| (2S,3R)-N'-[(3S)-1-Methyl-2-oxo-5-phenyl-3H-1,4-benzodiazepin-3-yl]-3-(2-methylpropyl)-2-propylbutanediamide | IC50 | 64.1 [1] |
| (2S,3R)-N'-[(3S)-7-Chloro-1-methyl-2-oxo-5-phenyl-3H-1,4-benzodiazepin-3-yl]-3-(2-methylpropyl)-2-prop-2-enylbutanediamide | IC50 | 42.4 [1] |
| (2S,3R)-3-(2-Methylpropyl)-N'-[(3S)-2-oxo-5-phenyl-1-propyl-3H-1,4-benzodiazepin-3-yl]-2-prop-2-enylbutanediamide | IC50 | 12.3 [1] |
| (2S,3R)-2-Butyl-N'-[(3S)-5-(4-chlorophenyl)-1-methyl-2-oxo-3H-1,4-benzodiazepin-3-yl]-3-(2-methylpropyl)butanediamide | IC50 | 5.1 [1] |
| Cyclohexyl 2,7,7-trimethyl-4-(4-nitrophenyl)-5-oxo-1,4,5,6,7,8-hexahydroquinoline-3-carboxylate | IC50 | 2510.0 [1] |
| (2S,3R)-3-(2,2-Dimethylpropyl)-N'-[(3S)-1-methyl-2-oxo-5-phenyl-3H-1,4-benzodiazepin-3-yl]-2-pentan-3-ylbutanediamide | IC50 | 3.0 [1] |
| (2S,3R)-N'-[(3S)-1-Methyl-2-oxo-5-phenyl-3H-1,4-benzodiazepin-3-yl]-2-pentan-3-yl-3-(3,3,3-trifluoropropyl)butanediamide | IC50 | 1.0 [1] |
| (2S,3R)-N'-[(3S)-1-Methyl-2-oxo-5-phenyl-3H-1,4-benzodiazepin-3-yl]-2-propyl-3-(2,2,2-trifluoroethyl)butanediamide | IC50 | 13.0 [1] |
| (2R,3R)-2-(1,2,4-Oxadiazol-3-yl)-N'-[(3S)-2-oxo-5-phenyl-1,3-dihydro-1,4-benzodiazepin-3-yl]-3-(3,3,3-trifluoropropyl)butanediamide | IC50 | 1190.0 [1] |
| (2R,3R)-2-(1,3-Oxazol-4-yl)-N'-[(3S)-2-oxo-5-phenyl-1,3-dihydro-1,4-benzodiazepin-3-yl]-3-(3,3,3-trifluoropropyl)butanediamide | IC50 | 231.0 [1] |
| (2R,3R)-2-(1,2-Oxazol-4-yl)-N'-[(3S)-2-oxo-5-phenyl-1,3-dihydro-1,4-benzodiazepin-3-yl]-3-(3,3,3-trifluoropropyl)butanediamide | IC50 | 32.0 [1] |
| (2R,3R)-2-(5-Methyl-1,2,4-oxadiazol-3-yl)-N'-[(3S)-1-methyl-2-oxo-5-phenyl-3H-1,4-benzodiazepin-3-yl]-3-(3,3,3-trifluoropropyl)butanediamide | IC50 | 169.0 [1] |
| (2R,3R)-2-(5-Methyl-1,2-oxazol-3-yl)-N'-[(3S)-1-methyl-2-oxo-5-phenyl-3H-1,4-benzodiazepin-3-yl]-3-(3,3,3-trifluoropropyl)butanediamide | IC50 | 54.0 [1] |
| (2R,3R)-N'-[(3S)-1-Methyl-2-oxo-5-phenyl-3H-1,4-benzodiazepin-3-yl]-2-(3-methylphenyl)-3-(3,3,3-trifluoropropyl)butanediamide | IC50 | 3.0 [1] |
| (2R,3R)-N'-[(3S)-1-Methyl-2-oxo-5-phenyl-3H-1,4-benzodiazepin-3-yl]-2-[3-(trifluoromethyl)phenyl]-3-(3,3,3-trifluoropropyl)butanediamide | IC50 | 1.0 [1] |
| (2R,3R)-N'-[(3S)-1-Methyl-2-oxo-5-phenyl-3H-1,4-benzodiazepin-3-yl]-2-[3-(trifluoromethoxy)phenyl]-3-(3,3,3-trifluoropropyl)butanediamide | IC50 | 3.0 [1] |
| (2R,3R)-N'-[(3S)-1-Methyl-2-oxo-5-phenyl-3H-1,4-benzodiazepin-3-yl]-2-(3-methylsulfonylphenyl)-3-(3,3,3-trifluoropropyl)butanediamide | IC50 | 2060.0 [1] |
| (2R,3R)-2-(4-Methoxyphenyl)-N'-[(3S)-1-methyl-2-oxo-5-phenyl-3H-1,4-benzodiazepin-3-yl]-3-(3,3,3-trifluoropropyl)butanediamide | IC50 | 9.0 [1] |
| (2R,3R)-2-(3,4-Difluorophenyl)-N'-[(3S)-1-methyl-2-oxo-5-phenyl-3H-1,4-benzodiazepin-3-yl]-3-(3,3,3-trifluoropropyl)butanediamide | IC50 | 2.0 [1] |
| (2R,3R)-2-(2,4-Difluorophenyl)-N'-[(3S)-1-methyl-2-oxo-5-phenyl-3H-1,4-benzodiazepin-3-yl]-3-(3,3,3-trifluoropropyl)butanediamide | IC50 | 1.0 [1] |
| (2R,3R)-2-(3,5-Difluorophenyl)-N'-[(3S)-1-methyl-2-oxo-5-phenyl-3H-1,4-benzodiazepin-3-yl]-3-(3,3,3-trifluoropropyl)butanediamide | IC50 | 2.0 [1] |
| [1-[(2-Methylpropan-2-yl)oxycarbonyl]piperidin-4-yl]methyl 2,7,7-trimethyl-5-oxo-4-(3-propan-2-ylphenyl)-1,4,6,8-tetrahydroquinoline-3-carboxylate | IC50 | 3320.0 [1] |
| [1-[(2-Methylpropan-2-yl)oxycarbonyl]piperidin-4-yl]methyl 2,7,7-trimethyl-5-oxo-4-quinolin-2-yl-1,4,6,8-tetrahydroquinoline-3-carboxylate | IC50 | 330.0 [1] |
| [1-[(2-Methylpropan-2-yl)oxycarbonyl]piperidin-4-yl] 4-(3-bromophenyl)-2,7,7-trimethyl-5-oxo-1,4,6,8-tetrahydroquinoline-3-carboxylate | IC50 | 10000.0 [1] |
| [1-[(2-Methylpropan-2-yl)oxycarbonyl]piperidin-4-yl]methyl 2,7,7-trimethyl-4-(3-nitrophenyl)-5-oxo-1,4,6,8-tetrahydroquinoline-3-carboxylate | IC50 | 10000.0 [1] |
| (4-Tert-butylphenyl)methyl 4-(3-bromophenyl)-2,7,7-trimethyl-5-oxo-1,4,6,8-tetrahydroquinoline-3-carboxylate | IC50 | 4270.0 [1] |
| Cyclohexyl 4-(3-cyanophenyl)-2,7,7-trimethyl-5-oxo-1,4,6,8-tetrahydroquinoline-3-carboxylate | IC50 | 43200.0 [1] |
| [1-[(2-Methylpropan-2-yl)oxycarbonyl]piperidin-4-yl]methyl 4-(2,3-dihydro-1,4-benzodioxin-6-yl)-2,7,7-trimethyl-5-oxo-1,4,6,8-tetrahydroquinoline-3-carboxylate | IC50 | 1520.0 [1] |
| [1-[(2-Methylpropan-2-yl)oxycarbonyl]piperidin-4-yl]methyl 4-(4-bromo-2-fluorophenyl)-2,7,7-trimethyl-5-oxo-1,4,6,8-tetrahydroquinoline-3-carboxylate | IC50 | 10000.0 [1] |
| 2-[1-[(2-Methylpropan-2-yl)oxycarbonyl]piperidin-4-yl]ethyl 4-(3-bromophenyl)-2,7,7-trimethyl-5-oxo-1,4,6,8-tetrahydroquinoline-3-carboxylate | IC50 | 2950.0 [1] |
| [1-[(2-Methylpropan-2-yl)oxycarbonyl]piperidin-4-yl]methyl (4S)-4-(3-bromophenyl)-2,7,7-trimethyl-5-oxo-1,4,6,8-tetrahydroquinoline-3-carboxylate | IC50 | 2590.0 [1] |
| [1-[(2-Methylpropan-2-yl)oxycarbonyl]piperidin-4-yl]methyl 2,7,7-trimethyl-5-oxo-4-[3-(trifluoromethyl)phenyl]-1,4,6,8-tetrahydroquinoline-3-carboxylate | IC50 | 760.0 [1] |
| [1-[(2-Methylpropan-2-yl)oxycarbonyl]piperidin-4-yl]methyl 4-[3-(1H-indol-5-yl)phenyl]-2,7,7-trimethyl-5-oxo-1,4,6,8-tetrahydroquinoline-3-carboxylate | IC50 | 770.0 [1] |
| Pyrazin-2-ylmethyl 4-(3-bromophenyl)-2,7,7-trimethyl-5-oxo-1,4,6,8-tetrahydroquinoline-3-carboxylate | IC50 | 860.0 [1] |
| 1-Adamantyl 4-(3-bromophenyl)-2,7,7-trimethyl-5-oxo-1,4,6,8-tetrahydroquinoline-3-carboxylate | IC50 | 10000.0 [1] |
| [1-[(2-Methylpropan-2-yl)oxycarbonyl]piperidin-4-yl]methyl 2,7,7-trimethyl-5-oxo-4-(4-phenylphenyl)-1,4,6,8-tetrahydroquinoline-3-carboxylate | IC50 | 10000.0 [1] |
| [1-[(2-Methylpropan-2-yl)oxycarbonyl]piperidin-4-yl]methyl 4-(3-cyanophenyl)-2,7,7-trimethyl-5-oxo-1,4,6,8-tetrahydroquinoline-3-carboxylate | IC50 | 220.0 [1] |
| [1-[(2-Methylpropan-2-yl)oxycarbonyl]piperidin-4-yl]methyl 4-(3-bromophenyl)-2,7,7-trimethyl-5-oxo-1,4,6,8-tetrahydroquinoline-3-carboxylate | IC50 | 360.0 [1] |
| [(1R)-2-Cyano-1-phenylethyl] 4-(3-bromophenyl)-2,7,7-trimethyl-5-oxo-1,4,6,8-tetrahydroquinoline-3-carboxylate | IC50 | 10000.0 [1] |
| [1-[(2-Methylpropan-2-yl)oxycarbonyl]piperidin-4-yl]methyl 4-(3,5-dichlorophenyl)-2,7,7-trimethyl-5-oxo-1,4,6,8-tetrahydroquinoline-3-carboxylate | IC50 | 640.0 [1] |
| [1-[(2-Methylpropan-2-yl)oxycarbonyl]piperidin-4-yl]methyl (4R)-4-(3-bromophenyl)-2,7,7-trimethyl-5-oxo-1,4,6,8-tetrahydroquinoline-3-carboxylate | IC50 | 130.0 [1] |
| Cyclohexyl 2,7,7-trimethyl-5-oxo-4-[3-(trifluoromethyl)phenyl]-1,4,6,8-tetrahydroquinoline-3-carboxylate | IC50 | 14700.0 [1] |
| Cyclohexyl 4-(2,3-dihydro-1,4-benzodioxin-6-yl)-2,7,7-trimethyl-5-oxo-1,4,6,8-tetrahydroquinoline-3-carboxylate | IC50 | 12300.0 [1] |
| Cyclohexyl 4-(3-bromophenyl)-2,7,7-trimethyl-5-oxo-1,4,5,6,7,8-hexahydroquinoline-3-carboxylate | IC50 | 4150.0 [1] |
| (2S,3R)-N'-[(3S)-1-Methyl-2-oxo-5-phenyl-3H-1,4-benzodiazepin-3-yl]-3-(2-methylpropyl)-2-pentan-3-ylbutanediamide | IC50 | 2.0 [1] |
| (2R,3R)-N'-[(3S)-1-Methyl-2-oxo-5-phenyl-3H-1,4-benzodiazepin-3-yl]-2-phenyl-3-(3,3,3-trifluoropropyl)butanediamide | IC50 | 4.0 [1] |
| Unii-lsk1L593UU | IC50 | 7.8 [1] |
| (2R,3R)-2-(4-Fluorophenyl)-N'-[(3S)-1-methyl-2-oxo-5-phenyl-3H-1,4-benzodiazepin-3-yl]-3-(3,3,3-trifluoropropyl)butanediamide | IC50 | 2.0 [1] |
| (2R,3R)-2-(3-Methyl-1,2-oxazol-4-yl)-N'-[(3S)-1-methyl-2-oxo-5-phenyl-3H-1,4-benzodiazepin-3-yl]-3-(3,3,3-trifluoropropyl)butanediamide | IC50 | 3.0 [1] |
| (2S,3R)-N'-[(3S)-9-Aminooxy-2-oxo-5-phenyl-1,3-dihydro-1,4-benzodiazepin-3-yl]-2-(3-fluoropropyl)-3-(3,3,3-trifluoropropyl)butanediamide | IC50 | 7.0 [1] |
| (2S,3R)-2-[(3,3-Difluorocyclobutyl)methyl]-N'-[(3S)-9-methyl-2-oxo-5-phenyl-1,3-dihydro-1,4-benzodiazepin-3-yl]-3-(3,3,3-trifluoropropyl)butanediamide | IC50 | 3.0 [1] |
| (2S,3R)-2-[(3,3-Difluorocyclobutyl)methyl]-N'-[(3S)-9-fluoro-2-oxo-5-phenyl-1,3-dihydro-1,4-benzodiazepin-3-yl]-3-(3,3,3-trifluoropropyl)butanediamide | IC50 | 4.5 [1] |
| (2S,3R)-2-(4,4-Difluorocyclohexyl)-N'-[(3S)-9-methoxy-2-oxo-5-phenyl-1,3-dihydro-1,4-benzodiazepin-3-yl]-3-(3,3,3-trifluoropropyl)butanediamide | IC50 | 7.0 [1] |
| (2S,3R)-N'-[(3S)-9-Cyclopropyloxy-5-(3-fluorophenyl)-2-oxo-1,3-dihydro-1,4-benzodiazepin-3-yl]-2-(4,4-difluorocyclohexyl)-3-(3,3,3-trifluoropropyl)butanediamide | IC50 | 4.2 [1] |
| (2S,3R)-N'-[(3S)-9-Chloro-2-oxo-5-phenyl-1,3-dihydro-1,4-benzodiazepin-3-yl]-2-[4-(trifluoromethyl)cyclohexyl]-3-(3,3,3-trifluoropropyl)butanediamide | IC50 | 11.9 [1] |
| (2S,3R)-N'-[(3S)-9-Chloro-2-oxo-5-phenyl-1,3-dihydro-1,4-benzodiazepin-3-yl]-2-(4,4-difluorocyclohexyl)-3-(3,3,3-trifluoropropyl)butanediamide | IC50 | 4.4 [1] |
| (2S,3R)-2-(3,3-Difluorocyclobutyl)-N'-[(3S)-2-oxo-5-phenyl-1,3-dihydro-1,4-benzodiazepin-3-yl]-3-(3,3,3-trifluoropropyl)butanediamide | IC50 | 14.0 [1] |
| (2S,3R)-N'-[(3S)-9-Cyclopropyloxy-2-oxo-5-phenyl-1,3-dihydro-1,4-benzodiazepin-3-yl]-2-[(3,3-difluorocyclobutyl)methyl]-3-(3,3,3-trifluoropropyl)butanediamide | IC50 | 3.9 [1] |
| (2S,3R)-2-[(3,3-Difluorocyclobutyl)methyl]-N'-[(3S)-9-methoxy-2-oxo-5-phenyl-1,3-dihydro-1,4-benzodiazepin-3-yl]-3-(3,3,3-trifluoropropyl)butanediamide | IC50 | 2.9 [1] |
| (2S,3R)-N'-[(3S)-9-Chloro-5-(3-methylphenyl)-2-oxo-1,3-dihydro-1,4-benzodiazepin-3-yl]-2-[(3,3-difluorocyclobutyl)methyl]-3-(3,3,3-trifluoropropyl)butanediamide | IC50 | 1.7 [1] |
| (2S,3R)-N'-[(3S)-9-Cyclopropyl-2-oxo-5-phenyl-1,3-dihydro-1,4-benzodiazepin-3-yl]-2-[(3,3-difluorocyclobutyl)methyl]-3-(3,3,3-trifluoropropyl)butanediamide | IC50 | 5.6 [1] |
| (2S,3R)-N'-[(3S)-9-Chloro-2-oxo-5-phenyl-1,3-dihydro-1,4-benzodiazepin-3-yl]-2-[(3,3-difluorocyclobutyl)methyl]-3-(3,3,3-trifluoropropyl)butanediamide | IC50 | 2.8 [1] |
| (2S,3R)-2-[(3,3-Difluorocyclobutyl)methyl]-N'-[(3S)-2-oxo-5-phenyl-1,3-dihydro-1,4-benzodiazepin-3-yl]-3-(3,3,3-trifluoropropyl)butanediamide | IC50 | 4.4 [1] |
| (2S,3R)-2-(3-Fluoropropyl)-N'-[(3S)-8-methoxy-2-oxo-5-phenyl-1,3-dihydro-1,4-benzodiazepin-3-yl]-3-(3,3,3-trifluoropropyl)butanediamide | IC50 | 5.8 [1] |
| (2S,3R)-2-(2,2-Difluoropropyl)-N'-[(3S)-2-oxo-5-phenyl-1,3-dihydro-1,4-benzodiazepin-3-yl]-3-(3,3,3-trifluoropropyl)butanediamide | IC50 | 2.7 [1] |
| (2S,3R)-N'-[(3S)-9-Fluoro-2-oxo-5-phenyl-1,3-dihydro-1,4-benzodiazepin-3-yl]-2-[(2S)-3,3,3-trifluoro-2-methylpropyl]-3-(3,3,3-trifluoropropyl)butanediamide | IC50 | 2.9 [1] |
| (2S,3R)-N'-[(3S)-9-Chloro-2-oxo-5-phenyl-1,3-dihydro-1,4-benzodiazepin-3-yl]-2-(3-fluoropropyl)-3-(3,3,3-trifluoropropyl)butanediamide | IC50 | 10.8 [1] |
| (2S,3R)-2-(3,3-Difluorobutyl)-N'-[(3S)-9-methoxy-2-oxo-5-phenyl-1,3-dihydro-1,4-benzodiazepin-3-yl]-3-(3,3,3-trifluoropropyl)butanediamide | IC50 | 7.5 [1] |
| (2S,3R)-N'-[(3S)-9-Chloro-2-oxo-5-phenyl-1,3-dihydro-1,4-benzodiazepin-3-yl]-2-[(2R)-3,3,3-trifluoro-2-methylpropyl]-3-(3,3,3-trifluoropropyl)butanediamide | IC50 | 3.2 [1] |
| (2S,3R)-N'-[(3S)-9-Chloro-2-oxo-5-phenyl-1,3-dihydro-1,4-benzodiazepin-3-yl]-2-[(2S)-3,3,3-trifluoro-2-methylpropyl]-3-(3,3,3-trifluoropropyl)butanediamide | IC50 | 5.1 [1] |
| (2S,3R)-N'-[(3S)-9-Chloro-2-oxo-5-phenyl-1,3-dihydro-1,4-benzodiazepin-3-yl]-2-(3,3-difluorobutyl)-3-(3,3,3-trifluoropropyl)butanediamide | IC50 | 3.9 [1] |
| (2S,3R)-2-[(1-Fluorocyclobutyl)methyl]-N'-[(3S)-9-methyl-2-oxo-5-phenyl-1,3-dihydro-1,4-benzodiazepin-3-yl]-3-(3,3,3-trifluoropropyl)butanediamide | IC50 | 3.8 [1] |
| (2S,3R)-N'-[(3S)-5-(3-Chlorophenyl)-9-ethyl-2-oxo-1,3-dihydro-1,4-benzodiazepin-3-yl]-2,3-bis(3,3,3-trifluoropropyl)butanediamide | IC50 | 4.9 [1] |
| (2S,3R)-N'-[(3S)-5-(3-Chlorophenyl)-2-oxo-9-propan-2-yl-1,3-dihydro-1,4-benzodiazepin-3-yl]-2,3-bis(3,3,3-trifluoropropyl)butanediamide | IC50 | 1.8 [1] |
| (2S,3R)-N'-[(3S)-9-Ethyl-5-(3-methylphenyl)-2-oxo-1,3-dihydro-1,4-benzodiazepin-3-yl]-2,3-bis(3,3,3-trifluoropropyl)butanediamide | IC50 | 7.2 [1] |
| (2S,3R)-N'-[(3S)-5-(3-Chlorophenyl)-9-methyl-2-oxo-1,3-dihydro-1,4-benzodiazepin-3-yl]-2,3-bis(3,3,3-trifluoropropyl)butanediamide | IC50 | 4.4 [1] |
| (2S,3R)-N'-[(3S)-5-(3-Chlorophenyl)-9-methyl-2-oxo-1,3-dihydro-1,4-benzodiazepin-3-yl]-2-(4,4,4-trifluorobutyl)-3-(3,3,3-trifluoropropyl)butanediamide | IC50 | 6.0 [1] |
| (2S,3R)-N'-[(3S)-5-(3-Methylphenyl)-2-oxo-9-(trifluoromethyl)-1,3-dihydro-1,4-benzodiazepin-3-yl]-2,3-bis(3,3,3-trifluoropropyl)butanediamide | IC50 | 8.2 [1] |
| (2S,3R)-N'-[(3S)-9-Chloro-5-(3,5-dimethylphenyl)-2-oxo-1,3-dihydro-1,4-benzodiazepin-3-yl]-2,3-bis(3,3,3-trifluoropropyl)butanediamide | IC50 | 2.5 [1] |
| (2S,3R)-N'-[(3S)-5-(3-Methylphenyl)-2-oxo-9-propan-2-yl-1,3-dihydro-1,4-benzodiazepin-3-yl]-2,3-bis(3,3,3-trifluoropropyl)butanediamide | IC50 | 3.0 [1] |
| (2S,3R)-N'-[(3S)-2-Oxo-5-phenyl-9-propan-2-yl-1,3-dihydro-1,4-benzodiazepin-3-yl]-2,3-bis(3,3,3-trifluoropropyl)butanediamide | IC50 | 3.4 [1] |
| (2S,3R)-N'-[(3S)-9-Cyclopropyloxy-5-(3-methylphenyl)-2-oxo-1,3-dihydro-1,4-benzodiazepin-3-yl]-2-(4,4,4-trifluorobutyl)-3-(3,3,3-trifluoropropyl)butanediamide | IC50 | 7.7 [1] |
| (2S,3R)-N'-[(3S)-9-Cyclopropyloxy-5-(3-methylphenyl)-2-oxo-1,3-dihydro-1,4-benzodiazepin-3-yl]-2,3-bis(3,3,3-trifluoropropyl)butanediamide | IC50 | 4.4 [1] |
| (2S,3R)-N'-[(3S)-9-Cyclopropyloxy-2-oxo-5-phenyl-1,3-dihydro-1,4-benzodiazepin-3-yl]-2-(4,4,4-trifluorobutyl)-3-(3,3,3-trifluoropropyl)butanediamide | IC50 | 5.8 [1] |
| (2S,3R)-N'-[(3S)-9-Chloro-5-(3-methylphenyl)-2-oxo-1,3-dihydro-1,4-benzodiazepin-3-yl]-2-(4,4,4-trifluorobutyl)-3-(3,3,3-trifluoropropyl)butanediamide | IC50 | 5.7 [1] |
| (2S,3R)-N'-[(3S)-9-Methyl-2-oxo-5-[3-(trifluoromethyl)phenyl]-1,3-dihydro-1,4-benzodiazepin-3-yl]-2-(4,4,4-trifluorobutyl)-3-(3,3,3-trifluoropropyl)butanediamide | IC50 | 4.6 [1] |
| (2S,3R)-N'-[(3S)-9-Cyclopropyloxy-2-oxo-5-phenyl-1,3-dihydro-1,4-benzodiazepin-3-yl]-2,3-bis(3,3,3-trifluoropropyl)butanediamide | IC50 | 4.8 [1] |
| (2S,3R)-N'-[(3S)-9-Methyl-2-oxo-5-[3-(trifluoromethyl)phenyl]-1,3-dihydro-1,4-benzodiazepin-3-yl]-2,3-bis(3,3,3-trifluoropropyl)butanediamide | IC50 | 1.6 [1] |
| (2S,3R)-N'-[(3S)-9-Chloro-5-(2-methylphenyl)-2-oxo-1,3-dihydro-1,4-benzodiazepin-3-yl]-2,3-bis(3,3,3-trifluoropropyl)butanediamide | IC50 | 3.3 [1] |
| (2S,3R)-N'-[(3S)-5-(4-Fluorophenyl)-9-methyl-2-oxo-1,3-dihydro-1,4-benzodiazepin-3-yl]-2,3-bis(3,3,3-trifluoropropyl)butanediamide | IC50 | 3.1 [1] |
| (2S,3R)-N'-[(3S)-9-Methyl-2-oxo-5-phenyl-1,3-dihydro-1,4-benzodiazepin-3-yl]-2,3-bis(3,3,3-trifluoropropyl)butanediamide | IC50 | 4.7 [1] |
| (2S,3R)-N'-[(3S)-9-Cyclopropyl-2-oxo-5-phenyl-1,3-dihydro-1,4-benzodiazepin-3-yl]-2,3-bis(3,3,3-trifluoropropyl)butanediamide | IC50 | 1.4 [1] |
| (2S,3R)-N'-[(3S)-9-Chloro-5-(3-cyclopropylphenyl)-2-oxo-1,3-dihydro-1,4-benzodiazepin-3-yl]-2,3-bis(3,3,3-trifluoropropyl)butanediamide | IC50 | 1.7 [1] |
| (2S,3R)-N'-[(3S)-5-(3-Chlorophenyl)-9-methoxy-2-oxo-1,3-dihydro-1,4-benzodiazepin-3-yl]-2,3-bis(3,3,3-trifluoropropyl)butanediamide | IC50 | 3.7 [1] |
| (2S,3R)-N'-[(3S)-5-(4-Chlorophenyl)-9-methoxy-2-oxo-1,3-dihydro-1,4-benzodiazepin-3-yl]-2,3-bis(3,3,3-trifluoropropyl)butanediamide | IC50 | 2.8 [1] |
| (2S,3R)-N'-[(3S)-9-Chloro-5-(3-methylphenyl)-2-oxo-1,3-dihydro-1,4-benzodiazepin-3-yl]-2,3-bis(3,3,3-trifluoropropyl)butanediamide | IC50 | 4.8 [1] |
| (2S,3R)-N'-[(3S)-9-Methoxy-5-(3-methylphenyl)-2-oxo-1,3-dihydro-1,4-benzodiazepin-3-yl]-2,3-bis(3,3,3-trifluoropropyl)butanediamide | IC50 | 3.9 [1] |
| (2S,3R)-N'-[(3S)-5-[4-(Hydroxymethyl)phenyl]-2-oxo-1,3-dihydro-1,4-benzodiazepin-3-yl]-2,3-bis(3,3,3-trifluoropropyl)butanediamide | IC50 | 4.8 [1] |
| (2S,3R)-N'-[(3S)-5-(2-Methylphenyl)-2-oxo-1,3-dihydro-1,4-benzodiazepin-3-yl]-2,3-bis(3,3,3-trifluoropropyl)butanediamide | IC50 | 2.8 [1] |
| (2S,3R)-N'-[(3S)-5-(3-Methylphenyl)-2-oxo-1,3-dihydro-1,4-benzodiazepin-3-yl]-2,3-bis(3,3,3-trifluoropropyl)butanediamide | IC50 | 6.4 [1] |