Mitogen-activated protein kinase kinase kinase 7-interacting protein 1 Inhibitors (IC50, Ki)

Structure ▲ ▼	Compound Name ▲ ▼	Standard Type ▲ ▼	Standard Values (in nM) ▲ ▼
	Staurosporine	IC50	35.0 [1]
	(E)-3-(4-Phenylmethoxy-7H-pyrrolo[2,3-d]pyrimidin-5-yl)prop-2-enenitrile	IC50	330.0 [1]
	(E)-3-[4-(2-Methylpropoxy)-7H-pyrrolo[2,3-d]pyrimidin-5-yl]prop-2-enenitrile	IC50	210.0 [1]
	(E)-3-[4-(2-Methylpropoxy)-7H-pyrrolo[2,3-d]pyrimidin-5-yl]prop-2-enoic acid	IC50	340.0 [1]
	1-[4-(2-Methylpropoxy)-7H-pyrrolo[2,3-d]pyrimidin-5-yl]ethanone	IC50	1700.0 [1]
	(E)-N-[(2R)-2-Hydroxypropyl]-3-[4-(2-methylpropoxy)-7H-pyrrolo[2,3-d]pyrimidin-5-yl]prop-2-enamide	IC50	2500.0 [1]
	(E)-3-(4-Phenylmethoxy-7H-pyrrolo[2,3-d]pyrimidin-5-yl)prop-2-enamide	IC50	730.0 [1]
	(Z)-2-Fluoro-3-[4-(2-methylpropoxy)-7H-pyrrolo[2,3-d]pyrimidin-5-yl]prop-2-enamide	IC50	860.0 [1]
	(E)-N-(Cyclopropylmethyl)-3-[4-(2-methylpropoxy)-7H-pyrrolo[2,3-d]pyrimidin-5-yl]prop-2-enamide	IC50	380.0 [1]
	(E)-1-[4-(2-Methylpropoxy)-7H-pyrrolo[2,3-d]pyrimidin-5-yl]pent-1-en-3-one	IC50	200.0 [1]
	(Z)-2-Chloro-3-[4-(2-methylpropoxy)-7H-pyrrolo[2,3-d]pyrimidin-5-yl]prop-2-enamide	IC50	360.0 [1]
	Methyl (E)-3-[4-(2-methylpropoxy)-7H-pyrrolo[2,3-d]pyrimidin-5-yl]prop-2-enoate	IC50	200.0 [1]
	Methyl (E)-3-(4-phenylmethoxy-7H-pyrrolo[2,3-d]pyrimidin-5-yl)prop-2-enoate	IC50	350.0 [1]
	(E)-N-[(2S)-2-Hydroxypropyl]-3-[4-(2-methylpropoxy)-7H-pyrrolo[2,3-d]pyrimidin-5-yl]prop-2-enamide	IC50	2500.0 [1]
	Methyl (E)-2-methyl-3-[4-(2-methylpropoxy)-7H-pyrrolo[2,3-d]pyrimidin-5-yl]prop-2-enoate	IC50	430.0 [1]
	2-Chloro-1-[4-(2-methylpropoxy)-7H-pyrrolo[2,3-d]pyrimidin-5-yl]ethanone	IC50	280.0 [1]
	2-[4-(2-Methylpropoxy)-7H-pyrrolo[2,3-d]pyrimidin-5-yl]prop-2-enenitrile	IC50	750.0 [1]
	4-(2-Methylpropoxy)-7H-pyrrolo[2,3-d]pyrimidine-5-carbonitrile	IC50	560.0 [1]
	(E)-3-[4-(2-Methylpropoxy)-7H-pyrrolo[2,3-d]pyrimidin-5-yl]prop-2-enamide	IC50	3.1 [1]
	(E)-3-(4-Butan-2-yloxy-7H-pyrrolo[2,3-d]pyrimidin-5-yl)prop-2-enamide	IC50	4.3 [1]
	(E)-3-(4-Propan-2-yloxy-7H-pyrrolo[2,3-d]pyrimidin-5-yl)prop-2-enamide	IC50	4.4 [1]
	(E)-3-(4-Propoxy-7H-pyrrolo[2,3-d]pyrimidin-5-yl)prop-2-enamide	IC50	19.0 [1]
	(E)-3-[4-(2,2,2-Trifluoroethoxy)-7H-pyrrolo[2,3-d]pyrimidin-5-yl]prop-2-enamide	IC50	33.0 [1]
	(E)-3-[4-(2,2-Dimethylpropoxy)-7H-pyrrolo[2,3-d]pyrimidin-5-yl]prop-2-enamide	IC50	5.2 [1]
	(E)-3-[4-(4,4-Difluorocyclohexyl)oxy-7H-pyrrolo[2,3-d]pyrimidin-5-yl]prop-2-enamide	IC50	16.0 [1]
	(E)-N-Methyl-3-[4-(2-methylpropoxy)-7H-pyrrolo[2,3-d]pyrimidin-5-yl]prop-2-enamide	IC50	41.0 [1]
	(E)-N-Ethyl-3-[4-(2-methylpropoxy)-7H-pyrrolo[2,3-d]pyrimidin-5-yl]prop-2-enamide	IC50	340.0 [1]
	(E)-N-Cyclopropyl-3-[4-(2-methylpropoxy)-7H-pyrrolo[2,3-d]pyrimidin-5-yl]prop-2-enamide	IC50	180.0 [1]
	(E)-N,N-Dimethyl-3-[4-(2-methylpropoxy)-7H-pyrrolo[2,3-d]pyrimidin-5-yl]prop-2-enamide	IC50	97.0 [1]
	(Z)-3-[4-(2-Methylpropoxy)-7H-pyrrolo[2,3-d]pyrimidin-5-yl]prop-2-enenitrile	IC50	170.0 [1]
	(E)-4-[4-(2-Methylpropoxy)-7H-pyrrolo[2,3-d]pyrimidin-5-yl]but-3-en-2-one	IC50	100.0 [1]
	3-[4-(2-Methylpropoxy)-7H-pyrrolo[2,3-d]pyrimidin-5-yl]prop-2-ynamide	IC50	7.0 [1]
	(E)-3-(4-Phenoxy-7H-pyrrolo[2,3-d]pyrimidin-5-yl)prop-2-enamide	IC50	170.0 [1]
	(E)-3-[4-(2-Hydroxy-2-methylpropoxy)-7H-pyrrolo[2,3-d]pyrimidin-5-yl]prop-2-enamide	IC50	75.0 [1]
	(E)-3-[4-[(3-Fluorophenyl)methoxy]-7H-pyrrolo[2,3-d]pyrimidin-5-yl]prop-2-enamide	IC50	51.0 [1]
	(E)-3-[4-[(2-Methylpropan-2-yl)oxy]-7H-pyrrolo[2,3-d]pyrimidin-5-yl]prop-2-enamide	IC50	13.0 [1]
	(E)-4-[4-(2-Methylpropoxy)-7H-pyrrolo[2,3-d]pyrimidin-5-yl]but-2-enamide	IC50	420.0 [1]

Entire TableStructureCompound NameStandard TypeStandard Values (in nM)

Items per page: 510All1 - 10 of 37 ⟨⟩

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References

This online tool may be cited as follows

MLA	"Quest Database™ Mitogen-activated protein kinase kinase kinase 7-interacting protein 1 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 21 Dec. 2024, https://www.aatbio.com/data-sets/mitogen-activated-protein-kinase-kinase-kinase-7-interacting-protein-1-inhibitors-ic50-ki.
APA	AAT Bioquest, Inc. (2024, December 21). Quest Database™ Mitogen-activated protein kinase kinase kinase 7-interacting protein 1 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/mitogen-activated-protein-kinase-kinase-kinase-7-interacting-protein-1-inhibitors-ic50-ki.
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