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Myosin light chain kinase, smooth muscle Inhibitors (IC50, Ki)

Structure
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▼
Compound Name
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▼
Standard Type
▲
▼
Standard Values (in nM)
▲
▼
WortmanninIC50170.0 [1], 1900.0 [2], 5000.0 [3]
StaurosporineIC5010.0 [1], 40.0 [2]
FasudilIC503600.0 [1]
FasudilKi36000.0 [1]
Antibiotic K 252aIC5022.0 [1]
Antibiotic K 252aKi20.0 [1]
PiceatannolIC5012000.0 [1]
ML-9 free baseKi3800.0 [1]
NifedipineIC502020.0 [1]
N-(2-(4-Bromocinnamylamino)ethyl)-5-isoquinolinesulfonamideKi28300.0 [1]
MyricetinKi1700.0 [1]
N-(6-Aminohexyl)-5-chloro-1-naphthalenesulfonamideKi110000.0 [1]
K252aKi17.0 [1]
Methyl (15S,16S,18R)-16-hydroxy-15-methyl-3-oxo-28-oxa-4,14,19-triazaoctacyclo[12.11.2.115,18.02,6.07,27.08,13.019,26.020,25]octacosa-1,6,8,10,12,20,22,24,26-nonaene-16-carboxylateIC5025.0 [1]
Go-6976IC505800.0 [1]
1H-1,4-Diazepine, hexahydro-1-((5-iodo-1-naphthalenyl)sulfonyl)-Ki300.0 [1]
N-(2-Guanidinoethyl)-5-isoquinolinesulfonamideKi150000.0 [1]
(S)-2-Methyl-1-[(4-methyl-5-isoquinoline)sulfonyl]-homopiperazineKi10100.0 [1]
Bisindolylmaleimide xi, HClIC5017800.0 [1]
3-[8-(Aminomethyl)-6,7,8,9-tetrahydropyrido[1,2-a]indol-10-yl]-4-(1-methylindol-3-yl)pyrrole-2,5-dioneIC503700.0 [1]
N-(2-Aminoethyl)-5-chloronaphthalene-1-sulfonamideKi7400.0 [1]
DehydroaltenusinIC50690.0 [1]
5,8-Dihydroxy-3-methyl-4-(9H)-naphtho(2,3-c)furanoneIC5010000.0 [1]
N-(4,6-Dimethyl-2-pyrimidinyl)-1,3-benzothiazol-2-amineIC50100000.0 [1]
CID 73442760IC501000000.0 [1]
1-[2-(1,3-Benzothiazol-2-ylamino)-4,6-dimethylpyrimidin-5-yl]ethanoneIC50100000.0 [1]
3-[3-(Dimethylamino)-2-hydroxypropyl]-7-methoxy-23-methyl-3,13,23-triazahexacyclo[14.7.0.02,10.04,9.011,15.017,22]tricosa-1,4(9),5,7,10,15,17,19,21-nonaene-12,14-dioneIC50120.0 [1]
CID 50898538IC5036000.0 [1]
Ethyl 2-methoxy-6-methyl-3-phenacyl-4-phenyl-2,4-dihydro-1H-pyrimidine-5-carboxylateIC504291904.01 [1]
Ethyl 3-[2-(4-chlorophenyl)-2-oxoethyl]-2-methoxy-6-methyl-4-phenyl-2,4-dihydro-1H-pyrimidine-5-carboxylateIC503003032.28 [1]
Ethyl 2-methoxy-3-[2-(4-methoxyphenyl)-2-oxoethyl]-6-methyl-4-phenyl-2,4-dihydro-1H-pyrimidine-5-carboxylateIC507518825.4 [1]
Ethyl 4-(4-chlorophenyl)-2-methoxy-6-methyl-3-phenacyl-2,4-dihydro-1H-pyrimidine-5-carboxylateIC503194920.09 [1]
Ethyl 4-(4-chlorophenyl)-3-[2-(4-chlorophenyl)-2-oxoethyl]-2-methoxy-6-methyl-2,4-dihydro-1H-pyrimidine-5-carboxylateIC502421307.79 [1]
Ethyl 3-[2-(4-chlorophenyl)-2-oxoethyl]-2-methoxy-4-(4-methoxyphenyl)-6-methyl-2,4-dihydro-1H-pyrimidine-5-carboxylateIC503300350.01 [1]
Ethyl 4-(4-hydroxyphenyl)-2-methoxy-6-methyl-3-phenacyl-2,4-dihydro-1H-pyrimidine-5-carboxylateIC509803925.45 [1]
Ethyl 3-[2-(4-chlorophenyl)-2-oxoethyl]-4-(4-hydroxyphenyl)-2-methoxy-6-methyl-2,4-dihydro-1H-pyrimidine-5-carboxylateIC506579001.72 [1]
Ethyl 4-(4-hydroxyphenyl)-2-methoxy-3-[2-(4-methoxyphenyl)-2-oxoethyl]-6-methyl-2,4-dihydro-1H-pyrimidine-5-carboxylateIC5010204224.39 [1]
Ethyl 2-methoxy-6-methyl-4-(4-methylphenyl)-3-phenacyl-2,4-dihydro-1H-pyrimidine-5-carboxylateIC505208348.07 [1]
Ethyl 3-[2-(4-chlorophenyl)-2-oxoethyl]-2-methoxy-6-methyl-4-(4-methylphenyl)-2,4-dihydro-1H-pyrimidine-5-carboxylateIC503424680.02 [1]
Ethyl 2-methoxy-3-[2-(4-methoxyphenyl)-2-oxoethyl]-6-methyl-4-(4-methylphenyl)-2,4-dihydro-1H-pyrimidine-5-carboxylateIC5019607851.09 [1]
Ethyl 2-methoxy-4-(4-methoxyphenyl)-6-methyl-3-phenacyl-2,4-dihydro-1H-pyrimidine-5-carboxylateIC5013513567.02 [1]
Ethyl 2-methoxy-4-(4-methoxyphenyl)-3-[2-(4-methoxyphenyl)-2-oxoethyl]-6-methyl-2,4-dihydro-1H-pyrimidine-5-carboxylateIC5024390460.5 [1]
6-(2,4-Difluorophenyl)sulfonyl-2-(1H-indol-5-ylamino)-8-methylpyrido[2,3-d]pyrimidin-7-oneIC5010000.0 [1]
8-(4-Ethylphenyl)-5-Methyl-2,5-Dihydropyrazolo[4,3-C][2,1]benzothiazine 4,4-DioxideIC504000.0 [1]
1-Ethyl-8-(4-Ethylphenyl)-5-Methyl-1,5-Dihydropyrazolo[4,3-C][2,1]benzothiazine 4,4-DioxideIC5010000.0 [1]
1-[4-(4-Chlorophenyl)-2-methyl-4H-pyrimido[2,1-b][1,3]benzothiazol-3-yl]ethanoneIC5010989046.22 [1]
Ethyl 4-(4-chlorophenyl)-2-methoxy-3-[2-(4-methoxyphenyl)-2-oxoethyl]-6-methyl-2,4-dihydro-1H-pyrimidine-5-carboxylateIC505494523.05 [1]
1-[4-(2-Chlorophenyl)-2-methyl-4H-pyrimido[2,1-b][1,3]benzothiazol-3-yl]ethanoneIC5010204224.39 [1]
1-[4-(4-Fluorophenyl)-2-methyl-4H-pyrimido[2,1-b][1,3]benzothiazol-3-yl]ethanoneIC5013698720.35 [1]
1-[4-(2-Hydroxyphenyl)-2-methyl-4H-pyrimido[2,1-b][1,3]benzothiazol-3-yl]ethanoneIC5023256266.74 [1]
1-[4-(4-Hydroxyphenyl)-2-methyl-4H-pyrimido[2,1-b][1,3]benzothiazol-3-yl]ethanoneIC5023753083.75 [1]
1-[4-(4-Methoxyphenyl)-2-methyl-4H-pyrimido[2,1-b][1,3]benzothiazol-3-yl]ethanoneIC5046729377.97 [1]
1-[2-Methyl-4-(3-nitrophenyl)-4H-pyrimido[2,1-b][1,3]benzothiazol-3-yl]ethanoneIC5049019626.74 [1]
1-[2-Methyl-4-(4-nitrophenyl)-4H-pyrimido[2,1-b][1,3]benzothiazol-3-yl]ethanoneIC5049023013.01 [1]
1-[4-[4-(Dimethylamino)phenyl]-2-methyl-4H-pyrimido[2,1-b][1,3]benzothiazol-3-yl]ethanoneIC5022883370.91 [1]
1-[4-(4-Hydroxy-3-methoxyphenyl)-2-methyl-4H-pyrimido[2,1-b][1,3]benzothiazol-3-yl]ethanoneIC5027248336.88 [1]
1-[4-(2-Chlorophenyl)-2-methyl-4H-pyrimido[2,1-b][1,3]benzothiazol-3-yl]propan-1-oneIC509259339.33 [1]
1-[4-(4-Chlorophenyl)-2-methyl-4H-pyrimido[2,1-b][1,3]benzothiazol-3-yl]propan-1-oneIC509009070.8 [1]
1-[4-(4-Fluorophenyl)-2-methyl-4H-pyrimido[2,1-b][1,3]benzothiazol-3-yl]propan-1-oneIC507518825.4 [1]
1-[4-(2-Hydroxyphenyl)-2-methyl-4H-pyrimido[2,1-b][1,3]benzothiazol-3-yl]propan-1-oneIC5021276980.72 [1]
1-[4-(4-Hydroxyphenyl)-2-methyl-4H-pyrimido[2,1-b][1,3]benzothiazol-3-yl]propan-1-oneIC5016949231.05 [1]
1-[4-(4-Methoxyphenyl)-2-methyl-4H-pyrimido[2,1-b][1,3]benzothiazol-3-yl]propan-1-oneIC5046083982.18 [1]
1-[2-Methyl-4-(3-nitrophenyl)-4H-pyrimido[2,1-b][1,3]benzothiazol-3-yl]propan-1-oneIC5047620066.77 [1]
1-[2-Methyl-4-(4-nitrophenyl)-4H-pyrimido[2,1-b][1,3]benzothiazol-3-yl]propan-1-oneIC5032895008.28 [1]
1-[4-[4-(Dimethylamino)phenyl]-2-methyl-4H-pyrimido[2,1-b][1,3]benzothiazol-3-yl]propan-1-oneIC5013568754.97 [1]
1-[4-(4-Hydroxy-3-methoxyphenyl)-2-methyl-4H-pyrimido[2,1-b][1,3]benzothiazol-3-yl]propan-1-oneIC5027248336.88 [1]
1-[2-(1,3-Benzothiazol-2-ylamino)-4-ethyl-6-methylpyrimidin-5-yl]ethanoneIC50100000.0 [1]
4-(2-Chloro-4-fluorophenyl)-8-(2,6-dichlorophenyl)-7-oxido-1,7-naphthyridin-7-iumIC5010000.0 [1]
N-[6-Benzyl-2-(2-phenylethylamino)-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-yl]naphthalene-2-sulfonamideIC50900.0 [1]
5-(Methoxymethyl)-4-[2,3,4-trihydroxy-6-(methoxymethyl)phenyl]benzene-1,2,3-triol;hydrochlorideIC5017800.0 [1]
3-[8-(Aminomethyl)-6,7,8,9-tetrahydropyrido[1,2-a]indol-3-yl]-4-(1-methylindol-3-yl)pyrrole-2,5-dione;hydrochlorideIC503700.0 [1]
4-Chloro-N-[2-(2-phenylethylamino)pyrimidin-4-yl]benzenesulfonamideIC5051000.0 [1]
(E)-N-[1-(3-Bromoanilino)-4-cyanoisoquinolin-7-yl]-4-(dimethylamino)but-2-enamideIC5023600.0 [1]
N-[1-(3-Bromoanilino)-4-cyanoisoquinolin-7-yl]-4-(dimethylamino)butanamideIC5025100.0 [1]
N-[1-(3-Bromoanilino)-4-cyanoisoquinolin-7-yl]-3-(4-methylpiperazin-1-yl)propanamideIC508700.0 [1]
1-[(3-Hydroxyphenyl)methyl]-3-(4-pyridin-4-yl-1,3-thiazol-2-yl)urea;methanesulfonic acidIC5015.63 [1]
4-(7-Methoxy-23-methyl-12,14-dioxo-3,13,23-triazahexacyclo[14.7.0.02,10.04,9.011,15.017,22]tricosa-1,4(9),5,7,10,15,17,19,21-nonaen-3-yl)butanenitrileIC5032.0 [1]
23-[3-(Dimethylamino)-2-hydroxypropyl]-19-methoxy-3-methyl-3,13,23-triazahexacyclo[14.7.0.02,10.04,9.011,15.017,22]tricosa-1,4,6,8,10,15,17(22),18,20-nonaen-12-oneIC509200.0 [1]
3-(7-Methoxy-23-methyl-12,14-dioxo-3,13,23-triazahexacyclo[14.7.0.02,10.04,9.011,15.017,22]tricosa-1,4(9),5,7,10,15,17,19,21-nonaen-3-yl)propanenitrileIC50200.0 [1]
Indolocarbazole deriv. 3bIC501600.0 [1]
Indolocarbazole deriv. 3cIC5030.0 [1]
Indolocarbazole deriv. 3dIC50390.0 [1]
Indolocarbazole deriv. 3eIC50220.0 [1]
Indolocarbazole deriv. 3fIC50310.0 [1]
Indolocarbazole deriv. 3gIC50250.0 [1]
Indolocarbazole deriv. 3hIC5018.0 [1]
23-[3-(Dimethylamino)-2-hydroxypropyl]-3-methyl-3,13,23-triazahexacyclo[14.7.0.02,10.04,9.011,15.017,22]tricosa-1,4,6,8,10,15,17,19,21-nonaen-12-oneIC505500.0 [1]
Indolocarbazole deriv. 3kIC5055.0 [1]
3-(19-Methoxy-23-methyl-12,14-dioxo-3,13,23-triazahexacyclo[14.7.0.02,10.04,9.011,15.017,22]tricosa-1,4,6,8,10,15,17(22),18,20-nonaen-3-yl)propanenitrileIC5049.0 [1]
Indolocarbazole deriv. 3nIC50180.0 [1]
Indolocarbazole deriv. 3pIC50120.0 [1]
Items per page: 1 - 10 of 91
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References

This online tool may be cited as follows

MLA

"Quest Database™ Myosin light chain kinase, smooth muscle Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 20 Nov. 2024, https://www.aatbio.com/data-sets/myosin-light-chain-kinase-smooth-muscle-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, November 20). Quest Database™ Myosin light chain kinase, smooth muscle Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/myosin-light-chain-kinase-smooth-muscle-inhibitors-ic50-ki.
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