![](https://images.aatbio.com/dataset/ic50/mitogen-activated-protein-kinase-kinase-kinase-10_308f46b4c40c812c872cfe130b3fc720.svg) | 3,9-Bis((ethylthio)methyl)-K-252a | IC50 | 2.0 [1], 51.0 [2] |
![](https://images.aatbio.com/dataset/ic50/mitogen-activated-protein-kinase-kinase-kinase-10_7a1d9fb4a82bc5ea68a5b57e2082aef5.svg) | K252a | IC50 | 45.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mitogen-activated-protein-kinase-kinase-kinase-10_7e037c210cad9a24b0c9ce116fb5b97c.svg) | CID 53469448 | IC50 | 452.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mitogen-activated-protein-kinase-kinase-kinase-10_4e8b5202a71aafe003ab207cc4576058.svg) | 3-(1H-Indol-5-yl)-5-(4-((4-methylpiperazin-1-yl)methyl)phenyl)-1H-pyrrolo[2,3-b]pyridine | IC50 | 42.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mitogen-activated-protein-kinase-kinase-kinase-10_d44bb541aaceb7d87194194110f1e1e1.svg) | CID 11634725 | Ki | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mitogen-activated-protein-kinase-kinase-kinase-10_8d08a07d2297c26adb17a3359934bc8c.svg) | CID 72547959 | IC50 | 767.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mitogen-activated-protein-kinase-kinase-kinase-10_9b77e0d646f6d1ac3a7ddedb939fdf94.svg) | 2-[[1-Cyclopentyl-5-[1-(Oxetan-3-Yl)piperidin-4-Yl]pyrazol-3-Yl]amino]pyridine-4-Carbonitrile | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mitogen-activated-protein-kinase-kinase-kinase-10_59f8e8493ac8cc4a8fa8d33eb818ed21.svg) | 3,13-Diazahexacyclo[14.7.0.02,10.04,9.011,15.017,22]tricosa-1(16),2(10),4,6,8,11(15),17,19,21-nonaen-12-one | IC50 | 2664.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mitogen-activated-protein-kinase-kinase-kinase-10_f046ae8812a77e5cb35fd8b53bebf05d.svg) | Ripk1-IN-7 | IC50 | 50.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mitogen-activated-protein-kinase-kinase-kinase-10_473049eaba0cda8ad169a5dcdf781925.svg) | 2-Methoxy-12-(2-hydroxyethyl)-13,14-dihydronaphthol[2,1-a]pyrrolo[3,4-c]carbazole-5-one | IC50 | 1582.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mitogen-activated-protein-kinase-kinase-kinase-10_51153882d3ab9f3566d96aeaf5c3eeab.svg) | 6-(2,4-Difluorophenyl)sulfonyl-2-(1H-indol-5-ylamino)-8-methylpyrido[2,3-d]pyrimidin-7-one | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mitogen-activated-protein-kinase-kinase-kinase-10_f5abe3234d4b41fad1784bb6b6683e98.svg) | 5-[1-(Cyclopropylmethyl)-5-[(1R,5S)-3-(oxetan-3-yl)-3-azabicyclo[3.1.0]hexan-6-yl]pyrazol-3-yl]-3-(trifluoromethyl)pyridin-2-amine | IC50 | 5150.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mitogen-activated-protein-kinase-kinase-kinase-10_ffb3f643c28315ae2654d18387c90755.svg) | 3,13-Diazahexacyclo[14.7.0.02,10.04,9.011,15.017,22]tricosa-1(16),2(10),4,6,8,11(15),17,19,21-nonaen-14-one | IC50 | 364.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mitogen-activated-protein-kinase-kinase-kinase-10_aaeb4e8768b7be5de894e0169a2f05d5.svg) | 2-Isopropoxy-12-(2-hydroxyethyl)-13,14-dihydronaphthol[2,1-a]pyrrolo[3,4-c]carbazole-5-one | IC50 | 1855.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mitogen-activated-protein-kinase-kinase-kinase-10_5aec4bb3eb103811bf187f792b18d464.svg) | Methyl (15S,16R,18R)-10,23-bis(butylsulfanylmethyl)-16-hydroxy-15-methyl-3-oxo-28-oxa-4,14,19-triazaoctacyclo[12.11.2.115,18.02,6.07,27.08,13.019,26.020,25]octacosa-1,6,8(13),9,11,20(25),21,23,26-nonaene-16-carboxylate | IC50 | 627.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mitogen-activated-protein-kinase-kinase-kinase-10_c65ea0d1878f60f6d493490cf5c589ae.svg) | Methyl (15S,16R,18R)-16-hydroxy-10,23-bis(methoxymethyl)-15-methyl-3-oxo-28-oxa-4,14,19-triazaoctacyclo[12.11.2.115,18.02,6.07,27.08,13.019,26.020,25]octacosa-1,6,8(13),9,11,20(25),21,23,26-nonaene-16-carboxylate | IC50 | 16.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mitogen-activated-protein-kinase-kinase-kinase-10_cb3bb7b1554677d919b57f20d8de29c3.svg) | Methyl (15S,16R,18R)-10,23-bis(ethoxymethyl)-16-hydroxy-15-methyl-3-oxo-28-oxa-4,14,19-triazaoctacyclo[12.11.2.115,18.02,6.07,27.08,13.019,26.020,25]octacosa-1,6,8(13),9,11,20(25),21,23,26-nonaene-16-carboxylate | IC50 | 20.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mitogen-activated-protein-kinase-kinase-kinase-10_0b43927816ebbc9be13e6e44e4f9f2e1.svg) | 5,5-Dimethyl-8-[[4-(2,2,2-trifluoroethylamino)furo[3,2-d]pyrimidin-2-yl]amino]-1H-4,1-benzoxazepin-2-one | IC50 | 4550.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mitogen-activated-protein-kinase-kinase-kinase-10_7b5c7e105f65c717f758d52b62cebcc3.svg) | 3-(2-Hydroxyethyl)-7-(propan-2-yloxymethyl)-3,13,23-triazahexacyclo[14.7.0.02,10.04,9.011,15.017,22]tricosa-1,4(9),5,7,10,15,17,19,21-nonaen-12-one | IC50 | 46.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mitogen-activated-protein-kinase-kinase-kinase-10_ce4a21853a3b06282a5b3d9a338a394d.svg) | 3,13-Diazahexacyclo[14.8.0.02,10.04,9.011,15.017,22]tetracosa-1(16),2(10),4,6,8,11(15),17,19,21-nonaen-12-one | IC50 | 3447.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mitogen-activated-protein-kinase-kinase-kinase-10_f9bf8fa4335782edad997ea9995f0ede.svg) | 3,13-Diazahexacyclo[14.8.0.02,10.04,9.011,15.017,22]tetracosa-1(16),2(10),4,6,8,11(15),17,19,21-nonaene-12,14-dione | IC50 | 339.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mitogen-activated-protein-kinase-kinase-kinase-10_570a23c02480e0f4f5b9482696944206.svg) | Methyl (15S,16R,18R)-10-(ethylsulfanylmethyl)-16-hydroxy-15-methyl-3-oxo-28-oxa-4,14,19-triazaoctacyclo[12.11.2.115,18.02,6.07,27.08,13.019,26.020,25]octacosa-1,6,8(13),9,11,20,22,24,26-nonaene-16-carboxylate | IC50 | 28.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mitogen-activated-protein-kinase-kinase-kinase-10_9c28dddff1b6f2d1e117b193b8ae13ce.svg) | Methyl (15S,16R,18R)-23-(ethylsulfanylmethyl)-16-hydroxy-15-methyl-3-oxo-28-oxa-4,14,19-triazaoctacyclo[12.11.2.115,18.02,6.07,27.08,13.019,26.020,25]octacosa-1,6,8,10,12,20(25),21,23,26-nonaene-16-carboxylate | IC50 | 140.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mitogen-activated-protein-kinase-kinase-kinase-10_6c34bcbf82f1b210364bfc6af4eddca3.svg) | 2-{3-[3-(Piperidin-4-Yl)propoxy]phenyl}-N-[4-(Pyridin-4-Yl)-1,3-Thiazol-2-Yl]acetamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mitogen-activated-protein-kinase-kinase-kinase-10_700247dab7b9fdcc2d81fe4984afa76c.svg) | 2-[3-(3-Piperazin-1-ylpropoxy)phenyl]-N-(4-pyridin-4-yl-1,3-thiazol-2-yl)acetamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mitogen-activated-protein-kinase-kinase-kinase-10_e23fa1bfdcc40f6f273a1efeafdbdbed.svg) | Dlk-IN-1 | IC50 | 7880.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mitogen-activated-protein-kinase-kinase-kinase-10_982eab592c51a6f88bce20abb8616513.svg) | 3-Thia-13,23-diazahexacyclo[14.7.0.02,10.04,9.011,15.017,22]tricosa-1,4,6,8,10,15,17,19,21-nonaen-12-one | IC50 | 2088.0 [1] |
![](https://images.aatbio.com/dataset/ic50/mitogen-activated-protein-kinase-kinase-kinase-10_9f7f20de4933fdf95496929588b27a3a.svg) | Methyl (15S,16R,18R)-16-hydroxy-15-methyl-3-oxo-10,23-bis(propan-2-ylsulfanylmethyl)-28-oxa-4,14,19-triazaoctacyclo[12.11.2.115,18.02,6.07,27.08,13.019,26.020,25]octacosa-1,6,8(13),9,11,20(25),21,23,26-nonaene-16-carboxylate | IC50 | 89.0 [1] |