Neuronal acetylcholine receptor subunit alpha-3 Inhibitors (IC50, Ki)

Structure ▲ ▼	Compound Name ▲ ▼	Standard Type ▲ ▼	Standard Values (in nM) ▲ ▼
	Nicotine	IC50	45.0 [1]
	Nicotine	Ki	220.0 [1]
	Imidacloprid	IC50	14000.0 [1]
	Tropisetron	Ki	16000.0 [1]
	Granisetron	Ki	67000.0 [1]
	4-Bromophenyl 1,4-diazabicyclo(3.2.2)nonane-4-carboxylate	IC50	6480.0 [1]
	(2z)-1-[(6-Chloropyridin-3-Yl)methyl]imidazolidin-2-Imine	IC50	14.0 [1]
	3-(1H-Indole-3-carbonyloxy)-8,8-dimethyl-8-azonia-bicyclo[3.2.1]octane	Ki	2300.0 [1]
	3-Bromocytisine	IC50	15.6 [1]
	1H-1,4-Diazepine-1-pentanamide, 4-acetylhexahydro-N-(5-(4-methoxyphenyl)-1H-pyrazol-3-yl)-	IC50	30000.0 [1]
	(1-Propan-2-ylpiperidin-3-yl)methyl 2-(3-methyl-2,5-dioxopyrrolidin-1-yl)benzoate	IC50	20000.0 [1]
	(1-Propan-2-ylpiperidin-3-yl)methyl 2-(2,5-dioxopyrrolidin-1-yl)benzoate	IC50	20000.0 [1]
	4-Bromo-3-chlorophenyl 1,4-diazabicyclo[3.2.2]nonane-4-carboxylate	IC50	2090.0 [1]
	(2Z)-1-[(6-Chloropyridin-3-yl)methyl]-2-(nitromethylidene)-1,3-diazinane	IC50	180.0 [1]
	N-[5-(4-Fluorophenyl)-1H-pyrazol-3-yl]-5-piperidin-1-ylpentanamide	IC50	3900.0 [1]
	N-[5-(4-Methoxyphenyl)-1H-pyrazol-3-yl]-5-morpholin-4-ylpentanamide	IC50	11610.0 [1]
	N-[5-(4-Methoxyphenyl)-1H-pyrazol-3-yl]-4-piperidin-1-ylbutanamide	IC50	31622.78 [1]
	4-Chlorophenyl 1,4-diazabicyclo[3.2.2]nonane-4-carboxylate	IC50	5000.0 [1]
	3-Benzoyl-4-bromophenyl 1,4-diazabicyclo[3.2.2]nonane-4-carboxylate	IC50	1390.0 [1]
	3,4-Dichlorophenyl 1,4-diazabicyclo[3.2.2]nonane-4-carboxylate	IC50	4750.0 [1]
	4-Chloro-3-fluorophenyl 1,4-diazabicyclo[3.2.2]nonane-4-carboxylate	IC50	9960.0 [1]
	2-[3-Cyclohexyl-5-(furan-2-ylmethyl)-6-oxopyridazin-1-yl]-N-(2,3-dihydro-1H-inden-2-yl)acetamide	IC50	1000.0 [1]
	N-[5-(4-Methoxyphenyl)-1H-pyrazol-3-yl]-5-piperidin-1-ylpentanamide	IC50	3250.0 [1]
	N-[5-(2-Methoxyphenyl)-1H-pyrazol-3-yl]-5-piperidin-1-ylpentanamide	IC50	6400.0 [1]
	N-[5-(4-Bromophenyl)-1H-pyrazol-3-yl]-5-piperidin-1-ylpentanamide	IC50	5800.0 [1]
	5-(Azepan-1-yl)-N-[5-(4-methoxyphenyl)-1H-pyrazol-3-yl]pentanamide	IC50	30000.0 [1]
	N-[5-(4-Methoxyphenyl)-1H-pyrazol-3-yl]-5-(1,4-oxazepan-4-yl)pentanamide	IC50	30000.0 [1]
	5-(4-Acetyl-1,4-diazepan-1-yl)-N-[5-(4-methoxyphenyl)-1H-pyrazol-3-yl]-2-methylpentanamide	IC50	30000.0 [1]
	4-(Azepan-1-yl)-N-[5-(4-methoxyphenyl)-1H-pyrazol-3-yl]butanamide	IC50	7943.28 [1]
	N-(2,4-Dimethylphenyl)-5-morpholin-4-yl-4-phenylthiophene-2-carboxamide	IC50	2511.89 [1]
	Naphthalen-2-yl 1,4-diazabicyclo[3.2.2]nonane-4-carboxylate	IC50	4910.0 [1]
	4-Bromo-3-methylphenyl 1,4-diazabicyclo[3.2.2]nonane-4-carboxylate	IC50	4020.0 [1]

Entire TableStructureCompound NameStandard TypeStandard Values (in nM)

Items per page: 510All1 - 10 of 32 ⟨⟩

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References

This online tool may be cited as follows

MLA	"Quest Database™ Neuronal acetylcholine receptor subunit alpha-3 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 21 Dec. 2024, https://www.aatbio.com/data-sets/neuronal-acetylcholine-receptor-subunit-alpha-3-inhibitors-ic50-ki.
APA	AAT Bioquest, Inc. (2024, December 21). Quest Database™ Neuronal acetylcholine receptor subunit alpha-3 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/neuronal-acetylcholine-receptor-subunit-alpha-3-inhibitors-ic50-ki.
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