![](https://images.aatbio.com/dataset/ic50/map-kinase-p38-alpha_b96c95589239aa5fc9b995c3e9055da0.svg) | 4-(4-Fluorophenyl)-2-(4-methylsulfinylphenyl)-5-(4-pyridyl)-1H-imidazole | IC50 | 48.0 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-p38-alpha_b96c95589239aa5fc9b995c3e9055da0.svg) | 4-(4-Fluorophenyl)-2-(4-methylsulfinylphenyl)-5-(4-pyridyl)-1H-imidazole | Ki | 18.0 [1], 57.0 [2] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-p38-alpha_0a83b01cf93719a90ccaeda771089c43.svg) | Doramapimod | IC50 | 17.0 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-p38-alpha_0a83b01cf93719a90ccaeda771089c43.svg) | Doramapimod | Ki | 0.1 [1], 6.4 [2], 22.0 [3], 46.0 [4] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-p38-alpha_3013791590a95a7fa1113a8967c19298.svg) | Neflamapimod | IC50 | 51.0 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-p38-alpha_398ba4ab0282ab056845b8e125351aa5.svg) | 4-(4-Fluorophenyl)-2-(4-hydroxyphenyl)-5-(4-pyridyl)-1H-imidazole | IC50 | 28.0 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-p38-alpha_2688d8bfa0592bfa6cd0f2033d501ca7.svg) | [5-Amino-1-(4-fluorophenyl)-1H-pyrazol-4-YL](3-{[(2R)-2,3-dihydroxypropyl]oxy}phenyl)methanone | IC50 | 400.0 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-p38-alpha_7cd07c14c9a6699a18c59379f39dd9e2.svg) | N~3~-Cyclopropyl-N~4~'-(Cyclopropylmethyl)-6-Methylbiphenyl-3,4'-Dicarboxamide | IC50 | 18.0 [1], 199.53 [2], 1584.89 [3] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-p38-alpha_7cd07c14c9a6699a18c59379f39dd9e2.svg) | N~3~-Cyclopropyl-N~4~'-(Cyclopropylmethyl)-6-Methylbiphenyl-3,4'-Dicarboxamide | Ki | 9.0 [1], 10.0 [2], 12.0 [3], 12.59 [4] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-p38-alpha_c8494007663098abb5d227cb27cc738b.svg) | Sorafenib | IC50 | 84.2 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-p38-alpha_461434bd943d10cbcd2b8085cc6a5221.svg) | 3-(3-Bromo-4-((2,4-difluorobenzyl)oxy)-6-methyl-2-oxopyridin-1(2H)-yl)-N,4-dimethylbenzamide | IC50 | 1.05 [1], 5.8 [2], 17.4 [3], 247.0 [4] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-p38-alpha_461434bd943d10cbcd2b8085cc6a5221.svg) | 3-(3-Bromo-4-((2,4-difluorobenzyl)oxy)-6-methyl-2-oxopyridin-1(2H)-yl)-N,4-dimethylbenzamide | Ki | 2.9 [1], 5.8 [2] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-p38-alpha_3d7fd13de900a9c7fee5495394736fdb.svg) | Benzamide, 3-((4-(6-methyl-2-pyridinyl)-5-(6-quinoxalinyl)-1H-imidazol-2-yl)methyl)- | IC50 | 480.0 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-p38-alpha_c022d5fe632b5699e5d9f02e9201a202.svg) | 4-(2-Cyanophenoxy)-N-(pyridin-4-ylmethyl)benzamide | IC50 | 600.0 [1], 5400.0 [2], 10000.0 [3], 21000.0 [4], 25000.0 [5] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-p38-alpha_c022d5fe632b5699e5d9f02e9201a202.svg) | 4-(2-Cyanophenoxy)-N-(pyridin-4-ylmethyl)benzamide | Ki | 290.0 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-p38-alpha_2b76387e020a39962bfa00976861b6d5.svg) | N-[5-(Dimethylsulfamoyl)-2-methylphenyl]-1-phenyl-5-propyl-1H-pyrazole-4-carboxamide | IC50 | 61.0 [1], 970.0 [2], 1500.0 [3], 9700.0 [4], 10000.0 [5] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-p38-alpha_2b76387e020a39962bfa00976861b6d5.svg) | N-[5-(Dimethylsulfamoyl)-2-methylphenyl]-1-phenyl-5-propyl-1H-pyrazole-4-carboxamide | Ki | 14.0 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-p38-alpha_d8c9f64db0b5aad78138a2dd34a08b59.svg) | 2-(4-(Benzo[d][1,3]dioxol-5-yl)-2-tert-butyl-1H-imidazol-5-yl)-6-methylpyridine | IC50 | 590.0 [1], 594.0 [2], 668.0 [3] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-p38-alpha_3767ea0199fd9fb4f2e8a75ca8ffc85c.svg) | Losmapimod | IC50 | 25.12 [1], 100.0 [2] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-p38-alpha_3767ea0199fd9fb4f2e8a75ca8ffc85c.svg) | Losmapimod | Ki | 7.94 [1], 63.1 [2] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-p38-alpha_07558cdb76f6c9279d40285cf5594a88.svg) | Talmapimod | IC50 | 9.0 [1], 10.0 [2], 36.0 [3], 96.0 [4] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-p38-alpha_1e7afdcf7ed1b7b6ec05c07f7a454e11.svg) | N-[4-Methyl-3-[[4-(1,3-thiazol-4-ylmethoxy)benzoyl]amino]phenyl]-3-morpholin-4-ylbenzamide | IC50 | 10.0 [1], 15.85 [2], 17.0 [3], 25.12 [4], 1258.93 [5] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-p38-alpha_5fbeb7be5a4397c2a476ca48e779f728.svg) | 7-(1-Tert-butylpiperidin-4-yl)-1-(2,6-dichlorophenyl)-5-(2,4-difluorophenyl)quinolin-2-one | IC50 | 0.08 [1], 0.14 [2], 1.7 [3], 2.4 [4], 28.0 [5] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-p38-alpha_2287ad8e3e282203ad2aacad5fc9c182.svg) | N-Cyclopropyl-3-(4'-hydroxy-2-oxospiro[1H-indole-3,1'-cyclohexane]-6-yl)-4-methylbenzamide | IC50 | 1.4 [1], 5.0 [2], 11.0 [3] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-p38-alpha_d1a554e9d8cdbc3e7b827e2772b17a0d.svg) | CK1 Inhibitor | IC50 | 4154.0 [1], 5800.0 [2], 12000.0 [3] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-p38-alpha_41880dd29cabf486dbc6f37e43a5ca93.svg) | 4-(4-Fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | IC50 | 19.0 [1], 20.0 [2] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-p38-alpha_0496776e10c2732c44d10545e177b210.svg) | Skepinone-L | IC50 | 5.0 [1], 40.0 [2] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-p38-alpha_6ad94dc26455bcde818c72b352ccec47.svg) | 4-(4-(4-Fluorophenyl)-1-(piperidin-4-yl)-1H-imidazol-5-yl)-2-methoxypyrimidine | IC50 | 19.0 [1], 40.0 [2], 130.0 [3] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-p38-alpha_6ad94dc26455bcde818c72b352ccec47.svg) | 4-(4-(4-Fluorophenyl)-1-(piperidin-4-yl)-1H-imidazol-5-yl)-2-methoxypyrimidine | Ki | 36.0 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-p38-alpha_e8faac28aa4780473e3d8d541a94acb6.svg) | N-[3-[4-(Cyclopropylmethylcarbamoyl)phenyl]-4-methylphenyl]furan-3-carboxamide | IC50 | 16.0 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-p38-alpha_e8faac28aa4780473e3d8d541a94acb6.svg) | N-[3-[4-(Cyclopropylmethylcarbamoyl)phenyl]-4-methylphenyl]furan-3-carboxamide | Ki | 6.0 [1], 15.0 [2] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-p38-alpha_358f0986945a73f2b266babf799f8794.svg) | 3-(2,4-Difluoroanilino)-6H-benzo[c][1]benzoxepin-11-one | IC50 | 239.0 [1], 240.0 [2], 22000.0 [3] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-p38-alpha_b938cdfc0f76d8ada82731c33b67b376.svg) | Methyl 5-(2-chlorophenyl)-1-(2,6-dichlorophenyl)-2-oxo-1,2,3,4-tetrahydroquinazoline-7-carboxylate | IC50 | 1.0 [1], 2.0 [2] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-p38-alpha_291b06385bacef5b4855d6889af62ea8.svg) | 1-(2,6-Dichlorophenyl)-5-(2-chlorophenyl)-7-methoxy-3,4-dihydro-2(1H)-quinazolinone | IC50 | 1.0 [1], 6.0 [2] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-p38-alpha_d89c41ad743193c7f8074cc3d3b6aaa3.svg) | 1-(2,6-Dichlorophenyl)-5-(2,4-difluorophenyl)-7-(4-piperidinyl)-1,2,3,4-tetrahydroquinazoline-2-one | IC50 | 0.2 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-p38-alpha_03cfc3a72db0322aa86332b598c19943.svg) | N-Cyclopropyl-4-Methyl-3-(2'-Oxo-1',2'-Dihydrospiro[cyclopentane-1,3'-Indol]-6'-Yl)benzamide | IC50 | 1.3 [1], 18.0 [2] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-p38-alpha_ab586e2a2df773b305311973f5d3abae.svg) | 4-[5-(4-Fluorophenyl)-2-methylsulfanyl-1H-imidazol-4-yl]-N-(oxan-4-yl)pyridin-2-amine | IC50 | 5.0 [1], 180.0 [2] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-p38-alpha_c76461a2a54d2da90f63ee5444e64ae1.svg) | 13-(2,4-Difluoroanilino)-5-(3-hydroxypropoxy)tricyclo[9.4.0.03,8]pentadeca-1(11),3(8),4,6,12,14-hexaen-2-one | IC50 | 8.0 [1], 13.0 [2], 190.0 [3], 191.0 [4] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-p38-alpha_b5c621124a998e3a4864ff4a09b7f3d3.svg) | 13-(2,4-Difluoroanilino)-5-hydroxytricyclo[9.4.0.03,8]pentadeca-1(11),3(8),4,6,12,14-hexaen-2-one | IC50 | 20.0 [1], 49.0 [2], 700.0 [3], 1247.0 [4] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-p38-alpha_b865d7d40eb8c1af1990915463355b9e.svg) | 13-(2,4-Difluoroanilino)-5-[(2S)-2,3-dihydroxypropoxy]tricyclo[9.4.0.03,8]pentadeca-1(11),3(8),4,6,12,14-hexaen-2-one | IC50 | 8.0 [1], 17.0 [2], 52.0 [3], 60.0 [4] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-p38-alpha_1a073f5a17bf34cd602cd7c9ce33164a.svg) | 13-(2,4-Difluoroanilino)-5-methoxytricyclo[9.4.0.03,8]pentadeca-1(11),3(8),4,6,12,14-hexaen-2-one | IC50 | 20.0 [1], 44.0 [2], 1200.0 [3], 1647.0 [4] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-p38-alpha_f41538f50a044146bd8a0aa18bb5efa1.svg) | 13-(2,4-Difluoroanilino)-5-(2-hydroxyethoxy)tricyclo[9.4.0.03,8]pentadeca-1(11),3(8),4,6,12,14-hexaen-2-one | IC50 | 10.0 [1], 19.0 [2], 480.0 [3], 583.0 [4] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-p38-alpha_6aa9cf2ea1733b23b9672f26521b02cc.svg) | 2-(4-Fluorophenyl)-N-[4-[5-(4-fluorophenyl)-2-methylsulfanyl-1H-imidazol-4-yl]pyridin-2-yl]acetamide | IC50 | 9.0 [1], 2980.0 [2] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-p38-alpha_a6691c074440f0145b963005e02d7b11.svg) | 13-(3-Benzamido-4-fluoroanilino)-N-(2-morpholin-4-ylethyl)-2-oxotricyclo[9.4.0.03,8]pentadeca-1(11),3(8),4,6,12,14-hexaene-5-carboxamide | IC50 | 0.2 [1], 31.0 [2], 38.0 [3] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-p38-alpha_ff87290449ba9d3323ddac98d6790a4e.svg) | N-Benzyl-4-(2-cyanophenoxy)benzamide | IC50 | 450.0 [1], 1400.0 [2], 10000.0 [3], 100000.0 [4] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-p38-alpha_2ab9354f611398d0e5d7bbc16f12ac04.svg) | 4-(2-Cyanophenoxy)-N-(pyridin-3-ylmethyl)benzamide | IC50 | 560.0 [1], 4700.0 [2], 10000.0 [3], 15000.0 [4] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-p38-alpha_00b5acc521e8646c2604f9f4f33e5ec5.svg) | 4-(2-Cyanophenoxy)-N-(pyrimidin-4-ylmethyl)benzamide | IC50 | 2800.0 [1], 7100.0 [2], 10000.0 [3], 100000.0 [4] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-p38-alpha_fd28bc49df7d7ccac0d5fc9efc79a3ba.svg) | N-(5-Cyano-2-methylphenyl)-1-phenyl-5-propylpyrazole-4-carboxamide | IC50 | 15.0 [1], 210.0 [2], 890.0 [3], 10000.0 [4] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-p38-alpha_8490671fd8598bf299b0138b3e7318ab.svg) | 4-Methyl-3-[(1-phenyl-5-propylpyrazole-4-carbonyl)amino]benzoic acid | IC50 | 86.0 [1], 4200.0 [2], 10000.0 [3], 21000.0 [4] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-p38-alpha_ae4f676a15c5016ae544acbc8d6cad98.svg) | N-[5-[[14-[(2S)-2,3-Dihydroxypropoxy]-2-oxo-6-tricyclo[9.4.0.03,8]pentadeca-1(11),3(8),4,6,12,14-hexaenyl]amino]-2-fluorophenyl]benzamide | IC50 | 1.0 [1], 3.0 [2], 280.0 [3] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-p38-alpha_2e4fe4208420c8b33e5ac8bf560c38da.svg) | 6-(4-Fluorophenyl)-2,3-dihydro-5-(4-pyridinyl)imidazo(2,1-b)thiazole | IC50 | 110.0 [1], 400.0 [2], 820.0 [3] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-p38-alpha_1760e4f1c30c41a3c0bdd7ae47cfa001.svg) | 1-(5-Tert-butyl-2-methyl-2H-pyrazol-3-YL)-3-(4-chloro-phenyl)-urea | IC50 | 794.33 [1], 16800.0 [2], 21000.0 [3] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-p38-alpha_0436ca6d274102f4500a83f1efa2f6fe.svg) | 4-(5-(4-Fluorophenyl)-3-(4-piperidyl)imidazol-4-yl)pyridine | IC50 | 38.0 [1], 60.0 [2] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-p38-alpha_0436ca6d274102f4500a83f1efa2f6fe.svg) | 4-(5-(4-Fluorophenyl)-3-(4-piperidyl)imidazol-4-yl)pyridine | Ki | 60.0 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-p38-alpha_de8afcc0ec0ff63df996c1f642d3883b.svg) | 2-Amino-Phenylamino-Dibenzosuberone | IC50 | 50.0 [1], 100.0 [2], 104.0 [3] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-p38-alpha_bf41e70c17a1e07746319c13984ebb6c.svg) | N-(3-Cyanophenyl)-2'-Methyl-5'-(5-Methyl-1,3,4-Oxadiazol-2-Yl)-4-Biphenylcarboxamide | Ki | 240.0 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-p38-alpha_fa01851622bb7f1f4cd0d71ede29af68.svg) | N-Cyclopropyl-4-methyl-3-[6-(4-methylpiperazin-1-yl)-4-oxoquinazolin-3(4H)-yl]benzamide | IC50 | 15.85 [1], 17.38 [2], 27.54 [3] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-p38-alpha_955ee68b75668dbe601bc47cf36a5834.svg) | 2-Phenoxy-4-[1-(piperidine-4-yl)-4-(4-fluorophenyl)-5-imidazolyl]pyrimidine | IC50 | 19.0 [1], 19.2 [2], 20.0 [3] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-p38-alpha_3a3590cd8b87a2cd33788ec6016110d4.svg) | 4-Phenoxy-N-(pyridin-4-ylmethyl)benzamide | IC50 | 2300.0 [1], 4000.0 [2], 10000.0 [3] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-p38-alpha_b25f98550f3c0c676c7ec478e5c86a49.svg) | 4-(4-Methylphenoxy)-N-(4-pyridinylmethyl)benzenecarboxamide | IC50 | 4700.0 [1], 10000.0 [2], 22000.0 [3] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-p38-alpha_612cc31d82aef72d2292d1f4829b1665.svg) | N-{4'-[(Cyclopropylmethyl)carbamoyl]-6-Methylbiphenyl-3-Yl}-2-Morpholin-4-Ylpyridine-4-Carboxamide | IC50 | 6.0 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-p38-alpha_612cc31d82aef72d2292d1f4829b1665.svg) | N-{4'-[(Cyclopropylmethyl)carbamoyl]-6-Methylbiphenyl-3-Yl}-2-Morpholin-4-Ylpyridine-4-Carboxamide | Ki | 4.4 [1], 6.0 [2] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-p38-alpha_39ceed0ad4ea5af71d276a234ff375b8.svg) | 4-[3-Methyl-2-piperidin-4-yl-5-[3-(trifluoromethyl)phenyl]imidazol-4-yl]-N-[(1S)-1-phenylethyl]pyridin-2-amine | IC50 | 0.1 [1], 2.0 [2], 34.0 [3] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-p38-alpha_b9f827ef1b2bfd816c726d1146451de8.svg) | N-[2-Methyl-5-(methylcarbamoyl)phenyl]-2-{[(1R)-1-methylpropyl]amino}-1,3-thiazole-5-carboxamide | IC50 | 3.5 [1], 4.0 [2] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-p38-alpha_969dba429fd4e580980eb0f30b530c40.svg) | 3-(2-Aminoquinazolin-6-Yl)-4-Methyl-N-[3-(Trifluoromethyl)phenyl]benzamide | IC50 | 6.0 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-p38-alpha_f020cbb4e686334360710d919818a328.svg) | N-(4-(2-(Phenylamino)pyridin-4-yl)pyridin-2-yl)-tetrahydrofuran-3-carboxamide | IC50 | 180.0 [1], 199.53 [2] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-p38-alpha_42496a2ac6869d2e8d7f76051d516e53.svg) | N-[4-[5-(4-Fluorophenyl)-3-methyl-2-methylsulfinylimidazol-4-yl]pyridin-2-yl]acetamide | IC50 | 500.0 [1], 710.0 [2], 1072.0 [3] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-p38-alpha_0c14876e228fcb8aee98a4b13e08928b.svg) | 4-[3-(4-Fluorophenyl)-5-isopropylisoxazol-4-yl]pyridine | IC50 | 450.0 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-p38-alpha_b10988c30da7aac7584f9b7d2ab1dae7.svg) | 4-[5-(4-Fluorophenyl)-3-isopropylisoxazol-4-yl]pyridine | IC50 | 2200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-p38-alpha_fa011acb3e00fab3b7e5df63dd0f03e6.svg) | N-(Cyclopropylmethyl)-2'-Methyl-5'-(5-Methyl-1,3,4-Oxadiazol-2-Yl)biphenyl-4-Carboxamide | Ki | 480.0 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-p38-alpha_7217c206f4ec15f1671e8eb53e0d04a1.svg) | 5-(2-Chlorophenyl)-1-(2,6-dichlorophenyl)-7-(piperidin-4-ylamino)-3,4-dihydroquinazolin-2(1H)-one | IC50 | 0.5 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-p38-alpha_b5f38a2a1c429f3a987267d99bcc9f7d.svg) | 1-Methyl-3-tert-butyl-5-[3-(2,3-dichlorophenyl)ureido]-1H-pyrazole | IC50 | 53.0 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-p38-alpha_688a326d0250790f3859af7c50a2c165.svg) | 6-(2,4-Difluoroanilino)tricyclo[9.4.0.03,8]pentadeca-1(15),3(8),4,6,11,13-hexaen-2-one | IC50 | 95.0 [1], 130.0 [2], 1907.0 [3] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-p38-alpha_3068d7735f2b149479d0348d5a341c5b.svg) | 1-(2,6-Dichlorophenyl)-5-(2,4-difluorophenyl)-7-piperazin-1-YL-3,4-dihydroquinazolin-2(1H)-one | IC50 | 2.6 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-p38-alpha_cecb544ee0b1385db075e679a45b012d.svg) | 5-(2-Chlorophenyl)-1-(2,6-dichlorophenyl)-7-piperazin-1-yl-3,4-dihydroquinazolin-2-one | IC50 | 1.4 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-p38-alpha_0fba6751444fffbe011ac2cb1ae23f60.svg) | 5-(2-Chlorophenyl)-1-(2,6-dichlorophenyl)-7-piperidin-4-yloxy-3,4-dihydroquinazolin-2-one | IC50 | 0.2 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-p38-alpha_3f3bfb56dae41c7d7d7da963d0e5ed5d.svg) | 5-(2-Chloro-4-fluorophenyl)-1-(2,6-dichlorophenyl)-7-(piperazine-1-carbonyl)-3,4-dihydroquinazolin-2-one | IC50 | 1.1 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-p38-alpha_1db504db5cdbd07b0e8cbab66ace4976.svg) | 2-(2-Chloro-4-fluorophenyl)sulfanyl-5-(2,6-dichlorophenyl)pyrimido[1,6-b]pyridazin-6-one | IC50 | 36.0 [1], 53.0 [2], 275.0 [3] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-p38-alpha_93a02f248c5d7cf3f93d2f99dc84c5fa.svg) | 5-(2,6-Dichlorophenyl)-2-(4-methylphenyl)sulfanylpyrimido[1,6-b]pyridazin-6-one | IC50 | 370.0 [1], 870.0 [2], 1400.0 [3] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-p38-alpha_1e3583a24db7c5a7ba67d5ba20f60241.svg) | 5-(2,6-Dichlorophenyl)-2-(phenylthio)-6H-pyrimido[1,6-b]pyridazin-6-one | IC50 | 250.0 [1], 400.0 [2], 460.0 [3] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-p38-alpha_778fd193b3ebc140a7ee6868f12eb3b3.svg) | 2-(3-Chlorophenyl)sulfanyl-5-(2,6-dichlorophenyl)pyrimido[1,6-b]pyridazin-6-one | IC50 | 280.0 [1], 350.0 [2], 900.0 [3] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-p38-alpha_3c147929dcd2ba0ddbfde0a2d1b14b31.svg) | 2-(4-Chloro-2-methylphenyl)sulfanyl-5-(2,6-dichlorophenyl)pyrimido[1,6-b]pyridazin-6-one | IC50 | 160.0 [1], 180.0 [2] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-p38-alpha_f2985021b5092e02b8193490ddf08195.svg) | 5-(2,6-Dichlorophenyl)-2-(3,4-dichlorophenyl)sulfanylpyrimido[1,6-b]pyridazin-6-one | IC50 | 800.0 [1], 970.0 [2], 1200.0 [3] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-p38-alpha_6670f102a578d3881be547fde9f0c38f.svg) | 5-(2,6-Dichlorophenyl)-2-(4-fluorophenyl)sulfanylpyrimido[1,6-b]pyridazin-6-one | IC50 | 99.0 [1], 123.0 [2], 293.0 [3] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-p38-alpha_863519447673986c682e08eb0f5dfe36.svg) | 5-(2,6-Dichlorophenyl)-2-(2,4-dimethylphenyl)sulfanylpyrimido[1,6-b]pyridazin-6-one | IC50 | 260.0 [1], 320.0 [2], 690.0 [3] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-p38-alpha_27e54ce67565472807d41081a156ebaf.svg) | 5-(2,6-Dichlorophenyl)-2-(2-hydroxyphenyl)sulfanylpyrimido[1,6-b]pyridazin-6-one | IC50 | 140.0 [1], 360.0 [2], 490.0 [3] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-p38-alpha_c013538d0a17474f8b36c28979c8b8b5.svg) | 5-(2,6-Dichlorophenyl)-2-(3,4-dimethylphenyl)sulfanylpyrimido[1,6-b]pyridazin-6-one | IC50 | 1900.0 [1], 2400.0 [2], 3500.0 [3] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-p38-alpha_9bc5391aa64fca5aab8852f872f8859f.svg) | 5-(2,6-Dichlorophenyl)-2-(3-fluorophenyl)sulfanylpyrimido[1,6-b]pyridazin-6-one | IC50 | 440.0 [1], 450.0 [2], 720.0 [3] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-p38-alpha_c017cfcf491aacce60f1572a5690c7d7.svg) | 5-(2,6-Dichlorophenyl)-2-(3-methylphenyl)sulfanylpyrimido[1,6-b]pyridazin-6-one | IC50 | 210.0 [1], 280.0 [2], 1400.0 [3] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-p38-alpha_ac25a2263376c11710a30a71db590254.svg) | 5-(2,6-Dichlorophenyl)-2-(2-methylphenyl)sulfanylpyrimido[1,6-b]pyridazin-6-one | IC50 | 200.0 [1], 330.0 [2], 3700.0 [3] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-p38-alpha_e9fca2917c414d638502f88600a9b7a9.svg) | 2-(2-Amino-4-fluorophenyl)sulfanyl-5-(2,6-dichlorophenyl)pyrimido[1,6-b]pyridazin-6-one | IC50 | 220.0 [1], 280.0 [2], 1200.0 [3] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-p38-alpha_b844ff2f47fc4d2bd7614b3a4f1c5326.svg) | 2-(3-Chloro-4-fluorophenyl)sulfanyl-5-(2,6-dichlorophenyl)pyrimido[1,6-b]pyridazin-6-one | IC50 | 180.0 [1], 480.0 [2], 500.0 [3] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-p38-alpha_6b892648075e69df7e5f1d26f1f7ddea.svg) | N-[4-Methyl-3-[6-(4-methylpiperazin-1-yl)-4-oxoquinazolin-3-yl]phenyl]-2-morpholin-4-ylpyridine-4-carboxamide | IC50 | 26.3 [1], 123.03 [2], 416.87 [3] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-p38-alpha_fa54b1c0b846c70b45e49551518d10e7.svg) | 1-(2,6-Dichlorophenyl)-5-(2,4-difluorophenyl)-7-methoxy-3,4-dihydro-2(1H)-quinazolinone | IC50 | 10.99 [1], 11.0 [2] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-p38-alpha_9c6ca5383a495b3c06f2bc85530224ee.svg) | 5-(2-Chloro-4-fluorophenyl)-1-(2,6-dichlorophenyl)-7-piperidin-4-yl-3,4-dihydroquinazolin-2-one | IC50 | 0.1 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-p38-alpha_d034b519d6fd7cbc710534f8ddf59f29.svg) | 1-(2,6-Dichlorophenyl)-5-(2-chloro-4-fluorophenyl)-7-methoxy-3,4-dihydro-2(1H)-quinazolinone | IC50 | 3.0 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-p38-alpha_2fcce0a95adbb4171989c8ccbf64f8ae.svg) | 1-(2,6-Dichlorophenyl)-5-(2,4-difluorophenyl)-7-(piperidin-4-ylamino)-3,4-dihydroquinazolin-2-one | IC50 | 0.6 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-p38-alpha_13fcb91932fb2565053344ba79d9fc56.svg) | 1-(2,6-Dichlorophenyl)-5-(2-chlorophenyl)-7-(4-piperidinyl)-1,2,3,4-tetrahydroquinazoline-2-one | IC50 | 0.9 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-p38-alpha_168a710a7898e824c586227fa593337a.svg) | Cyclohexyl-{4-[5-(4-fluorophenyl)-2-methylsulfanyl-1H-imidazol-4-yl]pyridin-2-yl}amine | IC50 | 20.0 [1], 27.0 [2], 170.0 [3] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-p38-alpha_2de502a134099a82df8e76c7a4934bee.svg) | 2-(4-Fluorophenyl)-3-[2-[[(1S)-1-phenylethyl]amino]pyrimidin-4-yl]imidazo[1,2-a]pyrimidin-7-amine | IC50 | 1.0 [1], 6.0 [2], 8.5 [3] |