![](https://images.aatbio.com/dataset/ic50/map-kinase-erk1_1d5eba4b4bb57896dda18b1604bab021.svg) | Staurosporine | IC50 | 5089.0 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-erk1_85bfeb5c1c0028708a30ec66fc1bbd21.svg) | Seliciclib | IC50 | 34000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-erk1_000b8ce6322fa44973ae7360b2e38f90.svg) | Olomoucine | IC50 | 25000.0 [1], 30000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-erk1_0a83b01cf93719a90ccaeda771089c43.svg) | Doramapimod | IC50 | 20000.0 [1], 30000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-erk1_26575b04a0a4cc9959845db9b7bd7b68.svg) | Purvalanol B | IC50 | 3300.0 [1], 3333.0 [2] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-erk1_e7902e795bb889d9776f6a7fbe9f7e96.svg) | Purvalanol A | IC50 | 9000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-erk1_0ee4cca9cb9a30297469dae72afaa1d1.svg) | CID 24866313 | IC50 | 4.0 [1], 8.0 [2] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-erk1_986a45a06f23aac579f61ed926220337.svg) | 5-(2-Phenylpyrazolo[1,5-A]pyridin-3-YL)-1H-pyrazolo[3,4-C]pyridazin-3-amine | Ki | 310.0 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-erk1_e31549449ac2e1990c406789dd9aeae1.svg) | Tanzisertib | IC50 | 480.0 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-erk1_c8494007663098abb5d227cb27cc738b.svg) | Sorafenib | IC50 | 18.1 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-erk1_b33d647a5a347bfb173a0ed912563556.svg) | (Z)-3-Amino-3-(4-aminophenylthio)-2-(2-(trifluoromethyl)phenyl)acrylonitrile | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-erk1_f888f082cfdd181caa483bbe675439bc.svg) | Kenpaullone | IC50 | 20000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-erk1_c74a1b9d6feb1def6b7e3f6834b5761b.svg) | Tak-285 | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-erk1_f3d0fcadcce0816240114937491b30f7.svg) | 1-(2,4-Difluorophenyl)-3-(4-(6,7-dimethoxyquinolin-4-yloxy)-2-fluorophenyl)urea | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-erk1_6218d7660845b31fc510a0466313fd99.svg) | Amg-458 | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-erk1_c71081a8619ec348ecd13cc61c9f2023.svg) | CID 46209401 | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-erk1_ab2268bff60761ec9560ebfb5b03f869.svg) | CID 6918852 | Ki | 50000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-erk1_ae7da5365c97b5164784d47f9074bd42.svg) | Benzamide, N-[4-[2-ethyl-4-(3-methylphenyl)-5-thiazolyl]-2-pyridinyl]- | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-erk1_298939ba2bdecf0f92f08e04bb796b27.svg) | 4-(7-Butyl-5H-pyrrolo[2,3-b]pyrazin-6-yl)phenol | IC50 | 18000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-erk1_f556b5bb65759c4a8d3410b88a5c8036.svg) | JNK Inhibitor V | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-erk1_478f8c74275fce83224a96edad0f0b1f.svg) | JNK Inhibitor VIII | Ki | 9200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-erk1_35d494726d3aaaac988a7ed448c35386.svg) | Bms-509744 | IC50 | 50000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-erk1_304d06e84e3237dcbaeea09a8542d685.svg) | Ravoxertinib | IC50 | 1.2 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-erk1_a97274caafef70d6423d3784397e9e54.svg) | Pyrimidone, 22 | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-erk1_c00f358adfafbd4bbc64f30e0249d7f9.svg) | (2S,3S)-3-((7-(Benzylamino)-3-isopropylpyrazolo[1,5-a]pyrimidin-5-yl)amino)butane-1,2,4-triol | IC50 | 3730.0 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-erk1_08cd44ca6baf1c92d36805c6a0f107ba.svg) | 3-Phenyl-1H-benzofuro[3,2-c]pyrazole | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-erk1_64f69317c84e5d1efc4211ef1e986fd2.svg) | 2-(4-Fluoroanilino)-5-[3-fluoro-4-[6-methoxy-7-(3-morpholin-4-ylpropoxy)quinolin-4-yl]oxyphenyl]-3-methylpyrimidin-4-one | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-erk1_941408e43c25b505975eab00c707db56.svg) | 1-[2-Fluoro-4-(5-methylpyrrolo[3,2-d]pyrimidin-4-yl)oxyphenyl]-3-[3-(trifluoromethyl)phenyl]urea | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-erk1_829d9468648eaacd7ae7ad912dac6a2f.svg) | N-[4-(6,7-Dimethoxyquinolin-4-yl)oxy-3-fluorophenyl]-1,5-dimethyl-3-oxo-2-phenylpyrazole-4-carboxamide | IC50 | 25000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-erk1_5a2f74ef53822d2a4766d321b6b50c36.svg) | MEK Inhibitor II | IC50 | 82900.0 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-erk1_3ab9460b7e7b1792127981364b5a6a2c.svg) | N'-(Pyrrolidino[2,1-B]isoindolin-4-ON-8-YL)-N-(pyridin-2-YL)urea | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-erk1_ea9d6c9c2bf0abdaf81032668de58db2.svg) | CID 46203864 | IC50 | 980.0 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-erk1_672e7998b8a2d8ffbf57a9a8fcc11921.svg) | (2R)-2-[(2S)-4-[3-Chloro-5-fluoro-6-(2H-pyrazolo[3,4-b]pyridin-3-yl)pyridin-2-yl]piperazin-2-yl]-3-methylbutan-2-ol | Ki | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-erk1_3ad10dc665b32d2dd5b178b07d0345b6.svg) | CID 58282870 | IC50 | 20.0 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-erk1_c4efceda17e53de30b363a8b6106fac2.svg) | N-(4-Amino-5-cyano-6-ethoxypyridin-2-yl)acetamide | Ki | 9200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-erk1_18ebff72d22a098c48d4abdeb13a4425.svg) | Lck Inhibitor | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-erk1_d89c41ad743193c7f8074cc3d3b6aaa3.svg) | 1-(2,6-Dichlorophenyl)-5-(2,4-difluorophenyl)-7-(4-piperidinyl)-1,2,3,4-tetrahydroquinazoline-2-one | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-erk1_7b6d64791d06a7e25ffce6c3c06aa871.svg) | 2,2-Dimethyl-7-(2-oxo-3H-imidazo[4,5-b]pyridin-1-yl)-1-[(1R)-1-phenylethyl]-3H-quinazolin-4-one | IC50 | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-erk1_e5c7a1e990d1af735a4c6d894ba6d642.svg) | Methyl 6-bromo-2-[(4-methylsulfonylphenyl)methyl]-1-oxo-4-phenylisoquinoline-3-carboxylate | IC50 | 11000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-erk1_3c615ad4ec6733825262ded1f3feba79.svg) | Meridianin E | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-erk1_25e94391e6ab6e12cda7b793ebb7c941.svg) | (E)-3-[4-[[[8-Carbamoyl-7-(3,5-dimethoxyanilino)imidazo[1,2-c]pyrimidin-5-yl]amino]methyl]phenyl]prop-2-enoic acid | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-erk1_c2aa7e0fb640ea7529d7330460976868.svg) | N-(4-Amino-5-cyano-6-ethoxypyridin-2-yl)-2-(2,5-dimethoxy-4-methylsulfonylphenyl)acetamide | Ki | 9200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-erk1_98598461b658b3f77425e67c797f8e2d.svg) | N-(4-Amino-5-chloro-6-ethoxypyridin-2-yl)-2-(4-methanesulfonyl-2,5-dimethoxyphenyl)acetamide | Ki | 9200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-erk1_a3bd9a5a28d4f4d2890ccf5cdf08d883.svg) | N-(4-Amino-5-cyano-6-isopropoxypyridin-2-yl)-2-(4-methanesulfonyl-2,5-dimethoxyphenyl)acetamide | Ki | 9200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-erk1_cde4e83180955e4849d8daba0837480d.svg) | N-(4-Amino-5-cyano-6-phenylpyridin-2-yl)acetamide | Ki | 9200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-erk1_7c30e90d304584aca2af8f794a12065e.svg) | 3-[2-(Pyridin-4-yl)-1,3-thiazol-4-yl]-1,2,3,4-tetrahydroquinazolin-2-one | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-erk1_dbc9774b4a10efc12e4d4309ee79f133.svg) | (13R,15S)-13-Methyl-16-oxa-8,9,12,22,24-pentazahexacyclo[15.6.2.16,9.112,15.02,7.021,25]heptacosa-1(24),2,4,6,17,19,21(25)-heptaene-23,27-dione | IC50 | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-erk1_8000c616960fd23cc7d5fdbb814a2f51.svg) | 3-[[[5-[1-(4-Methoxyphenyl)-1H-benzimidazol-6-yl]-1,3,4-oxadiazol-2-yl]thio]methyl]benzonitrile | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-erk1_58e0f004399fa00020a80ebd24cf76c1.svg) | [4-[[4-(3H-Benzimidazol-5-ylamino)-5-(trifluoromethyl)pyrimidin-2-yl]amino]-2-(cyanoamino)phenyl]cyanamide | IC50 | 300.0 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-erk1_622cd66903907f6e5eba8bda4305faf4.svg) | 2-N-(3H-Benzimidazol-5-yl)-4-N-(2-chlorophenyl)-5-(trifluoromethyl)pyrimidine-2,4-diamine | IC50 | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-erk1_a7ee75d4a7ce2e8d7ffa73cb444c324f.svg) | 5-(2-Amino-[1,2,4]triazolo[1,5-a]pyridin-7-yl)-N-tert-butylpyridine-3-sulfonamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-erk1_d53ca9729006e87596f190305485c7fe.svg) | 3-[1-(2-Imidazol-1-ylethyl)pyrazolo[3,4-b]pyridin-3-yl]-4-(1-methylindol-3-yl)pyrrole-2,5-dione | IC50 | 40000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-erk1_33e2eec82c4ed1aa33988b797bae80cc.svg) | 4-(4-Fluorophenyl)-N-[4-[3-[2-(methylamino)pyrimidin-4-yl]pyridin-2-yl]oxyphenyl]phthalazin-1-amine | IC50 | 25000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-erk1_400786f64062ecb5f10a9d3b11455207.svg) | 1-[5-Tert-butyl-3-[4-[2-(dimethylamino)ethyl]-5-oxo-1,4-diazepane-1-carbonyl]thiophen-2-yl]-3-(2,3-dichlorophenyl)urea | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-erk1_11d818e3086ce5d39d78d510661212e9.svg) | (3S)-N-[3-(4-Fluorophenyl)-1H-indazol-5-yl]-3-methylsulfanyl-1-[2-oxo-2-[4-(4-pyrimidin-2-ylphenyl)piperazin-1-yl]ethyl]pyrrolidine-3-carboxamide | IC50 | 25.0 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-erk1_75293a46b3079142e461cb328c482eda.svg) | Erk2 IN-1 | IC50 | 41.0 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-erk1_a69bed54275cb7e9f961910926c60794.svg) | N-[4-Chloro-3-(pyridin-3-yloxymethyl)phenyl]-3-fluoro-5-morpholin-4-ylbenzamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-erk1_51153882d3ab9f3566d96aeaf5c3eeab.svg) | 6-(2,4-Difluorophenyl)sulfonyl-2-(1H-indol-5-ylamino)-8-methylpyrido[2,3-d]pyrimidin-7-one | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-erk1_ef431bf27ff7842bbb4caafd947b43c7.svg) | Tilfrinib | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-erk1_b70290ebd844088252ff93f48253035f.svg) | [4-Amino-2-[4-(4-methylpiperazin-1-yl)anilino]-1,3-thiazol-5-yl]-(2,3-dihydro-1,4-benzodioxin-6-yl)methanone | IC50 | 100000000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-erk1_9cbc28ec8163d7ff921431afafc8af6c.svg) | Ethyl (E)-3-[4-[[[8-carbamoyl-7-(3,5-dimethoxyanilino)imidazo[1,2-c]pyrimidin-5-yl]amino]methyl]phenyl]prop-2-enoate | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-erk1_36aa00832b05a256d32e6330880d1520.svg) | 7-(Morpholin-4-ylmethyl)-3-[2-(pyridin-4-yl)-1,3-thiazol-4-yl]-1,2,3,4-tetrahydroquinazolin-2-one | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-erk1_e879126e9d744e7d1ff690817ee491a0.svg) | (4S,6Z,9S,10R,12E)-9,10,18-Trihydroxy-16-methoxy-4-methyl-3-oxabicyclo[12.4.0]octadeca-1(14),6,12,15,17-pentaene-2,8-dione | IC50 | 1400.0 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-erk1_da63de9d92c2d79ff40b1d8ee8ae24af.svg) | 3-[5-Chloro-4-[(2,4-difluorophenyl)methoxy]-6-oxopyrimidin-1-yl]-N-(2-hydroxyethyl)-4-methylbenzamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-erk1_61551f1612b1d03b33f689e3fdae85ae.svg) | 2-[3-(Methanesulfonamido)phenyl]-N-[4-(1H-pyrrolo[2,3-b]pyridin-3-yl)-1,3-thiazol-2-yl]acetamide | Ki | 2900.0 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-erk1_5b63ea15265b993819abd00ed6f2eee3.svg) | 2-[3-[3-(4-Methylpiperazin-1-yl)propoxy]phenyl]-N-[4-(1H-pyrrolo[2,3-b]pyridin-3-yl)-1,3-thiazol-2-yl]acetamide | Ki | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-erk1_af91a24eed916fe3d15fe15b067cac22.svg) | 2-[4-[(Z)-[1-(3-Methoxyphenyl)-5-oxo-2-phenylimidazol-4-ylidene]methyl]phenoxy]-N-phenylacetamide | IC50 | 65.0 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-erk1_519ab9602dc02666f62cfd91996215ce.svg) | 2-[4-[(Z)-[1-(3-Methoxyphenyl)-5-oxo-2-phenylimidazol-4-ylidene]methyl]phenoxy]-N-(2-methylphenyl)acetamide | IC50 | 43.0 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-erk1_253b9dec209663a66090ef7f25293b8e.svg) | 2-[4-[(Z)-[1-(3-Methoxyphenyl)-5-oxo-2-phenylimidazol-4-ylidene]methyl]phenoxy]-N-(3-methylphenyl)acetamide | IC50 | 20.0 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-erk1_bed65f01d22c0c738d153d617731bbf2.svg) | 2-[4-[(Z)-[1-(3-Methoxyphenyl)-5-oxo-2-phenylimidazol-4-ylidene]methyl]phenoxy]-N-(4-methylphenyl)acetamide | IC50 | 25.0 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-erk1_261c2a63fc6dde9ec34f017c5279ee80.svg) | N-(2-Methoxyphenyl)-2-[4-[(Z)-[1-(3-methoxyphenyl)-5-oxo-2-phenylimidazol-4-ylidene]methyl]phenoxy]acetamide | IC50 | 46.0 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-erk1_66e16232b364bba658e82470eeeb7804.svg) | N-(3-Methoxyphenyl)-2-[4-[(Z)-[1-(3-methoxyphenyl)-5-oxo-2-phenylimidazol-4-ylidene]methyl]phenoxy]acetamide | IC50 | 57.0 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-erk1_43bf930c5cc01b94e16b73043276b283.svg) | N-(4-Methoxyphenyl)-2-[4-[(Z)-[1-(3-methoxyphenyl)-5-oxo-2-phenylimidazol-4-ylidene]methyl]phenoxy]acetamide | IC50 | 76.0 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-erk1_0f9d09a18c6406a12e361b4fb58e571f.svg) | N-(2-Chlorophenyl)-2-[4-[(Z)-[1-(3-methoxyphenyl)-5-oxo-2-phenylimidazol-4-ylidene]methyl]phenoxy]acetamide | IC50 | 87.0 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-erk1_b5a05298b34e7a8a2b4ce28b96a1f053.svg) | N-(3-Chlorophenyl)-2-[4-[(Z)-[1-(3-methoxyphenyl)-5-oxo-2-phenylimidazol-4-ylidene]methyl]phenoxy]acetamide | IC50 | 89.0 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-erk1_cea478589564633353fd1ce58c86749b.svg) | N-(4-Chlorophenyl)-2-[4-[(Z)-[1-(3-methoxyphenyl)-5-oxo-2-phenylimidazol-4-ylidene]methyl]phenoxy]acetamide | IC50 | 95.0 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-erk1_8d837fd2526be26c613e1165ee61b164.svg) | 2-[4-[(Z)-[1-(4-Methoxyphenyl)-5-oxo-2-phenylimidazol-4-ylidene]methyl]phenoxy]-N-phenylacetamide | IC50 | 23.0 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-erk1_b1f777be64950cb4348288f124a21fce.svg) | 2-[4-[(Z)-[1-(4-Methoxyphenyl)-5-oxo-2-phenylimidazol-4-ylidene]methyl]phenoxy]-N-(2-methylphenyl)acetamide | IC50 | 32.0 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-erk1_d16be993f69f14d69e13ac68d76250ad.svg) | 2-[4-[(Z)-[1-(4-Methoxyphenyl)-5-oxo-2-phenylimidazol-4-ylidene]methyl]phenoxy]-N-(3-methylphenyl)acetamide | IC50 | 89.0 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-erk1_b9de6eb2ab34036dc35c720bac533cb9.svg) | 2-[4-[(Z)-[1-(4-Methoxyphenyl)-5-oxo-2-phenylimidazol-4-ylidene]methyl]phenoxy]-N-(4-methylphenyl)acetamide | IC50 | 23.0 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-erk1_45e72f62c769508d165c54901ad278e0.svg) | N-(2-Methoxyphenyl)-2-[4-[(Z)-[1-(4-methoxyphenyl)-5-oxo-2-phenylimidazol-4-ylidene]methyl]phenoxy]acetamide | IC50 | 43.0 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-erk1_b7e0a85602452fc76f1713570f8d8cb6.svg) | N-(3-Methoxyphenyl)-2-[4-[(Z)-[1-(4-methoxyphenyl)-5-oxo-2-phenylimidazol-4-ylidene]methyl]phenoxy]acetamide | IC50 | 21.0 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-erk1_82184f976d3ab2d0f2d3070f7a0ef667.svg) | N-(4-Methoxyphenyl)-2-[4-[(Z)-[1-(4-methoxyphenyl)-5-oxo-2-phenylimidazol-4-ylidene]methyl]phenoxy]acetamide | IC50 | 23.0 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-erk1_e8bc25cc3da75754e950cfb34364dd21.svg) | N-(2-Chlorophenyl)-2-[4-[(Z)-[1-(4-methoxyphenyl)-5-oxo-2-phenylimidazol-4-ylidene]methyl]phenoxy]acetamide | IC50 | 24.0 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-erk1_ad8f5f0efaf51fb046e98dcd47be915a.svg) | N-(3-Chlorophenyl)-2-[4-[(Z)-[1-(4-methoxyphenyl)-5-oxo-2-phenylimidazol-4-ylidene]methyl]phenoxy]acetamide | IC50 | 35.0 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-erk1_46b7d8a67d891b743cd0a6b4236d4c9d.svg) | N-(4-Chlorophenyl)-2-[4-[(Z)-[1-(4-methoxyphenyl)-5-oxo-2-phenylimidazol-4-ylidene]methyl]phenoxy]acetamide | IC50 | 47.0 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-erk1_a712b7503d03ee30b6a396b2ba67d9a2.svg) | 1-[4-Chloro-3-(trifluoromethyl)phenyl]-3-[2-methyl-4-[6-(methylamino)pyrimidin-4-yl]oxyphenyl]urea | IC50 | 3100.0 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-erk1_310f06cd6330b8ac8dea0294d98c11f3.svg) | 3-(2-Methylpyridin-4-yl)-N-[(2,3,5-trichloropyridin-4-yl)methyl]-1H-indazole-5-carboxamide | IC50 | 16.7 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-erk1_80a459834a533b4821cfa86c85d2067a.svg) | N-[(3-Chlorophenyl)methyl]-3-pyridin-4-yl-1H-indazole-5-carboxamide | IC50 | 74.2 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-erk1_ffeec205435c54cebc29a02901ee7894.svg) | N-[1-(3-Chlorophenyl)ethyl]-3-pyridin-4-yl-1H-indazole-5-carboxamide | IC50 | 154.0 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-erk1_7984c74398fadf15d4947ffe3ceb9857.svg) | N-[1-(3-Chlorophenyl)propyl]-3-pyridin-4-yl-1H-indazole-5-carboxamide | IC50 | 78.7 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-erk1_6507c5e17385f68ba377c0698dfe3ed8.svg) | N-[(1S)-1-(3-Chlorophenyl)-2-hydroxyethyl]-3-pyridin-4-yl-1H-indazole-5-carboxamide | IC50 | 26.3 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-erk1_0d826b48221a700cb51d23ad10b35ff2.svg) | N-[(1R)-1-(3-Chlorophenyl)-2-hydroxyethyl]-3-pyridin-4-yl-1H-indazole-5-carboxamide | IC50 | 833.0 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-erk1_059bd54d7e12dc52a8e1729c0f618f61.svg) | N-[(1S)-1-(2,6-Dichlorophenyl)ethyl]-3-(2-methylpyridin-4-yl)-1H-indazole-5-carboxamide | IC50 | 19.4 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-erk1_c50c08979c711c02bd47c03d6d9f407c.svg) | N-[1-(2-Chlorophenyl)ethyl]-3-pyridin-4-yl-1H-indazole-5-carboxamide | IC50 | 35.9 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-erk1_5af645dd772ccf22e189e07572c19deb.svg) | N-[(2-Chlorophenyl)methyl]-3-pyridin-4-yl-1H-indazole-5-carboxamide | IC50 | 46.3 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-erk1_db8c729fdaeca1ef9c8b36143c2624d1.svg) | N-[(2,4-Dichloro-3-fluorophenyl)methyl]-3-pyridin-4-yl-1H-indazole-5-carboxamide | IC50 | 29.2 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-erk1_7c72c07012331ed4e4243ec03a5db177.svg) | N-[1-(3-Chlorophenyl)-2-hydroxyethyl]-3-pyridin-4-yl-1H-indazole-5-carboxamide | IC50 | 72.4 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-erk1_8fc2fa1bb73bc7d85150391b7f8e4ab9.svg) | N-[1-(3-Chlorophenyl)-2-hydroxyethyl]-3-(2-methylpyridin-4-yl)-1H-indazole-5-carboxamide | IC50 | 53.4 [1] |
![](https://images.aatbio.com/dataset/ic50/map-kinase-erk1_a3779167401788fc337254fa56a17e4d.svg) | N-(3-Phenylpropyl)-3-pyridin-4-yl-1H-indazole-5-carboxamide | IC50 | 42.9 [1] |