![](https://images.aatbio.com/dataset/ic50/neuronal-acetylcholine-receptor-alpha3-beta4_86630ba4a7e4889b44175ac812cce53f.svg) | Nicotine | IC50 | 430.0 [1], 1000.0 [2], 10000.0 [3] |
![](https://images.aatbio.com/dataset/ic50/neuronal-acetylcholine-receptor-alpha3-beta4_86630ba4a7e4889b44175ac812cce53f.svg) | Nicotine | Ki | 530.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuronal-acetylcholine-receptor-alpha3-beta4_6da87654a41806f746deff10f04e816a.svg) | Cytisine | Ki | 840.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuronal-acetylcholine-receptor-alpha3-beta4_fcd3cfefde2b46eddadc801088ffc22a.svg) | Bupropion | IC50 | 1.8 [1], 1800.0 [2] |
![](https://images.aatbio.com/dataset/ic50/neuronal-acetylcholine-receptor-alpha3-beta4_f4b1d136c22b35f47b0361ed8a5f8191.svg) | Varenicline | IC50 | 110.0 [1], 1000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/neuronal-acetylcholine-receptor-alpha3-beta4_f4b1d136c22b35f47b0361ed8a5f8191.svg) | Varenicline | Ki | 74.7 [1], 86.0 [2] |
![](https://images.aatbio.com/dataset/ic50/neuronal-acetylcholine-receptor-alpha3-beta4_361ebe418f7f23487e23bc76f4bafd5f.svg) | Epibatidine | Ki | 0.15 [1], 0.19 [2], 0.22 [3], 0.46 [4] |
![](https://images.aatbio.com/dataset/ic50/neuronal-acetylcholine-receptor-alpha3-beta4_b9a73af7b9c5977535db0228e5a4eeb8.svg) | Mecamylamine | IC50 | 100.0 [1], 700.0 [2], 3400.0 [3] |
![](https://images.aatbio.com/dataset/ic50/neuronal-acetylcholine-receptor-alpha3-beta4_7f915764cafd78247516902505c7dc39.svg) | Piperidine, 1-(3,3-diphenylallyl)- | IC50 | 100.0 [1], 380.0 [2] |
![](https://images.aatbio.com/dataset/ic50/neuronal-acetylcholine-receptor-alpha3-beta4_7f915764cafd78247516902505c7dc39.svg) | Piperidine, 1-(3,3-diphenylallyl)- | Ki | 2200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuronal-acetylcholine-receptor-alpha3-beta4_47ab557b41e1ae998f426aac2b25ea20.svg) | 3-Benzhydrylquinuclidine | IC50 | 200.0 [1], 400.0 [2] |
![](https://images.aatbio.com/dataset/ic50/neuronal-acetylcholine-receptor-alpha3-beta4_47ab557b41e1ae998f426aac2b25ea20.svg) | 3-Benzhydrylquinuclidine | Ki | 1500.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuronal-acetylcholine-receptor-alpha3-beta4_361eef2caae464203911c6769911ba30.svg) | 3-Benzhydryl-1-benzyl-1-azoniabicyclo[2.2.2]octane | IC50 | 80.0 [1], 600.0 [2] |
![](https://images.aatbio.com/dataset/ic50/neuronal-acetylcholine-receptor-alpha3-beta4_361eef2caae464203911c6769911ba30.svg) | 3-Benzhydryl-1-benzyl-1-azoniabicyclo[2.2.2]octane | Ki | 2300.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuronal-acetylcholine-receptor-alpha3-beta4_f36665d48cf053dc7e38624549f06881.svg) | Tubocurarine chloride | IC50 | 2000.0 [1], 6800.0 [2] |
![](https://images.aatbio.com/dataset/ic50/neuronal-acetylcholine-receptor-alpha3-beta4_9bf567bfce4fef60f82160d0177552b0.svg) | 7,8,9,10-Tetrahydro-6,10-methano-6H-pyrazino(2,3-h)(3)benzazepine | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuronal-acetylcholine-receptor-alpha3-beta4_9bf567bfce4fef60f82160d0177552b0.svg) | 7,8,9,10-Tetrahydro-6,10-methano-6H-pyrazino(2,3-h)(3)benzazepine | Ki | 390.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuronal-acetylcholine-receptor-alpha3-beta4_b76189cabac5b949a1d3108e5ba7e808.svg) | Methyllycaconitine | IC50 | 1000.0 [1], 2600.0 [2] |
![](https://images.aatbio.com/dataset/ic50/neuronal-acetylcholine-receptor-alpha3-beta4_d7e372c4785415c85ac635995434e70b.svg) | 3-(2,4-Dimethoxybenzylidene)anabaseine | Ki | 2500.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuronal-acetylcholine-receptor-alpha3-beta4_06509802a287af8b4d6763b60cea549b.svg) | Benzamide, N-(3R)-1-azabicyclo[2.2.2]oct-3-yl-4-chloro- | IC50 | 60000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuronal-acetylcholine-receptor-alpha3-beta4_06509802a287af8b4d6763b60cea549b.svg) | Benzamide, N-(3R)-1-azabicyclo[2.2.2]oct-3-yl-4-chloro- | Ki | 60000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuronal-acetylcholine-receptor-alpha3-beta4_0f419d3719cf510be57b9e88deebdfd6.svg) | Sazetidine A | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuronal-acetylcholine-receptor-alpha3-beta4_0f419d3719cf510be57b9e88deebdfd6.svg) | Sazetidine A | Ki | 1900.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuronal-acetylcholine-receptor-alpha3-beta4_bcda24337f1f48f0e0f78a4fd27d888e.svg) | Radafaxine | IC50 | 3300.0 [1], 6500.0 [2] |
![](https://images.aatbio.com/dataset/ic50/neuronal-acetylcholine-receptor-alpha3-beta4_30c7310bb56e2677fe86efcbecf67a42.svg) | N-[(3R)-1-Azabicyclo[2.2.2]oct-3-yl]furo[2,3-c]pyridine-5-carboxamide | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuronal-acetylcholine-receptor-alpha3-beta4_644e2474d7ce27e7aacd11d418a8007b.svg) | 4-[(E)-5,6-Dihydro-2,3'-bipyridin-3(4H)-ylidenemethyl]-3-methoxyphenol | Ki | 970.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuronal-acetylcholine-receptor-alpha3-beta4_3c57e2725863f26a6d26d4591478a16d.svg) | N-(2-Fluorophenyl)-2-{4-[(4-fluorophenyl)sulfonyl]piperazin-1-yl}acetamide | IC50 | 9000.0 [1], 19600.0 [2] |
![](https://images.aatbio.com/dataset/ic50/neuronal-acetylcholine-receptor-alpha3-beta4_0a857010cf06d49165eb935f62cf08b0.svg) | 3-(5-Chloro-2-furoyl)-3,7-diazabicyclo[3.3.0]octane | Ki | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuronal-acetylcholine-receptor-alpha3-beta4_4f7e38e485ec780340b7e299df5bf0b4.svg) | Biphenyl-2-carboxylic acid 1-(3-phenyl-propyl)-piperidin-3-ylmethyl ester | IC50 | 1700.0 [1], 100000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/neuronal-acetylcholine-receptor-alpha3-beta4_6e6e3d234f9b8e188a2bed53146c8f34.svg) | 3-Benzylidenequinuclidine | IC50 | 6000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuronal-acetylcholine-receptor-alpha3-beta4_6e6e3d234f9b8e188a2bed53146c8f34.svg) | 3-Benzylidenequinuclidine | Ki | 2100.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuronal-acetylcholine-receptor-alpha3-beta4_69aaca6fe3f6c1e2f13a552e8b74d084.svg) | 3-[(Z)-(3-Pyridyl)methylene]-1-azabicyclo[2.2.2]octane | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuronal-acetylcholine-receptor-alpha3-beta4_69aaca6fe3f6c1e2f13a552e8b74d084.svg) | 3-[(Z)-(3-Pyridyl)methylene]-1-azabicyclo[2.2.2]octane | Ki | 1600.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuronal-acetylcholine-receptor-alpha3-beta4_818c8ddab8f39a886ae500e8225ccf59.svg) | 4-Methoxy-3-[[(2S)-1-methylpyrrolidin-2-yl]methoxy]phenol | Ki | 271.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuronal-acetylcholine-receptor-alpha3-beta4_7e68c0c789ba69b88258d607e599a65a.svg) | 3-[(1R)-1-[(2S)-1-Methylpyrrolidin-2-yl]ethoxy]phenol | Ki | 257.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuronal-acetylcholine-receptor-alpha3-beta4_c378772c0bb0db71ed12902503a5765f.svg) | Cyclopropyl(3,7-diazabicyclo[3.3.1]nonan-3-yl)methanone | Ki | 110.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuronal-acetylcholine-receptor-alpha3-beta4_f1e8c0ee2b67027176c81ab71af7983e.svg) | 2,3,3a,4,6,6a-Hexahydro-1H-pyrrolo[3,4-c]pyrrol-5-yl(cyclopropyl)methanone | Ki | 670.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuronal-acetylcholine-receptor-alpha3-beta4_43e9450cce1ed688ad05416a59f826b9.svg) | 2-Acetylamino-benzoic acid 1-(3-phenyl-propyl)-piperidin-3-ylmethyl ester | IC50 | 4265.8 [1], 8400.0 [2] |
![](https://images.aatbio.com/dataset/ic50/neuronal-acetylcholine-receptor-alpha3-beta4_fc11c7695bf81d7ed99681b4cafc1937.svg) | 2-Trifluoromethyl-benzoic acid 1-(3-phenyl-propyl)-piperidin-3-ylmethyl ester | IC50 | 3200.0 [1], 5500.0 [2] |
![](https://images.aatbio.com/dataset/ic50/neuronal-acetylcholine-receptor-alpha3-beta4_6b105b0949bcde4362013b49afa6e238.svg) | [1-(3-Phenylpropyl)piperidin-3-yl]methyl 2-(1,3-dioxoisoindol-2-yl)benzoate | IC50 | 1300.0 [1], 5888.44 [2] |
![](https://images.aatbio.com/dataset/ic50/neuronal-acetylcholine-receptor-alpha3-beta4_095cf78d5a918ed66e897d138f69e858.svg) | Biphenyl-4-carboxylic acid 1-(3-phenyl-propyl)-piperidin-3-ylmethyl ester | IC50 | 3000.0 [1], 18620.87 [2] |
![](https://images.aatbio.com/dataset/ic50/neuronal-acetylcholine-receptor-alpha3-beta4_7f2b5fcca88dfef10b20d6019ea8b36d.svg) | [1-(3-Phenylpropyl)piperidin-3-yl]methyl 2-(3,3-dimethyl-2,5-dioxopyrrolidin-1-yl)benzoate | IC50 | 5011.87 [1], 7500.0 [2] |
![](https://images.aatbio.com/dataset/ic50/neuronal-acetylcholine-receptor-alpha3-beta4_eae66a152833e1b4aca81271d47ede30.svg) | 2-Methoxy-benzoic acid 1-(3-phenyl-propyl)-piperidin-3-ylmethyl ester | IC50 | 3200.0 [1], 12022.64 [2] |
![](https://images.aatbio.com/dataset/ic50/neuronal-acetylcholine-receptor-alpha3-beta4_23cce5b70e28b7618cc21d1b71941e66.svg) | 2-Chloro-benzoic acid 1-(3-phenyl-propyl)-piperidin-3-ylmethyl ester | IC50 | 3400.0 [1], 22908.68 [2] |
![](https://images.aatbio.com/dataset/ic50/neuronal-acetylcholine-receptor-alpha3-beta4_33019aa9e472c1f0bc17685ebde1b1ad.svg) | (2S,3S)-2-(3-Fluorophenyl)-3,5,5-trimethylmorpholin-2-ol | IC50 | 5600.0 [1], 15000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/neuronal-acetylcholine-receptor-alpha3-beta4_6dd539c533459c86589f0bbeec6cfa06.svg) | (2S,3S)-2-(3-Bromophenyl)-3,5,5-trimethylmorpholin-2-ol | IC50 | 1400.0 [1], 3200.0 [2] |
![](https://images.aatbio.com/dataset/ic50/neuronal-acetylcholine-receptor-alpha3-beta4_f11f6184d360532feea2f8f0457b1f36.svg) | (2S,3S)-2-(3-Chlorophenyl)-3-ethyl-5,5-dimethylmorpholin-2-ol | IC50 | 4300.0 [1], 5600.0 [2] |
![](https://images.aatbio.com/dataset/ic50/neuronal-acetylcholine-receptor-alpha3-beta4_23a9fa7714ff1998e5d0500d5cfb3008.svg) | (2S,3S)-2-(3-Chlorophenyl)-5,5-dimethyl-3-propyl-morpholin-2-ol | IC50 | 3100.0 [1], 4800.0 [2] |
![](https://images.aatbio.com/dataset/ic50/neuronal-acetylcholine-receptor-alpha3-beta4_c136e181d6441da4465a5f56ff5542e3.svg) | (2S,3S)-2-(3-Chlorophenyl)-3,4,5,5-tetramethylmorpholin-2-ol | IC50 | 2800.0 [1], 6500.0 [2] |
![](https://images.aatbio.com/dataset/ic50/neuronal-acetylcholine-receptor-alpha3-beta4_b39c46aff515ad57b8d666b0021597b0.svg) | 1-Benzhydryl-4-aza-1-azoniabicyclo[2.2.2]octane | IC50 | 15000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuronal-acetylcholine-receptor-alpha3-beta4_b39c46aff515ad57b8d666b0021597b0.svg) | 1-Benzhydryl-4-aza-1-azoniabicyclo[2.2.2]octane | Ki | 8500.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuronal-acetylcholine-receptor-alpha3-beta4_079260af629afc451893d6f294a5fc46.svg) | (R,R)-Hydroxy Bupropion | IC50 | 1600.0 [1], 11000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/neuronal-acetylcholine-receptor-alpha3-beta4_6d877394c384ad94d74ad8aaf1979296.svg) | (R)-2-((2S)-1-Methyl-2-pyrrolidinyl)-1,4-benzodioxane | IC50 | 2780.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuronal-acetylcholine-receptor-alpha3-beta4_6d877394c384ad94d74ad8aaf1979296.svg) | (R)-2-((2S)-1-Methyl-2-pyrrolidinyl)-1,4-benzodioxane | Ki | 1200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuronal-acetylcholine-receptor-alpha3-beta4_b71ce768bf8820406b32aa670d522ec0.svg) | 3-[[(2S)-Azetidin-2-yl]methoxy]-5-hex-1-ynyl-2-methylpyridine | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuronal-acetylcholine-receptor-alpha3-beta4_b71ce768bf8820406b32aa670d522ec0.svg) | 3-[[(2S)-Azetidin-2-yl]methoxy]-5-hex-1-ynyl-2-methylpyridine | Ki | 230000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuronal-acetylcholine-receptor-alpha3-beta4_5b0e905c59f86ce8bb86f67e7c0a924d.svg) | 3-[[(2S)-Azetidin-2-yl]methoxy]-5-(6-fluorohex-1-ynyl)-2-methylpyridine | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuronal-acetylcholine-receptor-alpha3-beta4_5b0e905c59f86ce8bb86f67e7c0a924d.svg) | 3-[[(2S)-Azetidin-2-yl]methoxy]-5-(6-fluorohex-1-ynyl)-2-methylpyridine | Ki | 130000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuronal-acetylcholine-receptor-alpha3-beta4_1cb46d8ec1fd3e361ebd39de1eb91d97.svg) | 6-[5-[[(2S)-Azetidin-2-yl]methoxy]-6-methylpyridin-3-yl]hex-5-yn-1-ol | IC50 | 50000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuronal-acetylcholine-receptor-alpha3-beta4_1cb46d8ec1fd3e361ebd39de1eb91d97.svg) | 6-[5-[[(2S)-Azetidin-2-yl]methoxy]-6-methylpyridin-3-yl]hex-5-yn-1-ol | Ki | 250000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuronal-acetylcholine-receptor-alpha3-beta4_81138852c1ddf35c386e671d5d8b533b.svg) | 3-[[(2S)-Azetidin-2-yl]methoxy]-5-(6-chlorohex-1-ynyl)-2-methylpyridine | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuronal-acetylcholine-receptor-alpha3-beta4_81138852c1ddf35c386e671d5d8b533b.svg) | 3-[[(2S)-Azetidin-2-yl]methoxy]-5-(6-chlorohex-1-ynyl)-2-methylpyridine | Ki | 86000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuronal-acetylcholine-receptor-alpha3-beta4_891886f6dbb36cd12981ddbd4e3d45d4.svg) | 3-[[(2S)-Azetidin-2-yl]methoxy]-5-(2-cyclopropylethynyl)-2-methylpyridine | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuronal-acetylcholine-receptor-alpha3-beta4_891886f6dbb36cd12981ddbd4e3d45d4.svg) | 3-[[(2S)-Azetidin-2-yl]methoxy]-5-(2-cyclopropylethynyl)-2-methylpyridine | Ki | 150000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuronal-acetylcholine-receptor-alpha3-beta4_4790c2ed4aa68637e502beb23ab8d1bb.svg) | 5-Hex-1-ynyl-2-methyl-3-[[(2S)-pyrrolidin-2-yl]methoxy]pyridine | IC50 | 6400.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuronal-acetylcholine-receptor-alpha3-beta4_4790c2ed4aa68637e502beb23ab8d1bb.svg) | 5-Hex-1-ynyl-2-methyl-3-[[(2S)-pyrrolidin-2-yl]methoxy]pyridine | Ki | 94000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuronal-acetylcholine-receptor-alpha3-beta4_d2d9758783ff42eaccc6bbafe9095969.svg) | 2-(1-Azabicyclo[2.2.2]octan-3-yl)-2-phenylacetonitrile | IC50 | 23000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuronal-acetylcholine-receptor-alpha3-beta4_d2d9758783ff42eaccc6bbafe9095969.svg) | 2-(1-Azabicyclo[2.2.2]octan-3-yl)-2-phenylacetonitrile | Ki | 2100.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuronal-acetylcholine-receptor-alpha3-beta4_04cbfb18d4637aa7607c73b2f21de570.svg) | Ondansetron | IC50 | 27000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuronal-acetylcholine-receptor-alpha3-beta4_fe503d49f756ee0177fb46d02c8c9aca.svg) | Tropisetron | IC50 | 1800.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuronal-acetylcholine-receptor-alpha3-beta4_14035e126a8a9aaf49d9a09d42373790.svg) | Decamethonium | IC50 | 1700.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuronal-acetylcholine-receptor-alpha3-beta4_0cb317d7cb5776f7efc05f9c6766c452.svg) | Benzamide, N-(3R)-1-azabicyclo(2.2.2)oct-3-yl-4-chloro-, monohydrochloride | IC50 | 60000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuronal-acetylcholine-receptor-alpha3-beta4_f4447b2edb88e5ef4694b6b26776dda0.svg) | Polygodial | IC50 | 48200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuronal-acetylcholine-receptor-alpha3-beta4_889c75941cc4ae0a55b6d028f9169fbd.svg) | alpha-Methyltryptamine | Ki | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuronal-acetylcholine-receptor-alpha3-beta4_45d6e90fcd2b7827bf0fea3f667ce1eb.svg) | Rivanicline | Ki | 5400.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuronal-acetylcholine-receptor-alpha3-beta4_cdf24b636f44308fd836ed426670b1be.svg) | 18-Methoxycoronaridine | Ki | 700.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuronal-acetylcholine-receptor-alpha3-beta4_c77de99dec26af64c24ff26105ceddc1.svg) | (5S)-Spiro[1,3-oxazolidine-5,3'-1-azabicyclo[2.2.2]octane]-2-one | IC50 | 1000000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuronal-acetylcholine-receptor-alpha3-beta4_5b9eab44496be35c12fe90f7d96dd5f4.svg) | Anabaseine | Ki | 107.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuronal-acetylcholine-receptor-alpha3-beta4_c0c6df8450ab00c131d728b537100462.svg) | CID 9823180 | Ki | 7000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuronal-acetylcholine-receptor-alpha3-beta4_7e67dc53b9dda9b460fb3afbfa5076d7.svg) | N,N-Diallyl-5-methoxytryptamine | Ki | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuronal-acetylcholine-receptor-alpha3-beta4_ba6c26e69a828c39b9229453f4f9adf1.svg) | 4-(6-Fluoro-5,5-dioxido-3-dibenzothienyl)-1,4-diazabicyclo(3.2.2)nonane | Ki | 709.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuronal-acetylcholine-receptor-alpha3-beta4_9ab3a675d11cd378b16a92a061958fbc.svg) | 3-Bromocytisine | IC50 | 15.6 [1] |
![](https://images.aatbio.com/dataset/ic50/neuronal-acetylcholine-receptor-alpha3-beta4_337d343ac05001d0b2b0851f83a6cf09.svg) | (S)-1-(2-Fluorophenyl)ethyl (S)-quinuclidin-3-ylcarbamate | IC50 | 19952.62 [1] |
![](https://images.aatbio.com/dataset/ic50/neuronal-acetylcholine-receptor-alpha3-beta4_8b4d77cb27f5f9273b6a6a6db557abed.svg) | (1R,2R,4S)-N,2,3,3-Tetramethylbicyclo[2.2.1]heptan-2-amine | IC50 | 50.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuronal-acetylcholine-receptor-alpha3-beta4_645744e0fd17c4d697ef803008888a33.svg) | Cinnamolide | IC50 | 2620.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuronal-acetylcholine-receptor-alpha3-beta4_4ebae5232d796166b252ddecd40b430a.svg) | Phantasmidine | Ki | 390.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuronal-acetylcholine-receptor-alpha3-beta4_daee457496b948ec4286caf125b46a10.svg) | 2-(4-Morpholinyl)-5-[(2-thienylmethyl)amino]benzoic acid | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuronal-acetylcholine-receptor-alpha3-beta4_fa8450992c39aee44232c2a8b15adb57.svg) | Rac-7-(3-pyridinyl)-1,7-diazaspiro[4.4]nonane | Ki | 1200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuronal-acetylcholine-receptor-alpha3-beta4_d85b744fe1b6d5c99d5f50b8e973a612.svg) | Dendocarbin A | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuronal-acetylcholine-receptor-alpha3-beta4_452bd3b499a61f2b4f896c42746f77e3.svg) | 1,4-Diazabicyclo(3.2.2)nonane, 4-(5-methyloxazolo(4,5-b)pyridin-2-yl)- | Ki | 5370.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuronal-acetylcholine-receptor-alpha3-beta4_2bc42c23863bb21d5ccbc032ecdaa52a.svg) | A-582941 Free base | Ki | 4700.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuronal-acetylcholine-receptor-alpha3-beta4_85db2f1a1be1ddf59cfa27190d1682ba.svg) | 1,5-Methano-1H-3-benzazepine, 2,3,4,5-tetrahydro- | Ki | 2850.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuronal-acetylcholine-receptor-alpha3-beta4_438220d42319e0ffca8be5b2625d1f41.svg) | 3-(3-Pyridinyl)-3,7-diazabicyclo[3.3.1]nonane | Ki | 6.6 [1] |
![](https://images.aatbio.com/dataset/ic50/neuronal-acetylcholine-receptor-alpha3-beta4_1c8e1bddcd306ac38f0b6838c2ee3467.svg) | CID 10107234 | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuronal-acetylcholine-receptor-alpha3-beta4_ffb7ec3db158effee1a626dcd8d2faf4.svg) | N-[(3R)-1-Azabicyclo[2.2.2]oct-3-yl]-1-benzofuran-6-carboxamide | IC50 | 81000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuronal-acetylcholine-receptor-alpha3-beta4_43082b20f49dd474be56b949cd75bff5.svg) | N-[(3R)-1-Azabicyclo[2.2.2]oct-3-yl]-1-benzothiophene-6-carboxamide | IC50 | 38000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuronal-acetylcholine-receptor-alpha3-beta4_566982896c31f240c40713e080e4492f.svg) | 2-(Tert-butyl(methyl)amino)-1-(3-chlorophenyl)propan-1-one | IC50 | 1.2 [1] |
![](https://images.aatbio.com/dataset/ic50/neuronal-acetylcholine-receptor-alpha3-beta4_66a0ea464877ef00ef0bdb152a04c888.svg) | 2-(Tert-butylamino)-1-(3-fluorophenyl)propan-1-one | IC50 | 4.4 [1] |
![](https://images.aatbio.com/dataset/ic50/neuronal-acetylcholine-receptor-alpha3-beta4_1696bb8d62226d33ebc46b9df3cf2749.svg) | 4-Allyloxy-N-pyridin-2-yl-benzamide | IC50 | 61400.0 [1] |
![](https://images.aatbio.com/dataset/ic50/neuronal-acetylcholine-receptor-alpha3-beta4_1e91f8e719e4711865dbd459b58b8a59.svg) | Laburnamine | Ki | 37000.0 [1] |