![](https://images.aatbio.com/dataset/ic50/macrophage-stimulating-protein-receptor_173905a1d8206fe6271a8ee9486c99d9.svg) | Foretinib | IC50 | 3.0 [1] |
![](https://images.aatbio.com/dataset/ic50/macrophage-stimulating-protein-receptor_008b82bfee0baa55c0bab6b3c3e488d2.svg) | N-[3-Fluoro-4-[2-(1-methylimidazol-4-yl)thieno[3,2-b]pyridin-7-yl]oxyphenyl]-1-phenyl-5-(trifluoromethyl)pyrazole-4-carboxamide | IC50 | 12.0 [1] |
![](https://images.aatbio.com/dataset/ic50/macrophage-stimulating-protein-receptor_1d5eba4b4bb57896dda18b1604bab021.svg) | Staurosporine | IC50 | 102.7 [1], 326.0 [2], 442.5 [3] |
![](https://images.aatbio.com/dataset/ic50/macrophage-stimulating-protein-receptor_35e47530605128bdf6619cacfd802af2.svg) | N-[3-Fluoro-4-[2-(1-methylimidazol-4-yl)thieno[3,2-b]pyridin-7-yl]oxyphenyl]-N-methyl-1-phenyl-5-(trifluoromethyl)pyrazole-4-carboxamide | IC50 | 575.0 [1], 580.0 [2] |
![](https://images.aatbio.com/dataset/ic50/macrophage-stimulating-protein-receptor_4af080018fcfdd3453abbbc05a2c39a3.svg) | N-[4-(6,7-Dimethoxyquinolin-4-yl)oxy-3-fluorophenyl]-1-phenyl-5-(trifluoromethyl)pyrazole-4-carboxamide | IC50 | 16.0 [1], 80.0 [2] |
![](https://images.aatbio.com/dataset/ic50/macrophage-stimulating-protein-receptor_44aa3a6da7f2767bb07774343291b239.svg) | 4-[6-Amino-7-[(1R)-1-(2,6-dichloro-3-fluorophenyl)ethoxy]furo[3,2-c]pyridin-3-yl]-3,6-dihydro-2H-pyridine-1-carboxamide | IC50 | 25.0 [1], 200.0 [2] |
![](https://images.aatbio.com/dataset/ic50/macrophage-stimulating-protein-receptor_a840767d7ddb2c27c40164419a996160.svg) | Infigratinib phosphate | IC50 | 2891.0 [1], 10000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/macrophage-stimulating-protein-receptor_c77eb69f87d46b4d00314a6bfb851cf8.svg) | Crizotinib | IC50 | 300.0 [1] |
![](https://images.aatbio.com/dataset/ic50/macrophage-stimulating-protein-receptor_7c1f47f3c7bae38fb065c983ece631c1.svg) | Vandetanib | IC50 | 3370.0 [1] |
![](https://images.aatbio.com/dataset/ic50/macrophage-stimulating-protein-receptor_9d111ca31c6b5557bbe95cc7cad92c76.svg) | Vatalanib | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/macrophage-stimulating-protein-receptor_8a69b3902a36c5bcb114db8f49f8eabe.svg) | Semaxanib | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/macrophage-stimulating-protein-receptor_34ec291e290db2e13648ccc8dee7e3a5.svg) | Cabozantinib | IC50 | 69.0 [1] |
![](https://images.aatbio.com/dataset/ic50/macrophage-stimulating-protein-receptor_0a83b01cf93719a90ccaeda771089c43.svg) | Doramapimod | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/macrophage-stimulating-protein-receptor_088eb7e3c0fbd58f12adde928af7d44f.svg) | Pha-665752 | IC50 | 68.0 [1] |
![](https://images.aatbio.com/dataset/ic50/macrophage-stimulating-protein-receptor_c38cbdee4404993837adfc282c860ec1.svg) | Nvp-tae 684 | IC50 | 1634.0 [1] |
![](https://images.aatbio.com/dataset/ic50/macrophage-stimulating-protein-receptor_e7ecb06887875f4d78baf892d82c33a5.svg) | Bms-777607 | IC50 | 1.8 [1] |
![](https://images.aatbio.com/dataset/ic50/macrophage-stimulating-protein-receptor_6218d7660845b31fc510a0466313fd99.svg) | Amg-458 | IC50 | 10.0 [1] |
![](https://images.aatbio.com/dataset/ic50/macrophage-stimulating-protein-receptor_aa4ae66a17e1730306dedb6ebaeee891.svg) | 2-(Pyridin-4-Ylmethylamino)-~{n}-[3-(Trifluoromethyl)phenyl]benzamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/macrophage-stimulating-protein-receptor_179888a64edb35ddee0be2a16e245b3a.svg) | MK-2461 | IC50 | 7.0 [1] |
![](https://images.aatbio.com/dataset/ic50/macrophage-stimulating-protein-receptor_a97274caafef70d6423d3784397e9e54.svg) | Pyrimidone, 22 | Ki | 195.0 [1] |
![](https://images.aatbio.com/dataset/ic50/macrophage-stimulating-protein-receptor_c1834625131d0c2ad0228dc67b109c54.svg) | MK-8033 | IC50 | 7.0 [1] |
![](https://images.aatbio.com/dataset/ic50/macrophage-stimulating-protein-receptor_64f69317c84e5d1efc4211ef1e986fd2.svg) | 2-(4-Fluoroanilino)-5-[3-fluoro-4-[6-methoxy-7-(3-morpholin-4-ylpropoxy)quinolin-4-yl]oxyphenyl]-3-methylpyrimidin-4-one | Ki | 28.0 [1] |
![](https://images.aatbio.com/dataset/ic50/macrophage-stimulating-protein-receptor_dced13dbc2c667b8afa41c93b72d7d74.svg) | 5'-Fluoroindirubinoxime | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/macrophage-stimulating-protein-receptor_5fdad235d88d47467d429d2ef1d29e33.svg) | CID 44155856 | IC50 | 3.0 [1] |
![](https://images.aatbio.com/dataset/ic50/macrophage-stimulating-protein-receptor_829d9468648eaacd7ae7ad912dac6a2f.svg) | N-[4-(6,7-Dimethoxyquinolin-4-yl)oxy-3-fluorophenyl]-1,5-dimethyl-3-oxo-2-phenylpyrazole-4-carboxamide | Ki | 1.0 [1] |
![](https://images.aatbio.com/dataset/ic50/macrophage-stimulating-protein-receptor_e07c8cd6f81fa23b777a36d7d9709688.svg) | 4-Tert-Butyl-N-[6-(1h-Imidazol-1-Yl)imidazo[1,2-A]pyridin-2-Yl]benzamide | IC50 | 19952.62 [1] |
![](https://images.aatbio.com/dataset/ic50/macrophage-stimulating-protein-receptor_aa78cc3183c29821fe7c015c8320a3ff.svg) | CID 44814409 | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/macrophage-stimulating-protein-receptor_0d9863ed59ccd1ba92b866d4ff4460aa.svg) | N-[3-Fluoro-4-[2-(1-methylimidazol-4-yl)thieno[3,2-b]pyridin-7-yl]oxyphenyl]-2-oxo-3-phenylimidazolidine-1-carboxamide | IC50 | 170.0 [1] |
![](https://images.aatbio.com/dataset/ic50/macrophage-stimulating-protein-receptor_5e317ff1d4c29361137032616d2a8b14.svg) | 2-Benzyl-5-{4-[(6,7-dimethoxyquinolin-4-yl)oxy]-3-fluorophenyl}-3-methylpyrimidin-4(3H)-one | Ki | 581.0 [1] |
![](https://images.aatbio.com/dataset/ic50/macrophage-stimulating-protein-receptor_628e796c331326ac7d59e9f8e229eaa5.svg) | 6,6-Dimethyl-8-[1-(oxan-4-ylmethyl)piperidin-4-yl]-11-oxo-5H-benzo[b]carbazole-3-carbonitrile | IC50 | 93.4 [1] |
![](https://images.aatbio.com/dataset/ic50/macrophage-stimulating-protein-receptor_0f45e39d61abf0ed403c69c6706b0181.svg) | 5-[4-(6,7-Dimethoxyquinolin-4-yl)oxy-3-fluorophenyl]-2-(4-fluoroanilino)-3-methylpyrimidin-4-one | Ki | 80.0 [1] |
![](https://images.aatbio.com/dataset/ic50/macrophage-stimulating-protein-receptor_3530c4babc83bff493a56acf99df81b0.svg) | 5-[3-Fluoro-4-[6-methoxy-7-(3-morpholin-4-ylpropoxy)quinolin-4-yl]oxyphenyl]-2-[(4-fluorophenyl)methyl]-3-methylpyrimidin-4-one | Ki | 706.0 [1] |
![](https://images.aatbio.com/dataset/ic50/macrophage-stimulating-protein-receptor_3967f1261f1958810b393b6f50ce9b27.svg) | 14-(Dimethylsulfamoylamino)-5-(1-methylpyrazol-4-yl)-2-oxo-7-azatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),4,6,9,12,14-heptaene | IC50 | 7.0 [1] |
![](https://images.aatbio.com/dataset/ic50/macrophage-stimulating-protein-receptor_482caccce5577424472b4f30ef45663d.svg) | [6-Chloro-4-methyl-3-[[3-(methylsulfamoylamino)phenyl]methyl]-2-oxochromen-7-yl] N,N-dimethylcarbamate | IC50 | 50000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/macrophage-stimulating-protein-receptor_95a0bd49e8f0995cb52a25e6fd825622.svg) | 4,4,4-Trifluoro-3-[3-fluoro-4-[2-(1-methylimidazol-4-yl)thieno[3,2-b]pyridin-7-yl]oxyanilino]-N-phenylbutanamide | IC50 | 1030.0 [1] |
![](https://images.aatbio.com/dataset/ic50/macrophage-stimulating-protein-receptor_65e02195d34f10978d83a4d3018943d5.svg) | 3-Anilino-4,4,4-trifluoro-N-[3-fluoro-4-[2-(1-methylimidazol-4-yl)thieno[3,2-b]pyridin-7-yl]oxyphenyl]butanamide | IC50 | 410.0 [1] |
![](https://images.aatbio.com/dataset/ic50/macrophage-stimulating-protein-receptor_a7ee75d4a7ce2e8d7ffa73cb444c324f.svg) | 5-(2-Amino-[1,2,4]triazolo[1,5-a]pyridin-7-yl)-N-tert-butylpyridine-3-sulfonamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/macrophage-stimulating-protein-receptor_fcca6043b08d60b7934c389a846b207f.svg) | 3-(4-Acetylpiperazin-1-yl)-5-(3-nitrobenzylamino)-7-(trifluoromethyl)quinoline | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/macrophage-stimulating-protein-receptor_dcf1cd66de7c1bdcab62160a0a9db4e0.svg) | N-[5-Amino-1-[(4-methoxyphenyl)methyl]pyrazol-4-yl]-5-[[4-chloro-3-(trifluoromethyl)phenyl]carbamoylamino]-2-methylbenzamide | IC50 | 277.1 [1] |
![](https://images.aatbio.com/dataset/ic50/macrophage-stimulating-protein-receptor_b47eb0b10c004af2684a6d610b4c991d.svg) | Ethyl 8-oxo-8H-acenaphtho[1,2-b]pyrrole-9-carboxylate | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/macrophage-stimulating-protein-receptor_f83aeef223e4cffa787f7bf871c66dc3.svg) | 1-(4-Fluorophenyl)-N-[3-fluoro-4-(5-phenylthieno[2,3-d]pyrimidin-4-yl)oxyphenyl]-2-oxopyridine-3-carboxamide | IC50 | 50.4 [1] |
![](https://images.aatbio.com/dataset/ic50/macrophage-stimulating-protein-receptor_400786f64062ecb5f10a9d3b11455207.svg) | 1-[5-Tert-butyl-3-[4-[2-(dimethylamino)ethyl]-5-oxo-1,4-diazepane-1-carbonyl]thiophen-2-yl]-3-(2,3-dichlorophenyl)urea | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/macrophage-stimulating-protein-receptor_bd7ab61fd74e87578c2dfefbcc47d031.svg) | 7,8-Dichloro-9-methyl-1-oxospiro[2,4-dihydropyrido[3,4-b]indole-3,4'-piperidine]-4-carbonitrile | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/macrophage-stimulating-protein-receptor_84ad2ce5fbf306770a6c850a5b17125a.svg) | 9-Cyclopentyl-N2-[4-(4-methylpiperazin-1-yl)phenyl]-N8-phenyl-purine-2,8-diamine | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/macrophage-stimulating-protein-receptor_5c1c042b05f26ce92f172346c957e7d0.svg) | N-(7-Methoxyquinolin-6-yl)thieno[3,2-d]pyrimidine-7-carboxamide | IC50 | 50000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/macrophage-stimulating-protein-receptor_51153882d3ab9f3566d96aeaf5c3eeab.svg) | 6-(2,4-Difluorophenyl)sulfonyl-2-(1H-indol-5-ylamino)-8-methylpyrido[2,3-d]pyrimidin-7-one | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/macrophage-stimulating-protein-receptor_77f4b74dc836b9bdb4b558af6f5da27f.svg) | 6-(6-Fluoroindol-1-yl)-2-[2-[7-(3-morpholin-4-ylpropoxy)quinolin-4-yl]oxyethyl]pyridazin-3-one | IC50 | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/macrophage-stimulating-protein-receptor_1eb9f67be328781c5c0ecf7e4b407b2b.svg) | 1-(2-Chlorophenyl)-N-[3-fluoro-4-[6-methoxy-7-(3-piperidin-1-ylpropoxy)quinolin-4-yl]oxyphenyl]triazole-4-carboxamide | IC50 | 345.7 [1] |
![](https://images.aatbio.com/dataset/ic50/macrophage-stimulating-protein-receptor_5b5057f07ba36d969b42e83280bc9205.svg) | 2-[3-(3-Piperidin-4-ylpropoxy)phenyl]-N-[4-(1H-pyrrolo[2,3-b]pyridin-3-yl)-1,3-thiazol-2-yl]acetamide | Ki | 2000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/macrophage-stimulating-protein-receptor_61551f1612b1d03b33f689e3fdae85ae.svg) | 2-[3-(Methanesulfonamido)phenyl]-N-[4-(1H-pyrrolo[2,3-b]pyridin-3-yl)-1,3-thiazol-2-yl]acetamide | Ki | 2000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/macrophage-stimulating-protein-receptor_9e00becee6f355fe8fb384fe33c8c3e7.svg) | 4-[4-(6-Benzyl-pyridazin-3-yl)-2-fluoro-phenoxy]-6,7-dimethoxy-quinoline | Ki | 79.0 [1] |
![](https://images.aatbio.com/dataset/ic50/macrophage-stimulating-protein-receptor_cd27a3b0136fe5b91b6c49045230013c.svg) | 2-[3-Fluoro-4-[6-methoxy-7-(3-pyrrolidin-1-ylpropoxy)quinolin-4-yl]oxyphenyl]-N-[(E)-[4-(trifluoromethyl)phenyl]methylideneamino]acetamide | IC50 | 28.6 [1] |
![](https://images.aatbio.com/dataset/ic50/macrophage-stimulating-protein-receptor_fc8fdbb1a10b7ab64261226840ec00c1.svg) | N-[3-Fluoro-4-[2-(1-methylimidazol-4-yl)thieno[3,2-b]pyridin-7-yl]oxyphenyl]-1-phenyl-2-(trifluoromethyl)pyrrole-3-carboxamide | IC50 | 10.0 [1] |
![](https://images.aatbio.com/dataset/ic50/macrophage-stimulating-protein-receptor_019fc703d3399d580d6ce5709c309ff0.svg) | N-[3-Fluoro-4-[2-(1-methylimidazol-4-yl)thieno[3,2-b]pyridin-7-yl]oxyphenyl]-1-phenyl-5-(trifluoromethyl)imidazole-4-carboxamide | IC50 | 13.0 [1] |
![](https://images.aatbio.com/dataset/ic50/macrophage-stimulating-protein-receptor_bc3d75a4a41b9ce86555a7ffb4313cf7.svg) | N-[3-Fluoro-4-[2-(1-methylimidazol-4-yl)thieno[3,2-b]pyridin-7-yl]oxyphenyl]-1-phenyl-5-(trifluoromethyl)triazole-4-carboxamide | IC50 | 17.0 [1] |
![](https://images.aatbio.com/dataset/ic50/macrophage-stimulating-protein-receptor_33bb2ae60d1db1156db30426f2ab075b.svg) | N-[3-Fluoro-4-[2-(1-methylimidazol-4-yl)thieno[3,2-b]pyridin-7-yl]oxyphenyl]-1-phenyl-3-(trifluoromethyl)pyrazole-4-carboxamide | IC50 | 95.0 [1] |
![](https://images.aatbio.com/dataset/ic50/macrophage-stimulating-protein-receptor_d4dcb90de9d4313a829148276af523b0.svg) | N-[3-Fluoro-4-[2-(1-methylimidazol-4-yl)thieno[3,2-b]pyridin-7-yl]oxyphenyl]-1-(4-fluorophenyl)-5-(trifluoromethyl)pyrazole-4-carboxamide | IC50 | 44.0 [1] |
![](https://images.aatbio.com/dataset/ic50/macrophage-stimulating-protein-receptor_b6faf72dfa81ac6f5cbbee7518dcb7f6.svg) | 4-[6-(Benzylamino)imidazo[1,2-B]pyridazin-3-Yl]benzonitrile | IC50 | 6100.0 [1] |
![](https://images.aatbio.com/dataset/ic50/macrophage-stimulating-protein-receptor_07f245678e6fcc2d52455f8c1a6544d0.svg) | 2-[4-[4-[6-[(2R)-2-(3-Fluorophenyl)pyrrolidin-1-yl]imidazo[1,2-b]pyridazin-3-yl]pyridin-2-yl]piperazin-1-yl]acetic acid | IC50 | 5000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/macrophage-stimulating-protein-receptor_cadcfe40c75731fb4d071e8664de359c.svg) | 1-[4-[6-[(2R)-2-(3-Fluorophenyl)pyrrolidin-1-yl]imidazo[1,2-b]pyridazin-3-yl]pyridin-2-yl]piperidin-4-ol | IC50 | 4800.0 [1] |
![](https://images.aatbio.com/dataset/ic50/macrophage-stimulating-protein-receptor_9d0079a827d9ee8e20f8d60ef6b71b04.svg) | 3-(2-Chlorophenyl)-N-[3-fluoro-4-[6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinolin-4-yl]oxyphenyl]-4-methyl-2-oxo-1H-imidazole-5-carboxamide | IC50 | 270.0 [1] |
![](https://images.aatbio.com/dataset/ic50/macrophage-stimulating-protein-receptor_ce57f652e429810e18086b4ce709d38a.svg) | N-[3-Fluoro-4-[2-(1-methylimidazol-4-yl)thieno[3,2-b]pyridin-7-yl]oxyphenyl]-1,5-diphenylpyrazole-4-carboxamide | IC50 | 23.0 [1] |
![](https://images.aatbio.com/dataset/ic50/macrophage-stimulating-protein-receptor_49e79a52654f6745b95a75363b629e6e.svg) | N-[3-Fluoro-4-[2-(1-methylimidazol-4-yl)thieno[3,2-b]pyridin-7-yl]oxyphenyl]-1,3-diphenylpyrazole-4-carboxamide | IC50 | 32.0 [1] |
![](https://images.aatbio.com/dataset/ic50/macrophage-stimulating-protein-receptor_cbea69b7d7587a81745b8820dc641354.svg) | N-[3-Fluoro-4-[2-(1-methylimidazol-4-yl)thieno[3,2-b]pyridin-7-yl]oxyphenyl]-2,4-diphenyl-1,3-thiazole-5-carboxamide | IC50 | 45.0 [1] |
![](https://images.aatbio.com/dataset/ic50/macrophage-stimulating-protein-receptor_937d13a4663bbca11a25b1ac62eda422.svg) | N-[3-Fluoro-4-[2-(1-methylimidazol-4-yl)thieno[3,2-b]pyridin-7-yl]oxyphenyl]-1,5-diphenylpyrrole-3-carboxamide | IC50 | 101.0 [1] |
![](https://images.aatbio.com/dataset/ic50/macrophage-stimulating-protein-receptor_dce93bb0a333cde14607bf7fecab190f.svg) | N-[3-Fluoro-4-[2-(1-methylimidazol-4-yl)thieno[3,2-b]pyridin-7-yl]oxyphenyl]-5-(2-fluorophenyl)-1-phenylpyrazole-4-carboxamide | IC50 | 25.0 [1] |
![](https://images.aatbio.com/dataset/ic50/macrophage-stimulating-protein-receptor_a392144d06e28871e645fb2ab9eece76.svg) | N-[3-Fluoro-4-[2-(1-methylimidazol-4-yl)thieno[3,2-b]pyridin-7-yl]oxyphenyl]-1-phenyl-5-pyridin-2-ylpyrazole-4-carboxamide | IC50 | 23.0 [1] |
![](https://images.aatbio.com/dataset/ic50/macrophage-stimulating-protein-receptor_7b455461f114dda50ec7394f0a707465.svg) | N-[3-Fluoro-4-[2-(1-methylimidazol-4-yl)thieno[3,2-b]pyridin-7-yl]oxyphenyl]-5-(3-methoxyphenyl)-1-phenylpyrazole-4-carboxamide | IC50 | 27.0 [1] |
![](https://images.aatbio.com/dataset/ic50/macrophage-stimulating-protein-receptor_bca8a9efcfb4c5eb3dd7245b3a68c747.svg) | N-[3-Fluoro-4-[2-(1-methylimidazol-4-yl)thieno[3,2-b]pyridin-7-yl]oxyphenyl]-1-phenyl-5-pyridin-3-ylpyrazole-4-carboxamide | IC50 | 14.0 [1] |
![](https://images.aatbio.com/dataset/ic50/macrophage-stimulating-protein-receptor_64c6fa795c5f161c8c61c274348d5340.svg) | 5-[3-Fluoro-4-[2-(1-methylimidazol-4-yl)thieno[3,2-b]pyridin-7-yl]oxyphenyl]-1-phenyl-6H-pyrazolo[4,3-c]azepin-4-one | IC50 | 49.0 [1] |
![](https://images.aatbio.com/dataset/ic50/macrophage-stimulating-protein-receptor_d8cdd1cfcb8cfe08a6efe38eb8f48150.svg) | 5-[3-Fluoro-4-[2-(1-methylimidazol-4-yl)thieno[3,2-b]pyridin-7-yl]oxyphenyl]-1-phenyl-7,8-dihydro-6H-pyrazolo[4,3-c]azepin-4-one | IC50 | 34.0 [1] |
![](https://images.aatbio.com/dataset/ic50/macrophage-stimulating-protein-receptor_870e48430d670623c62a9b1fba164eb9.svg) | 5-[3-Fluoro-4-[2-(1-methylimidazol-4-yl)thieno[3,2-b]pyridin-7-yl]oxyphenyl]-1-phenyl-6,7-dihydropyrazolo[4,3-c]pyridin-4-one | IC50 | 30.0 [1] |
![](https://images.aatbio.com/dataset/ic50/macrophage-stimulating-protein-receptor_574a45544e8cb1fe403e1c65b194818e.svg) | 6-(1-Methylpyrazol-4-yl)-2-[[3-[[5-(1-methylpyrazol-4-yl)pyrimidin-2-yl]amino]phenyl]methyl]pyridazin-3-one | IC50 | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/macrophage-stimulating-protein-receptor_095fdd82a4a20d96c83b3b6059843827.svg) | N-[3-Fluoro-4-[6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinolin-4-yl]oxyphenyl]-4-(4-fluorophenyl)-3-oxoquinoxaline-2-carboxamide | IC50 | 82.56 [1] |
![](https://images.aatbio.com/dataset/ic50/macrophage-stimulating-protein-receptor_1a1d2c0e05cf497a481bc9bdb9924538.svg) | N-[3-Fluoro-4-[6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinolin-4-yl]oxyphenyl]-1-(2-fluorophenyl)-4-methyl-5-oxo-1,2,4-triazole-3-carboxamide | IC50 | 140.72 [1] |
![](https://images.aatbio.com/dataset/ic50/macrophage-stimulating-protein-receptor_c4b2bbc8da3445973fd48f1caf9c3c0a.svg) | c-Met-IN-2 | IC50 | 731.0 [1] |
![](https://images.aatbio.com/dataset/ic50/macrophage-stimulating-protein-receptor_d17996d869706c9d32d18da9e09eca11.svg) | 1-[3-Fluoro-4-[6-methoxy-7-(3-piperidin-1-ylpropoxy)quinolin-4-yl]oxyphenyl]-3-[(E)-(2-hydroxy-3-prop-2-enylphenyl)methylideneamino]urea | IC50 | 14.5 [1] |
![](https://images.aatbio.com/dataset/ic50/macrophage-stimulating-protein-receptor_da047ffc419503aaf95a9fdc33a2b601.svg) | 5-[3-Fluoro-4-[2-(1-methylimidazol-4-yl)thieno[3,2-b]pyridin-7-yl]oxyphenyl]-1-phenyl-6,8-dihydropyrazolo[3,4-e][1,4]diazepine-4,7-dione | IC50 | 361.0 [1] |
![](https://images.aatbio.com/dataset/ic50/macrophage-stimulating-protein-receptor_757cdf5ddd5e72c0e265b6e51e4dab1b.svg) | N-[1-(2-Methoxyethyl)pyrazol-4-yl]-2-(4-propan-2-yl-1,2,4-triazol-3-yl)-1,3-thiazole-4-carboxamide | IC50 | 19952.62 [1] |
![](https://images.aatbio.com/dataset/ic50/macrophage-stimulating-protein-receptor_18dfe79111a4a456aa52f2e484e47921.svg) | 1-[2-(2,6-Difluorophenyl)-4-oxo-1,3-thiazolidin-3-yl]-3-[2-fluoro-4-[6-methoxy-7-(3-pyrrolidin-1-ylpropoxy)quinolin-4-yl]oxyphenyl]urea | IC50 | 3.1 [1] |
![](https://images.aatbio.com/dataset/ic50/macrophage-stimulating-protein-receptor_a0af8d0e22a6427fec980f348a0adf45.svg) | 2-Methyl-N-[2-[4-(4-methylpiperazin-1-yl)anilino]pyrimidin-5-yl]-5-[[3-(trifluoromethyl)benzoyl]amino]benzamide | IC50 | 25000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/macrophage-stimulating-protein-receptor_a6a4c7f2143c80500bf54f909f9074c9.svg) | 2-(4-Fluoroanilino)-5-[5-[6-methoxy-7-(3-morpholin-4-ylpropoxy)quinolin-4-yl]oxypyridin-2-yl]-3-methylpyrimidin-4-one | Ki | 1.3 [1] |
![](https://images.aatbio.com/dataset/ic50/macrophage-stimulating-protein-receptor_581faf9c3edc19cf2627b4526aa02d17.svg) | N-[3-Fluoro-4-[2-(1-methylimidazol-2-yl)thieno[3,2-b]pyridin-7-yl]oxyphenyl]-1-phenyl-5-(trifluoromethyl)pyrazole-4-carboxamide | IC50 | 60.0 [1] |
![](https://images.aatbio.com/dataset/ic50/macrophage-stimulating-protein-receptor_3744f98eb62cad5ba77ae3fb4e3eeb08.svg) | N-[3-Fluoro-4-[2-(1-methylimidazol-4-yl)thieno[3,2-b]pyridin-7-yl]oxyphenyl]-5-methyl-1-phenylpyrazole-4-carboxamide | IC50 | 150.0 [1] |
![](https://images.aatbio.com/dataset/ic50/macrophage-stimulating-protein-receptor_5b830edc926b2120187bc7b936ddcd55.svg) | N-[3-Fluoro-4-[2-(1-methylimidazol-4-yl)thieno[3,2-b]pyridin-7-yl]oxyphenyl]-1-phenylpyrazole-4-carboxamide | IC50 | 590.0 [1] |
![](https://images.aatbio.com/dataset/ic50/macrophage-stimulating-protein-receptor_7ed40b44e2a306748b3d1093575009ac.svg) | N-[3-Fluoro-4-[2-(1-methylimidazol-4-yl)thieno[3,2-b]pyridin-7-yl]oxyphenyl]-1-methyl-5-(trifluoromethyl)pyrazole-4-carboxamide | IC50 | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/macrophage-stimulating-protein-receptor_58018f60837f6817eb1a823ec52c51eb.svg) | 5-Amino-N-[3-fluoro-4-[2-(1-methylimidazol-4-yl)thieno[3,2-b]pyridin-7-yl]oxyphenyl]-1-phenylpyrazole-4-carboxamide | IC50 | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/macrophage-stimulating-protein-receptor_d6402ff78ab6cfe13b10229e239b9dee.svg) | N-[4-[2-[4-[[Acetyl-[(2S)-1-methoxypropan-2-yl]amino]methyl]phenyl]thieno[3,2-b]pyridin-7-yl]oxy-3-fluorophenyl]-1-phenyl-5-(trifluoromethyl)pyrazole-4-carboxamide | IC50 | 60.0 [1] |
![](https://images.aatbio.com/dataset/ic50/macrophage-stimulating-protein-receptor_1ae9a65fd5679eef9354305aebe41f5e.svg) | N-(3-Isoquinolin-4-yl-phenyl)-2-[(pyridin-4-ylmethyl)-amino]-benzamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/macrophage-stimulating-protein-receptor_04dbcf7af04440bd78309a37caffa5d5.svg) | (R)-6-(1-(2,6-Dichloro-3-fluorophenyl)ethoxy)quinoline | IC50 | 3600.0 [1] |
![](https://images.aatbio.com/dataset/ic50/macrophage-stimulating-protein-receptor_e9567a5f3376da1cdb468430ffe1f86a.svg) | (E)-3-[6-[(1R)-1-(2,6-Dichloro-3-fluorophenyl)ethoxy]quinolin-3-yl]prop-2-enamide | IC50 | 450.0 [1] |
![](https://images.aatbio.com/dataset/ic50/macrophage-stimulating-protein-receptor_072c551bbafb20960465c20cfbd4e5d9.svg) | 2-(6-((R)-1-(2,6-Dichloro-3-fluorophenyl)ethoxy)quinolin-3-yl)cyclopropanecarboxamide | IC50 | 230.0 [1] |
![](https://images.aatbio.com/dataset/ic50/macrophage-stimulating-protein-receptor_df55b9ba10508e517acb9c3a2aa4cc02.svg) | 1-Tert-butyl-N-[3-fluoro-4-[2-(1-methylimidazol-4-yl)thieno[3,2-b]pyridin-7-yl]oxyphenyl]-5-(trifluoromethyl)pyrazole-4-carboxamide | IC50 | 200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/macrophage-stimulating-protein-receptor_01efc63ce344c81020ac9e088c1c88e5.svg) | N-[3-Fluoro-4-[2-[4-[(2-methylsulfonylethylamino)methyl]phenyl]thieno[3,2-b]pyridin-7-yl]oxyphenyl]-1-phenyl-5-(trifluoromethyl)pyrazole-4-carboxamide | IC50 | 80.0 [1] |
![](https://images.aatbio.com/dataset/ic50/macrophage-stimulating-protein-receptor_1e194ebe61a7230d69aa071560c44aed.svg) | N-[4-[2-[4-(Dimethylcarbamoyl)phenyl]thieno[3,2-b]pyridin-7-yl]oxy-3-fluorophenyl]-1-phenyl-5-(trifluoromethyl)pyrazole-4-carboxamide | IC50 | 30.0 [1] |
![](https://images.aatbio.com/dataset/ic50/macrophage-stimulating-protein-receptor_ca237125180ba5b54895a9e9d25aa2d9.svg) | N-[4-[2-[4-[2-(Dimethylamino)ethyl-methylcarbamoyl]phenyl]thieno[3,2-b]pyridin-7-yl]oxy-3-fluorophenyl]-1-phenyl-5-(trifluoromethyl)pyrazole-4-carboxamide | IC50 | 90.0 [1] |
![](https://images.aatbio.com/dataset/ic50/macrophage-stimulating-protein-receptor_913fcb5c44fcdba4a75a96891f7634ac.svg) | N-[4-[2-[4-[(3S)-3-(Dimethylamino)pyrrolidine-1-carbonyl]phenyl]thieno[3,2-b]pyridin-7-yl]oxy-3-fluorophenyl]-1-phenyl-5-(trifluoromethyl)pyrazole-4-carboxamide | IC50 | 100.0 [1] |
![](https://images.aatbio.com/dataset/ic50/macrophage-stimulating-protein-receptor_62dfd094ea8ed7dbdd80d4280f065d99.svg) | 6-[7-[2-Fluoro-4-[[1-phenyl-5-(trifluoromethyl)pyrazole-4-carbonyl]amino]phenoxy]thieno[3,2-b]pyridin-2-yl]-N,N-dimethylpyridine-3-carboxamide | IC50 | 30.0 [1] |
![](https://images.aatbio.com/dataset/ic50/macrophage-stimulating-protein-receptor_0845ff6c6c03381935a2b2e011eba3a9.svg) | 6-[7-[2-Fluoro-4-[[1-phenyl-5-(trifluoromethyl)pyrazole-4-carbonyl]amino]phenoxy]thieno[3,2-b]pyridin-2-yl]-N-(2-methoxyethyl)pyridine-3-carboxamide | IC50 | 40.0 [1] |
![](https://images.aatbio.com/dataset/ic50/macrophage-stimulating-protein-receptor_edc44538eedfe45a101aacb1dadf77bb.svg) | N-[4-[2-(1-Acetyl-3,6-dihydro-2H-pyridin-4-yl)thieno[3,2-b]pyridin-7-yl]oxy-3-fluorophenyl]-1-phenyl-5-(trifluoromethyl)pyrazole-4-carboxamide | IC50 | 90.0 [1] |