![](https://images.aatbio.com/dataset/ic50/mitogen-activated-protein-kinase-kinase-kinase-kinase-2_b5f9e60dc2b2b7e76e07307c1d8f7888.svg) | Bosutinib | IC50 | 9.9 [1] |
![](https://images.aatbio.com/dataset/ic50/mitogen-activated-protein-kinase-kinase-kinase-kinase-2_b59db0701363c3c70952517bffcea5fd.svg) | Pluripotin | IC50 | 5.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mitogen-activated-protein-kinase-kinase-kinase-kinase-2_27d3a5b4d06517b7e7f7d0e79a2b07e5.svg) | CID 44219749 | IC50 | 50000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mitogen-activated-protein-kinase-kinase-kinase-kinase-2_11867fb79821176b92958b384e879689.svg) | CID 11478363 | IC50 | 8.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mitogen-activated-protein-kinase-kinase-kinase-kinase-2_836d58634120a742d63c1602f26addff.svg) | CID 59604787 | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mitogen-activated-protein-kinase-kinase-kinase-kinase-2_801b71b496c9e614d27c57f59ce0b9c5.svg) | (1S,2S,3R,4R)-3-[[5-Chloro-2-[[(7S)-4-methoxy-7-morpholin-4-yl-6,7,8,9-tetrahydro-5H-benzo[7]annulen-3-yl]amino]pyrimidin-4-yl]amino]bicyclo[2.2.1]hept-5-ene-2-carboxamide | IC50 | 60.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mitogen-activated-protein-kinase-kinase-kinase-kinase-2_8a081faabc28a2a6ff42b6477d7bcf26.svg) | N-[3-(7-Amino-1-methyl-2-oxo-4H-pyrimido[4,5-d]pyrimidin-3-yl)-4-methylphenyl]-3-(trifluoromethyl)benzamide | IC50 | 28.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mitogen-activated-protein-kinase-kinase-kinase-kinase-2_99d590530c99b53efc4907213bcd8b23.svg) | 7-Chloro-3-oxo-8-(1,3-thiazol-5-ylmethylamino)-11,16-dioxa-2,4,19,21-tetrazatricyclo[15.3.1.05,10]henicosa-1(20),5,7,9,17(21),18-hexaene-18-carbonitrile | Ki | 6516.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mitogen-activated-protein-kinase-kinase-kinase-kinase-2_21aa752395444707db3d7c65ae53dc35.svg) | 1-({4-[(3,4-Dichlorophenyl)methoxy]phenyl}methyl)azetidine-3-carboxylic acid | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mitogen-activated-protein-kinase-kinase-kinase-kinase-2_f64ae507fb96828f441cbfe1c221da9b.svg) | 1-[5-Amino-4-(3,4-dichlorophenyl)-3-methylpyrazol-1-yl]ethanone | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mitogen-activated-protein-kinase-kinase-kinase-kinase-2_f046ae8812a77e5cb35fd8b53bebf05d.svg) | Ripk1-IN-7 | IC50 | 387.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mitogen-activated-protein-kinase-kinase-kinase-kinase-2_b076cdaba7bb8b7d9a4e8120c86a34a8.svg) | N-Propyl-4-({4-[(2,2,2-trifluoroethyl)amino]-1H-pyrrolo[2,3-d]pyrimidin-2-yl}amino)benzamide | IC50 | 115.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mitogen-activated-protein-kinase-kinase-kinase-kinase-2_4d6874c80e57f5096b5a429fd0508716.svg) | N-(3-(2-(Pyridin-4-yl)pyrazolo[1,5-a]pyrimidin-7-yl)phenyl)-3-(trifluoromethyl)benzamide | IC50 | 50000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mitogen-activated-protein-kinase-kinase-kinase-kinase-2_420c640ab3d9d5b9acd6e7f999ac08f0.svg) | CID 27666048 | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mitogen-activated-protein-kinase-kinase-kinase-kinase-2_a7ee75d4a7ce2e8d7ffa73cb444c324f.svg) | 5-(2-Amino-[1,2,4]triazolo[1,5-a]pyridin-7-yl)-N-tert-butylpyridine-3-sulfonamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mitogen-activated-protein-kinase-kinase-kinase-kinase-2_a393d807e71b1e743502e2b63e78a618.svg) | 3-[7-[4-[(1S,4S)-5-Methyl-2,5-diazabicyclo[2.2.1]heptan-2-yl]phenyl]-2-pyridin-4-ylpyrazolo[1,5-a]pyrimidin-3-yl]phenol | IC50 | 4100.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mitogen-activated-protein-kinase-kinase-kinase-kinase-2_e92d8b13a8ce53f076211343eda30eb3.svg) | N-[3-(7-Anilino-1-methyl-2-oxo-4H-pyrimido[4,5-d]pyrimidin-3-yl)-4-methylphenyl]-3-(trifluoromethyl)benzamide | IC50 | 47.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mitogen-activated-protein-kinase-kinase-kinase-kinase-2_51153882d3ab9f3566d96aeaf5c3eeab.svg) | 6-(2,4-Difluorophenyl)sulfonyl-2-(1H-indol-5-ylamino)-8-methylpyrido[2,3-d]pyrimidin-7-one | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mitogen-activated-protein-kinase-kinase-kinase-kinase-2_ea5eb9d28ea73c1459251ec3ca29dbf2.svg) | 8-(4-Ethylphenyl)-5-Methyl-2,5-Dihydropyrazolo[4,3-C][2,1]benzothiazine 4,4-Dioxide | IC50 | 3000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mitogen-activated-protein-kinase-kinase-kinase-kinase-2_fb2996a255e5f9696d221b04a92bff1c.svg) | 1-Ethyl-8-(4-Ethylphenyl)-5-Methyl-1,5-Dihydropyrazolo[4,3-C][2,1]benzothiazine 4,4-Dioxide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mitogen-activated-protein-kinase-kinase-kinase-kinase-2_dd977b4ed27c8b0261f86e32605a6f69.svg) | N-[3-[7-(Cyclopropylamino)-1-methyl-2-oxo-4H-pyrimido[4,5-d]pyrimidin-3-yl]-4-methylphenyl]-3-(trifluoromethyl)benzamide | IC50 | 42.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mitogen-activated-protein-kinase-kinase-kinase-kinase-2_1c0473dfbc1be5975a9d2f806082e709.svg) | N-[3-[7-[4-(4-Ethylpiperazin-1-yl)anilino]-1-methyl-2-oxo-4H-pyrimido[4,5-d]pyrimidin-3-yl]-4-methylphenyl]-3-(trifluoromethyl)benzamide | IC50 | 8.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mitogen-activated-protein-kinase-kinase-kinase-kinase-2_fc35583a4d15434d654ab81810797660.svg) | N-[3-[7-(2-Hydroxyethylamino)-1-methyl-2-oxo-4H-pyrimido[4,5-d]pyrimidin-3-yl]-4-methylphenyl]-3-(trifluoromethyl)benzamide | IC50 | 33.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mitogen-activated-protein-kinase-kinase-kinase-kinase-2_6a93a96578de91b6a771fe3415fec659.svg) | N-[3-[7-[[6-(4-Ethylpiperazin-1-yl)pyridin-3-yl]amino]-1-methyl-2-oxo-4H-pyrimido[4,5-d]pyrimidin-3-yl]-4-methylphenyl]-3-(trifluoromethyl)benzamide | IC50 | 7.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mitogen-activated-protein-kinase-kinase-kinase-kinase-2_fe3fdfb9521ad25e272c3f4289b3aa44.svg) | N-[4-Methyl-3-[1-methyl-7-[(1-methylpyrazol-4-yl)amino]-2-oxo-4H-pyrimido[4,5-d]pyrimidin-3-yl]phenyl]-3-(trifluoromethyl)benzamide | IC50 | 6.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mitogen-activated-protein-kinase-kinase-kinase-kinase-2_b6aefd059d89e70e4183546bea05b913.svg) | N-[3-[7-[[6-(4-Acetylpiperazin-1-yl)pyridin-3-yl]amino]-1-methyl-2-oxo-4H-pyrimido[4,5-d]pyrimidin-3-yl]-4-methylphenyl]-3-(trifluoromethyl)benzamide | IC50 | 1.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mitogen-activated-protein-kinase-kinase-kinase-kinase-2_0b43927816ebbc9be13e6e44e4f9f2e1.svg) | 5,5-Dimethyl-8-[[4-(2,2,2-trifluoroethylamino)furo[3,2-d]pyrimidin-2-yl]amino]-1H-4,1-benzoxazepin-2-one | IC50 | 2940.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mitogen-activated-protein-kinase-kinase-kinase-kinase-2_ab3f0733db57234abb9178e327241b14.svg) | N-[4-Methyl-3-[1-methyl-7-[(6-methylpyridin-3-yl)amino]-2-oxo-4H-pyrimido[4,5-d]pyrimidin-3-yl]phenyl]-4-pyrrol-1-yl-3-(trifluoromethyl)benzamide | IC50 | 24.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mitogen-activated-protein-kinase-kinase-kinase-kinase-2_6f45287cd96a2a6915f488168e883a3b.svg) | 3-(4-Methylimidazol-1-yl)-N-[4-methyl-3-[1-methyl-7-[(6-methylpyridin-3-yl)amino]-2-oxo-4H-pyrimido[4,5-d]pyrimidin-3-yl]phenyl]-5-(trifluoromethyl)benzamide | IC50 | 27.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mitogen-activated-protein-kinase-kinase-kinase-kinase-2_0bd8059cc7ac34fdff7d305304570700.svg) | N-[4-Methyl-3-[1-methyl-7-[(6-methylpyridin-3-yl)amino]-2-oxo-4H-pyrimido[4,5-d]pyrimidin-3-yl]phenyl]-4-(4-methylpiperazin-1-yl)-3-(trifluoromethyl)benzamide | IC50 | 10.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mitogen-activated-protein-kinase-kinase-kinase-kinase-2_1a52c607c3ea6f31129932d9fd0c43bf.svg) | 4-Methyl-N-[4-methyl-3-[1-methyl-7-[(6-methylpyridin-3-yl)amino]-2-oxo-4H-pyrimido[4,5-d]pyrimidin-3-yl]phenyl]-3-(trifluoromethyl)benzamide | IC50 | 39.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mitogen-activated-protein-kinase-kinase-kinase-kinase-2_245f447aa1cfc6568210f125d5daac40.svg) | N-[3-[1-Cyclopropyl-7-[(6-methylpyridin-3-yl)amino]-2-oxo-4H-pyrimido[4,5-d]pyrimidin-3-yl]-4-methylphenyl]-4-methyl-3-(trifluoromethyl)benzamide | IC50 | 63.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mitogen-activated-protein-kinase-kinase-kinase-kinase-2_3963a48e53d00085a552a5b2d8ff74ed.svg) | N-[4-Methyl-3-[1-methyl-7-[(6-methylpyridin-3-yl)amino]-2-oxo-4H-pyrimido[4,5-d]pyrimidin-3-yl]phenyl]benzamide | IC50 | 1080.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mitogen-activated-protein-kinase-kinase-kinase-kinase-2_4608c420ce4fb27bfe024702c594ead6.svg) | 4-[[3-(Dimethylamino)pyrrolidin-1-yl]methyl]-N-[3-[7-[[6-(4-ethylpiperazine-1-carbonyl)pyridin-3-yl]amino]-1-methyl-2-oxo-4H-pyrimido[4,5-d]pyrimidin-3-yl]-4-methylphenyl]-3-(trifluoromethyl)benzamide | IC50 | 14.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mitogen-activated-protein-kinase-kinase-kinase-kinase-2_5c6d38e9097e7d907a1491edea2ef20e.svg) | 4-[[3-(Dimethylamino)pyrrolidin-1-yl]methyl]-N-[3-[7-[(2,5-dimethylpyrazol-3-yl)amino]-1-methyl-2-oxo-4H-pyrimido[4,5-d]pyrimidin-3-yl]-4-methylphenyl]-3-(trifluoromethyl)benzamide | IC50 | 17.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mitogen-activated-protein-kinase-kinase-kinase-kinase-2_1355f6586f7126183de765a5126e209d.svg) | N-[3-[1-Cyclohexyl-7-[(6-methylpyridin-3-yl)amino]-2-oxo-4H-pyrimido[4,5-d]pyrimidin-3-yl]-4-methylphenyl]-4-methyl-3-(trifluoromethyl)benzamide | IC50 | 497.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mitogen-activated-protein-kinase-kinase-kinase-kinase-2_7cf0db9f30313634b9e133b97ebf3773.svg) | N-[4-Methyl-3-[1-methyl-7-[(6-methylpyridin-3-yl)amino]-2-oxo-4H-pyrimido[4,5-d]pyrimidin-3-yl]phenyl]-3-morpholin-4-yl-5-(trifluoromethyl)benzamide | IC50 | 45.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mitogen-activated-protein-kinase-kinase-kinase-kinase-2_1522b6755814d34695c597c03fb92855.svg) | 4-Methyl-N-[4-methyl-3-[7-[(6-methylpyridin-3-yl)amino]-2-oxo-1-phenyl-4H-pyrimido[4,5-d]pyrimidin-3-yl]phenyl]-3-(trifluoromethyl)benzamide | IC50 | 55.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mitogen-activated-protein-kinase-kinase-kinase-kinase-2_34e2ce71e9fefb7c82804297ab9b560b.svg) | N-[3-[7-[[6-(4-Acetylpiperazin-1-yl)pyridin-3-yl]amino]-1-methyl-2-oxo-4H-pyrimido[4,5-d]pyrimidin-3-yl]-4-methylphenyl]-4-[[3-(dimethylamino)pyrrolidin-1-yl]methyl]-3-(trifluoromethyl)benzamide | IC50 | 16.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mitogen-activated-protein-kinase-kinase-kinase-kinase-2_8e87e0fea014032576294a35c192a858.svg) | 4-[[3-(Dimethylamino)pyrrolidin-1-yl]methyl]-N-[4-methyl-3-[1-methyl-7-[(1-methylpyrazol-4-yl)amino]-2-oxo-4H-pyrimido[4,5-d]pyrimidin-3-yl]phenyl]-3-(trifluoromethyl)benzamide | IC50 | 8.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mitogen-activated-protein-kinase-kinase-kinase-kinase-2_9b02df793e457742fc4383cf691c6acc.svg) | N-[3-[1-Ethyl-7-[(6-methylpyridin-3-yl)amino]-2-oxo-4H-pyrimido[4,5-d]pyrimidin-3-yl]-4-methylphenyl]-4-methyl-3-(trifluoromethyl)benzamide | IC50 | 34.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mitogen-activated-protein-kinase-kinase-kinase-kinase-2_b5a012eaa24b85e232df2fe5e6664f14.svg) | N-[4-Methyl-3-[1-methyl-7-[(6-methylpyridin-3-yl)amino]-2-oxo-4H-pyrimido[4,5-d]pyrimidin-3-yl]phenyl]-4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)benzamide | IC50 | 5.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mitogen-activated-protein-kinase-kinase-kinase-kinase-2_c0e90f0b8872a5501958dd1d2ea84b5d.svg) | 3-(4-Hydroxypiperidin-1-yl)-N-[4-methyl-3-[1-methyl-7-[(6-methylpyridin-3-yl)amino]-2-oxo-4H-pyrimido[4,5-d]pyrimidin-3-yl]phenyl]-5-(trifluoromethyl)benzamide | IC50 | 72.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mitogen-activated-protein-kinase-kinase-kinase-kinase-2_dbe6a9d05decfc89f8873c99512d77fd.svg) | N-[3-[7-[[6-(4-Ethylpiperazine-1-carbonyl)pyridin-3-yl]amino]-1-methyl-2-oxo-4H-pyrimido[4,5-d]pyrimidin-3-yl]-4-methylphenyl]-3-(trifluoromethyl)benzamide | IC50 | 2.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mitogen-activated-protein-kinase-kinase-kinase-kinase-2_ece372a475b481df4c84b5f8094d6669.svg) | N-[3-[1-Benzyl-7-[(6-methylpyridin-3-yl)amino]-2-oxo-4H-pyrimido[4,5-d]pyrimidin-3-yl]-4-methylphenyl]-4-methyl-3-(trifluoromethyl)benzamide | IC50 | 165.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mitogen-activated-protein-kinase-kinase-kinase-kinase-2_d71cca53ad28051b959b962997c464fe.svg) | 4-[[3-(Dimethylamino)pyrrolidin-1-yl]methyl]-N-[4-methyl-3-[1-methyl-7-[(6-methylpyridin-3-yl)amino]-2-oxo-4H-pyrimido[4,5-d]pyrimidin-3-yl]phenyl]-3-(trifluoromethyl)benzamide | IC50 | 2.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mitogen-activated-protein-kinase-kinase-kinase-kinase-2_fe36d92f25988fc0fb64ee4465475cb6.svg) | 5-[(E)-4-[(3R)-3-Aminopiperidin-1-yl]but-1-enyl]-4-[(4-methyl-1H-indol-5-yl)amino]pyridine-3-carbonitrile | IC50 | 2600.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mitogen-activated-protein-kinase-kinase-kinase-kinase-2_68e0b5867fb9bf360f7aed3ad8804faf.svg) | N-(2-Hydroxyethyl)-4-[3-[(Z)-(4-hydroxy-3-oxo-1-benzofuran-2-ylidene)methyl]-1-methylpyrrolo[2,3-b]pyridin-4-yl]benzamide | IC50 | 50000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mitogen-activated-protein-kinase-kinase-kinase-kinase-2_eb6227e6c3f665cde5788efe127c843a.svg) | Methyl 4-(6-(4-aminophenyl)-4-morpholino-1H-pyrazolo[3,4-d]pyrimidin-1-yl)piperidine-1-carboxylate | IC50 | 50000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mitogen-activated-protein-kinase-kinase-kinase-kinase-2_603383508252a1d5c473147ffda04752.svg) | Tert-butyl 4-[6-(4-aminophenyl)-4-morpholin-4-ylpyrazolo[3,4-d]pyrimidin-1-yl]piperidine-1-carboxylate | IC50 | 50000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mitogen-activated-protein-kinase-kinase-kinase-kinase-2_94e89e9705ce8e01fe931a014495c355.svg) | Atropisomer 1 | Ki | 340.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mitogen-activated-protein-kinase-kinase-kinase-kinase-2_793d8427574718310b36bfc2f5b0ef6e.svg) | 4-(4-Methyl-1H-indol-5-ylamino)-5-(3-(4-methylpiperazin-1-ylsulfonyl)styryl)nicotinonitrile | IC50 | 1300.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mitogen-activated-protein-kinase-kinase-kinase-kinase-2_e504da47f712ca636f26a8738cbed8f0.svg) | 6-Methyl-4-(4-methyl-1H-indol-5-ylamino)-5-(3-(4-methylpiperazin-1-ylsulfonyl)styryl)nicotinonitrile | IC50 | 50000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mitogen-activated-protein-kinase-kinase-kinase-kinase-2_856f48d6d8e8440f40e1ed1695d741b8.svg) | CID 46179972 | IC50 | 24.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mitogen-activated-protein-kinase-kinase-kinase-kinase-2_59c709e56f1adb4cd0a96f4865747914.svg) | 1-[4-[4-(3-Oxa-8-azabicyclo[3.2.1]octan-8-yl)-6-(oxan-4-yl)-1,3,5-triazin-2-yl]phenyl]-3-[4-(4-propan-2-ylpiperazine-1-carbonyl)phenyl]urea | IC50 | 50000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mitogen-activated-protein-kinase-kinase-kinase-kinase-2_14ffc8aab4232c3ddf73be9c15f0e03d.svg) | N-[3-[7-(Cyclohexylamino)-1-methyl-2-oxo-4H-pyrimido[4,5-d]pyrimidin-3-yl]-4-methylphenyl]-3-(trifluoromethyl)benzamide | IC50 | 925.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mitogen-activated-protein-kinase-kinase-kinase-kinase-2_6c34bcbf82f1b210364bfc6af4eddca3.svg) | 2-{3-[3-(Piperidin-4-Yl)propoxy]phenyl}-N-[4-(Pyridin-4-Yl)-1,3-Thiazol-2-Yl]acetamide | IC50 | 5000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mitogen-activated-protein-kinase-kinase-kinase-kinase-2_700247dab7b9fdcc2d81fe4984afa76c.svg) | 2-[3-(3-Piperazin-1-ylpropoxy)phenyl]-N-(4-pyridin-4-yl-1,3-thiazol-2-yl)acetamide | IC50 | 2500.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mitogen-activated-protein-kinase-kinase-kinase-kinase-2_f980e35cc5a89e33324ed62d29bf7e45.svg) | 2-N-(1H-Indazol-6-yl)-4-N-(2,2,2-trifluoroethyl)furo[3,2-d]pyrimidine-2,4-diamine | IC50 | 4760.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mitogen-activated-protein-kinase-kinase-kinase-kinase-2_ea7d68d5631badf4d76195468cfe148a.svg) | N~4~-Cyclopropyl-N~2~-(3-Methyl-1h-Indazol-6-Yl)furo[3,2-D]pyrimidine-2,4-Diamine | IC50 | 6240.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mitogen-activated-protein-kinase-kinase-kinase-kinase-2_f8ee55f6cac6bc1babf9b394bab747fe.svg) | 2-N-(3-Chloro-4-morpholin-4-ylphenyl)-4-N-(2,2,2-trifluoroethyl)furo[3,2-d]pyrimidine-2,4-diamine | IC50 | 1570.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mitogen-activated-protein-kinase-kinase-kinase-kinase-2_7001927caad7c36762b0d4d34597955f.svg) | (2R)-N-[5-(6-Aminopyridin-3-yl)-4-methyl-1,3-thiazol-2-yl]-4,4,4-trifluoro-2-methylbutanamide | IC50 | 9700.0 [1] |