| Rimonabant | IC50 | 10100.0 [1] |
| 5-(1,1-Dimethylheptyl)-2-[5-hydroxy-2-(3-hydroxypropyl)cyclohexyl]phenol | IC50 | 5990.0 [1] |
| N-Arachidonoylglycine | IC50 | 10000.0 [1] |
| Psb-SB1202 | IC50 | 10000.0 [1] |
| 5-Hydroxy-3-[(2-hydroxyphenyl)methyl]-7-(2-methyloctan-2-yl)chromen-2-one | IC50 | 15900.0 [1] |
| 3-Benzyl-5-isopropyl-8-methylchromen-2-one | IC50 | 10000.0 [1] |
| 3-Benzyl-5-methoxy-7-methylchromen-2-one | IC50 | 10000.0 [1] |
| 5-Isopropyl-3,8-dimethylchromen-2-one | IC50 | 10000.0 [1] |
| (1S,2S,5S,7R,9S,10R,13S)-1,2,9-Trimethyl-7-(2-methylprop-1-enyl)-6-oxa-22-azahexacyclo[11.10.0.02,10.05,9.015,23.016,21]tricosa-15(23),16,18,20-tetraene | IC50 | 9910.0 [1] |
| 3-[(2-Hydroxyphenyl)methyl]-8-methyl-5-propan-2-ylchromen-2-one | IC50 | 10000.0 [1] |
| 7-Bromo-5-methoxy-3-[(3-methoxyphenyl)methyl]chromen-2-one | IC50 | 10000.0 [1] |
| 5-Methoxy-3-[(3-methoxyphenyl)methyl]-7-pentylchromen-2-one | IC50 | 10000.0 [1] |
| 5-Hydroxy-3-[(3-hydroxyphenyl)methyl]-7-pentylchromen-2-one | IC50 | 10000.0 [1] |
| 5-Methoxy-3-[(2-methylphenyl)methyl]-7-pentylchromen-2-one | IC50 | 10000.0 [1] |
| 5-Hydroxy-3-[(2-methylphenyl)methyl]-7-pentylchromen-2-one | IC50 | 10000.0 [1] |
| 3-[(2-Chlorophenyl)methyl]-5-methoxy-7-pentylchromen-2-one | IC50 | 10000.0 [1] |
| 3-[(2-Chlorophenyl)methyl]-5-hydroxy-7-pentylchromen-2-one | IC50 | 10000.0 [1] |
| 3-Benzyl-5-methoxy-7-(2-methyloctan-2-yl)chromen-2-one | IC50 | 10000.0 [1] |
| 3-Benzyl-5-hydroxy-7-(2-methyloctan-2-yl)chromen-2-one | IC50 | 8100.0 [1] |
| 5-Methoxy-3-[(2-methoxyphenyl)methyl]-7-(2-methyloctan-2-yl)chromen-2-one | IC50 | 10000.0 [1] |
| 5-Methoxy-3-[(2-methoxyphenyl)methyl]-7-(2-methylnonan-2-yl)chromen-2-one | IC50 | 10000.0 [1] |
| Psb-SB-487 | IC50 | 12500.0 [1] |
| 7-(1-Butylcyclopentyl)-5-methoxy-3-[(2-methoxyphenyl)methyl]chromen-2-one | IC50 | 10000.0 [1] |
| 7-(1-Butylcyclopentyl)-5-hydroxy-3-[(2-hydroxyphenyl)methyl]chromen-2-one | IC50 | 10000.0 [1] |
| 7-(1-Butylcyclohexyl)-5-methoxy-3-[(2-methoxyphenyl)methyl]chromen-2-one | IC50 | 10000.0 [1] |
| 7-(1-Butylcyclohexyl)-5-hydroxy-3-[(2-hydroxyphenyl)methyl]chromen-2-one | IC50 | 10000.0 [1] |
| (1S,12S,15R,16S,17S,20S)-16-[(E)-4-Methoxy-4-methylpent-2-enyl]-1,16,20-trimethyl-3-azapentacyclo[10.8.0.02,10.04,9.015,20]icosa-2(10),4,6,8-tetraen-17-ol | IC50 | 13400.0 [1] |
| (2Z)-2-[[3-[6-(4-Propan-2-ylphenoxy)hexoxy]phenyl]methylidene]-6,7-dihydro-5H-imidazo[2,1-b][1,3]thiazin-3-one | IC50 | 10000.0 [1] |
| (5Z)-5-[[3-[(4-Chlorophenyl)methoxy]phenyl]methylidene]-3-methyl-2-methylsulfanylimidazol-4-one | IC50 | 10000.0 [1] |
| (4Z)-4-[[3-[(4-Chlorophenyl)methoxy]phenyl]methylidene]-2-[(4-methylphenyl)methylsulfanyl]-1H-imidazol-5-one | IC50 | 10000.0 [1] |
| (5Z)-5-[[3-[(4-Chlorophenyl)methoxy]phenyl]methylidene]-2-imino-1-methylimidazolidin-4-one | IC50 | 10000.0 [1] |
| (4Z)-2-Benzylsulfanyl-4-[[3-[(4-chlorophenyl)methoxy]phenyl]methylidene]-1H-imidazol-5-one | IC50 | 10000.0 [1] |
| (4Z)-4-[[3-[(4-Chlorophenyl)methoxy]phenyl]methylidene]-2-[(4-chlorophenyl)methylsulfanyl]-1H-imidazol-5-one | IC50 | 10000.0 [1] |
| (2Z)-2-[[3-[6-(2-Chlorophenoxy)hexoxy]phenyl]methylidene]-6,7-dihydro-5H-imidazo[2,1-b][1,3]thiazin-3-one | IC50 | 10000.0 [1] |
| (4Z)-4-[[3-[(4-Chlorophenyl)methoxy]phenyl]methylidene]-2-[(4-fluorophenyl)methylsulfanyl]-1H-imidazol-5-one | IC50 | 10000.0 [1] |
| (2Z)-2-[[3-[(4-Fluorophenyl)methoxy]phenyl]methylidene]-6,7-dihydro-5H-imidazo[2,1-b][1,3]thiazin-3-one | IC50 | 10000.0 [1] |
| (5Z)-5-{3-[(4-Chlorobenzyl)oxy]benzylidene}-2-thioxo-1,3-thiazolidin-4-one | IC50 | 10000.0 [1] |
| (5Z)-5-[[3-[(4-Chlorophenyl)methoxy]phenyl]methylidene]-1,3-thiazolidine-2,4-dione | IC50 | 10000.0 [1] |
| 3-[(2-Methoxyphenyl)methyl]-5,8-dimethylchromen-2-one | IC50 | 10000.0 [1] |
| 3-[(2-Methoxyphenyl)methyl]-5-methyl-8-propan-2-ylchromen-2-one | IC50 | 11300.0 [1] |
| 6-Methoxy-3-[(2-methoxyphenyl)methyl]-5,7,8-trimethylchromen-2-one | IC50 | 10000.0 [1] |
| 3-Benzyl-6-methoxy-5,7,8-trimethylchromen-2-one | IC50 | 10000.0 [1] |
| 3-Benzyl-6-hydroxy-5,7,8-trimethylchromen-2-one | IC50 | 10000.0 [1] |
| 3-[(4-Fluorophenyl)methyl]-6-methoxy-5,7,8-trimethylchromen-2-one | IC50 | 10000.0 [1] |
| 3-[(4-Fluorophenyl)methyl]-6-hydroxy-5,7,8-trimethylchromen-2-one | IC50 | 10000.0 [1] |
| 6-Methoxy-5,7,8-trimethyl-3-[(2-methylphenyl)methyl]chromen-2-one | IC50 | 10000.0 [1] |
| 6-Hydroxy-5,7,8-trimethyl-3-[(2-methylphenyl)methyl]chromen-2-one | IC50 | 10000.0 [1] |
| 3-[(4-Chlorophenyl)methyl]-5-methoxy-7-pentylchromen-2-one | IC50 | 10000.0 [1] |
| 3-[(4-Bromophenyl)methyl]-5-methoxy-7-pentylchromen-2-one | IC50 | 10000.0 [1] |
| (2Z)-2-[(3-Chlorophenyl)methylidene]-6,7-dihydro-5H-imidazo[2,1-b][1,3]thiazin-3-one | IC50 | 10000.0 [1] |
| (2Z)-2-[(E)-3-Phenylprop-2-enylidene]-6,7-dihydro-5H-imidazo[2,1-b][1,3]thiazin-3-one | IC50 | 10000.0 [1] |
| (2Z)-2-[(4-Propan-2-ylphenyl)methylidene]-6,7-dihydro-5H-imidazo[2,1-b][1,3]thiazin-3-one | IC50 | 10000.0 [1] |
| (2Z)-2-[(2,3-Dichlorophenyl)methylidene]-6,7-dihydro-5H-imidazo[2,1-b][1,3]thiazin-3-one | IC50 | 10000.0 [1] |
| (3Z)-3-[(E)-3-Phenylprop-2-enylidene]-6,7-dihydro-5H-imidazo[2,1-b][1,3]thiazin-2-one | IC50 | 10000.0 [1] |
| (2Z)-2-[(3-Phenoxyphenyl)methylidene]-5,6,7,8-tetrahydroimidazo[2,1-b][1,3]thiazepin-3-one | IC50 | 14100.0 [1] |
| Ethyl 2-[3-[(Z)-(3-oxo-5,6,7,8-tetrahydroimidazo[2,1-b][1,3]thiazepin-2-ylidene)methyl]phenoxy]acetate | IC50 | 10000.0 [1] |
| (2Z)-2-[(4-Phenylphenyl)methylidene]-5,6,7,8-tetrahydroimidazo[2,1-b][1,3]thiazepin-3-one | IC50 | 10000.0 [1] |
| 2-[3-(4-Chlorobenzyloxy)benzylidene]-2,3,5,6,7,8-hexahydroimidazo[2,1-b][1,3]thiazepine-3-one | IC50 | 10000.0 [1] |
| (2Z)-2-(1-Phenylethylidene)-5,6,7,8-tetrahydroimidazo[2,1-b][1,3]thiazepin-3-one | IC50 | 10000.0 [1] |
| 2-[3-(2,4-Dichlorobenzyloxy)benzylidene]-2,3,5,6,7,8-hexahydroimidazo[2,1-b][1,3]thiazepine-3-one | IC50 | 4610.0 [1] |
| 2-(2,4-Dimethoxybenzylidene)-2,3,6,7-tetrahydro-5H-imidazo[2,1-b][1,3]thiazine-3-one | IC50 | 10000.0 [1] |
| (2Z)-2-[(2-Methoxyphenyl)methylidene]-6,7-dihydro-5H-imidazo[2,1-b][1,3]thiazin-3-one | IC50 | 10000.0 [1] |
| 2-(2-Chlorobenzylidene)-2,3,6,7-tetrahydro-5H-imidazo[2,1-b][1,3]thiazine-3-one | IC50 | 10000.0 [1] |
| (2Z)-2-[(3,4-Dimethoxyphenyl)methylidene]-6,7-dihydro-5H-imidazo[2,1-b][1,3]thiazin-3-one | IC50 | 10000.0 [1] |
| (2Z)-2-[(3-Phenoxyphenyl)methylidene]-6,7-dihydro-5H-imidazo[2,1-b][1,3]thiazin-3-one | IC50 | 10000.0 [1] |
| 3,3-Diphenyl-5,6,7,8-tetrahydroimidazo[2,1-b][1,3]thiazepin-2-one | IC50 | 10000.0 [1] |
| 2,2-Diphenyl-2,3,5,6,7,8-hexahydroimidazo[2,1-b][1,3]thiazepine-3-one | IC50 | 10000.0 [1] |
| (2Z)-2-Benzylidene-6,7-dihydro-5H-imidazo[2,1-b][1,3]thiazin-3-one | IC50 | 10000.0 [1] |
| (2Z)-2-[(4-Chlorophenyl)methylidene]-6,7-dihydro-5H-imidazo[2,1-b][1,3]thiazin-3-one | IC50 | 10000.0 [1] |
| (2Z)-2-[(4-Bromophenyl)methylidene]-6,7-dihydro-5H-imidazo[2,1-b][1,3]thiazin-3-one | IC50 | 10000.0 [1] |
| (2Z)-2-[[4-(Dimethylamino)phenyl]methylidene]-6,7-dihydro-5H-imidazo[2,1-b][1,3]thiazin-3-one | IC50 | 10000.0 [1] |
| (2Z)-2-[(4-Methoxyphenyl)methylidene]-6,7-dihydro-5H-imidazo[2,1-b][1,3]thiazin-3-one | IC50 | 10000.0 [1] |
| 5,5-Diphenyl-6-oxo-2,3,5,6-tetrahydroimidazo[2,1-b]thiazole-2-carboxylic acid ethyl ester | IC50 | 10000.0 [1] |
| 5-Oxo-6,6-diphenyl-2,3,5,6-tetrahydroimidazo[2,1-b]thiazole-2-carboxylic acid ethyl ester | IC50 | 10000.0 [1] |
| 6,6-Diphenyl-2,3-dihydroimidazo[2,1-b][1,3]thiazol-5-one | IC50 | 10000.0 [1] |
| 5,5-Diphenyl-2,3-dihydroimidazo[2,1-b][1,3]thiazol-6(5H)-one | IC50 | 10000.0 [1] |
| 3,3-Diphenyl-6,7-dihydro-5H-imidazo[2,1-b][1,3]thiazin-2-one | IC50 | 10000.0 [1] |
| 2,2-Diphenyl-6,7-dihydro-5H-imidazo[2,1-b][1,3]thiazin-3-one | IC50 | 10000.0 [1] |
| (2Z)-2-[(3-Nitrophenyl)methylidene]-6,7-dihydro-5H-imidazo[2,1-b][1,3]thiazin-3-one | IC50 | 10000.0 [1] |
| (2Z)-2-[(4-Nitrophenyl)methylidene]-6,7-dihydro-5H-imidazo[2,1-b][1,3]thiazin-3-one | IC50 | 10000.0 [1] |
| 2-(2,3-Difluorobenzylidene)-2,3,6,7-tetrahydro-5H-imidazo[2,1-b][1,3]thiazine-3-one | IC50 | 10000.0 [1] |
| (2Z)-2-[[3-[(4-Chlorophenyl)methoxy]phenyl]methylidene]-6,7-dihydro-5H-imidazo[2,1-b][1,3]thiazin-3-one | IC50 | 279.0 [1] |
| [3-[(Z)-(3-Oxo-5,6,7,8-tetrahydroimidazo[2,1-b][1,3]thiazepin-2-ylidene)methyl]phenyl] 4-methylbenzoate | IC50 | 6450.0 [1] |
| (2Z)-2-[(2-Fluorophenyl)methylidene]-6,7-dihydro-5H-imidazo[2,1-b][1,3]thiazin-3-one | IC50 | 10000.0 [1] |
| 2-(2,4-Difluorobenzylidene)-2,3,6,7-tetrahydro-5H-imidazo[2,1-b][1,3]thiazine-3-one | IC50 | 10000.0 [1] |
| (2Z)-2-[(2,3-Dimethoxyphenyl)methylidene]-6,7-dihydro-5H-imidazo[2,1-b][1,3]thiazin-3-one | IC50 | 10000.0 [1] |
| 2-[3-(Benzyloxy)benzylidene]-2,3,6,7-tetrahydro-5H-imidazo[2,1-b][1,3]thiazine-3-one | IC50 | 7220.0 [1] |
| 2-[3-(2-Chlorobenzyloxy)benzylidene]-2,3,6,7-tetrahydro-5H-imidazo[2,1-b][1,3]thiazine-3-one | IC50 | 1650.0 [1] |
| 2-[3-(2,4-Dichlorobenzyloxy)benzylidene]-2,3,6,7-tetrahydro-5H-imidazo[2,1-b][1,3]thiazine-3-one | IC50 | 2550.0 [1] |
| (2Z)-2-[[3-[(3,4-Dichlorophenyl)methoxy]phenyl]methylidene]-6,7-dihydro-5H-imidazo[2,1-b][1,3]thiazin-3-one | IC50 | 6160.0 [1] |
| [3-[(Z)-(3-Oxo-6,7-dihydro-5H-imidazo[2,1-b][1,3]thiazin-2-ylidene)methyl]phenyl] benzoate | IC50 | 6350.0 [1] |
| [3-[(Z)-(3-Oxo-6,7-dihydro-5H-imidazo[2,1-b][1,3]thiazin-2-ylidene)methyl]phenyl] 4-chlorobenzoate | IC50 | 14300.0 [1] |
| 2-[3-(Benzyloxy)benzylidene]-2,3,5,6,7,8-hexahydroimidazo[2,1-b][1,3]thiazepine-3-one | IC50 | 10000.0 [1] |
| (2Z)-2-[[3-[(3-Chlorophenyl)methoxy]phenyl]methylidene]-5,6,7,8-tetrahydroimidazo[2,1-b][1,3]thiazepin-3-one | IC50 | 10000.0 [1] |
| (2Z)-2-[[3-[(2-Chlorophenyl)methoxy]phenyl]methylidene]-5,6,7,8-tetrahydroimidazo[2,1-b][1,3]thiazepin-3-one | IC50 | 6480.0 [1] |
| 2-[3-(4-Fluorobenzyloxy)benzylidene]-2,3,5,6,7,8-hexahydroimidazo[2,1-b][1,3]thiazepine-3-one | IC50 | 10000.0 [1] |
| [(2R)-1-Hydroxy-3-[hydroxy-[(2S,3R,5S,6S)-2,3,4,5,6-pentahydroxycyclohexyl]oxyphosphoryl]oxypropan-2-yl] (5Z,8Z,11Z,14Z)-icosa-5,8,11,14-tetraenoate | IC50 | 10000.0 [1] |
| (2Z)-2-[(2,4-Dichlorophenyl)methylidene]-6,7-dihydro-5H-imidazo[2,1-b][1,3]thiazin-3-one | IC50 | 10000.0 [1] |
| (2Z)-2-[(2,6-Dichlorophenyl)methylidene]-6,7-dihydro-5H-imidazo[2,1-b][1,3]thiazin-3-one | IC50 | 10000.0 [1] |