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Lysine-specific histone demethylase 1 Inhibitors (IC50, Ki)

Structure
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Compound Name
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Standard Type
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Standard Values (in nM)
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(1S,2R)-2-Phenylcyclopropan-1-amine;(1R,2S)-2-phenylcyclopropan-1-amineIC5027800.0 [1]
(1S,2R)-2-Phenylcyclopropan-1-amine;(1R,2S)-2-phenylcyclopropan-1-amineKi21000.0 [1], 25000.0 [2], 357000.0 [3]
ParnateIC5025000.0 [1]
ParnateKi28100.0 [1], 243000.0 [2], 284000.0 [3]
(E)-N'-(1-(5-Chloro-2-hydroxyphenyl)ethylidene)-3-(morpholinosulfonyl)benzohydrazideIC5013.0 [1]
(E)-N'-(1-(5-Chloro-2-hydroxyphenyl)ethylidene)-3-(morpholinosulfonyl)benzohydrazideKi13.5 [1], 31.92 [2], 35.17 [3], 35.32 [4], 54.66 [5]
N-[(2S)-4-[3-(2-Aminocyclopropyl)phenoxy]-1-(benzylamino)-1-oxobutan-2-yl]benzamideIC502500.0 [1]
N-[(2S)-4-[3-(2-Aminocyclopropyl)phenoxy]-1-(benzylamino)-1-oxobutan-2-yl]benzamideKi5700.0 [1]
Benzyl N-[1-[4-(2-aminocyclopropyl)anilino]-1-oxo-3-phenylpropan-2-yl]carbamateIC50150.0 [1], 1300.0 [2]
Benzyl N-[1-[4-(2-aminocyclopropyl)anilino]-1-oxo-3-phenylpropan-2-yl]carbamateKi1000.0 [1], 1300.0 [2], 2100.0 [3]
trans-2-PhenylcyclopropylamineIC503600.0 [1], 6300.0 [2], 6500.0 [3]
trans-2-PhenylcyclopropylamineKi28100.0 [1], 284000.0 [2]
N-[(2S)-4-[4-[(1S,2R)-2-Aminocyclopropyl]phenoxy]-1-(benzylamino)-1-oxobutan-2-yl]benzamideIC501900.0 [1], 2000.0 [2]
N-[(2S)-4-[4-[(1S,2R)-2-Aminocyclopropyl]phenoxy]-1-(benzylamino)-1-oxobutan-2-yl]benzamideKi3100.0 [1]
2-(3,5-Difluoro-2-phenylmethoxyphenyl)cyclopropan-1-amineIC50990.0 [1]
2-(3,5-Difluoro-2-phenylmethoxyphenyl)cyclopropan-1-amineKi610.0 [1], 2000.0 [2]
[[5-Cyano-2-prop-2-ynylsulfanyl-6-(3,4,5-trimethoxyphenyl)pyrimidin-4-yl]amino]thioureaIC50650.0 [1], 650.13 [2]
CID 46830247IC5019.0 [1]
CID 46830247Ki1000.0 [1], 1100.0 [2]
PhenelzineKi5600.0 [1], 17600.0 [2], 18000.0 [3]
4-((4-((((1R,2S)-2-Phenylcyclopropyl)amino)methyl)piperidin-1-yl)methyl)benzoic acidIC5024.0 [1], 41.0 [2]
4-((4-((((1R,2S)-2-Phenylcyclopropyl)amino)methyl)piperidin-1-yl)methyl)benzoic acidKi1700.0 [1]
IadademstatIC5014.0 [1], 15.0 [2], 33.0 [3]
(2S)-2-[[(2S)-2-[[(2S)-5-Amino-2-[[(2S)-6-amino-2-[[(2S)-2-[[(2S)-1-[(2S)-2-[[(2S)-6-amino-2-[[2-[[2-[[(2S,3R)-2-[[(2S)-2-[[(2S)-6-amino-2-[[(2S)-2-[[(2S)-2-[[(2S,3R)-2-[[(2S)-5-amino-2-[[(2S)-2-[[(2S,3R)-2-[[(2S)-2-[[(2S)-2-aminopropanoyl]amino]-5-carbamimidamidopentanoyl]amino]-3-hydroxybutanoyl]amino]-6-(prop-2-ynylamino)hexanoyl]amino]-5-oxopentanoyl]amino]-3-hydroxybutanoyl]amino]propanoyl]amino]-5-carbamimidamidopentanoyl]amino]hexanoyl]amino]-3-hydroxypropanoyl]amino]-3-hydroxybutanoyl]amino]acetyl]amino]acetyl]amino]hexanoyl]amino]propanoyl]pyrrolidine-2-carbonyl]amino]-5-carbamimidamidopentanoyl]amino]hexanoyl]amino]-5-oxopentanoyl]amino]-4-methylpentanoyl]amino]propanoic acidKi290.0 [1], 16600.0 [2]
(2S)-2-[[(2S)-2-[[(2S)-5-Amino-2-[[(2S)-6-amino-2-[[(2S)-2-[[(2S)-1-[(2S)-2-[[(2S)-6-amino-2-[[2-[[2-[[(2S,3R)-2-[[(2S)-2-[[(2S)-6-amino-2-[[(2S)-2-[[(2S)-2-[[(2S,3R)-2-[[(2S)-5-amino-2-[[(2S)-2-[[(2S,3R)-2-[[(2S)-2-[[(2S)-2-aminopropanoyl]amino]-5-carbamimidamidopentanoyl]amino]-3-hydroxybutanoyl]amino]-6-hydrazinylhexanoyl]amino]-5-oxopentanoyl]amino]-3-hydroxybutanoyl]amino]propanoyl]amino]-5-carbamimidamidopentanoyl]amino]hexanoyl]amino]-3-hydroxypropanoyl]amino]-3-hydroxybutanoyl]amino]acetyl]amino]acetyl]amino]hexanoyl]amino]propanoyl]pyrrolidine-2-carbonyl]amino]-5-carbamimidamidopentanoyl]amino]hexanoyl]amino]-5-oxopentanoyl]amino]-4-methylpentanoyl]amino]propanoic acidKi4.35 [1], 4400.0 [2]
3-Chloro-6-nitro-2-(trifluoromethyl)chromoneIC5051000.0 [1]
(2S)-2-[[(2S)-2-[[(2S)-5-Amino-2-[[(2S)-6-amino-2-[[(2S)-2-[[(2S)-1-[(2S)-2-[[(2S)-6-amino-2-[[2-[[2-[[(2S,3R)-2-[[(2S)-2-[[(2S)-6-amino-2-[[(2S)-2-[[(2S)-2-[[(2S,3R)-2-[[(2S)-5-amino-2-[[(2S)-2-[[(2S,3R)-2-[[(2S)-2-[[(2S)-2-aminopropanoyl]amino]-5-carbamimidamidopentanoyl]amino]-3-hydroxybutanoyl]amino]-6-(aziridin-1-yl)hexanoyl]amino]-5-oxopentanoyl]amino]-3-hydroxybutanoyl]amino]propanoyl]amino]-5-carbamimidamidopentanoyl]amino]hexanoyl]amino]-3-hydroxypropanoyl]amino]-3-hydroxybutanoyl]amino]acetyl]amino]acetyl]amino]hexanoyl]amino]propanoyl]pyrrolidine-2-carbonyl]amino]-5-carbamimidamidopentanoyl]amino]hexanoyl]amino]-5-oxopentanoyl]amino]-4-methylpentanoyl]amino]propanoic acidIC5015600.0 [1]
(2S)-2-[[(2S)-2-[[(2S)-5-Amino-2-[[(2S)-6-amino-2-[[(2S)-2-[[(2S)-1-[(2S)-2-[[(2S)-6-amino-2-[[2-[[2-[[(2S,3R)-2-[[(2S)-2-[[(2S)-6-amino-2-[[(2S)-2-[[(2S)-2-[[(2S,3R)-2-[[(2S)-5-amino-2-[[(2S)-2-[[(2S,3R)-2-[[(2S)-2-[[(2S)-2-aminopropanoyl]amino]-5-carbamimidamidopentanoyl]amino]-3-hydroxybutanoyl]amino]-6-(aziridin-1-yl)hexanoyl]amino]-5-oxopentanoyl]amino]-3-hydroxybutanoyl]amino]propanoyl]amino]-5-carbamimidamidopentanoyl]amino]hexanoyl]amino]-3-hydroxypropanoyl]amino]-3-hydroxybutanoyl]amino]acetyl]amino]acetyl]amino]hexanoyl]amino]propanoyl]pyrrolidine-2-carbonyl]amino]-5-carbamimidamidopentanoyl]amino]hexanoyl]amino]-5-oxopentanoyl]amino]-4-methylpentanoyl]amino]propanoic acidKi15600.0 [1]
(2S)-2-[[(2S)-2-[[(2S)-5-Amino-2-[[(2S)-6-amino-2-[[(2S)-2-[[(2S)-1-[(2S)-2-[[(2S)-6-amino-2-[[2-[[2-[[(2S,3R)-2-[[(2S)-2-[[(2S)-6-amino-2-[[(2S)-2-[[(2S)-2-[[(2S,3R)-2-[[(2S)-5-amino-2-[[(2S)-2-[[(2S,3R)-2-[[(2S)-2-[[(2S)-2-aminopropanoyl]amino]-5-carbamimidamidopentanoyl]amino]-3-hydroxybutanoyl]amino]-4-methylsulfanylbutanoyl]amino]-5-oxopentanoyl]amino]-3-hydroxybutanoyl]amino]propanoyl]amino]-5-carbamimidamidopentanoyl]amino]hexanoyl]amino]-3-hydroxypropanoyl]amino]-3-hydroxybutanoyl]amino]acetyl]amino]acetyl]amino]hexanoyl]amino]propanoyl]pyrrolidine-2-carbonyl]amino]-5-carbamimidamidopentanoyl]amino]hexanoyl]amino]-5-oxopentanoyl]amino]-4-methylpentanoyl]amino]propanoic acidKi40.0 [1], 50.0 [2]
Benzyl 4-(2-Aminocyclopropyl)PhenylcarbamateKi1000.0 [1], 1900.0 [2], 2000.0 [3]
1-(4-Methylpiperazin-1-yl)-2-[[(1S,2R)-2-(4-phenylmethoxyphenyl)cyclopropyl]amino]ethanoneIC508.0 [1], 70.0 [2]
1-(4-Methylpiperazin-1-yl)-2-[[(1S,2R)-2-(4-phenylmethoxyphenyl)cyclopropyl]amino]ethanoneKi30.0 [1]
4-[3-[(3R)-3-Aminopiperidine-1-carbonyl]-5-(pyridin-2-ylmethoxy)pyrazol-1-yl]benzonitrileIC50100.0 [1], 230.0 [2], 2300.0 [3]
(2S)-1-[(17S,20S,23S,26S,29S,32S,35S,38S)-29-Benzyl-20,35-bis[3-(diaminomethylideneamino)propyl]-32-(hydroxymethyl)-26-(2-methylpropyl)-2,11,19,22,25,28,31,34,37-nonaoxo-23-propan-2-yl-3,10-dioxa-6,7-dithia-1,12,18,21,24,27,30,33,36-nonazabicyclo[36.3.0]hentetracontane-17-carbonyl]pyrrolidine-2-carboxamideKi1600.0 [1], 37000.0 [2], 44000.0 [3]
4-[2-(4-Methylphenyl)-5-[[(3R)-pyrrolidin-3-yl]methoxy]pyridin-3-yl]benzonitrileIC5030.0 [1], 41.0 [2], 1400.0 [3]
4-N-[(1S,2R)-2-[4-[3-(Trifluoromethyl)phenyl]phenyl]cyclopropyl]cyclohexane-1,4-diamineIC5048.0 [1], 86.0 [2], 94.0 [3]
TranylcypromineIC5022300.0 [1], 29310.0 [2]
Tranylcypromine hydrochlorideIC502100.0 [1], 27800.0 [2]
1-[N'-[3-[7-[3-[[Amino-[[N'-(3,3-diphenylpropyl)carbamimidoyl]amino]methylidene]amino]propylamino]heptylamino]propyl]carbamimidoyl]-2-(3,3-diphenylpropyl)guanidineIC50500.0 [1], 1000.0 [2]
CID 6476700IC50500.0 [1], 5000.0 [2]
4-(4-Chloroanilino)-6-phenyl-2-prop-2-ynylsulfanylpyrimidine-5-carbonitrileIC50125000.0 [1], 125025.9 [2]
1-[2-(2-Chloroanilino)thiazole-4-yl]ethanoneIC50188000.0 [1], 437000.0 [2]
(2S)-2-[[(2S)-2-[[(2S)-5-Amino-2-[[(2S)-6-amino-2-[[(2S)-2-[[(2S)-1-[(2S)-2-[[(2S)-6-amino-2-[[2-[[2-[[(2S,3R)-2-[[(2S)-2-[[(2S)-6-amino-2-[[(2S)-2-[[(2S)-2-[[(2S,3R)-2-[[(2S)-5-amino-2-[[(2S)-2-[[(2S,3R)-2-[[(2S)-2-[[(2S)-2-aminopropanoyl]amino]-5-carbamimidamidopentanoyl]amino]-3-hydroxybutanoyl]amino]-6-[methyl(prop-2-ynyl)amino]hexanoyl]amino]-5-oxopentanoyl]amino]-3-hydroxybutanoyl]amino]propanoyl]amino]-5-carbamimidamidopentanoyl]amino]hexanoyl]amino]-3-hydroxypropanoyl]amino]-3-hydroxybutanoyl]amino]acetyl]amino]acetyl]amino]hexanoyl]amino]propanoyl]pyrrolidine-2-carbonyl]amino]-5-carbamimidamidopentanoyl]amino]hexanoyl]amino]-5-oxopentanoyl]amino]-4-methylpentanoyl]amino]propanoic acidKi107.0 [1]
4-Hydroxybenzoic (2-hydroxybenzylidene)hydrazideIC50218.0 [1]
3-N-[(2-Chloro-6-phenoxyphenyl)methyl]-1H-1,2,4-triazole-3,5-diamineIC501200.0 [1]
3-N-[(2-Chloro-6-phenoxyphenyl)methyl]-1H-1,2,4-triazole-3,5-diamineKi2200.0 [1]
(2S)-2-[[(2S)-2-[[(2S)-5-Amino-2-[[(2S)-6-amino-2-[[(2S)-2-[[(2S)-1-[(2S)-2-[[(2S)-6-amino-2-[[2-[[2-[[(2S,3R)-2-[[(2S)-2-[[(2S)-6-amino-2-[[(2S)-2-[[(2S)-2-[[(2S,3R)-2-[[(2S)-5-amino-2-[[(2S)-6-amino-2-[[(2S,3R)-2-[[(2S)-2-[[(2S)-2-aminopropanoyl]amino]-5-carbamimidamidopentanoyl]amino]-3-hydroxybutanoyl]amino]hexanoyl]amino]-5-oxopentanoyl]amino]-3-hydroxybutanoyl]amino]propanoyl]amino]-5-carbamimidamidopentanoyl]amino]hexanoyl]amino]-3-hydroxypropanoyl]amino]-3-hydroxybutanoyl]amino]acetyl]amino]acetyl]amino]hexanoyl]amino]propanoyl]pyrrolidine-2-carbonyl]amino]-5-carbamimidamidopentanoyl]amino]hexanoyl]amino]-5-oxopentanoyl]amino]-4-methylpentanoyl]amino]propanoic acidKi1800.0 [1]
Tert-butyl 4-[[1-[(4-methylphenyl)methyl]triazol-4-yl]methylsulfanylcarbothioyl]piperazine-1-carboxylateIC502100.0 [1]
4-[[4-[[[(1S,2R)-2-Phenylcyclopropyl]amino]methyl]piperidin-1-yl]methyl]benzoic acidIC50610.0 [1], 1700.0 [2]
[[5-Cyano-6-(4-fluorophenyl)-2-prop-2-ynylsulfanylpyrimidin-4-yl]amino]thioureaIC501820.0 [1], 1823.9 [2]
4-(4-Fluoroanilino)-6-phenyl-2-prop-2-ynylsulfanylpyrimidine-5-carbonitrileIC50125000.0 [1], 125025.9 [2]
4-(4-Nitroanilino)-6-phenyl-2-prop-2-ynylsulfanylpyrimidine-5-carbonitrileIC50123310.48 [1], 125000.0 [2]
4-Chloro-2-[[1-[(2-chlorophenyl)methyl]triazol-4-yl]methylsulfanyl]-6-phenylpyrimidine-5-carbonitrileIC5097274.72 [1], 125000.0 [2]
4-Chloro-6-(4-chlorophenyl)-2-[[1-[(2-chlorophenyl)methyl]triazol-4-yl]methylsulfanyl]pyrimidine-5-carbonitrileIC50125000.0 [1], 125025.9 [2]
[[5-Cyano-2-[(3,4-dichlorophenyl)methylsulfanyl]-6-(3,4,5-trimethoxyphenyl)pyrimidin-4-yl]amino]thioureaIC5098174.79 [1], 98570.0 [2]
[[5-Cyano-2-[(4-fluorophenyl)methylsulfanyl]-6-(3,4,5-trimethoxyphenyl)pyrimidin-4-yl]amino]thioureaIC50125000.0 [1], 125025.9 [2]
4-[2-(4-Methylphenyl)-5-(piperidin-4-ylmethoxy)pyridin-3-yl]benzonitrileKi29.0 [1]
N-[(2S)-1-[(3-Chlorophenyl)methylamino]-1-oxo-6-[[(1R,2S)-2-phenylcyclopropyl]amino]hexan-2-yl]-4-phenylbenzamideIC50132.0 [1], 770.0 [2]
(2S)-1-[(2S)-6-Amino-2-[[(2S)-5-(diaminomethylideneamino)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-5-(diaminomethylideneamino)-2-[[(2S)-pyrrolidine-2-carbonyl]amino]pentanoyl]amino]-3-hydroxypropanoyl]amino]-3-phenylpropanoyl]amino]-4-methylpentanoyl]amino]-3-methylbutanoyl]amino]pentanoyl]amino]hexanoyl]pyrrolidine-2-carboxamideKi140.0 [1], 1900.0 [2]
N-[(E)-(5-Chloro-2-hydroxyphenyl)methylideneamino]-4-hydroxybenzamideIC50275.0 [1]
4-[3-[(3R)-3-Aminopiperidine-1-carbonyl]-5-[(3-ethyl-1,2-oxazol-5-yl)methoxy]pyrazol-1-yl]benzonitrileIC5079.0 [1], 520.0 [2]
N-[(2S)-4-[3-[(1R,2S)-2-Aminocyclopropyl]phenoxy]-1-(benzylamino)-1-oxobutan-2-yl]benzamideIC501600.0 [1], 1900.0 [2]
2-(Perfluorophenyl)CyclopropanamineIC509000.0 [1]
2-(Perfluorophenyl)CyclopropanamineKi8900.0 [1]
(2S)-2-[[(2S)-2-[[(2S)-5-Amino-2-[[(2S)-6-amino-2-[[(2S)-2-[[(2S)-1-[(2S)-2-[[(2S)-6-amino-2-[[2-[[2-[[(2S,3R)-2-[[(2S)-2-[[(2S)-6-amino-2-[[(2S)-2-[[(2S)-2-[[(2S,3R)-2-[[(2S)-5-amino-2-[[(2S)-2-[[(2S,3R)-2-[[(2S)-2-[[(2S)-2-aminopropanoyl]amino]-5-carbamimidamidopentanoyl]amino]-3-hydroxybutanoyl]amino]-6-(cyclopropylamino)hexanoyl]amino]-5-oxopentanoyl]amino]-3-hydroxybutanoyl]amino]propanoyl]amino]-5-carbamimidamidopentanoyl]amino]hexanoyl]amino]-3-hydroxypropanoyl]amino]-3-hydroxybutanoyl]amino]acetyl]amino]acetyl]amino]hexanoyl]amino]propanoyl]pyrrolidine-2-carbonyl]amino]-5-carbamimidamidopentanoyl]amino]hexanoyl]amino]-5-oxopentanoyl]amino]-4-methylpentanoyl]amino]propanoic acidKi2700.0 [1], 2800.0 [2]
(2S)-2-[[(2S)-6-Amino-2-[[(2S)-2-[[(2S)-1-[(2S)-2-[[(2S)-6-amino-2-[[2-[[2-[[(2S,3R)-2-[[(2S,5S,8S,11S,14S,23S)-11-(4-aminobutyl)-23-[[(2S)-2-[[(2S,3R)-2-[[(2S)-2-[[(2S)-2-aminopropanoyl]amino]-5-carbamimidamidopentanoyl]amino]-3-hydroxybutanoyl]amino]-4-methylsulfanylbutanoyl]amino]-8-(3-carbamimidamidopropyl)-2-[(1R)-1-hydroxyethyl]-5-methyl-3,6,9,12,17,24-hexaoxo-1,4,7,10,13,18-hexazacyclotetracosane-14-carbonyl]amino]-3-hydroxybutanoyl]amino]acetyl]amino]acetyl]amino]hexanoyl]amino]propanoyl]pyrrolidine-2-carbonyl]amino]-5-carbamimidamidopentanoyl]amino]hexanoyl]amino]-N-[(2S)-1-[[(2S)-1-amino-1-oxopropan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]pentanediamideIC502100.0 [1]
(2S)-2-[[(2S)-6-Amino-2-[[(2S)-2-[[(2S)-1-[(2S)-2-[[(2S)-6-amino-2-[[2-[[2-[[(2S,3R)-2-[[(2S,5S,8S,11S,14S,23S)-11-(4-aminobutyl)-23-[[(2S)-2-[[(2S,3R)-2-[[(2S)-2-[[(2S)-2-aminopropanoyl]amino]-5-carbamimidamidopentanoyl]amino]-3-hydroxybutanoyl]amino]-4-methylsulfanylbutanoyl]amino]-8-(3-carbamimidamidopropyl)-2-[(1R)-1-hydroxyethyl]-5-methyl-3,6,9,12,17,24-hexaoxo-1,4,7,10,13,18-hexazacyclotetracosane-14-carbonyl]amino]-3-hydroxybutanoyl]amino]acetyl]amino]acetyl]amino]hexanoyl]amino]propanoyl]pyrrolidine-2-carbonyl]amino]-5-carbamimidamidopentanoyl]amino]hexanoyl]amino]-N-[(2S)-1-[[(2S)-1-amino-1-oxopropan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]pentanediamideKi385.0 [1]
N-[(2S)-1-(Benzylamino)-1-oxo-6-[(2-phenylcyclopropyl)amino]hexan-2-yl]benzamideIC50300.0 [1]
Tert-butyl [4-[(1S,2R)-2-[(2-methylpropan-2-yl)oxycarbonylamino]cyclopropyl]phenyl] carbonateIC5021250.0 [1]
[[6-(4-Bromophenyl)-5-cyano-2-prop-2-ynylsulfanylpyrimidin-4-yl]amino]ureaIC5041495.4 [1], 41510.0 [2]
[[5-Cyano-6-(4-methylphenyl)-2-prop-2-ynylsulfanylpyrimidin-4-yl]amino]ureaIC503160.0 [1], 3162.28 [2]
[[5-Cyano-6-(4-nitrophenyl)-2-prop-2-ynylsulfanylpyrimidin-4-yl]amino]ureaIC5011190.0 [1], 11194.38 [2]
[[6-(3-Chlorophenyl)-5-cyano-2-prop-2-ynylsulfanylpyrimidin-4-yl]amino]ureaIC505060.0 [1], 5069.91 [2]
4-Chloro-6-phenyl-2-prop-2-ynylsulfanylpyrimidine-5-carbonitrileIC5045708.82 [1], 45750.0 [2]
4-Chloro-6-(4-chlorophenyl)-2-prop-2-ynylsulfanylpyrimidine-5-carbonitrileIC508330.0 [1], 8336.81 [2]
4-Chloro-2-prop-2-ynylsulfanyl-6-(3,4,5-trimethoxyphenyl)pyrimidine-5-carbonitrileIC503130.0 [1], 3133.29 [2]
4-Chloro-6-(3,4-difluorophenyl)-2-prop-2-ynylsulfanylpyrimidine-5-carbonitrileIC5024370.0 [1], 24378.11 [2]
4-(4-Bromophenyl)-6-chloro-2-prop-2-ynylsulfanylpyrimidine-5-carbonitrileIC5024710.0 [1], 24717.24 [2]
4-Chloro-6-(4-fluorophenyl)-2-prop-2-ynylsulfanylpyrimidine-5-carbonitrileIC5021820.0 [1], 21827.3 [2]
4-Chloro-6-(4-methylphenyl)-2-prop-2-ynylsulfanylpyrimidine-5-carbonitrileIC5059160.0 [1], 59292.53 [2]
4-Chloro-6-(4-nitrophenyl)-2-prop-2-ynylsulfanylpyrimidine-5-carbonitrileIC50125000.0 [1], 125025.9 [2]
[(5-Cyano-6-phenyl-2-prop-2-ynylsulfanylpyrimidin-4-yl)amino]thioureaIC501590.0 [1], 1592.21 [2]
[[6-(4-Chlorophenyl)-5-cyano-2-prop-2-ynylsulfanylpyrimidin-4-yl]amino]thioureaIC501590.0 [1], 1592.21 [2]
[[5-Cyano-6-(3,4-difluorophenyl)-2-prop-2-ynylsulfanylpyrimidin-4-yl]amino]thioureaIC501660.0 [1], 1663.41 [2]
[[6-(4-Bromophenyl)-5-cyano-2-prop-2-ynylsulfanylpyrimidin-4-yl]amino]thioureaIC501590.0 [1], 1592.21 [2]
[[5-Cyano-6-(4-methylphenyl)-2-prop-2-ynylsulfanylpyrimidin-4-yl]amino]thioureaIC501100.0 [1], 1101.54 [2]
[[5-Cyano-6-(4-nitrophenyl)-2-prop-2-ynylsulfanylpyrimidin-4-yl]amino]thioureaIC502580.0 [1], 2582.26 [2]
[[6-(3-Chlorophenyl)-5-cyano-2-prop-2-ynylsulfanylpyrimidin-4-yl]amino]thioureaIC503580.0 [1], 3580.96 [2]
[[5-Cyano-6-(3-methoxyphenyl)-2-prop-2-ynylsulfanylpyrimidin-4-yl]amino]thioureaIC502610.0 [1], 2612.16 [2]
[[6-(4-Chlorophenyl)-5-cyano-2-prop-2-ynylsulfanylpyrimidin-4-yl]amino]ureaIC502640.0 [1], 2642.41 [2]
4-[5-(4-Methylphenyl)-2-[[(3S)-pyrrolidin-3-yl]methylamino]pyrimidin-4-yl]benzonitrileIC5010.0 [1]
1-(3,3-Diphenylpropyl)-3-[3-[5-[3-(3,3-diphenylpropylcarbamothioylamino)propylamino]pentylamino]propyl]thiourea;hydrochlorideIC504800.0 [1]
1-(3,3-Diphenylpropyl)-3-[3-[5-[3-(3,3-diphenylpropylcarbamothioylamino)propylamino]pentylamino]propyl]thiourea;hydrochlorideKi2400.0 [1]
4-[2-Phenyl-5-(piperidin-4-ylmethoxy)pyridin-3-yl]benzonitrileKi1800.0 [1], 2300.0 [2]
(2S)-1-[(17S,20S,23S,26S,29S,32S,35S,38S)-29-Benzyl-20,35-bis[3-(diaminomethylideneamino)propyl]-32-(hydroxymethyl)-26-(2-methylpropyl)-2,11,19,22,25,28,31,34,37-nonaoxo-23-propan-2-yl-3,10-dioxa-1,12,18,21,24,27,30,33,36-nonazabicyclo[36.3.0]hentetracontane-17-carbonyl]pyrrolidine-2-carboxamideKi300000.0 [1]
(E)-4-Bromo-N'-(2-hydroxybenzylidene)benzohydrazideIC50196.0 [1]
4-Hydroxy-N-[(E)-1-(2-hydroxyphenyl)ethylideneamino]benzamideIC50291.0 [1]
3-Chloro-N'-(2-hydroxybenzylidene)benzohydrazideIC50333.0 [1]
N'-[(1E)-1-(5-Chloro-2-hydroxyphenyl)ethylidene]benzohydrazideIC50128.0 [1]
(1S,2R)-N-[(2-Methoxypyridin-3-yl)methyl]-2-phenylcyclopropan-1-amineIC5065.5 [1], 98.0 [2]
Items per page: 1 - 10 of 100
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References

This online tool may be cited as follows

MLA

"Quest Database™ Lysine-specific histone demethylase 1 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 22 Feb. 2025, https://www.aatbio.com/data-sets/lysine-specific-histone-demethylase-1-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2025, February 22). Quest Database™ Lysine-specific histone demethylase 1 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/lysine-specific-histone-demethylase-1-inhibitors-ic50-ki.
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