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Membrane-bound transcription factor site-1 protease Inhibitors (IC50, Ki)

Structure
▲
▼
Compound Name
▲
▼
Standard Type
▲
▼
Standard Values (in nM)
▲
▼
(R)-4-((Diethylamino)methyl)-N-(2-methoxyphenethyl)-N-(pyrrolidin-3-yl)benzamideIC50170.0 [1]
CID 44433047IC508.0 [1]
N-(2-Chlorophenethyl)-4-isopropoxy-N-(pyrrolidin-3-yl)benzamideIC501400.0 [1]
N-(2-Fluorophenethyl)-4-isopropoxy-N-(pyrrolidin-3-yl)benzamideIC509000.0 [1]
N-(3-Chlorophenethyl)-4-isopropoxy-N-(pyrrolidin-3-yl)benzamideIC509600.0 [1]
N-(2-Methoxyphenethyl)-4-((diethylamino)methyl)-N-(pyrrolidin-3-yl)benzamideIC50540.0 [1]
N-(2-Methoxyphenethyl)-4-(benzyloxy)-N-(pyrrolidin-3-yl)benzamideIC50310.0 [1]
N-(2-Chlorophenethyl)-4-((diethylamino)methyl)-N-(pyrrolidin-3-yl)benzamideIC50840.0 [1]
N-(2-Chlorophenethyl)-4-(benzyloxy)-N-(pyrrolidin-3-yl)benzamideIC50590.0 [1]
N-(2-Chlorobenzyl)-4-isopropoxy-N-(pyrrolidin-3-yl)benzamideIC505000.0 [1]
N-(2,6-Dichlorophenethyl)-4-((diethylamino)methyl)-N-(pyrrolidin-3-yl)benzamideIC50430.0 [1]
N-(4-Chlorophenethyl)-4-((diethylamino)methyl)-N-(pyrrolidin-3-yl)benzamideIC503700.0 [1]
N-(3-Chlorophenethyl)-4-(benzyloxy)-N-(pyrrolidin-3-yl)benzamideIC50510.0 [1]
4-Diethylaminomethyl-N-pyrrolidin-3-yl-N-(2-o-tolyl-ethyl)-benzamideIC501600.0 [1]
N-(2-Ethoxyphenethyl)-4-((diethylamino)methyl)-N-(pyrrolidin-3-yl)benzamideIC5016000.0 [1]
N-(2-Chlorophenethyl)-4-isopropoxy-N-(1-methylpyrrolidin-3-yl)benzamideIC5030000.0 [1]
N-(2-Chlorophenethyl)-4-isopropoxy-N-(tetrahydrothiophen-3-yl)benzamideIC5030000.0 [1]
N-(2-Chlorophenethyl)-N-(1-formylpyrrolidin-3-yl)-4-isopropoxybenzamideIC5030000.0 [1]
N-(2-Chlorophenethyl)-4-isopropoxy-N-(piperidin-3-yl)benzamideIC5030000.0 [1]
N-(2-Chlorophenethyl)-N-(azetidin-3-yl)-4-isopropoxybenzamideIC5030000.0 [1]
N-(2-Chlorophenethyl)-4-(piperidin-1-ylmethyl)-N-(tetrahydrofuran-3-yl)benzamideIC5030000.0 [1]
N-[2-(2-Methoxyphenyl)ethyl]-4-[[3-(2-methylphenyl)piperidin-1-yl]methyl]-N-pyrrolidin-3-ylbenzamideIC5037.0 [1]
4-(6-Azabicyclo[3.2.1]octan-6-ylmethyl)-N-[2-(2-methoxyphenyl)ethyl]-N-pyrrolidin-3-ylbenzamideIC5029.0 [1]
4-(2-Azabicyclo[2.2.1]heptan-2-ylmethyl)-N-[2-(2-methoxyphenyl)ethyl]-N-pyrrolidin-3-ylbenzamideIC5095.0 [1]
4-[[[(1S,2S)-2-Hydroxycyclohexyl]amino]methyl]-N-[2-(2-methoxyphenyl)ethyl]-N-pyrrolidin-3-ylbenzamideIC50100.0 [1]
N-(2-Methoxyphenethyl)-4-(piperidin-1-ylmethyl)-N-(pyrrolidin-3-yl)benzamideIC50250.0 [1]
4-[[(2S)-2-(Methoxymethyl)pyrrolidin-1-yl]methyl]-N-[2-(2-methoxyphenyl)ethyl]-N-pyrrolidin-3-ylbenzamideIC50140.0 [1]
1-[[4-[2-(2-Methoxyphenyl)ethyl-pyrrolidin-3-ylcarbamoyl]phenyl]methyl]piperidine-3-carboxamideIC50160.0 [1]
(S)-N-(2-Methoxyphenethyl)-4-((diethylamino)methyl)-N-(pyrrolidin-3-yl)benzamideIC50970.0 [1]
Benzyl (2S)-3-methyl-2-[[2-[2-[[2-[2-[[(2S)-3-methyl-1-oxo-1-phenylmethoxybutan-2-yl]amino]-2-oxoethoxy]phenyl]diazenyl]phenoxy]acetyl]amino]butanoateKi125000.0 [1]
Benzyl (2S)-2-[[2-[2-[[2-[2-oxo-2-[[(2S)-1-oxo-3-phenyl-1-phenylmethoxypropan-2-yl]amino]ethoxy]phenyl]diazenyl]phenoxy]acetyl]amino]-3-phenylpropanoateKi11800.0 [1]
(2S)-2-[[2-[2-[[2-[2-[[(1S)-1-Carboxy-2-methylpropyl]amino]-2-oxoethoxy]phenyl]diazenyl]phenoxy]acetyl]amino]-3-methylbutanoic acidKi75000.0 [1]
(2S)-2-[[2-[2-[[2-[2-[[(1S)-1-Carboxy-2-phenylethyl]amino]-2-oxoethoxy]phenyl]diazenyl]phenoxy]acetyl]amino]-3-phenylpropanoic acidKi225000.0 [1]
2-[[2-[2-[[2-[2-(Carboxymethylamino)-2-oxoethoxy]phenyl]diazenyl]phenoxy]acetyl]amino]acetic acidKi265000.0 [1]
(2S)-2-[[(2S)-2-[[2-[2-[[2-[2-[[(2S)-1-[[(1S)-1-Carboxy-2-phenylethyl]amino]-1-oxo-3-phenylpropan-2-yl]amino]-2-oxoethoxy]phenyl]diazenyl]phenoxy]acetyl]amino]-3-phenylpropanoyl]amino]-3-phenylpropanoic acidKi140000.0 [1]
Items per page: 1 - 10 of 35
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References

This online tool may be cited as follows

MLA

"Quest Database™ Membrane-bound transcription factor site-1 protease Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 20 Feb. 2025, https://www.aatbio.com/data-sets/membrane-bound-transcription-factor-site-1-protease-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2025, February 20). Quest Database™ Membrane-bound transcription factor site-1 protease Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/membrane-bound-transcription-factor-site-1-protease-inhibitors-ic50-ki.
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