![](https://images.aatbio.com/dataset/ic50/melatonin-receptor-1a_f49643c3e5855473bdcde726c343e778.svg) | Melatonin | Ki | 0.08 [1], 0.12 [2], 0.29 [3], 0.3 [4] |
![](https://images.aatbio.com/dataset/ic50/melatonin-receptor-1a_c44948b090d42e84488f27346327bded.svg) | N-(2-(5-Methoxybenzofuran-3-yl)ethyl)acetamide | IC50 | 0.6 [1], 1.58 [2] |
![](https://images.aatbio.com/dataset/ic50/melatonin-receptor-1a_c44948b090d42e84488f27346327bded.svg) | N-(2-(5-Methoxybenzofuran-3-yl)ethyl)acetamide | Ki | 0.15 [1] |
![](https://images.aatbio.com/dataset/ic50/melatonin-receptor-1a_80443e492c1445fbac67782c8a98c48c.svg) | N-[2-[7-[4-[8-(2-Acetamidoethyl)naphthalen-2-yl]oxybutoxy]naphthalen-1-yl]ethyl]acetamide | Ki | 0.6 [1], 3.1 [2] |
![](https://images.aatbio.com/dataset/ic50/melatonin-receptor-1a_9496a94fd94151cd7dd45b2b66f6bc63.svg) | N-[2-[7-[3-[8-(2-Acetamidoethyl)naphthalen-2-yl]oxypropoxy]naphthalen-1-yl]ethyl]acetamide | Ki | 0.5 [1], 3.9 [2], 112.0 [3] |
![](https://images.aatbio.com/dataset/ic50/melatonin-receptor-1a_e9ee179bd352304e7e09277c926eb686.svg) | 2-Iodomelatonin | IC50 | 1.0 [1] |
![](https://images.aatbio.com/dataset/ic50/melatonin-receptor-1a_e9ee179bd352304e7e09277c926eb686.svg) | 2-Iodomelatonin | Ki | 0.01 [1], 0.07 [2], 0.08 [3] |
![](https://images.aatbio.com/dataset/ic50/melatonin-receptor-1a_ebddad8cbaf90b8707dba39c077b1b6f.svg) | N-[2-(11-Methoxy-6,7-dihydro-5H-indolo[2,1-a][2]benzazepin-13-yl)ethyl]butanamide | Ki | 66.0 [1], 66.07 [2], 66.1 [3] |
![](https://images.aatbio.com/dataset/ic50/melatonin-receptor-1a_b699463291e385894eb82c38012c8931.svg) | CID 10428383 | Ki | 1288.25 [1], 1290.0 [2] |
![](https://images.aatbio.com/dataset/ic50/melatonin-receptor-1a_95cdcac29414daffd65bda1cb8a19ed2.svg) | CID 9998187 | Ki | 27.0 [1], 40.6 [2], 40.74 [3] |
![](https://images.aatbio.com/dataset/ic50/melatonin-receptor-1a_556f47ad534a2f260eeb597263314e71.svg) | N-[2-(2-Benzyl-5-methoxy-benzofuran-3-yl)-ethyl]-acetamide | IC50 | 0.02 [1] |
![](https://images.aatbio.com/dataset/ic50/melatonin-receptor-1a_556f47ad534a2f260eeb597263314e71.svg) | N-[2-(2-Benzyl-5-methoxy-benzofuran-3-yl)-ethyl]-acetamide | Ki | 1.27 [1] |
![](https://images.aatbio.com/dataset/ic50/melatonin-receptor-1a_fc48dc2f850e64f709f105e31cf8bac5.svg) | N-[2-(7,17-Dimethoxy-3,13-diazapentacyclo[11.7.0.03,11.04,9.014,19]icosa-4(9),5,7,10,14(19),15,17-heptaen-10-yl)ethyl]acetamide | Ki | 1800.0 [1], 1819.7 [2] |
![](https://images.aatbio.com/dataset/ic50/melatonin-receptor-1a_d47a8902652d1e055746d1256a577b54.svg) | Luzindole | Ki | 158.0 [1], 603.0 [2], 794.33 [3] |
![](https://images.aatbio.com/dataset/ic50/melatonin-receptor-1a_1a521a61b28e17948e4df1af817ebcaa.svg) | 4-P-Pdot | Ki | 59.0 [1], 104.71 [2], 501.0 [3] |
![](https://images.aatbio.com/dataset/ic50/melatonin-receptor-1a_349223c5ae60001cd145d74a2c8dc564.svg) | N-[(6-Methoxy-9-tricyclo[9.4.0.03,8]pentadeca-1(15),3(8),4,6,11,13-hexaenyl)methyl]acetamide | Ki | 6.17 [1], 27.0 [2] |
![](https://images.aatbio.com/dataset/ic50/melatonin-receptor-1a_5a315ec46675d5cd7a4d100a3e7c74f5.svg) | 7-Azamelatonin | IC50 | 125.89 [1] |
![](https://images.aatbio.com/dataset/ic50/melatonin-receptor-1a_5a315ec46675d5cd7a4d100a3e7c74f5.svg) | 7-Azamelatonin | Ki | 40.0 [1] |
![](https://images.aatbio.com/dataset/ic50/melatonin-receptor-1a_dbba3ceccdb762369dbf147fb1358838.svg) | 4-Azamelatonin | Ki | 0.2 [1], 0.24 [2] |
![](https://images.aatbio.com/dataset/ic50/melatonin-receptor-1a_30defceefd6b9e817bbf0d8e86707e25.svg) | N-[2-(7-Methoxy-3,13-diazapentacyclo[11.7.0.03,11.04,9.014,19]icosa-4(9),5,7,10,14,16,18-heptaen-10-yl)ethyl]acetamide | Ki | 316.23 [1], 319.3 [2], 320.0 [3] |
![](https://images.aatbio.com/dataset/ic50/melatonin-receptor-1a_4d31b93323be749cf52ebf36aa299a7f.svg) | 1-[1-(2,2-Diphenyl-ethyl)-6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl]-ethanone | IC50 | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/melatonin-receptor-1a_4d31b93323be749cf52ebf36aa299a7f.svg) | 1-[1-(2,2-Diphenyl-ethyl)-6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl]-ethanone | Ki | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/melatonin-receptor-1a_df028b23d3c2fe96f0f83d086c1763be.svg) | N-[3-[5-Methoxy-2-[(3-methoxyphenyl)methoxy]phenyl]propyl]propanamide | Ki | 121.0 [1], 1348.96 [2], 1350.0 [3] |
![](https://images.aatbio.com/dataset/ic50/melatonin-receptor-1a_86b5f55acca53c45a6d9f892e86b7cdb.svg) | 5-Methoxycarbonylamino-N-acetyltryptamine | IC50 | 100.0 [1], 1000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/melatonin-receptor-1a_8a261a3c5ce63e37fbbb62c96223b18d.svg) | N-[2-(2-Methoxy-6H-isoindolo[2,1-a]indol-11-yl)ethyl]butanamide | Ki | 4.47 [1] |
![](https://images.aatbio.com/dataset/ic50/melatonin-receptor-1a_f0f0bbca2d0969168c6f792a42f847f6.svg) | N-[2-(5-Methoxy-1-methyl-1H-indol-3-yl)-ethyl]-acetamide | Ki | 2.24 [1], 2.6 [2] |
![](https://images.aatbio.com/dataset/ic50/melatonin-receptor-1a_d1eaaef40cea68213cae464b2407df58.svg) | N-[2-(2,7-Dimethoxy-naphthalen-1-yl)-ethyl]-propionamide | Ki | 0.1 [1] |
![](https://images.aatbio.com/dataset/ic50/melatonin-receptor-1a_2ec34fa4e2d5207a2e59a7a42f478905.svg) | N-[(6-Methoxy-9-tricyclo[9.4.0.03,8]pentadeca-1(15),3(8),4,6,11,13-hexaenyl)methyl]propanamide | Ki | 1.35 [1], 1.4 [2] |
![](https://images.aatbio.com/dataset/ic50/melatonin-receptor-1a_1ffd16e7440cc39f78035b07583cbce2.svg) | N-[(4-Methoxy-1H-indol-2-yl)methyl]propanamide | Ki | 407.38 [1] |
![](https://images.aatbio.com/dataset/ic50/melatonin-receptor-1a_0774f0fd96f4e294a582afd116ddce00.svg) | N-[2-(5-Methoxy-2-phenyl-benzofuran-3-yl)-ethyl]-acetamide | Ki | 0.01 [1] |
![](https://images.aatbio.com/dataset/ic50/melatonin-receptor-1a_6d1cdedd1118d4dda4ce9bd5f0fe8fc2.svg) | N-[2-[5-Methoxy-2-[(3-methoxyphenyl)methyl]-1-benzofuran-3-yl]ethyl]but-3-enamide | Ki | 21.6 [1] |
![](https://images.aatbio.com/dataset/ic50/melatonin-receptor-1a_75f32e4f6e8eca21b597270c4e564561.svg) | N-[2-(5-Methoxy-1H-indol-2-yl)ethyl]acetamide | Ki | 16218.1 [1] |
![](https://images.aatbio.com/dataset/ic50/melatonin-receptor-1a_ad6eddf95c691b5312959063f618d586.svg) | N-[(4-Methoxy-1H-indol-2-yl)methyl]cyclobutanecarboxamide | Ki | 524.81 [1] |
![](https://images.aatbio.com/dataset/ic50/melatonin-receptor-1a_4ee31e26436741227ac6544a5c2a0756.svg) | N-[(1-Benzyl-4-methoxyindol-2-yl)methyl]propanamide | Ki | 630.96 [1] |
![](https://images.aatbio.com/dataset/ic50/melatonin-receptor-1a_ea8037b742a38e25451579fb5be32f25.svg) | N-[2-(1-Benzyl-5-methoxyindol-3-yl)ethyl]acetamide | Ki | 141.25 [1] |
![](https://images.aatbio.com/dataset/ic50/melatonin-receptor-1a_3b8986d125f573a7c0cd24b4cc8fffe3.svg) | Acetylaminoethyl-methyl-phenylbutoxyphenyl-amine | Ki | 1.17 [1] |
![](https://images.aatbio.com/dataset/ic50/melatonin-receptor-1a_512d08cc96bf76fc99859e564a733c1d.svg) | Acetamide, N-[2-(1H-indol-2-yl)ethyl]- | Ki | 2454.71 [1] |
![](https://images.aatbio.com/dataset/ic50/melatonin-receptor-1a_43ab23e1c5ad6bce2422a27a70ca9173.svg) | N-[2-(4-Methoxy-1H-indol-2-yl)ethyl]acetamide | Ki | 630.96 [1] |
![](https://images.aatbio.com/dataset/ic50/melatonin-receptor-1a_9122c004554c3983f3d55b2435a19e87.svg) | N-[2-(4-Methoxy-1-phenylindol-2-yl)ethyl]acetamide | Ki | 87.1 [1] |
![](https://images.aatbio.com/dataset/ic50/melatonin-receptor-1a_585be5930729b4e60bb3bca71a1d45a6.svg) | N-[2-(4-Methoxy-1-phenylindol-2-yl)ethyl]propanamide | Ki | 63.1 [1] |
![](https://images.aatbio.com/dataset/ic50/melatonin-receptor-1a_04fb7af1d2e3e8c29611203ebb8eb1bc.svg) | N-[2-(6-Methoxy-1H-indol-2-yl)ethyl]acetamide | Ki | 8511.38 [1] |
![](https://images.aatbio.com/dataset/ic50/melatonin-receptor-1a_82ad15c0111aa36763e69b8b1ae39c5a.svg) | N-[2-(4-Methoxy-1H-indol-2-yl)ethyl]propanamide | Ki | 134.9 [1] |
![](https://images.aatbio.com/dataset/ic50/melatonin-receptor-1a_6017bca80bfaf4a2f8028f4ef83edc33.svg) | N-[2-(3-Bromo-6-methoxy-1H-indol-2-yl)ethyl]acetamide | Ki | 3981.07 [1] |
![](https://images.aatbio.com/dataset/ic50/melatonin-receptor-1a_6334e041e4e23a060001927549ef8d11.svg) | N-[2-(1-Benzyl-4-methoxyindol-2-yl)ethyl]propanamide | Ki | 831.76 [1] |
![](https://images.aatbio.com/dataset/ic50/melatonin-receptor-1a_482f80bb6625d89a8328165351064bf9.svg) | Acetamide, N-[(4-methoxy-1H-indol-2-yl)methyl]- | Ki | 1230.27 [1] |
![](https://images.aatbio.com/dataset/ic50/melatonin-receptor-1a_58daa3b8ba402b60855272f7b015e33e.svg) | N-[3-(5-Methoxy-1H-indol-2-yl)propyl]acetamide | Ki | 2951.21 [1] |
![](https://images.aatbio.com/dataset/ic50/melatonin-receptor-1a_c4db08218d060c5258c9ff1e6cd2b700.svg) | N-[2-(7-Methoxy-1H-indol-2-yl)ethyl]acetamide | Ki | 3801.89 [1] |
![](https://images.aatbio.com/dataset/ic50/melatonin-receptor-1a_cb65bbe210636b99be1e193240730075.svg) | N-[2-(6-Methoxy-1-methylindol-2-yl)ethyl]acetamide | Ki | 1819.7 [1] |
![](https://images.aatbio.com/dataset/ic50/melatonin-receptor-1a_d24c3a767379cdb1540e6418879f8bb5.svg) | N-(3-(3-Methoxyphenyl)-3-phenylallyl)acetamide | Ki | 2.69 [1], 230.0 [2] |
![](https://images.aatbio.com/dataset/ic50/melatonin-receptor-1a_ed6e2bd28d35993ac3558a07bc0ebcf0.svg) | N-[2-(3,13-Diazapentacyclo[11.7.0.03,11.04,9.014,19]icosa-4,6,8,10,14,16,18-heptaen-10-yl)ethyl]acetamide | Ki | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/melatonin-receptor-1a_1f8a9c473d0ec52ce0645f963e40be15.svg) | N-[2-(7-Phenyl-2,6-dihydro-1H-cyclopenta[e][1]benzofuran-8-yl)ethyl]acetamide | Ki | 0.01 [1] |
![](https://images.aatbio.com/dataset/ic50/melatonin-receptor-1a_4e9c4398d28bb5280da9515841cf9b68.svg) | N-[3-[2-(4-Phenylbutyl)-1,3-benzoxazol-7-yl]propyl]cyclopropanecarboxamide | Ki | 0.63 [1] |
![](https://images.aatbio.com/dataset/ic50/melatonin-receptor-1a_84a38459ff72dbcd22013154bb4527ea.svg) | 1-[6,7-Dimethoxy-1-(2-phenylethyl)-3,4-dihydro-1H-isoquinolin-2-yl]ethanone | IC50 | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/melatonin-receptor-1a_a60eb608d330657681ac64aa606c50fb.svg) | CID 44436051 | Ki | 7.24 [1], 40.74 [2] |
![](https://images.aatbio.com/dataset/ic50/melatonin-receptor-1a_8dbe32d1d9aad984f3609814e64b8c0b.svg) | N-(2-(6-Methoxy-1H-pyrrolo[2,3-b]pyridin-1-yl)ethyl)acetamide | Ki | 1.4 [1] |
![](https://images.aatbio.com/dataset/ic50/melatonin-receptor-1a_71dd6acaa1c7005d2165a82fc376b2f4.svg) | N-[2-[7-[8-(2-Acetamidoethyl)naphthalen-2-yl]naphthalen-1-yl]ethyl]acetamide | Ki | 5.2 [1] |
![](https://images.aatbio.com/dataset/ic50/melatonin-receptor-1a_6736fb21863be64fb2e01d8a5040a221.svg) | N-[2-(8-Methoxy-2-methyl-3,4-dihydro-1H-pyrazino[1,2-a]indol-10-yl)ethyl]butanamide | IC50 | 3.14 [1] |
![](https://images.aatbio.com/dataset/ic50/melatonin-receptor-1a_6736fb21863be64fb2e01d8a5040a221.svg) | N-[2-(8-Methoxy-2-methyl-3,4-dihydro-1H-pyrazino[1,2-a]indol-10-yl)ethyl]butanamide | Ki | 6.61 [1] |
![](https://images.aatbio.com/dataset/ic50/melatonin-receptor-1a_3bcf561ca5f81a0a2b20e27bbef03656.svg) | N-[3-Hydroxy-2-(7-methoxynaphthalen-1-yl)propyl]acetamide | IC50 | 19.95 [1] |
![](https://images.aatbio.com/dataset/ic50/melatonin-receptor-1a_3bcf561ca5f81a0a2b20e27bbef03656.svg) | N-[3-Hydroxy-2-(7-methoxynaphthalen-1-yl)propyl]acetamide | Ki | 10.96 [1] |
![](https://images.aatbio.com/dataset/ic50/melatonin-receptor-1a_8b6ab9141ce3fbe328ce44cde9cd3b14.svg) | N-[2-[5-(3-Phenoxypropoxy)-1H-indol-3-yl]ethyl]acetamide | Ki | 7.9 [1] |
![](https://images.aatbio.com/dataset/ic50/melatonin-receptor-1a_ae86a5a6e255bdd00ff343e5a64e75b7.svg) | N-[2-(6-Hexoxy-3,4-dihydro-2H-chromen-4-yl)ethyl]acetamide | Ki | 1.2 [1], 3.4 [2] |
![](https://images.aatbio.com/dataset/ic50/melatonin-receptor-1a_822b68838fffd6964517f5b8f84eafba.svg) | Dopamine | Ki | 7100.0 [1] |
![](https://images.aatbio.com/dataset/ic50/melatonin-receptor-1a_d18403d0f5d9853ddeee0383ca83ab4a.svg) | Serotonin | Ki | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/melatonin-receptor-1a_04e54d33c1a0ab3fa178d3a4be227b23.svg) | Ramelteon | Ki | 0.01 [1] |
![](https://images.aatbio.com/dataset/ic50/melatonin-receptor-1a_817c99ecd9284aad4f56c483d81e9768.svg) | N,N-Dimethyl-5-methoxytryptamine | Ki | 210.0 [1] |
![](https://images.aatbio.com/dataset/ic50/melatonin-receptor-1a_1aabafc80e3d3623452d58e846b702c7.svg) | Auraptene | Ki | 1900.0 [1] |
![](https://images.aatbio.com/dataset/ic50/melatonin-receptor-1a_098048eeb11ab3c84085ce36c084da30.svg) | 6-Chloromelatonin | Ki | 11.4 [1] |
![](https://images.aatbio.com/dataset/ic50/melatonin-receptor-1a_90fb2a3a66730e2f70a5255e06106c8e.svg) | 4-(4-Butylpiperidin-1-yl)-1-o-tolylbutan-1-one | Ki | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/melatonin-receptor-1a_86a887389e40a5334a3fd70722654349.svg) | 4-[[(E)-3,7-Dimethyl-2,6-octadienyl]oxy]-3-methoxycinnamic acid | Ki | 59000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/melatonin-receptor-1a_f6a025ec0ca3b8b08182a391fe09ed7e.svg) | 7-Prenyloxycoumarin | Ki | 5200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/melatonin-receptor-1a_c756ec9a7693a92edfb7586a38469d5f.svg) | 7-(Benzyloxy)-2H-chromen-2-one | Ki | 445.0 [1] |
![](https://images.aatbio.com/dataset/ic50/melatonin-receptor-1a_32005c8db107cbcf0ffd7d856a96acea.svg) | n-[(2r)-2-(6-Chloro-5-methoxy-1h-indol-3-yl)propyl]acetamide | Ki | 0.08 [1] |
![](https://images.aatbio.com/dataset/ic50/melatonin-receptor-1a_1b1100f95f7e05081468fe14121dbfa1.svg) | N-[2-(N-(4-Methoxyphenyl)anilino)ethyl]acetamide | Ki | 776.25 [1] |
![](https://images.aatbio.com/dataset/ic50/melatonin-receptor-1a_9a440f264f7f7a9d74b61c9a9ffdb8ca.svg) | CID 44208891 | Ki | 90.4 [1] |
![](https://images.aatbio.com/dataset/ic50/melatonin-receptor-1a_73919bad13f99f16d328ab9e60ce1bcd.svg) | 5-Methoxyluzindole | Ki | 32.7 [1] |
![](https://images.aatbio.com/dataset/ic50/melatonin-receptor-1a_4febcd17193d4fb3ad48309541eba599.svg) | N-Cyclopropylcarbonyl-2-(7-methoxy-1-naphthyl)ethylamine | IC50 | 1.26 [1] |
![](https://images.aatbio.com/dataset/ic50/melatonin-receptor-1a_fea97911fa84b15343dc6d5220a2180e.svg) | n-[2-(5,6-Dimethoxy-1h-indol-3-yl)ethyl]acetamide | Ki | 207.0 [1] |
![](https://images.aatbio.com/dataset/ic50/melatonin-receptor-1a_9d247348f9fa86863c920ac877d23134.svg) | N-(2,3-Dihydro-benzo[1,4]dioxin-2-ylmethyl)-acetamide | IC50 | 1995.26 [1] |
![](https://images.aatbio.com/dataset/ic50/melatonin-receptor-1a_30ae04f73fb83a21ca3b4763a49111d6.svg) | Propanamide, N-(2-(7-methoxy-1-naphthalenyl)ethyl)- | IC50 | 2.0 [1] |
![](https://images.aatbio.com/dataset/ic50/melatonin-receptor-1a_f4050af134925eaa4ffb394663110e32.svg) | N-[2-(2-Phenyl-1H-indol-3-yl)ethyl]cyclobutanecarboxamide | Ki | 199.53 [1] |
![](https://images.aatbio.com/dataset/ic50/melatonin-receptor-1a_c7597eb084d4cc7db53ad7a6d435536a.svg) | Acetamide,n-[2-(2-iodo-5-methoxy-1-methyl-4-nitro-1h-indol-3-yl)ethyl]- | Ki | 1880.0 [1] |
![](https://images.aatbio.com/dataset/ic50/melatonin-receptor-1a_45b57079108e1855cc01d784dd841461.svg) | N-[(1-Benzyl-5-methoxy-3,4-dihydro-2H-quinolin-2-yl)methyl]propanamide | Ki | 17.0 [1] |
![](https://images.aatbio.com/dataset/ic50/melatonin-receptor-1a_dbe9eaf8db3006fde0bcb4153f434d01.svg) | N-[2-(N-(3-Methoxyphenyl)anilino)ethyl]acetamide | Ki | 4.17 [1] |
![](https://images.aatbio.com/dataset/ic50/melatonin-receptor-1a_0bfe405be3ae87808a0923ee6484643e.svg) | Propanamide, N-(2-(7-methoxy-1-naphthalenyl)ethyl)-2-methyl- | IC50 | 2.51 [1] |
![](https://images.aatbio.com/dataset/ic50/melatonin-receptor-1a_110d3565d392ce0ee789548d93187df4.svg) | N-[1-[3-(3-Oxo-1,4-benzoxazin-4-yl)propyl]piperidin-4-yl]-2-phenylacetamide | Ki | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/melatonin-receptor-1a_10c3ccce5b1fc70a01b2919de4e88f9b.svg) | N-[2-(6-Fluoro-5-methoxy-1H-indol-3-yl)ethyl]cyclopropanecarboxamide | IC50 | 2.0 [1] |
![](https://images.aatbio.com/dataset/ic50/melatonin-receptor-1a_574d2484e852fa388faf7a13a1e16d1a.svg) | N-(3-(3-Methoxyphenyl)propyl)propionamide | Ki | 85.4 [1] |
![](https://images.aatbio.com/dataset/ic50/melatonin-receptor-1a_7b300bff0005026b9470e4b58d2b3d42.svg) | N-[3-(3-Methoxyphenyl)propyl]acetamide | Ki | 23.3 [1] |
![](https://images.aatbio.com/dataset/ic50/melatonin-receptor-1a_f92ac4dac3a704f759dbbd57f02a005a.svg) | N-[2-(5-Methoxy-1-methyl-4-nitro-1H-indol-3-yl)-ethyl]-acetamide | Ki | 8560.0 [1] |
![](https://images.aatbio.com/dataset/ic50/melatonin-receptor-1a_8010f814e357b625cb762e4a2ec34593.svg) | N-(2-Phenoxyethyl)Acetamide | Ki | 11481.54 [1] |
![](https://images.aatbio.com/dataset/ic50/melatonin-receptor-1a_fb9ec30c68ae0344ddc23fcdb29a5406.svg) | N-[2-(7-Methoxynaphthalen-1-yl)ethyl]hexanamide | IC50 | 1995.26 [1] |
![](https://images.aatbio.com/dataset/ic50/melatonin-receptor-1a_99ec266c80a3e7ce91ad6c2f608b4ecb.svg) | N-[2-(7-Methoxynaphthalen-1-yl)ethyl]heptanamide | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/melatonin-receptor-1a_260006abfbffb635ab0461c6f564362b.svg) | N-[2-[3-(3-Aminophenyl)-7-methoxynaphthalen-1-yl]ethyl]acetamide | Ki | 82.0 [1] |
![](https://images.aatbio.com/dataset/ic50/melatonin-receptor-1a_50c3e633563ffc5b62c5639377b89081.svg) | N-[2-(3-Methoxy-N-methylanilino)ethyl]acetamide | Ki | 0.81 [1] |
![](https://images.aatbio.com/dataset/ic50/melatonin-receptor-1a_4005a7a22b79d550c43063753781c1c9.svg) | Efppea | Ki | 0.06 [1] |
![](https://images.aatbio.com/dataset/ic50/melatonin-receptor-1a_e7028e7306e6787ccbd43a340033549d.svg) | N-(2-(7-Methoxynaphth-1-yl)ethyl)pyrrolidin-2-one | IC50 | 100.0 [1] |
![](https://images.aatbio.com/dataset/ic50/melatonin-receptor-1a_6c7f83adc683c35aed3c0c2cecb28733.svg) | 1H-Indole-2-carboxamide, N-(2-(7-methoxy-1-naphthalenyl)ethyl)- | IC50 | 2511.89 [1] |
![](https://images.aatbio.com/dataset/ic50/melatonin-receptor-1a_3c49351d89e5184b83fa1a493737e204.svg) | ACETAMIDE, N-(2-(5-METHOXYBENZO(b)THIEN-3-YL)ETHYL)- | IC50 | 1.26 [1] |