N(G),N(G)-dimethylarginine dimethylaminohydrolase 1 Inhibitors (IC50, Ki)

Structure ▲ ▼	Compound Name ▲ ▼	Standard Type ▲ ▼	Standard Values (in nM) ▲ ▼
	1,2-Benzisothiazol-3(2H)-one	IC50	13200.0 [1]
	2-Ethylbenzimidazole	IC50	1400000.0 [1]
	2-Ethylbenzimidazole	Ki	800000.0 [1]
	3-(5-p-Tolyl-furan-2-yl)-propionic acid	IC50	45800.0 [1]
	4-(2,5-Dioxo-2,5-dihydro-1H-pyrrol-1-yl)benzoic acid	IC50	23300.0 [1]
	N~5~-{Imino[(2-Methoxyethyl)amino]methyl}-L-Ornithine	IC50	29000.0 [1]
	2-(4,6-Dimethyl-3-oxo-[1,2]thiazolo[5,4-b]pyridin-2-yl)-N-[2-(4-ethoxyphenyl)ethyl]acetamide	IC50	10500.0 [1]
	3-Aminomethylene-5-phenyl-3H-furan-2-thione	IC50	17700.0 [1]
	2-(1,3-Benzoxazol-2-ylsulfanyl)ethanamine	IC50	2700000.0 [1]
	2-(1,3-Benzoxazol-2-ylsulfanyl)ethanamine	Ki	1700000.0 [1]
	N-[2-(2,5-Dimethoxyphenyl)ethyl]-2-(4,6-dimethyl-3-oxo-[1,2]thiazolo[5,4-b]pyridin-2-yl)acetamide	IC50	9900.0 [1]
	2-(4,6-Dimethyl-3-oxo-[1,2]thiazolo[5,4-b]pyridin-2-yl)-N-(1-phenylethyl)acetamide	IC50	13700.0 [1]
	N-[2-(4-Chlorophenyl)ethyl]-2-(4,6-dimethyl-3-oxo-[1,2]thiazolo[5,4-b]pyridin-2-yl)acetamide	IC50	13400.0 [1]
	N-Butyl-2-(4,6-dimethyl-3-oxo-[1,2]thiazolo[5,4-b]pyridin-2-yl)acetamide	IC50	5100.0 [1]
	2-(4,6-Dimethyl-3-oxo-[1,2]thiazolo[5,4-b]pyridin-2-yl)-N-(3-ethoxypropyl)acetamide	IC50	7100.0 [1]
	N-(1,3-Benzodioxol-5-ylmethyl)-2-(4,6-dimethyl-3-oxo-[1,2]thiazolo[5,4-b]pyridin-2-yl)acetamide	IC50	11000.0 [1]
	N-(2,3-Dimethylcyclohexyl)-2-(4,6-dimethyl-3-oxo-[1,2]thiazolo[5,4-b]pyridin-2-yl)acetamide	IC50	8600.0 [1]
	N-[2-(Cyclohexen-1-yl)ethyl]-2-(4,6-dimethyl-3-oxo-[1,2]thiazolo[5,4-b]pyridin-2-yl)acetamide	IC50	11800.0 [1]
	2-(4,6-Dimethyl-3-oxo-[1,2]thiazolo[5,4-b]pyridin-2-yl)-N-(2-methoxyethyl)acetamide	IC50	3300.0 [1]
	Methyl(2-benzothiazolyl)phosphinic acid	IC50	9900.0 [1]
	3-(Azepan-1-yl)-1-naphthalen-1-ylpyrrolidine-2,5-dione	IC50	13100.0 [1]
	N-[(2-Chlorophenyl)methyl]-2-(4,6-dimethyl-3-oxo-[1,2]thiazolo[5,4-b]pyridin-2-yl)acetamide	IC50	39900.0 [1]
	(2E)-N-(4-Methylphenyl)but-2-enediamide	IC50	21200.0 [1]
	N-(3-Cyclohexylsulfanylpropyl)-2-(4,6-dimethyl-3-oxo-[1,2]thiazolo[5,4-b]pyridin-2-yl)acetamide	IC50	12800.0 [1]
	2-(4,6-Dimethyl-3-oxo-[1,2]thiazolo[5,4-b]pyridin-2-yl)-N-(4-phenylbutan-2-yl)acetamide	IC50	14100.0 [1]
	L-Homocysteine	IC50	640000.0 [1]
	N-omega-Propyl-L-arginine	IC50	283000.0 [1]
	(2S)-2-Amino-5-(1-aminobut-3-enylideneamino)pentanoic Acid	IC50	13000.0 [1]
	delta-N-Methylarginine	IC50	5000000.0 [1]
	SCH-202676 hydrobromide	IC50	13250.0 [1]
	omega-N-Allylarginine	IC50	207000.0 [1]
	N-omega-Propargyl-L-arginine	IC50	55000.0 [1]
	N-(2,6-Dimethyl-4-oxocyclohexa-2,5-dien-1-ylidene)benzenesulfonamide	IC50	9030.0 [1]
	N5-(1-Iminopropyl)-L-ornithine	IC50	300000.0 [1]
	N5-(1-Iminobutyl)-L-ornithine	IC50	70000.0 [1]
	L-N5-(1-Imino-3-pentenyl) ornithine	IC50	79000.0 [1]
	(2S)-2-Amino-5-[(N'-but-3-enylcarbamimidoyl)amino]pentanoic acid	IC50	189000.0 [1]
	(2S)-2-Amino-5-[carbamoyl(methyl)amino]pentanoic acid	IC50	5000000.0 [1]
	(2S)-2-Amino-5-[[(Z)-N,N'-dihydroxycarbamimidoyl]-methylamino]pentanoic acid	IC50	5000000.0 [1]
	Pyridazin-3(2H)-one, 4-mercapto-5-methoxy-2-phenyl-	IC50	12700.0 [1]
	Hddah-1-IN-1	IC50	70000.0 [1]
	(NE)-N-(3-chloro-2,6-dimethyl-4-oxocyclohexa-2,5-dien-1-ylidene)-4-methylbenzenesulfonamide	IC50	5500.0 [1]

Entire TableStructureCompound NameStandard TypeStandard Values (in nM)

Items per page: 510All1 - 10 of 42 ⟨⟩

---

---

References

This online tool may be cited as follows

MLA	"Quest Database™ N(G),N(G)-dimethylarginine dimethylaminohydrolase 1 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 21 Nov. 2024, https://www.aatbio.com/data-sets/n-g-n-g-dimethylarginine-dimethylaminohydrolase-1-inhibitors-ic50-ki.
APA	AAT Bioquest, Inc. (2024, November 21). Quest Database™ N(G),N(G)-dimethylarginine dimethylaminohydrolase 1 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/n-g-n-g-dimethylarginine-dimethylaminohydrolase-1-inhibitors-ic50-ki.
BibTeX	EndNote	RefMan