| 1,5-Bis[(E)-2-(3,4-dichlorophenyl)ethenyl]-2,4-dinitrobenzene | IC50 | 9300.0 [1] |
| 1,5-Bis[(E)-2-(3,4-dichlorophenyl)ethenyl]-2,4-dinitrobenzene | Ki | 3000.0 [1] |
| N-(4-Pyridin-2-yl-thiazol-2-yl)-benzamide | IC50 | 12100.0 [1] |
| 2-{5-[(4-Chloro-2-Methylphenyl)methoxy]-1h-Pyrazol-1-Yl}pyridine-4-Carboxylic Acid | IC50 | 170.0 [1] |
| CID 127030711 | IC50 | 10.0 [1] |
| 8-Hydroxy-3-[4-(2-naphthalen-1-ylethyl)-1,4-diazepan-1-yl]quinoline-5-carboxylic acid | IC50 | 1000.0 [1] |
| N-[6-(Dimethylamino)hexyl]-3-(8-hydroxyquinolin-6-yl)benzamide | IC50 | 1000.0 [1] |
| 3-[[(1R)-6-(N-Methylanilino)-1,2,3,4-tetrahydronaphthalen-1-yl]methylamino]pyridine-4-carboxylic acid | IC50 | 56.0 [1] |
| Pyrido[3,4-d]pyrimidin-4(3H)-one | IC50 | 1000.0 [1] |
| 3-Ethylsulfonyl-N-(4-pyridin-2-yl-1,3-thiazol-2-yl)benzamide | IC50 | 10900.0 [1] |
| 2-(((2-((2-(Dimethylamino)ethyl)(ethyl)amino)-2-oxoethyl)amino)methyl)isonicotinic acid | IC50 | 100.0 [1] |
| 2-(2-Azanyl-1,3-Thiazol-4-Yl)pyridine-4-Carboxamide | IC50 | 32700.0 [1] |
| 2-(2-Benzamido-1,3-thiazol-4-yl)pyridine-4-carboxylic acid | IC50 | 17000.0 [1] |
| Lithium;2-[(furan-2-ylmethylamino)methyl]pyridine-4-carboxylate | IC50 | 170.0 [1] |
| Lithium;2-[(benzylamino)methyl]pyridine-4-carboxylate | IC50 | 1200.0 [1] |
| 8-(2-Azanyl-1,3-Thiazol-4-Yl)-3~{h}-Pyrido[3,4-D]pyrimidin-4-One | IC50 | 5000.0 [1] |
| 8-(1,3-Thiazol-4-Yl)-3~{h}-Pyrido[3,4-D]pyrimidin-4-One | IC50 | 3100.0 [1] |
| 8-[4-[2-[(4-Fluorophenyl)methyl-Methyl-Amino]ethyl]pyrazol-1-Yl]-3~{h}-Pyrido[3,4-D]pyrimidin-4-One | IC50 | 390.0 [1] |
| 8-[4-[2-(Dimethylamino)ethyl]pyrazol-1-yl]-3H-pyrido[3,4-d]pyrimidin-4-one | IC50 | 2300.0 [1] |
| 8-[4-[2-[4-(4-Chlorophenyl)piperidin-1-Yl]ethyl]pyrazol-1-Yl]-3~{h}-Pyrido[3,4-D]pyrimidin-4-One | IC50 | 86.0 [1] |
| 8-[4-[2-[4-[(4-Chlorophenyl)methyl]piperidin-1-yl]ethyl]pyrazol-1-yl]-3H-pyrido[3,4-d]pyrimidin-4-one | IC50 | 50.0 [1] |
| 8-Pyrazol-1-yl-3H-pyrido[3,4-d]pyrimidin-4-one | IC50 | 4600.0 [1] |
| 8-[4-[2-[4-(3,5-Dichlorophenyl)piperidin-1-yl]ethyl]pyrazol-1-yl]-3H-pyrido[3,4-d]pyrimidin-4-one | IC50 | 17.0 [1] |
| 8-[[(Phenylmethyl)amino]methyl]-1~{h}-Pyrido[3,4-D]pyrimidin-4-One | IC50 | 6500.0 [1] |
| 8-[4-(2-Hydroxyethyl)pyrazol-1-yl]-3H-pyrido[3,4-d]pyrimidin-4-one | IC50 | 8800.0 [1] |
| 8-(1H-Pyrazol-5-yl)-3H-pyrido[3,4-d]pyrimidin-4-one | IC50 | 2800.0 [1] |
| 8-[4-(2-Pyrrolidin-1-ylethyl)pyrazol-1-yl]-3H-pyrido[3,4-d]pyrimidin-4-one | IC50 | 750.0 [1] |
| 8-[4-(2-Piperidin-1-ylethyl)pyrazol-1-yl]-3H-pyrido[3,4-d]pyrimidin-4-one | IC50 | 650.0 [1] |
| 8-[4-[2-[(3,4-Dichlorophenyl)methyl-methylamino]ethyl]pyrazol-1-yl]-3H-pyrido[3,4-d]pyrimidin-4-one | IC50 | 165.0 [1] |
| 8-[4-[2-[Methyl-[(4-methylsulfonylphenyl)methyl]amino]ethyl]pyrazol-1-yl]-3H-pyrido[3,4-d]pyrimidin-4-one | IC50 | 400.0 [1] |
| 4-[[Methyl-[2-[1-(4-oxo-3H-pyrido[3,4-d]pyrimidin-8-yl)pyrazol-4-yl]ethyl]amino]methyl]benzonitrile | IC50 | 340.0 [1] |
| 4-[[Methyl-[3-[1-(4-oxo-3H-pyrido[3,4-d]pyrimidin-8-yl)pyrazol-4-yl]propyl]amino]methyl]benzonitrile | IC50 | 260.0 [1] |
| 8-(1-Methylpyrazol-3-yl)-3H-pyrido[3,4-d]pyrimidin-4-one | IC50 | 9200.0 [1] |
| 8-[(Furan-2-ylmethylamino)methyl]-3H-pyrido[3,4-d]pyrimidin-4-one | IC50 | 3100.0 [1] |
| 8-[(4-Methylpiperazin-1-yl)methyl]-3H-pyrido[3,4-d]pyrimidin-4-one | IC50 | 8500.0 [1] |
| 8-[(4-Phenylpiperazin-1-yl)methyl]-3H-pyrido[3,4-d]pyrimidin-4-one | IC50 | 81500.0 [1] |
| 8-[(4-Pyridin-2-ylpiperazin-1-yl)methyl]-3H-pyrido[3,4-d]pyrimidin-4-one | IC50 | 24600.0 [1] |
| 8-[4-[2-[4-(3-Chlorophenyl)piperidin-1-yl]ethyl]pyrazol-1-yl]-3~{H}-pyrido[3,4-d]pyrimidin-4-one | IC50 | 31.0 [1] |
| 8-[4-[2-[4-(3,5-Difluorophenyl)piperidin-1-yl]ethyl]pyrazol-1-yl]-3H-pyrido[3,4-d]pyrimidin-4-one | IC50 | 41.0 [1] |
| 8-[4-[2-[4-(2,4-Difluorophenyl)piperidin-1-yl]ethyl]pyrazol-1-yl]-3H-pyrido[3,4-d]pyrimidin-4-one | IC50 | 36.0 [1] |
| 8-[4-[2-[4-[3-(Trifluoromethyl)phenyl]piperidin-1-yl]ethyl]pyrazol-1-yl]-3H-pyrido[3,4-d]pyrimidin-4-one | IC50 | 39.0 [1] |
| 8-[4-[2-[4-(1,3-Benzodioxol-5-ylmethyl)piperidin-1-yl]ethyl]pyrazol-1-yl]-3H-pyrido[3,4-d]pyrimidin-4-one | IC50 | 72.0 [1] |
| 8-[4-[2-[4-(Pyridin-3-ylmethyl)piperidin-1-yl]ethyl]pyrazol-1-yl]-3H-pyrido[3,4-d]pyrimidin-4-one | IC50 | 207.0 [1] |
| 8-[4-[2-[4-[(5-Cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]piperidin-1-yl]ethyl]pyrazol-1-yl]-3H-pyrido[3,4-d]pyrimidin-4-one | IC50 | 247.0 [1] |
| 8-[4-[2-[4-(4-Fluorophenyl)piperidin-1-yl]ethyl]pyrazol-1-yl]-3H-pyrido[3,4-d]pyrimidin-4-one | IC50 | 61.0 [1] |
| 8-[4-[2-[4-(4-Methoxyphenyl)piperidin-1-yl]ethyl]pyrazol-1-yl]-3H-pyrido[3,4-d]pyrimidin-4-one | IC50 | 39.0 [1] |
| 8-[4-[2-[4-(2-Chlorophenyl)piperidin-1-yl]ethyl]pyrazol-1-yl]-3H-pyrido[3,4-d]pyrimidin-4-one | IC50 | 179.0 [1] |
| 8-[4-[2-(4-Phenylpiperidin-1-yl)ethyl]pyrazol-1-yl]-3H-pyrido[3,4-d]pyrimidin-4-one | IC50 | 274.0 [1] |
| 8-[4-[2-(4-Pyridin-4-ylpiperidin-1-yl)ethyl]pyrazol-1-yl]-3H-pyrido[3,4-d]pyrimidin-4-one | IC50 | 55.0 [1] |
| 8-[4-[2-(4-Thiophen-2-ylpiperidin-1-yl)ethyl]pyrazol-1-yl]-3H-pyrido[3,4-d]pyrimidin-4-one | IC50 | 29.0 [1] |
| 8-(Piperidin-1-ylmethyl)-3H-pyrido[3,4-d]pyrimidin-4-one | IC50 | 100000.0 [1] |
| 8-[(Dimethylamino)methyl]-3H-pyrido[3,4-d]pyrimidin-4-one | IC50 | 7800.0 [1] |
| 8-[4-[2-(4-Benzylpiperidin-1-yl)ethyl]pyrazol-1-yl]-3H-pyrido[3,4-d]pyrimidin-4-one | IC50 | 118.0 [1] |
| 8-[4-[2-[4-[(4-Fluorophenyl)methyl]piperidin-1-yl]ethyl]pyrazol-1-yl]-3H-pyrido[3,4-d]pyrimidin-4-one | IC50 | 79.0 [1] |
| 8-[4-[2-[4-[[4-(Trifluoromethyl)phenyl]methyl]piperidin-1-yl]ethyl]pyrazol-1-yl]-3H-pyrido[3,4-d]pyrimidin-4-one | IC50 | 62.0 [1] |
| 8-[4-[2-[4-[(3,4-Dichlorophenyl)methyl]piperidin-1-yl]ethyl]pyrazol-1-yl]-3H-pyrido[3,4-d]pyrimidin-4-one | IC50 | 68.0 [1] |
| 8-[4-[2-[4-[(3-Methoxyphenyl)methyl]piperidin-1-yl]ethyl]pyrazol-1-yl]-3H-pyrido[3,4-d]pyrimidin-4-one | IC50 | 149.0 [1] |
| 8-[4-[2-[4-(4-Methylsulfonylphenyl)piperidin-1-yl]ethyl]pyrazol-1-yl]-3H-pyrido[3,4-d]pyrimidin-4-one | IC50 | 69.0 [1] |
| 4-[1-[2-[1-(4-Oxo-3H-pyrido[3,4-d]pyrimidin-8-yl)pyrazol-4-yl]ethyl]piperidin-4-yl]benzonitrile | IC50 | 69.0 [1] |
| 3-Methylsulfonyl-N-(4-pyridin-2-yl-1,3-thiazol-2-yl)benzamide | IC50 | 11300.0 [1] |
| Tcmdc-142577 | IC50 | 6400.0 [1] |
| N-[[2-[[[2-[2-(Dimethylamino)ethyl-ethylamino]-2-oxoethyl]amino]methyl]pyridin-4-yl]methyl]-2,2,2-trifluoroacetamide | IC50 | 2500.0 [1] |
| 2-[[4-(Diethylamino)butylamino]methyl]pyridine-4-carbaldehyde | IC50 | 250.0 [1] |
| 2-(2-Azanyl-1,3-Thiazol-4-Yl)pyridine-4-Carboxylic Acid | IC50 | 83.0 [1] |
| 2-(2-Methyl-1,3-thiazol-4-yl)pyridine-4-carboxylic acid | IC50 | 2300.0 [1] |
| 2-(1,3-Thiazol-4-yl)pyridine-4-carboxylic acid | IC50 | 350.0 [1] |