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Melanin-concentrating hormone receptor Inhibitors (IC50, Ki)

Structure
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▼
Compound Name
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Standard Type
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▼
Standard Values (in nM)
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▼
2-(4-(Benzyloxy)phenyl)-N-(1-(2-(pyrrolidin-1-yl)ethyl)-1H-indazol-6-yl)acetamideIC5011.0 [1]
7-Fluorochromone-2-carboxamideIC5029.0 [1]
6-Benzyloxymethyl-5-[4-(4-chloro-benzylamino)-phenyl]-pyrimidine-2,4-diamineIC5010000.0 [1]
N-(4-Phenoxyphenyl)-N'-[1-(2-pyrrolidin-1-ylethyl)-1H-indazol-5-yl]ureaIC50104.0 [1]
MCHr1 antagonist 2IC5025.0 [1]
N-(1-(4-Acetamidobenzyl)piperidin-4-yl)-7-fluoro-4-oxo-4H-chromene-2-carboxamideIC5010000.0 [1]
1-(2-{5-[3-(4-Phenoxy-phenyl)-ureido]-indazol-1-yl}-ethyl)-piperidine-4-carboxylic acid amideIC50171.0 [1]
1-(4-Phenoxy-benzyl)-3-[1-(2-pyrrolidin-1-yl-ethyl)-1H-indazol-6-yl]-ureaIC50626.0 [1]
1-[1-[2-[(2S)-2-(Methoxymethyl)pyrrolidin-1-yl]ethyl]indazol-5-yl]-3-(4-phenoxyphenyl)ureaIC50516.0 [1]
1-[2-(4-Phenoxyphenyl)ethyl]-3-[1-(2-pyrrolidin-1-ylethyl)indazol-6-yl]ureaIC50178.0 [1]
N-(1-((1H-Indol-6-yl)methyl)piperidin-4-yl)-7-fluoro-4-oxo-4H-chromene-2-carboxamideIC5066.0 [1]
N-(1-(Benzo[b]thiophen-5-ylmethyl)piperidin-4-yl)-7-fluoro-4-oxo-4H-chromene-2-carboxamideIC5057.0 [1]
1-(4-Benzyloxy-phenyl)-3-[1-(2-pyrrolidin-1-yl-ethyl)-1H-indazol-6-yl]-ureaIC507140.0 [1]
1-(4-Phenoxyphenyl)-3-[1-(2-pyrrolidin-1-ylethyl)-1H-indazol-5-yl]imidazolidin-2-oneIC501120.0 [1]
7-Fluoro-N-[1-[(1-methyl-2-oxoquinolin-7-yl)methyl]piperidin-4-yl]-4-oxochromene-2-carboxamideIC5044.0 [1]
7-Fluoro-4-oxo-N-(1-((2-oxo-2H-chromen-7-yl)methyl)piperidin-4-yl)-4H-chromene-2-carboxamideIC5046.0 [1]
N-(1-((1H-Indol-5-yl)methyl)piperidin-4-yl)-7-fluoro-4-oxo-4H-chromene-2-carboxamideIC50110.0 [1]
1-(4-Phenoxy-phenyl)-3-[1-(2-pyrrolidin-1-yl-ethyl)-1H-indazol-5-yl]-1,3-dihydro-imidazol-2-oneIC50654.0 [1]
N-(1-(Benzo[d]oxazol-6-ylmethyl)piperidin-4-yl)-7-fluoro-4-oxo-4H-chromene-2-carboxamideIC50106.0 [1]
N-[1-(6-Acetamido-2,3-dihydro-1H-inden-1-yl)piperidin-4-yl]-7-fluoro-4-oxochromene-2-carboxamideIC5010000.0 [1]
N-(1-(Benzofuran-5-ylmethyl)piperidin-4-yl)-7-fluoro-4-oxo-4H-chromene-2-carboxamideIC5035.0 [1]
7-Fluoro-4-oxo-N-[1-[(2-oxo-1H-quinolin-7-yl)methyl]piperidin-4-yl]chromene-2-carboxamideIC50162.0 [1]
N-[1-(6,7-Dihydro-5H-cyclopenta[f][1,3]benzodioxol-7-yl)piperidin-4-yl]-6-fluoro-4-oxochromene-2-carboxamideIC5010000.0 [1]
1-[1-[3-(Cyclopentylamino)propyl]indazol-5-yl]-3-(4-phenoxyphenyl)ureaIC50275.0 [1]
1-[3-[5-[(4-Phenoxyphenyl)carbamoylamino]indazol-1-yl]propyl]piperidine-4-carboxamideIC502880.0 [1]
1-[1-[2-(4-Hydroxypiperidin-1-yl)ethyl]indazol-5-yl]-3-(4-phenoxyphenyl)ureaIC5010000.0 [1]
1-[2-(4-Phenoxyphenyl)ethyl]-3-[1-(2-pyrrolidin-1-ylethyl)indazol-5-yl]ureaIC5010000.0 [1]
1-(4-Phenoxyphenyl)-3-[1-(2-pyrrolidin-1-ylethyl)indazol-4-yl]ureaIC5010000.0 [1]
1-(4-Phenoxyphenyl)-3-[1-(2-pyrrolidin-1-ylethyl)indazol-6-yl]ureaIC5010000.0 [1]
1-(4-Phenylmethoxyphenyl)-3-[1-(2-pyrrolidin-1-ylethyl)indazol-5-yl]ureaIC5010000.0 [1]
1-[1-[3-[(2S)-2-(Methoxymethyl)pyrrolidin-1-yl]propyl]indazol-5-yl]-3-(4-phenoxyphenyl)ureaIC501177.0 [1]
1-(4-Phenylmethoxyphenyl)-3-[1-(2-pyrrolidin-1-ylethyl)indazol-4-yl]ureaIC5010000.0 [1]
1-[(4-Phenoxyphenyl)methyl]-3-[1-(2-pyrrolidin-1-ylethyl)indazol-5-yl]ureaIC5010000.0 [1]
1-[1-[2-(2-Methylpropylamino)ethyl]indazol-5-yl]-3-(4-phenoxyphenyl)ureaIC50751.0 [1]
1-[1-[3-(4-Hydroxypiperidin-1-yl)propyl]indazol-5-yl]-3-(4-phenoxyphenyl)ureaIC50894.0 [1]
1-[1-[2-(3,3-Difluoropyrrolidin-1-yl)ethyl]indazol-5-yl]-3-(4-phenoxyphenyl)ureaIC5010000.0 [1]
1-(1-Benzylpiperidin-4-yl)-3-[1-(2-pyrrolidin-1-ylethyl)indazol-6-yl]ureaIC5010000.0 [1]
1-(1-Benzylpiperidin-4-yl)-3-[1-(2-pyrrolidin-1-ylethyl)indazol-5-yl]ureaIC5010000.0 [1]
1-[1-[2-(Cyclopentylamino)ethyl]indazol-5-yl]-3-(4-phenoxyphenyl)ureaIC50147.0 [1]
2-[(4-Phenoxyphenyl)methylamino]-N-[1-(2-pyrrolidin-1-ylethyl)indol-6-yl]acetamideIC501810.0 [1]
N-[1-(7,8-Dihydro-6H-cyclopenta[g][1,3]benzodioxol-6-yl)piperidin-4-yl]-6-fluoro-4-oxochromene-2-carboxamideIC502750.0 [1]
7-Fluoro-4-oxo-N-[1-(2-oxo-3,5,6,7-tetrahydrocyclopenta[f][1,3]benzoxazol-5-yl)piperidin-4-yl]chromene-2-carboxamideIC50173.0 [1]
7-Fluoro-4-oxo-N-[1-(3-oxo-4,6,7,8-tetrahydrocyclopenta[g][1,4]benzoxazin-6-yl)piperidin-4-yl]chromene-2-carboxamideIC5095.0 [1]
N-[1-[(2-Ethyl-1,3-benzoxazol-6-yl)methyl]piperidin-4-yl]-7-fluoro-4-oxochromene-2-carboxamideIC5010000.0 [1]
N-[1-[(2-Ethyl-1,3-benzoxazol-5-yl)methyl]piperidin-4-yl]-7-fluoro-4-oxochromene-2-carboxamideIC501380.0 [1]
7-Fluoro-4-oxo-N-[1-[(2-oxo-3H-1,3-benzoxazol-5-yl)methyl]piperidin-4-yl]chromene-2-carboxamideIC50569.0 [1]
7-Fluoro-4-oxo-N-[1-[(2-oxo-1,3-benzodioxol-5-yl)methyl]piperidin-4-yl]chromene-2-carboxamideIC505590.0 [1]
7-Fluoro-4-oxo-N-[1-[(3-oxo-4H-1,4-benzoxazin-7-yl)methyl]piperidin-4-yl]chromene-2-carboxamideIC502410.0 [1]
N-[1-[(3-Acetamidophenyl)methyl]piperidin-4-yl]-7-fluoro-4-oxochromene-2-carboxamideIC50551.0 [1]
7-Fluoro-4-oxo-N-[1-[(3-oxo-4H-1,4-benzoxazin-6-yl)methyl]piperidin-4-yl]chromene-2-carboxamideIC50233.0 [1]
Items per page: 1 - 10 of 50
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References

This online tool may be cited as follows

MLA

"Quest Database™ Melanin-concentrating hormone receptor Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 21 Dec. 2024, https://www.aatbio.com/data-sets/melanin-concentrating-hormone-receptor-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, December 21). Quest Database™ Melanin-concentrating hormone receptor Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/melanin-concentrating-hormone-receptor-inhibitors-ic50-ki.
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