(piperidine-1-carbonyl)phenyl]benzamide | IC50 | 251.19 [1] |
![](https://images.aatbio.com/dataset/ic50/neuropeptide-s-receptor_4772f72a244c3e95dc98794ebda0da95.svg) | 5-Phenyl-N-[2-(piperidine-1-carbonyl)phenyl]-1H-pyrrole-2-carboxamide | IC50 | 5011.87 [1] |
![](https://images.aatbio.com/dataset/ic50/neuropeptide-s-receptor_fbe6b9af650b8e2d8a7bf2644bf69c8b.svg) | 7-Phenyl-2-[2-(piperidine-1-carbonyl)phenyl]-4,5-dihydro-3H-pyrrolo[1,2-a][1,4]diazepin-1-one | IC50 | 5011.87 [1] |
![](https://images.aatbio.com/dataset/ic50/neuropeptide-s-receptor_b76e7c4dfca57a30bfc02e1d1d746f13.svg) | 5-(4-Bromophenyl)-5-[2-(oxan-4-yl)ethyl]imidazo[2,1-a]isoindole | IC50 | 154.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuropeptide-s-receptor_6326cde98baca569db8edad6726f810f.svg) | 5-Benzyl-5-(4-chlorophenyl)imidazo[2,1-a]isoindole | IC50 | 358.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuropeptide-s-receptor_1fc9e105cbb01153ed0b3ab7fcafb596.svg) | 5-(4-Chlorophenyl)-5-(oxan-4-ylmethyl)imidazo[2,1-a]isoindole | IC50 | 134.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuropeptide-s-receptor_56c2533180936998ea8e8bfb577bc1ad.svg) | 3-[5-(4-Chlorophenyl)imidazo[1,2-b]isoindol-5-yl]-N,N-di(propan-2-yl)propanamide | IC50 | 96.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuropeptide-s-receptor_6de2294ca0b50617aaa7dabb817f7bd0.svg) | 3-[5-(4-Chlorophenyl)-7-methoxyimidazo[1,2-b]isoindol-5-yl]-1-[(2R,5S)-2,5-dimethylpyrrolidin-1-yl]propan-1-one | IC50 | 50.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuropeptide-s-receptor_f1e97f7e1740febe0e4ad97e50cb05ce.svg) | 3-[5-(4-Chlorophenyl)imidazo[1,2-b]isoindol-5-yl]-1-[(2R,5S)-2,5-dimethylpyrrolidin-1-yl]propan-1-one | IC50 | 92.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuropeptide-s-receptor_a4c646827fe81c3e87f9e36ca2470d92.svg) | 3-[5-(4-Chlorophenyl)imidazo[1,2-b]isoindol-5-yl]-N,N-diethylpropanamide | IC50 | 90.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuropeptide-s-receptor_7a5235b1295707db3fcc0b89db7e4b7c.svg) | 3-(5-Benzylimidazo[1,2-b]isoindol-5-yl)benzonitrile | IC50 | 3166.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuropeptide-s-receptor_54500ec502f3256032217de5c8e27964.svg) | 3-[5-(4-Chlorophenyl)imidazo[1,2-b]isoindol-5-yl]-1-[4-[1-(3,3-difluoropyrrolidin-1-yl)ethyl]piperidin-1-yl]propan-1-one | IC50 | 239.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuropeptide-s-receptor_fc34cbda2310c6fa2f7afe256fdffe0e.svg) | 7-Benzyl-7-(4-bromophenyl)-3,6,12-triazatricyclo[6.4.0.02,6]dodeca-1(8),2,4,9,11-pentaene | IC50 | 1458.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuropeptide-s-receptor_8afa42240885d6922a30058dcf1068d7.svg) | 5-Benzyl-5-(6-bromopyridin-3-yl)imidazo[2,1-a]isoindole | IC50 | 1500.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuropeptide-s-receptor_a6cc9a985423f126adb9710a63fa3478.svg) | 5-(4-Bromophenyl)-5-(oxan-4-ylmethyl)imidazo[2,1-a]isoindole | IC50 | 92.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuropeptide-s-receptor_2c871808b60bba7d68a4fabdeb265b04.svg) | 5-Benzyl-5-(4-fluorophenyl)imidazo[2,1-a]isoindole | IC50 | 336.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuropeptide-s-receptor_8bd256f4596b847da955b44b021e7437.svg) | 4-[5-(Oxan-4-ylmethyl)imidazo[1,2-b]isoindol-5-yl]benzonitrile | IC50 | 635.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuropeptide-s-receptor_5a5bc4a6300c50998fc25a5d34f7fa04.svg) | 3-[5-(4-Chlorophenyl)imidazo[1,2-b]isoindol-5-yl]-1-(2-ethylpiperidin-1-yl)propan-1-one | IC50 | 131.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuropeptide-s-receptor_140a0a63edddbe70e81177515a7064d1.svg) | 3-[5-(4-Chlorophenyl)imidazo[1,2-b]isoindol-5-yl]-1-[4-(1-pyrrolidin-1-ylethyl)piperidin-1-yl]propan-1-one | IC50 | 126.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuropeptide-s-receptor_a061f3205cd8cd97e71ca0784e76230e.svg) | 5-(4-Fluorophenyl)-5-(oxan-4-ylmethyl)imidazo[2,1-a]isoindole | IC50 | 660.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuropeptide-s-receptor_9588bf9c63fd30af99698d95c1b87247.svg) | 5-Benzyl-5-(3-bromophenyl)imidazo[2,1-a]isoindole | IC50 | 1725.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuropeptide-s-receptor_b2aec4a1bdadade9b45a6b3643f7fba7.svg) | 3-[5-(4-Chlorophenyl)imidazo[1,2-b]isoindol-5-yl]-N-ethyl-N-propan-2-ylpropanamide | IC50 | 138.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuropeptide-s-receptor_6d0a4e03b99175dc90f96c9f5275cd21.svg) | 1-(8-Azabicyclo[3.2.1]octan-8-yl)-3-[5-(4-chlorophenyl)imidazo[1,2-b]isoindol-5-yl]propan-1-one | IC50 | 95.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuropeptide-s-receptor_30d3b8744293d81744eaeb769d8ef992.svg) | 2-(4-Benzylpiperazino)-2-phenyl-1H-indene-1,3(2H)-dione | IC50 | 27.0 [1] |