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MAP kinase p38 delta Inhibitors (IC50, Ki)

Structure
▲
▼
Compound Name
▲
▼
Standard Type
▲
▼
Standard Values (in nM)
▲
▼
DoramapimodIC50300.0 [1], 1968.0 [2]
4-(4-Fluorophenyl)-2-(4-methylsulfinylphenyl)-5-(4-pyridyl)-1H-imidazoleIC5087600000.0 [1]
TofacitinibIC5010000.0 [1]
Cyclohexanol, 4-(4-(4-fluorophenyl)-5-(2-methoxy-4-pyrimidinyl)-1H-imidazol-1-yl)-, trans-IC50100000.0 [1]
Benzamide, N-[4-[2-ethyl-4-(3-methylphenyl)-5-thiazolyl]-2-pyridinyl]-IC5010000.0 [1]
JNK Inhibitor VIIIKi6900.0 [1]
6-[(6R)-2-(4-Fluorophenyl)-6-(hydroxymethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-3-yl]-2-(2-methylphenyl)pyridazin-3-oneIC5011.0 [1]
Amg-548IC507736.0 [1]
3-(3-Tert-butyl-6,8-difluoro-[1,2,4]triazolo[4,3-a]pyridin-7-yl)-N-cyclopropyl-5-fluoro-4-methylbenzamideIC506.2 [1]
N-[2-Methyl-5-(methylcarbamoyl)phenyl]-2-{[(1R)-1-methylpropyl]amino}-1,3-thiazole-5-carboxamideIC5030000.0 [1]
N-(4-Amino-5-cyano-6-ethoxypyridin-2-yl)acetamideKi6900.0 [1]
4-Amino-5-chloro-6-ethoxy-pyridine-2-carboxylic acid 4-methanesulfonyl-benzylamideKi6800.0 [1]
7-Chloro-3-oxo-8-(1,3-thiazol-5-ylmethylamino)-11,16-dioxa-2,4,19,21-tetrazatricyclo[15.3.1.05,10]henicosa-1(20),5,7,9,17(21),18-hexaene-18-carbonitrileKi6812.0 [1]
1-({4-[(3,4-Dichlorophenyl)methoxy]phenyl}methyl)azetidine-3-carboxylic acidIC5010000.0 [1]
6-Acetyl-8-cyclopentyl-5-methyl-2-(4-piperazin-1-yl-phenylamino)-8H-pyrido[2,3-d]pyrimidin-7-oneIC5010000.0 [1]
Khk-IN-1IC5040000.0 [1]
3-[[5-Cyano-6-(cyclopentylamino)pyrimidin-4-yl]amino]-4-methyl-N-(1,2-oxazol-3-yl)benzamideIC5030000.0 [1]
7-Chloro-8-(3-hydroxypropoxy)-3-oxo-11,17-dioxa-2,4,20,22-tetrazatricyclo[16.3.1.05,10]docosa-1(21),5,7,9,18(22),19-hexaene-19-carbonitrileKi10000.0 [1]
7-Chloro-8-(3-hydroxypropyl)-3-oxo-11,17-dioxa-2,4,20,22-tetrazatricyclo[16.3.1.05,10]docosa-1(21),5(10),6,8,18(22),19-hexaene-19-carbonitrileKi10000.0 [1]
N-(7-Chloro-19-cyano-3-oxo-11,17-dioxa-2,4,20,22-tetrazatricyclo[16.3.1.05,10]docosa-1(21),5,7,9,18(22),19-hexaen-8-yl)methanesulfonamideKi10000.0 [1]
N-(4-Amino-5-cyano-6-ethoxypyridin-2-yl)-2-(2,5-dimethoxy-4-methylsulfonylphenyl)acetamideKi6900.0 [1]
N-(4-Amino-5-chloro-6-ethoxypyridin-2-yl)-2-(4-methanesulfonyl-2,5-dimethoxyphenyl)acetamideKi6900.0 [1]
N-(4-Amino-5-cyano-6-isopropoxypyridin-2-yl)-2-(4-methanesulfonyl-2,5-dimethoxyphenyl)acetamideKi6900.0 [1]
N-(4-Amino-5-cyano-6-phenylpyridin-2-yl)acetamideKi6900.0 [1]
Ripk1-IN-7IC50347.0 [1]
(13R,15S)-13-Methyl-16-oxa-8,9,12,22,24-pentazahexacyclo[15.6.2.16,9.112,15.02,7.021,25]heptacosa-1(24),2,4,6,17,19,21(25)-heptaene-23,27-dioneIC501000.0 [1]
1-(3-Tert-Butyl-1-Methyl-1h-Pyrazol-5-Yl)-3-[4-(Pyridin-4-Yloxy)phenyl]ureaIC5082.72 [1]
N-Cyclopropyl-3-[1-(2,6-difluorophenyl)-7-methyl-6-oxopyrazolo[3,4-b]pyridin-5-yl]-4-methylbenzamideKi2100.0 [1]
CID 25060878IC500.64 [1]
5-(2-Aminoethyl)-7-(7-(benzo[b]thiophen-2-yl)-1H-indazol-5-yl)-5H-pyrrolo[3,2-d]pyrimidin-2-amineIC507400.0 [1]
N-[3-[5-[2-(3-Morpholin-4-ylanilino)pyrimidin-4-yl]imidazo[2,1-b][1,3]thiazol-6-yl]phenyl]-2-phenylacetamideIC501000.0 [1]
1-[5-Tert-butyl-3-[4-[2-(dimethylamino)ethyl]-5-oxo-1,4-diazepane-1-carbonyl]thiophen-2-yl]-3-(2,3-dichlorophenyl)ureaIC5030000.0 [1]
6-(2,4-Difluorophenyl)sulfonyl-2-(1H-indol-5-ylamino)-8-methylpyrido[2,3-d]pyrimidin-7-oneIC5010000.0 [1]
2-Anilino-7-[(1S)-4-hydroxy-2,3-dihydro-1H-inden-1-yl]-5,5-dimethylpyrrolo[2,3-d]pyrimidin-6-oneIC5010000.0 [1]
CID 9811100IC5010000.0 [1]
2-(1-Methyl-4-hydroxy-4-piperidinyl)-4-(4-fluorophenyl)-5-(4-pyridinyl)oxazoleIC5010000.0 [1]
3-[(6-Benzoyl-5-Methylpyrrolo[2,1-F][1,2,4]triazin-4-Yl)amino]-N-Cyclopropyl-4-MethylbenzamideIC5025000.0 [1]
5-(3-Tert-butyl-[1,2,4]triazolo[4,3-a]pyridin-6-yl)-4-(2,4-difluorophenyl)-1,3-oxazoleIC5010000.0 [1]
5-(3-Propan-2-yl-[1,2,4]triazolo[4,3-a]pyridin-6-yl)-4-(2,4,5-trifluorophenyl)-1,3-oxazoleIC5010000.0 [1]
2-[3-(3-Piperidin-4-ylpropoxy)phenyl]-N-[4-(1H-pyrrolo[2,3-b]pyridin-3-yl)-1,3-thiazol-2-yl]acetamideKi2000.0 [1]
2-[3-(Methanesulfonamido)phenyl]-N-[4-(1H-pyrrolo[2,3-b]pyridin-3-yl)-1,3-thiazol-2-yl]acetamideKi2000.0 [1]
3-Tert-butyl-6-(2,4-difluorophenyl)sulfanyl-[1,2,4]triazolo[4,3-a]pyridineIC5062.0 [1]
N,4-Dimethyl-3-[[6-(methylamino)-1-phenylpyrazolo[3,4-d]pyrimidin-4-yl]amino]benzamideIC5030000.0 [1]
4-(2-Chloro-4-fluorophenyl)-5-(3-propan-2-yl-[1,2,4]triazolo[4,3-a]pyridin-6-yl)-1,3-oxazoleIC5010000.0 [1]
N-Ethyl-6-[4-(4-fluorophenyl)-1,3-oxazol-5-yl]-[1,2,4]triazolo[4,3-a]pyridin-3-amineIC5010000.0 [1]
6-[5-(2,5-Difluorophenyl)-1H-pyrazol-4-yl]-3-propan-2-yl-[1,2,4]triazolo[4,3-a]pyridineIC5010000.0 [1]
3-[3-(3-Chloropyridin-4-yl)-[1,2,4]triazolo[4,3-a]pyridin-7-yl]-N-cyclopropyl-5-fluoro-4-methylbenzamideIC500.83 [1]
4-(2-Chloro-4-fluorophenyl)-8-(2,6-dichlorophenyl)-7-oxido-1,7-naphthyridin-7-iumIC5010000.0 [1]
N-Cyclopropyl-4-methyl-3-(3-propan-2-yl-[1,2,4]triazolo[4,3-a]pyridin-7-yl)benzamideIC5027.0 [1]
3-(3-Tert-butyl-[1,2,4]triazolo[4,3-a]pyridin-7-yl)-N-cyclopropyl-5-fluoro-4-methylbenzamideIC502.0 [1]
3-[3-(2-Chlorophenyl)-[1,2,4]triazolo[4,3-a]pyridin-7-yl]-N-cyclopropyl-5-fluoro-4-methylbenzamideIC501.6 [1]
3-[3-(3-Chloropyridin-4-yl)-[1,2,4]triazolo[4,3-a]pyridin-7-yl]-N-cyclopropyl-4-methylbenzamideIC5038.0 [1]
3-[3-(2-Chlorophenyl)-[1,2,4]triazolo[4,3-a]pyridin-7-yl]-N-cyclopropyl-4-methylbenzamideIC506.3 [1]
3-(3-Tert-Butyl[1,2,4]triazolo[4,3-A]pyridin-7-Yl)-N-Cyclopropyl-4-MethylbenzamideIC5016.0 [1]
N-Cyclopropyl-3-(3-cyclopropyl-[1,2,4]triazolo[4,3-a]pyridin-7-yl)-4-methylbenzamideIC5026.0 [1]
N-Cyclopropyl-4-methyl-3-[3-(1-methylcyclopropyl)-[1,2,4]triazolo[4,3-a]pyridin-7-yl]benzamideIC5012.0 [1]
3-(3-Cyclobutyl-[1,2,4]triazolo[4,3-a]pyridin-7-yl)-N-cyclopropyl-4-methylbenzamideIC5020.0 [1]
3-(3-Tert-butyl-6,8-difluoro-[1,2,4]triazolo[4,3-a]pyridin-7-yl)-N-cyclopropyl-4-methylbenzamideIC5049.0 [1]
N-Cyclopropyl-3-(6,8-difluoro-3-propan-2-yl-[1,2,4]triazolo[4,3-a]pyridin-7-yl)-5-fluoro-4-methylbenzamideIC506.7 [1]
N-Cyclopropyl-3-(3-cyclopropyl-6,8-difluoro-[1,2,4]triazolo[4,3-a]pyridin-7-yl)-5-fluoro-4-methylbenzamideIC5010.0 [1]
3-[3-(3-Chloropyridin-4-yl)-6,8-difluoro-[1,2,4]triazolo[4,3-a]pyridin-7-yl]-N-cyclopropyl-5-fluoro-4-methylbenzamideIC5023.0 [1]
N-Cyclopropyl-3-(3-cyclopropyl-[1,2,4]triazolo[4,3-a]pyridin-7-yl)-5-fluoro-4-methylbenzamideIC506.7 [1]
N-Cyclopropyl-3-fluoro-4-methyl-5-(3-propan-2-yl-[1,2,4]triazolo[4,3-a]pyridin-7-yl)benzamideIC503.0 [1]
3-(3-Cyclobutyl-[1,2,4]triazolo[4,3-a]pyridin-7-yl)-N-cyclopropyl-5-fluoro-4-methylbenzamideIC501.9 [1]
N-Cyclopropyl-3-fluoro-4-methyl-5-[3-(oxan-4-yl)-[1,2,4]triazolo[4,3-a]pyridin-7-yl]benzamideIC5030.0 [1]
3-[3-(2-Aminopropan-2-yl)-[1,2,4]triazolo[4,3-a]pyridin-7-yl]-N-cyclopropyl-5-fluoro-4-methylbenzamideIC5015.4 [1]
N-Cyclopropyl-3-fluoro-5-[3-(2-methoxypropan-2-yl)-[1,2,4]triazolo[4,3-a]pyridin-7-yl]-4-methylbenzamideIC509.4 [1]
N-Cyclopropyl-3-fluoro-4-methyl-5-[3-(trifluoromethyl)-[1,2,4]triazolo[4,3-a]pyridin-7-yl]benzamideIC5085.0 [1]
3-[3-(2-Acetamidopropan-2-yl)-[1,2,4]triazolo[4,3-a]pyridin-7-yl]-N-cyclopropyl-5-fluoro-4-methylbenzamideIC50253.0 [1]
N-Cyclopropyl-3-fluoro-5-[3-(2-hydroxypropan-2-yl)-[1,2,4]triazolo[4,3-a]pyridin-7-yl]-4-methylbenzamideIC503.1 [1]
3-[3-(2-Aminopropan-2-yl)-6,8-difluoro-[1,2,4]triazolo[4,3-a]pyridin-7-yl]-N-cyclopropyl-5-fluoro-4-methylbenzamideIC5012.0 [1]
N-Cyclopropyl-4-methyl-3-[3-(trifluoromethyl)-[1,2,4]triazolo[4,3-a]pyridin-7-yl]benzamideIC50853.0 [1]
7-[5-(Cyclopropylcarbamoyl)-3-fluoro-2-methylphenyl]-[1,2,4]triazolo[4,3-a]pyridine-3-carboxamideIC50102.0 [1]
N-Cyclopropyl-4-methyl-3-[3-(oxan-4-yl)-[1,2,4]triazolo[4,3-a]pyridin-7-yl]benzamideIC5056.0 [1]
N-{4-[(6-Oxo-5,6-Dihydrobenzo[c][1,8]naphthyridin-1-Yl)amino]phenyl}benzamideIC50411.0 [1]
4-Chloro-N-cyclopropyl-3-[[1-(4-fluorophenyl)-7-methyl-6-oxopyrazolo[3,4-b]pyridin-4-yl]amino]benzamideIC504.0 [1]
4-(4-(2-(Cyclopentylamino)pyrimidin-4-yl)-1H-pyrazol-3-yl)cyclohexanolIC501200.0 [1]
N-Cyclopropyl-3-[3-[2-(dimethylamino)propan-2-yl]-6,8-difluoro-[1,2,4]triazolo[4,3-a]pyridin-7-yl]-5-fluoro-4-methylbenzamideIC5015.0 [1]
N-Cyclopropyl-3-fluoro-5-[3-[2-(methanesulfonamido)propan-2-yl]-[1,2,4]triazolo[4,3-a]pyridin-7-yl]-4-methylbenzamideIC5017.0 [1]
N-Cyclopropyl-3-[3-[2-(dimethylamino)propan-2-yl]-[1,2,4]triazolo[4,3-a]pyridin-7-yl]-5-fluoro-4-methylbenzamideIC501.7 [1]
2-[3-(3-Piperazin-1-ylpropoxy)phenyl]-N-(4-pyridin-4-yl-1,3-thiazol-2-yl)acetamideIC5010000.0 [1]
8-N-(Cyclopropylmethyl)-4-N-(2-methylsulfanylphenyl)-2-(4-piperidin-4-ylpiperazin-1-yl)pyrimido[5,4-d]pyrimidine-4,8-diamineIC5010000.0 [1]
2-(Morpholin-4-Yl)-N-[4-(Pyridin-4-Yloxy)phenyl]pyridine-4-CarboxamideIC5098747.0 [1]
N-Cyclopropyl-3-[3-(1-methoxyethyl)-[1,2,4]triazolo[4,3-a]pyridin-7-yl]-4-methylbenzamideIC5043.0 [1]
N-Cyclopropyl-3-fluoro-5-[3-(1-methoxyethyl)-[1,2,4]triazolo[4,3-a]pyridin-7-yl]-4-methylbenzamideIC5018.0 [1]
N-Cyclopropyl-4-methyl-3-(3-piperidin-1-yl-1,2-benzoxazol-6-yl)benzamideIC5014.0 [1]
3-(Tert-butylamino)-4-[[2-(4-pyridin-4-ylanilino)pyrimidin-4-yl]amino]cyclobut-3-ene-1,2-dioneKi5900.0 [1]
3-Isopropyl-6-(4-phenyl-oxazol-5-yl)-[1,2,4]triazolo[4,3-a]pyridineIC5010000.0 [1]
5-(3-Tert-butyl-[1,2,4]triazolo[4,3-a]pyridin-6-yl)-4-(2,4,5-trifluorophenyl)-1,3-oxazoleIC5010000.0 [1]
1-[5-Tert-butyl-2-(4-methylphenyl)pyrazol-3-yl]-3-[2-(oxane-4-carbonyl)-1,3-dihydroisoindol-5-yl]ureaIC508650.0 [1]
3-(4-Methyl-1h-Imidazol-1-Yl)-N-[4-(Pyridin-4-Yloxy)phenyl]benzamideIC5010200.0 [1]
1-[5-Tert-butyl-2-(4-methylphenyl)pyrazol-3-yl]-3-[5-(2-morpholin-4-ylethyl)-1,3-thiazol-2-yl]ureaIC5027.54 [1]
1-[5-Tert-butyl-2-(4-methylphenyl)pyrazol-3-yl]-3-(4-pyridin-4-yloxyphenyl)ureaIC50280.5 [1]
Items per page: 1 - 10 of 93
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References

This online tool may be cited as follows

MLA

"Quest Database™ MAP kinase p38 delta Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 21 Nov. 2024, https://www.aatbio.com/data-sets/map-kinase-p38-delta-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, November 21). Quest Database™ MAP kinase p38 delta Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/map-kinase-p38-delta-inhibitors-ic50-ki.
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