| Clorgiline | IC50 | 4.46 [1] |
| Clorgiline | Ki | 0.3 [1], 12.0 [2] |
| Iproniazid | IC50 | 6560.0 [1] |
| Selegiline | IC50 | 67250.0 [1] |
| Selegiline | Ki | 3600.0 [1], 9060.0 [2], 16890.0 [3], 67250.0 [4] |
| Moclobemide | IC50 | 361380.0 [1] |
| Moclobemide | Ki | 5.0 [1], 14.0 [2], 102.0 [3], 110.0 [4] |
| Rasagiline | IC50 | 1420.0 [1] |
| Rasagiline | Ki | 9700.0 [1] |
| Toloxatone | IC50 | 3920.0 [1] |
| Toloxatone | Ki | 1500.0 [1] |
| Pargyline | IC50 | 3520.0 [1] |
| (1S,2R)-2-Phenylcyclopropan-1-amine;(1R,2S)-2-phenylcyclopropan-1-amine | IC50 | 2100.0 [1] |
| Parnate | IC50 | 6000.0 [1] |
| Parnate | Ki | 102000.0 [1] |
| Isatin | IC50 | 40000.0 [1], 56234.13 [2] |
| Isatin | Ki | 15000.0 [1] |
| Safinamide | IC50 | 50000.0 [1] |
| Safinamide | Ki | 365000.0 [1] |
| 4-(1-Benzylpiperidin-4-yl)-2-[(8-hydroxyquinolin-2-yl)methyl-prop-2-ynylamino]butanenitrile | IC50 | 3800.0 [1] |
| Iadademstat | IC50 | 48380.0 [1] |
| Linezolid | IC50 | 46000.0 [1] |
| Linezolid | Ki | 7900.0 [1], 20000.0 [2], 53000.0 [3], 55000.0 [4] |
| Apigenin | IC50 | 640.0 [1], 1550.0 [2], 1700.0 [3] |
| Acacetin | IC50 | 121.0 [1], 190.0 [2] |
| Acacetin | Ki | 59.2 [1] |
| Benzyl N-[1-[4-(2-aminocyclopropyl)anilino]-1-oxo-3-phenylpropan-2-yl]carbamate | IC50 | 320.0 [1], 1200.0 [2] |
| Benzyl N-[1-[4-(2-aminocyclopropyl)anilino]-1-oxo-3-phenylpropan-2-yl]carbamate | Ki | 1200.0 [1], 4000.0 [2] |
| 1-[3-(2,4-Dichloro-phenoxy)-propyl]-1,2,3,6-tetrahydro-pyridine | IC50 | 2600.0 [1] |
| 1-[3-(2,4-Dichloro-phenoxy)-propyl]-1,2,3,6-tetrahydro-pyridine | Ki | 900.0 [1], 2200.0 [2], 7400.0 [3] |
| Harmine | Ki | 5.0 [1], 16.9 [2], 17.0 [3] |
| Purpurin | IC50 | 2500.0 [1] |
| Purpurin | Ki | 422.0 [1] |
| Ladostigil | IC50 | 85000.0 [1], 100000.0 [2] |
| Ladostigil | Ki | 227000.0 [1] |
| Tranylcypromine hydrochloride | IC50 | 4500.0 [1], 10600.0 [2], 20000.0 [3] |
| 1-Phenethylpiperidine | IC50 | 757300.0 [1] |
| 1-Phenethylpiperidine | Ki | 121400.0 [1], 3681000.0 [2] |
| Aplysinopsin | IC50 | 35.0 [1], 10017.0 [2] |
| 4-Imidazolidinone, 5-((6-bromo-1H-indol-3-yl)methylene)-2-imino-1,3-dimethyl- | IC50 | 5.6 [1], 447.0 [2] |
| 5-Benzyloxyphthalimide | IC50 | 4170.0 [1] |
| 5-Benzyloxyphthalimide | Ki | 1100.0 [1] |
| 6-[(4-Chlorophenyl)methoxy]-1,3-benzoxathiol-2-one | IC50 | 189.0 [1] |
| 6-[(4-Chlorophenyl)methoxy]-1,3-benzoxathiol-2-one | Ki | 360.0 [1], 560.0 [2] |
| 6-(3-Phenylpropoxy)-3H-2-benzofuran-1-one | IC50 | 96.0 [1] |
| 6-(3-Phenylpropoxy)-3H-2-benzofuran-1-one | Ki | 25.0 [1], 62.0 [2] |
| 4-Methyl-1-(2-phenylethyl)-3,6-dihydro-2H-pyridine | IC50 | 623400.0 [1] |
| 4-Methyl-1-(2-phenylethyl)-3,6-dihydro-2H-pyridine | Ki | 407900.0 [1], 2587000.0 [2] |
| 7-[[4-(Trifluoromethyl)phenyl]methoxy]chromen-4-one | IC50 | 1970.0 [1], 18940.0 [2] |
| 4-N-[(1S,2R)-2-[4-[3-(Trifluoromethyl)phenyl]phenyl]cyclopropyl]cyclohexane-1,4-diamine | IC50 | 10700.0 [1], 14640.0 [2], 50000.0 [3] |
| Quercetin | IC50 | 2440.0 [1], 2800.0 [2] |
| 1,4-Benzoquinone | IC50 | 4820.0 [1] |
| 1,4-Benzoquinone | Ki | 9620.0 [1] |
| Donepezil | IC50 | 850000.0 [1], 1000000.0 [2] |
| Chelerythrine | IC50 | 550.0 [1] |
| Chelerythrine | Ki | 220.0 [1] |
| Deprenyl | IC50 | 67250.0 [1] |
| Tranylcypromine | IC50 | 4720.0 [1], 11500.0 [2] |
| Phenelzine | IC50 | 238.0 [1] |
| Phenelzine | Ki | 163.0 [1] |
| N-Propargyl-1(S)-aminoindan | IC50 | 17700.0 [1] |
| N-Propargyl-1(S)-aminoindan | Ki | 112000.0 [1] |
| Decursin | IC50 | 1760.0 [1] |
| Alternariol monomethyl ether | IC50 | 1710.0 [1] |
| Tedizolid | IC50 | 8700.0 [1] |
| Tedizolid | Ki | 2000.0 [1] |
| Mofegiline | IC50 | 1780.0 [1] |
| Mofegiline | Ki | 1100.0 [1] |
| 2-(Phenylazo)pyridine | IC50 | 18000.0 [1] |
| 2-(Phenylazo)pyridine | Ki | 5100.0 [1] |
| N-[(5-Phenylmethoxy-1H-indol-2-yl)methyl]prop-2-yn-1-amine | IC50 | 287.3 [1], 790.0 [2] |
| CID 53378764 | IC50 | 4.2 [1], 58.2 [2] |
| (E)-N'-(1-(5-Chloro-2-hydroxyphenyl)ethylidene)-3-(morpholinosulfonyl)benzohydrazide | IC50 | 300000.0 [1] |
| Hispidol | IC50 | 260.0 [1] |
| Hispidol | Ki | 100.0 [1] |
| 1,4-Naphthalenedione, 2,3,6-trimethyl- | Ki | 3000.0 [1], 6000.0 [2] |
| 4-(2-Pyridylazo)-N,N-dimethylaniline | IC50 | 7900.0 [1] |
| 4-(2-Pyridylazo)-N,N-dimethylaniline | Ki | 2300.0 [1] |
| N-[(2S)-4-[3-(2-Aminocyclopropyl)phenoxy]-1-(benzylamino)-1-oxobutan-2-yl]benzamide | IC50 | 230000.0 [1] |
| N-[(2S)-4-[3-(2-Aminocyclopropyl)phenoxy]-1-(benzylamino)-1-oxobutan-2-yl]benzamide | Ki | 230000.0 [1] |
| N-Phenylpyridine-2-methylamine | IC50 | 20000.0 [1] |
| N-Phenylpyridine-2-methylamine | Ki | 5700.0 [1] |
| 3,4-Dimethyl-7-(3,4-difluorobenzyloxy)coumarin | IC50 | 123.0 [1], 100000.0 [2] |
| N-[(2S)-4-[4-[(1S,2R)-2-Aminocyclopropyl]phenoxy]-1-(benzylamino)-1-oxobutan-2-yl]benzamide | IC50 | 290000.0 [1] |
| N-[(2S)-4-[4-[(1S,2R)-2-Aminocyclopropyl]phenoxy]-1-(benzylamino)-1-oxobutan-2-yl]benzamide | Ki | 250000.0 [1] |
| N-(4-Chlorophenyl)-4-oxochromene-3-carboxamide | IC50 | 10000.0 [1], 100000.0 [2] |
| N,N-Dimethyl-4-(pyridin-2-ylmethylideneamino)aniline | IC50 | 360.0 [1] |
| N,N-Dimethyl-4-(pyridin-2-ylmethylideneamino)aniline | Ki | 100.0 [1] |
| Pyridine, 2-(N-phenylformimidoyl)- | IC50 | 129000.0 [1] |
| Pyridine, 2-(N-phenylformimidoyl)- | Ki | 37000.0 [1] |
| 4-Hydroxybenzoic (2-hydroxybenzylidene)hydrazide | IC50 | 88500.0 [1] |
| N-(3,4-Dihydroxyphenyl)-4-oxochromene-2-carboxamide | IC50 | 190.0 [1], 190.55 [2] |
| N-[(E)-(2-Methylcyclohexylidene)amino]-4-phenyl-1,3-thiazol-2-amine | IC50 | 41230.0 [1], 41236.0 [2] |
| 4-(4-Methoxyphenyl)-N-[(E)-(2-methylcyclohexylidene)amino]-1,3-thiazol-2-amine | IC50 | 2760.0 [1], 2762.0 [2] |
| 4-(4-Chlorophenyl)-N-[(E)-(2-methylcyclohexylidene)amino]-1,3-thiazol-2-amine | IC50 | 35220.0 [1] |
| 7-Methoxy-3-(3-trifluoromethyl-phenyl)-indeno[1,2-c]pyridazin-5-one | IC50 | 38.0 [1], 1000.0 [2] |
| 8-Methoxy-3-[3-(trifluoromethyl)phenyl]indeno[1,2-c]pyridazin-5-one | IC50 | 0.1 [1], 1000.0 [2] |
| 7-Acetonyloxy-3-acetylamino-8-methoxycoumarin | IC50 | 5310.0 [1], 6430.0 [2] |
| N-[(2S)-1-[(3-Chlorophenyl)methylamino]-1-oxo-6-[[(1R,2S)-2-phenylcyclopropyl]amino]hexan-2-yl]-4-phenylbenzamide | IC50 | 100000.0 [1] |
| 6-((4-Chlorobenzyl)oxy)-3,4-dihydronaphthalen-1(2H)-one | IC50 | 238.0 [1], 340.0 [2] |