![](https://images.aatbio.com/dataset/ic50/mixed-lineage-kinase-7_b0f6535d633b24658defe8380c006aae.svg) | Vemurafenib | IC50 | 23.0 [1], 31.4 [2] |
![](https://images.aatbio.com/dataset/ic50/mixed-lineage-kinase-7_e9ddbfd3b6f07208dc97db4e7ef39cb0.svg) | 4-(3-Pyridin-2-YL-1H-pyrazol-4-YL)quinoline | IC50 | 1400.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mixed-lineage-kinase-7_c212e894513b08a44a48498579ea742a.svg) | LY-2090314 | IC50 | 20000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mixed-lineage-kinase-7_777898ba417f4e875e6f3109cad807ee.svg) | LY-3009120 | IC50 | 39.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mixed-lineage-kinase-7_f0a154106aee26d2cb409ff4c746c070.svg) | 3-Imidazo[1,2-a]pyridin-3-yl-4-[10-(morpholine-4-carbonyl)-1,10-diazatricyclo[6.4.1.04,13]trideca-2,4,6,8(13)-tetraen-3-yl]pyrrole-2,5-dione | IC50 | 13400.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mixed-lineage-kinase-7_498d85cce39dd7384f7a0bb29cf8216c.svg) | 3-(4-Imidazo[1,2-a]pyridin-3-yl-2,5-dioxopyrrol-3-yl)-N,N-dimethyl-1,10-diazatricyclo[6.4.1.04,13]trideca-2,4,6,8(13)-tetraene-10-carboxamide | IC50 | 20000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mixed-lineage-kinase-7_99d590530c99b53efc4907213bcd8b23.svg) | 7-Chloro-3-oxo-8-(1,3-thiazol-5-ylmethylamino)-11,16-dioxa-2,4,19,21-tetrazatricyclo[15.3.1.05,10]henicosa-1(20),5,7,9,17(21),18-hexaene-18-carbonitrile | Ki | 8573.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mixed-lineage-kinase-7_21aa752395444707db3d7c65ae53dc35.svg) | 1-({4-[(3,4-Dichlorophenyl)methoxy]phenyl}methyl)azetidine-3-carboxylic acid | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mixed-lineage-kinase-7_135745c63ed912627deefccdab2cf518.svg) | 3-[6-(2-Pyridin-2-yl-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl)benzimidazol-1-yl]propan-1-ol | IC50 | 708.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mixed-lineage-kinase-7_6bad3df0a8f4743f2718943d69c2c4f6.svg) | 4-[3-[6-[2-(6-Methylpyridin-2-yl)-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl]benzimidazol-1-yl]propyl]morpholine | IC50 | 8480.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mixed-lineage-kinase-7_ed98d3f7c09ac11edc8356dc5b0faed9.svg) | 3-Imidazo[1,2-a]pyridin-3-yl-4-[10-(piperidine-1-carbonyl)-1,10-diazatricyclo[6.4.1.04,13]trideca-2,4,6,8(13)-tetraen-3-yl]pyrrole-2,5-dione | IC50 | 20000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mixed-lineage-kinase-7_08529250ec2ce2c613602b3955d91e73.svg) | 3-[6-[2-(6-Methylpyridin-2-yl)-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl]benzimidazol-1-yl]propan-1-ol | IC50 | 2810.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mixed-lineage-kinase-7_f046ae8812a77e5cb35fd8b53bebf05d.svg) | Ripk1-IN-7 | IC50 | 457.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mixed-lineage-kinase-7_679cfd0590ae1f0d16e0c64b14500fbe.svg) | N,N-Diethyl-3-[6-[2-(6-methylpyridin-2-yl)-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl]benzimidazol-1-yl]propan-1-amine | IC50 | 20000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mixed-lineage-kinase-7_32260304c881c7e9a838fa55a76af1ee.svg) | 6-(2-Pyridin-2-yl-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl)-1-(3-pyrrolidin-1-ylpropyl)benzimidazole | IC50 | 4880.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mixed-lineage-kinase-7_a7ee75d4a7ce2e8d7ffa73cb444c324f.svg) | 5-(2-Amino-[1,2,4]triazolo[1,5-a]pyridin-7-yl)-N-tert-butylpyridine-3-sulfonamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mixed-lineage-kinase-7_51153882d3ab9f3566d96aeaf5c3eeab.svg) | 6-(2,4-Difluorophenyl)sulfonyl-2-(1H-indol-5-ylamino)-8-methylpyrido[2,3-d]pyrimidin-7-one | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mixed-lineage-kinase-7_59c6aab724852b8d67b99c2de32605b3.svg) | 6-(2-Pyridin-2-yl-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl)-1H-benzimidazole | IC50 | 20000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mixed-lineage-kinase-7_c04fbddbc0ab9108e3eb71dae12a8a8d.svg) | 6-[2-(6-Methylpyridin-2-yl)-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl]-1-(3-pyrrolidin-1-ylpropyl)benzimidazole | IC50 | 20000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mixed-lineage-kinase-7_c1026b7908f4e5db836f77ab3d7edfde.svg) | 5-[2-(6-Methylpyridin-2-yl)-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl]-1-[3-(oxan-2-yloxy)propyl]benzimidazole | IC50 | 20000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mixed-lineage-kinase-7_6f471ec8d26cc3f90ae463ae0799ae2d.svg) | 1-Methyl-6-(2-pyridin-2-yl-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl)benzimidazole | IC50 | 1310.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mixed-lineage-kinase-7_fcfcb9f09c76afcf95bfeac6aed6c031.svg) | 1-[3-(Oxan-2-yloxy)propyl]-5-(2-pyridin-2-yl-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl)benzimidazole | IC50 | 20000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mixed-lineage-kinase-7_5552e6487f0ab3659321a0f425845e04.svg) | 6-[2-(6-Methylpyridin-2-yl)-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl]-1-(3-piperidin-1-ylpropyl)benzimidazole | IC50 | 20000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mixed-lineage-kinase-7_ae92bb23f717566f8e8e99089aa41b22.svg) | 1-Methyl-6-[2-(6-methylpyridin-2-yl)-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl]benzimidazole | IC50 | 2340.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mixed-lineage-kinase-7_5715f628b864353ae465bb7190af2e4e.svg) | Propan-2-yl 3-(4-imidazo[1,2-a]pyridin-3-yl-2,5-dioxopyrrol-3-yl)-1,10-diazatricyclo[6.4.1.04,13]trideca-2,4,6,8(13)-tetraene-10-carboxylate | IC50 | 20000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mixed-lineage-kinase-7_7b77b20b9648173942886c5c04d36a35.svg) | 5-(2-Pyridin-2-yl-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl)-1H-indole | IC50 | 20000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mixed-lineage-kinase-7_a9be5c77c459be6a3988366cde650110.svg) | 6-[2-(6-Methylpyridin-2-yl)-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl]-1H-benzimidazole | IC50 | 15940.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mixed-lineage-kinase-7_79d4dc5e2a9950b673379798d4bdb5b1.svg) | 3-Bromo-N-[2,4-difluoro-3-[2-(3-methoxy-1H-pyrazolo[3,4-b]pyridin-5-yl)ethynyl]phenyl]benzenesulfonamide | IC50 | 5.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mixed-lineage-kinase-7_ce2fe90a5c55f4807bba224440e942fa.svg) | 3-Chloro-N-[2,4-difluoro-3-[2-(1-methylpyrazolo[3,4-b]pyridin-5-yl)ethynyl]phenyl]benzenesulfonamide | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mixed-lineage-kinase-7_6706cc2dedbd16c6908c75f6e1108e4c.svg) | 4-Chloro-N-[2,4-difluoro-3-[2-(3-methoxy-1H-pyrazolo[3,4-b]pyridin-5-yl)ethynyl]phenyl]benzenesulfonamide | IC50 | 16.8 [1] |
![](https://images.aatbio.com/dataset/ic50/mixed-lineage-kinase-7_19e03d33c15ee022ea7839f883d507cf.svg) | 3-Chloro-N-[2,4-difluoro-3-[2-(1H-pyrrolo[2,3-b]pyridin-5-yl)ethynyl]phenyl]benzenesulfonamide | IC50 | 22.6 [1] |
![](https://images.aatbio.com/dataset/ic50/mixed-lineage-kinase-7_8d2c6bdb823075d34dfe45928f6c6720.svg) | 3-Chloro-N-[2,4-difluoro-3-[2-(3-propan-2-yloxy-1H-pyrazolo[3,4-b]pyridin-5-yl)ethynyl]phenyl]benzenesulfonamide | IC50 | 42.7 [1] |
![](https://images.aatbio.com/dataset/ic50/mixed-lineage-kinase-7_b0d7c7db5b827b64ce6e8581452fc2ca.svg) | 2,3-Dichloro-N-[2,4-difluoro-3-[2-(3-methoxy-1H-pyrazolo[3,4-b]pyridin-5-yl)ethynyl]phenyl]benzenesulfonamide | IC50 | 9.6 [1] |
![](https://images.aatbio.com/dataset/ic50/mixed-lineage-kinase-7_92c44f937b53c338109d97b7cb9c231e.svg) | 3-Chloro-N-[2,4-difluoro-3-[2-(1H-pyrazolo[3,4-b]pyridin-5-yl)ethynyl]phenyl]benzenesulfonamide | IC50 | 5.1 [1] |
![](https://images.aatbio.com/dataset/ic50/mixed-lineage-kinase-7_41e700fa55f10a77f9f97fa5f3595a8e.svg) | 3-Chloro-N-[2,4-difluoro-3-[2-(1H-indazol-5-yl)ethynyl]phenyl]benzenesulfonamide | IC50 | 994.1 [1] |
![](https://images.aatbio.com/dataset/ic50/mixed-lineage-kinase-7_32c8b34e1dc883198c7c4e0ccb444030.svg) | N-[2,4-Difluoro-3-[2-(3-methoxy-1H-pyrazolo[3,4-b]pyridin-5-yl)ethynyl]phenyl]benzenesulfonamide | IC50 | 19.2 [1] |
![](https://images.aatbio.com/dataset/ic50/mixed-lineage-kinase-7_abee97892484e54af63ba61f634275bc.svg) | N-[2,4-Difluoro-3-[2-(3-methoxy-1H-pyrazolo[3,4-b]pyridin-5-yl)ethynyl]phenyl]-3-methoxybenzenesulfonamide | IC50 | 7.5 [1] |
![](https://images.aatbio.com/dataset/ic50/mixed-lineage-kinase-7_aa0948d2b439ba579b311c14ebc3f7ee.svg) | 3-Chloro-N-[3-[2-(3-cyclopentyloxy-1H-pyrazolo[3,4-b]pyridin-5-yl)ethynyl]-2,4-difluorophenyl]benzenesulfonamide | IC50 | 143.7 [1] |
![](https://images.aatbio.com/dataset/ic50/mixed-lineage-kinase-7_1701465051c97c28a4bc2b15eeb25bb9.svg) | 3-Chloro-N-[2,4-difluoro-3-[2-(3-methoxy-1H-pyrazolo[3,4-b]pyridin-5-yl)ethynyl]phenyl]benzenesulfonamide | IC50 | 4.2 [1] |
![](https://images.aatbio.com/dataset/ic50/mixed-lineage-kinase-7_ce58e19ae964a112d6c2f51e4a9a8e69.svg) | 2-Chloro-N-[2,4-difluoro-3-[2-(3-methoxy-1H-pyrazolo[3,4-b]pyridin-5-yl)ethynyl]phenyl]benzenesulfonamide | IC50 | 5.1 [1] |
![](https://images.aatbio.com/dataset/ic50/mixed-lineage-kinase-7_42059abe4dcfb562a910f7ee4c3b6767.svg) | N-[2,4-Difluoro-3-[2-(3-methoxy-1H-pyrazolo[3,4-b]pyridin-5-yl)ethynyl]phenyl]-3-methylbenzenesulfonamide | IC50 | 12.1 [1] |
![](https://images.aatbio.com/dataset/ic50/mixed-lineage-kinase-7_cead7f65283c61797278fffe237c13ae.svg) | 3-Cyano-N-[2,4-difluoro-3-[2-(3-methoxy-1H-pyrazolo[3,4-b]pyridin-5-yl)ethynyl]phenyl]benzenesulfonamide | IC50 | 3.3 [1] |
![](https://images.aatbio.com/dataset/ic50/mixed-lineage-kinase-7_da569f46166fb5a4efb41e6800f2a157.svg) | N,N-Dimethyl-3-[6-[2-(6-methylpyridin-2-yl)-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl]benzimidazol-1-yl]propan-1-amine | IC50 | 20000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mixed-lineage-kinase-7_f29c45ad374a44e3cd2130f61df14c63.svg) | N,N-Dimethyl-3-[6-(2-pyridin-2-yl-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl)benzimidazol-1-yl]propan-1-amine | IC50 | 15880.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mixed-lineage-kinase-7_7042a2bfb0bfc3bafa0ee59fb6233e6a.svg) | Indolocarbazole deriv. 14m | IC50 | 9970.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mixed-lineage-kinase-7_d6e994bac1fa2a4f14247f9dd25b96a5.svg) | 1-Methyl-5-(2-pyridin-2-yl-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl)indole | IC50 | 16610.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mixed-lineage-kinase-7_6a2a42109fb182b2e0710d7ba72ecaa7.svg) | 1-Methyl-5-[2-(6-methylpyridin-2-yl)-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl]indole | IC50 | 20000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mixed-lineage-kinase-7_8ade20c058c32991163979fbe107d3bc.svg) | 1-Methyl-5-(2-pyridin-2-yl-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl)benzimidazole | IC50 | 20000.0 [1] |