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Mas-related G-protein coupled receptor member X1 Inhibitors (IC50, Ki)

Structure
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Compound Name
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Standard Type
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▼
Standard Values (in nM)
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▼
2-[2-(Diphenylmethyl)-1-azabicyclo[2.2.2]oct-3-ylidene]-1-(2-methoxyphenyl)-ethanoneIC5050.0 [1], 320.0 [2], 800.0 [3]
2-[4-[2-[2-(4-Chlorophenyl)ethylamino]pyrimidin-4-yl]piperazin-1-yl]-N-[(3,5-dichloropyridin-4-yl)methyl]-N-(3-morpholin-4-ylpropyl)acetamideIC5014.0 [1], 50.0 [2]
4-(2-Benzhydryl-1-aza-bicyclo[2.2.2]oct-3-yloxymethyl)-benzonitrileIC50556.0 [1], 1850.0 [2]
[(3R)-2-Benzhydryl-1-azabicyclo[2.2.2]octan-3-yl] N-(3-nitrophenyl)carbamateIC50290.0 [1], 1850.0 [2]
[(3S)-2-Benzhydryl-1-azabicyclo[2.2.2]octan-3-yl] N-(2-chlorophenyl)carbamateIC50375.0 [1], 1180.0 [2]
(3E)-2-Benzhydryl-3-(2-phenylethylidene)-1-azabicyclo[2.2.2]octaneIC50163.0 [1], 1430.0 [2]
[(3R)-2-Benzhydryl-1-azabicyclo[2.2.2]octan-3-yl] N-(2-chlorophenyl)carbamateIC50140.0 [1], 607.0 [2]
(2E)-2-(2-Benzhydryl-1-azabicyclo[2.2.2]octan-3-ylidene)-1-(4-fluorophenyl)ethanolIC50165.0 [1], 630.0 [2]
[(3R)-2-Benzhydryl-1-azabicyclo[2.2.2]octan-3-yl] N-naphthalen-1-ylcarbamateIC50124.0 [1], 1220.0 [2]
1-[(3R)-2-Benzhydryl-1-azabicyclo[2.2.2]octan-3-yl]-3-(2-methoxyphenyl)thioureaIC50418.0 [1], 2510.0 [2]
(2E)-2-(2-Benzhydryl-1-azabicyclo[2.2.2]octan-3-ylidene)-1-(2-methoxyphenyl)ethanolIC5080.0 [1], 182.0 [2]
[(3R)-2-Benzhydryl-1-azabicyclo[2.2.2]octan-3-yl] 2-(trifluoromethyl)benzoateIC50252.0 [1], 2400.0 [2]
(3R)-2-Benzhydryl-N-[[2-(trifluoromethyl)phenyl]methyl]-1-azabicyclo[2.2.2]octan-3-amineIC50244.0 [1], 1290.0 [2]
N-[2-(4-Chlorophenyl)ethyl]-4-pyrrolidin-1-ylquinazolin-2-amineIC508060.0 [1]
2-[4-[2-[2-(4-Chlorophenyl)ethylamino]pyrimidin-4-yl]piperazin-1-yl]-N-(oxolan-2-ylmethyl)-N-(pyridin-4-ylmethyl)acetamideIC5040.0 [1]
2-[4-[2-[2-(4-Chlorophenyl)ethylamino]pyrimidin-4-yl]piperazin-1-yl]-N-(3-methoxypropyl)-N-(pyridin-4-ylmethyl)acetamideIC5088.0 [1]
2-[4-[2-[2-(4-Chlorophenyl)ethylamino]pyrimidin-4-yl]piperazin-1-yl]-N-[(3,5-dichloropyridin-4-yl)methyl]-N-(pyridin-4-ylmethyl)acetamideIC5024.0 [1]
2-[4-[2-[2-(4-Chlorophenyl)ethylamino]pyrimidin-4-yl]piperazin-1-yl]-N-(cyclopropylmethyl)-N-(pyridin-4-ylmethyl)acetamideIC50295.0 [1]
N-[(3-Bromopyridin-4-yl)methyl]-2-[4-[2-[2-(4-chlorophenyl)ethylamino]pyrimidin-4-yl]piperazin-1-yl]-N-ethylacetamideIC50108.0 [1]
4-(2-(2-(4-Chlorophenethylamino)quinazolin-4-ylamino)ethyl)benzenesulfonamideIC50640.0 [1]
4-(2-(2-(4-Chlorophenethylamino)pyrimidin-4-ylamino)ethyl)benzenesulfonamideIC50301.0 [1]
2-[4-[2-[2-(4-Chlorophenyl)ethylamino]pyrimidin-4-yl]piperazin-1-yl]-1-piperidin-1-ylethanoneIC50758.0 [1]
2-[4-[2-[2-(4-Chlorophenyl)ethylamino]pyrimidin-4-yl]piperazin-1-yl]-N-(furan-2-ylmethyl)-N-(pyridin-4-ylmethyl)acetamideIC5020.0 [1]
N-Benzyl-2-[4-[2-[2-(4-chlorophenyl)ethylamino]pyrimidin-4-yl]piperazin-1-yl]-N-(pyridin-4-ylmethyl)acetamideIC5022.0 [1]
2-[4-[2-[2-(4-Chlorophenyl)ethylamino]pyrimidin-4-yl]piperazin-1-yl]-N-ethyl-N-(pyridin-4-ylmethyl)acetamideIC50244.0 [1]
1-[2-[2-(4-Chlorophenyl)ethylamino]-4-pyrrolidin-1-ylquinazolin-6-yl]sulfonyl-N-[1-(dimethylamino)propan-2-yl]piperidine-4-carboxamideIC50530.0 [1]
N-Benzyl-2-[4-[2-[2-(4-chlorophenyl)ethylamino]pyrimidin-4-yl]piperazin-1-yl]-N-ethylacetamideIC50330.0 [1]
2-[4-[2-[2-(4-Chlorophenyl)ethylamino]pyrimidin-4-yl]piperazin-1-yl]-N-[(3,5-dichloropyridin-4-yl)methyl]-N-ethylacetamideIC5077.0 [1]
(2E)-2-(2-Benzhydryl-1-azabicyclo[2.2.2]octan-3-ylidene)-1-[3-(trifluoromethyl)phenyl]ethanolIC5090.0 [1]
[(3S)-2-Benzhydryl-1-azabicyclo[2.2.2]octan-3-yl] 3,4-dimethoxybenzoateIC5064.0 [1]
(2E)-2-(2-Benzhydryl-1-azabicyclo[2.2.2]octan-3-ylidene)-1-(3,5-dimethylphenyl)ethanolIC50200.0 [1]
3-[[(3R)-2-Benzhydryl-1-azabicyclo[2.2.2]octan-3-yl]oxymethyl]benzonitrileIC50209.0 [1]
Items per page: 1 - 10 of 32
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References

This online tool may be cited as follows

MLA

"Quest Database™ Mas-related G-protein coupled receptor member X1 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 22 Feb. 2025, https://www.aatbio.com/data-sets/mas-related-g-protein-coupled-receptor-member-x1-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2025, February 22). Quest Database™ Mas-related G-protein coupled receptor member X1 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/mas-related-g-protein-coupled-receptor-member-x1-inhibitors-ic50-ki.
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