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Methionine aminopeptidase 1 Inhibitors (IC50, Ki)

Structure
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▼
Compound Name
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▼
Standard Type
▲
▼
Standard Values (in nM)
▲
▼
8-HydroxyquinolineIC5012900.0 [1], 15000.0 [2], 21500.0 [3]
8-HydroxyquinaldineIC5015000.0 [1]
5-Chloro-8-hydroxyquinolineIC5012900.0 [1], 15000.0 [2]
Bengamide AIC50700.0 [1], 2000.0 [2]
Tert-Butyl {2-[(1,3-Thiazol-2-Ylamino)carbonyl]pyridin-3-Yl}carbamateIC50400.0 [1], 2000.0 [2]
ThiabendazoleIC5047800.0 [1]
NitroxolineIC5015000.0 [1]
8-Hydroxyquinoline-5-sulfonic acidIC5015000.0 [1]
2-(2-Pyridyl)benzimidazoleIC5028400.0 [1]
4-(p-Tolyl)-1H-1,2,3-triazoleIC507100.0 [1]
BenzoxiquineIC5042800.0 [1]
N-(1,3-Thiazol-2-yl)pyridine-2-carboxamideIC508100.0 [1]
8-(4-Benzenesulfonylamino)quinolineIC5044900.0 [1]
4,5-Dimethylaminobenzylidene-2-thiobarbituric acidKi100000.0 [1]
5-Benzylidenebarbituric acidKi162000.0 [1]
4,6(1H,5H)-Pyrimidinedione, dihydro-5-((4-methoxyphenyl)methylene)-2-thioxo-Ki100000.0 [1]
5-Chloro-6-methyl-N-(2-phenylethyl)-2-pyridin-2-ylpyrimidin-4-amineIC50860.0 [1]
5-Methyl-2-pyridin-2-yl-1H-benzoimidazoleIC5032600.0 [1]
2,4,6(1H,3H,5H)-Pyrimidinetrione, 5-[[4-(dimethylamino)phenyl]methylene]-Ki10000.0 [1]
[(3R,6S)-7-Oxo-6-[[(E,2R,3R,4S,5R)-3,4,5-trihydroxy-2-methoxy-8,8-dimethylnon-6-enoyl]amino]azepan-3-yl] cyclohexanecarboxylateIC50700.0 [1]
5-Nitro-2-(2-pyridinyl)-1H-benzimidazoleIC5028800.0 [1]
BARBITURIC ACID, 5-(p-METHOXYBENZYLIDENE)-Ki2000.0 [1]
N'-((2S,3R)-3-Amino-2-hydroxy-5-(isopropylsulfanyl)pentanoyl)-N-3-chlorobenzoyl hydrazideIC5056000.0 [1]
5-(4-Hydroxybenzylidene)pyrimidine-2,4,6(1H,3H,5H)-trioneKi10000.0 [1]
5-Benzylidene-2-thioxodihydropyrimidine-4,6(1h,5h)-dioneKi100000.0 [1]
(alpha-Aminobenzyl)phosphonic acidKi111600.0 [1]
1,3-Dimethyl-5-(phenylmethylidene)-1,3-diazinane-2,4,6-trioneKi100000.0 [1]
5-(4-Methoxybenzylidene)-1,3-dimethyl-2,4,6(1H,3H,5H)-pyrimidinetrioneKi100000.0 [1]
Quinolin-8-yl benzenesulfonateIC5041200.0 [1]
N'-(5-Chloro-6-methyl-2-pyridin-2-ylpyrimidin-4-yl)-N-[5-(trifluoromethyl)pyridin-2-yl]ethane-1,2-diamineIC502000.0 [1]
2-{4-[5-Chloro-6-Methyl-2-(Pyridin-2-Yl)pyrimidin-4-Yl]piperazin-1-Yl}ethanolIC501100.0 [1]
5-Chloro-N-[1-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]piperidin-4-yl]-6-methyl-2-pyridin-2-ylpyrimidin-4-amineIC50360.0 [1]
5-(4-Hydroxybenzylidene)-2-thioxodihydro-4,6(1H,5H)-pyrimidinedioneKi100000.0 [1]
5-(4-Hydroxybenzylidene)-1,3-dimethylpyrimidine-2,4,6(1H,3H,5H)-trioneKi100000.0 [1]
2-(Pyridin-2-yl)-3H-imidazo[4,5-b]pyridineIC5027600.0 [1]
1,3-Dimethyl-5-(3-phenyl-allylidene)-pyrimidine-2,4,6-trioneKi100000.0 [1]
5-Chloro-7-(morpholin-4-ylmethyl)quinolin-8-olIC5050000.0 [1]
5-Cinnamylidenebarbituric acidKi9000.0 [1]
2-(2-Pyridinyl)-1H-imidazo[4,5-c]pyridineIC5010300.0 [1]
1H-Benzimidazole, 6-methyl-2-(4-thiazolyl)-IC5035500.0 [1]
4-(5-Nitro-1H-benzo[d]imidazol-2-yl)thiazoleIC5048500.0 [1]
Phenyl-(2-thiazol-4-yl-1H-benzoimidazol-5-yl)-methanoneIC5041000.0 [1]
5-ChlorothiabendazoleIC5047000.0 [1]
1-Phosphono-3-cyclohexylpropylamineKi9900.0 [1]
4-(5,6-Dimethyl-1H-benzo[d]imidazol-2-yl)thiazoleIC5038800.0 [1]
5-Fluoro-2-(thiazol-4-yl)-1H-benzimidazoleIC5045800.0 [1]
2-(Thiazol-4-yl)-1H-imidazo[4,5-c]pyridineIC5019000.0 [1]
6-Chloro-2-(pyridin-2-yl)-1H-1,3-benzodiazoleIC5048800.0 [1]
(E,2R,3R,4S,5R)-N-(2-Amino-2-oxo-ethyl)-3,4,5-trihydroxy-2-methoxy-8,8-dimethyl-non-6-enamideIC503590.0 [1]
(E,2R,3R,4S,5R)-3,4,5-Trihydroxy-N-indan-2-yl-2-methoxy-8,8-dimethyl-non-6-enamideIC505580.0 [1]
n-MethylthiabendazoleIC5032400.0 [1]
5-Chloro-7-(piperidin-1-ylmethyl)quinolin-8-olIC5050000.0 [1]
2,3-Dihydro-5-(3-phenyl-2-propenylidene)-2-thioxo-4,6(1H,5H)-pyrimidinedioneKi98000.0 [1]
5-((4-(Dimethylamino)phenyl)methylene)-1,3-dimethylbarbituric acidKi100000.0 [1]
2-[2-Amino-4-(methylthio)butyryl]pyridineIC5016000.0 [1]
2-Amino-4-methylsulfanyl-1-(1,3-thiazol-2-yl)butan-1-oneIC5019000.0 [1]
5-Methoxy-2-methyleneindan-1-oneIC5030100.0 [1]
1H-Imidazo[4,5-b]pyrazine, 2-(2-pyridinyl)-IC5040100.0 [1]
2-(Pyridin-2-yl)-1H-1,3-benzodiazole-5-carbonitrileIC5037300.0 [1]
5,6-Dimethyl-2-(pyridin-2-yl)-1H-benzo[d]imidazoleIC5032600.0 [1]
5-Fluoro-2-(2-pyridyl)-1H-benzimidazoleIC5034700.0 [1]
9H-Purine, 8-(2-pyridinyl)-IC5033900.0 [1]
1-Phosphono-2-cyclohexylethanamineKi500000.0 [1]
N'-(5-Chloro-6-methyl-2-pyridin-2-ylpyrimidin-4-yl)-N-[6-(trifluoromethyl)pyridin-2-yl]ethane-1,2-diamineIC501000.0 [1]
N-Benzyl-5-chloro-6-methyl-2-pyridin-3-ylpyrimidin-4-amineIC50100000.0 [1]
4-Benzylsulfanyl-5-chloro-6-methyl-2-pyridin-2-ylpyrimidineIC5011000.0 [1]
N-Benzyl-5-chloro-N,6-dimethyl-2-pyridin-2-ylpyrimidin-4-amineIC501500.0 [1]
4-(2,4,6-Trioxohexahydropyrimidine-5-ylidenemethyl)benzoic acidKi5000.0 [1]
3-[(4-Tert-butylphenyl)methylsulfanyl]-1H-1,2,4-triazol-5-amineIC5015000.0 [1]
5-Chloro-7-[(4-methylpiperazinyl)methyl]quinolin-8-olIC5050000.0 [1]
6-Methyl-N-(2-phenylethyl)-2-pyridin-2-ylpyrimidin-4-amineIC50100000.0 [1]
1-Phosphono-2-methylpentylamineKi54800.0 [1]
(E,2R,3R,4S,5R)-N-[3-(Furan-2-yl)-3-phenylpropyl]-3,4,5-trihydroxy-2-methoxy-8,8-dimethylnon-6-enamideIC505140.0 [1]
3-Anilino-5-benzylthio-1,2,4-triazoleKi3900.0 [1]
[(3R,6S)-7-Oxo-6-[[(E,2R,3R,4S,5R)-3,4,5-trihydroxy-2-methoxy-6,8,8-trimethylnon-6-enoyl]amino]azepan-3-yl] cyclohexanecarboxylateIC5010000.0 [1]
3-Amino-1-(cyclopropylamino)heptan-2-oneIC507000.0 [1]
(2S)-2-Amino-N-hydroxy-N-[2-oxo-2-(2-pyridin-2-ylethylamino)ethyl]hexanamideKi33000.0 [1]
[(3S,6S)-7-Oxo-6-[[(E,2R,3R,4S,5R)-3,4,5-trihydroxy-2-methoxy-8-methylnon-6-enoyl]amino]azepan-3-yl] 12-methyltridecanoateIC503000.0 [1]
6-Methoxy-2-methylene-2,3-dihydro-1H-inden-1-oneIC5018800.0 [1]
5-Bromo-2-methyleneindan-1-oneIC503500.0 [1]
1-Phosphono-2-propylpentylamineKi4900.0 [1]
1-Naphthalenecarboxylic acid, 2-[(phenylsulfonyl)amino]-IC5047000.0 [1]
2-[(Dimethylamino)methyl]-6-methyl-2,3-dihydroinden-1-one;hydrochlorideIC5016200.0 [1]
2-[(Dimethylamino)methyl]-5-methoxy-2,3-dihydroinden-1-one;hydrochlorideIC5053700.0 [1]
5-Chloro-2-methylidene-3H-inden-1-oneIC501000.0 [1]
1,3-Dimethyl-5-[3-[4-(dimethylamino)phenyl]-2-propene-1-ylidene]pyrimidine-2,4,6(1H,3H,5H)-trioneKi100000.0 [1]
(S)-2-((R)-3-Amino-2-hydroxy-5-methylsulfanyl-pentanoylamino)-propionic acid ethyl esterIC5063000.0 [1]
(S)-2-((R)-3-Amino-2-hydroxy-heptanoylamino)-propionic acid ethyl esterIC50100000.0 [1]
2-((Dimethylamino)methyl)-2,3-dihydro-1H-inden-1-one hydrochlorideIC5023400.0 [1]
(S)-2-((R)-3-Amino-5-ethylsulfanyl-2-hydroxy-pentanoylamino)-propionic acid ethyl esterIC5069000.0 [1]
1,3-Dimethyl-5-(4-fluorobenzylidene)pyrimidine-2,4,6(1H,3H,5H)-trioneKi100000.0 [1]
4-(1,3-Dimethyl-2,4,6-trioxo-tetrahydro-pyrimidin-5-ylidenemethyl)-benzoic acidKi100000.0 [1]
1,3-Dimethyl-5-(4-nitrobenzylidene)pyrimidine-2,4,6(1H,3H,5H)-trioneKi100000.0 [1]
(2S,3S)-3-Amino-2-hydroxy-4-(2-methylpropylsulfanyl)-N-[(1S)-1-naphthalen-1-ylethyl]butanamideIC502200.0 [1]
(2S,3R)-3-Amino-2-hydroxy-N-[(1S)-1-naphthalen-1-ylethyl]-5-propan-2-ylsulfanylpentanamideIC5012000.0 [1]
N'-[(2S,3R)-3-Amino-5-ethylsulfanyl-2-hydroxypentanoyl]-3-chlorobenzohydrazideIC508700.0 [1]
N'-[(2S,3S)-3-Amino-2-hydroxy-4-(2-methylpropylsulfanyl)butanoyl]-3-chlorobenzohydrazideIC508100.0 [1]
5-(3-Nitro-benzylidene)-pyrimidine-2,4,6-trioneKi2000.0 [1]
5-Chloro-N,6-dimethyl-2-pyridin-2-ylpyrimidin-4-amineIC508900.0 [1]
1,3-Dimethyl-5-[(3-nitrophenyl)methylidene]-1,3-diazinane-2,4,6-trioneKi100000.0 [1]
Items per page: 1 - 10 of 100
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References

This online tool may be cited as follows

MLA

"Quest Database™ Methionine aminopeptidase 1 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 20 Feb. 2025, https://www.aatbio.com/data-sets/methionine-aminopeptidase-1-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2025, February 20). Quest Database™ Methionine aminopeptidase 1 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/methionine-aminopeptidase-1-inhibitors-ic50-ki.
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