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Lysine-specific demethylase 4A Inhibitors (IC50, Ki)

Structure
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▼
Compound Name
▲
▼
Standard Type
▲
▼
Standard Values (in nM)
▲
▼
N-OxalylglycineIC50250000.0 [1]
Pyridine-2,4-dicarboxylic acidIC50700.0 [1], 4200.0 [2]
8-Hydroxy-5-quinolinecarboxylic acidIC501700.0 [1], 3200.0 [2], 86500.0 [3]
3-[9-(Dimethylamino)nonanoyl-hydroxyamino]propanoic acidIC50800.0 [1], 3000.0 [2]
4-Oxo-4-[4-[4-(1-naphthylcarbamoyloxymethyl)benzylamino]butylhydroxyamino]-2-butenoic acidIC503300.0 [1], 4300.0 [2]
Tetrazole-5-acetohydrazideIC502400.0 [1], 46600.0 [2]
Tetrazole-5-acetohydrazideKi1940.0 [1]
LutiramIC503300.0 [1]
(R)-3-(4-(4-Bromophenylsulfonyloxy)phenyl)-2-(carboxyformamido)propanoic acidIC5012000.0 [1]
1,5-Bis[(E)-2-(3,4-dichlorophenyl)ethenyl]-2,4-dinitrobenzeneIC506400.0 [1]
1,5-Bis[(E)-2-(3,4-dichlorophenyl)ethenyl]-2,4-dinitrobenzeneKi5500.0 [1]
2-(1-Methylimidazol-4-yl)pyridine-4-carboxylic acidIC50100.0 [1]
2-(1-Methylimidazol-4-yl)-4-(2H-tetrazol-5-yl)pyridineIC5010000.0 [1]
(2R)-2-Hydroxypentanedioic acidIC5024000.0 [1]
DaminozideIC503300000.0 [1]
3-[[2-Pyridin-2-Yl-6-(1,2,4,5-Tetrahydro-3-Benzazepin-3-Yl)pyrimidin-4-Yl]amino]propanoic AcidIC50400000.0 [1]
N-(4-Pyridin-2-yl-thiazol-2-yl)-benzamideIC5020900.0 [1]
3-Aminoisonicotinic acidIC50501.19 [1]
Di-N-desethylamiodaroneIC5072000.0 [1]
(2S)-2-Hydroxypentanedioic acidIC5026000.0 [1]
2-{5-[(4-Chloro-2-Methylphenyl)methoxy]-1h-Pyrazol-1-Yl}pyridine-4-Carboxylic AcidIC5099.0 [1]
CID 127030711IC501000.0 [1]
8-Hydroxy-3-[4-(2-naphthalen-1-ylethyl)-1,4-diazepan-1-yl]quinoline-5-carboxylic acidIC501000.0 [1]
N-[6-(4-Acryloyl-1,4-diazepan-1-yl)-2-(pyridin-2-yl)pyrimidin-4-yl]-beta-alanineIC50230000.0 [1]
2-[[3-[[(E)-4-(Dimethylamino)but-2-enoyl]amino]phenyl]-(2-piperidin-1-ylethoxy)methyl]thieno[3,2-b]pyridine-7-carboxylic acidIC505300.0 [1]
N-[6-(Dimethylamino)hexyl]-3-(8-hydroxyquinolin-6-yl)benzamideIC501000.0 [1]
8-Hydroxyquinoline-4-carboxylic acidIC501700.0 [1]
3-[[(1R)-6-(N-Methylanilino)-1,2,3,4-tetrahydronaphthalen-1-yl]methylamino]pyridine-4-carboxylic acidIC50104.0 [1]
Pyrido[3,4-d]pyrimidin-4(3H)-oneIC501700.0 [1]
2-[(1-Benzyl-1h-Pyrazol-4-Yl)oxy]pyrido[3,4-D]pyrimidin-4(3h)-OneIC50630.96 [1]
3-Ethylsulfonyl-N-(4-pyridin-2-yl-1,3-thiazol-2-yl)benzamideIC5013200.0 [1]
(R)-2-(Carboxyformamido)-3-(4-(4-fluorophenylsulfonyloxy)phenyl)propanoic acidIC5020000.0 [1]
(R)-3-(4-(4-Tert-butylphenylsulfonyloxy)phenyl)-2-(carboxyformamido)propanoic acidIC5013000.0 [1]
2-(((2-((2-(Dimethylamino)ethyl)(ethyl)amino)-2-oxoethyl)amino)methyl)isonicotinic acidIC50100.0 [1]
2,2'-Bipyridine-4-carboxylic acidIC501258.93 [1]
2-[1-[(3R)-1-Benzoylpiperidin-3-yl]triazol-4-yl]pyridine-4-carboxylic acidIC5015848.93 [1]
2-(2-Azanyl-1,3-Thiazol-4-Yl)pyridine-4-CarboxamideIC50104200.0 [1]
2-[(3-Methylthiophen-2-yl)methylamino]pyridine-3-carboxylic acidIC50100000.0 [1]
2-[1-(2-Phenylethyl)triazol-4-yl]pyridine-4-carboxylic acidIC5063095.73 [1]
2-[1-(2-Phenoxyethyl)triazol-4-yl]pyridine-4-carboxylic acidIC50100000.0 [1]
2-[1-(1-Ethoxycarbonylpiperidin-4-yl)triazol-4-yl]pyridine-4-carboxylic acidIC50100000.0 [1]
2-[1-(1-Benzoylpiperidin-4-yl)triazol-4-yl]pyridine-4-carboxylic acidIC5050118.72 [1]
2-[1-[1-(2-Phenylacetyl)piperidin-4-yl]triazol-4-yl]pyridine-4-carboxylic acidIC5039810.72 [1]
2-[1-[1-(3-Phenylpropanoyl)piperidin-4-yl]triazol-4-yl]pyridine-4-carboxylic acidIC5079432.82 [1]
2-[1-(1-Acetylazetidin-3-yl)triazol-4-yl]pyridine-4-carboxylic acidIC502511.89 [1]
2-[1-(1-Propanoylazetidin-3-yl)triazol-4-yl]pyridine-4-carboxylic acidIC505011.87 [1]
2-[1-(1-Butanoylazetidin-3-yl)triazol-4-yl]pyridine-4-carboxylic acidIC505011.87 [1]
2-[1-(1-Benzoylazetidin-3-yl)triazol-4-yl]pyridine-4-carboxylic acidIC50100000.0 [1]
2-[1-[1-(3-Phenylpropanoyl)azetidin-3-yl]triazol-4-yl]pyridine-4-carboxylic acidIC506309.57 [1]
2-[1-(1-Acetylpiperidin-3-yl)triazol-4-yl]pyridine-4-carboxylic acidIC5039810.72 [1]
2-[1-(1-Benzoylpiperidin-3-yl)triazol-4-yl]pyridine-4-carboxylic acidIC5063095.73 [1]
8-Hydroxy-2-(pyridin-2-ylcarbamoyl)quinoline-5-carboxylic acidIC502800.0 [1]
8-Hydroxy-2-(phenylcarbamoyl)quinoline-5-carboxylic acidIC50100000.0 [1]
8-Hydroxy-2-(naphthalen-1-ylcarbamoyl)quinoline-5-carboxylic acidIC50100000.0 [1]
2-(Dimethylcarbamoyl)-8-hydroxyquinoline-5-carboxylic acidIC503700.0 [1]
2-(Cyclohexylcarbamoyl)-8-hydroxyquinoline-5-carboxylic acidIC50100000.0 [1]
8-Hydroxy-2-[(4-methoxyphenyl)carbamoyl]quinoline-5-carboxylic acidIC50100000.0 [1]
8-Hydroxy-2-[(3-methoxyphenyl)carbamoyl]quinoline-5-carboxylic acidIC50100000.0 [1]
8-Hydroxy-2-[(3-methylphenyl)carbamoyl]quinoline-5-carboxylic acidIC50100000.0 [1]
8-Hydroxy-2-[(2-methylphenyl)carbamoyl]quinoline-5-carboxylic acidIC50100000.0 [1]
8-Hydroxy-2-[(4-methylphenyl)carbamoyl]quinoline-5-carboxylic acidIC50100000.0 [1]
2-[(4-Fluorophenyl)carbamoyl]-8-hydroxyquinoline-5-carboxylic acidIC50100000.0 [1]
2-[(2-Fluorophenyl)carbamoyl]-8-hydroxyquinoline-5-carboxylic acidIC50100000.0 [1]
2-[[4-(Dimethylamino)phenyl]carbamoyl]-8-hydroxyquinoline-5-carboxylic acidIC50100000.0 [1]
8-Hydroxy-2-[[4-(trifluoromethoxy)phenyl]carbamoyl]quinoline-5-carboxylic acidIC50100000.0 [1]
2-(Benzylcarbamoyl)-8-hydroxyquinoline-5-carboxylic acidIC50100000.0 [1]
2-(1H-Benzimidazol-2-ylcarbamoyl)-8-hydroxyquinoline-5-carboxylic acidIC5019000.0 [1]
8-Hydroxy-2-[(5-methylpyridin-2-yl)carbamoyl]quinoline-5-carboxylic acidIC506200.0 [1]
8-Hydroxy-2-[2-(1H-indol-3-yl)ethylcarbamoyl]quinoline-5-carboxylic acidIC5024000.0 [1]
2-(Diethylcarbamoyl)-8-hydroxyquinoline-5-carboxylic acidIC501800.0 [1]
8-Hydroxy-2-(3-morpholin-4-ylpropylcarbamoyl)quinoline-5-carboxylic acidIC5082000.0 [1]
8-Hydroxy-2-(4-methylpiperazine-1-carbonyl)quinoline-5-carboxylic acidIC501600.0 [1]
8-Hydroxy-2-(morpholine-4-carbonyl)quinoline-5-carboxylic acidIC505100.0 [1]
8-Hydroxy-2-(1-methylpiperidine-4-carbonyl)quinoline-5-carboxylic acidIC5050000.0 [1]
4-[(E)-2-(1-Hexylpyridin-1-ium-4-yl)ethenyl]-N,N-dimethylaniline;iodideKi420.0 [1]
2-[[4-Chloro-3-(cyclopropylmethoxy)phenyl]methoxy]-1H-pyrrolo[3,2-b]pyridine-7-carboxylic acidIC501000.0 [1]
2-(2-Benzamido-1,3-thiazol-4-yl)pyridine-4-carboxylic acidIC5030600.0 [1]
Lithium;2-[(furan-2-ylmethylamino)methyl]pyridine-4-carboxylateIC50300.0 [1]
Lithium;2-[(benzylamino)methyl]pyridine-4-carboxylateIC50950.0 [1]
2-[(4-Chloro-3-methoxyphenyl)methoxy]-1H-pyrrolo[3,2-b]pyridine-7-carboxylic acidIC50100.0 [1]
2-[[4-Chloro-3-(trifluoromethoxy)phenyl]methoxy]-1H-pyrrolo[3,2-b]pyridine-7-carboxylic acidIC50100.0 [1]
8-(2-Azanyl-1,3-Thiazol-4-Yl)-3~{h}-Pyrido[3,4-D]pyrimidin-4-OneIC5011500.0 [1]
8-(1,3-Thiazol-4-Yl)-3~{h}-Pyrido[3,4-D]pyrimidin-4-OneIC508000.0 [1]
8-[4-[2-[(4-Fluorophenyl)methyl-Methyl-Amino]ethyl]pyrazol-1-Yl]-3~{h}-Pyrido[3,4-D]pyrimidin-4-OneIC50900.0 [1]
8-[4-[2-(Dimethylamino)ethyl]pyrazol-1-yl]-3H-pyrido[3,4-d]pyrimidin-4-oneIC504100.0 [1]
8-[4-[2-[4-(4-Chlorophenyl)piperidin-1-Yl]ethyl]pyrazol-1-Yl]-3~{h}-Pyrido[3,4-D]pyrimidin-4-OneIC50138.0 [1]
8-[4-[2-[4-[(4-Chlorophenyl)methyl]piperidin-1-yl]ethyl]pyrazol-1-yl]-3H-pyrido[3,4-d]pyrimidin-4-oneIC50126.0 [1]
8-Pyrazol-1-yl-3H-pyrido[3,4-d]pyrimidin-4-oneIC5016700.0 [1]
8-[4-[2-[4-(3,5-Dichlorophenyl)piperidin-1-yl]ethyl]pyrazol-1-yl]-3H-pyrido[3,4-d]pyrimidin-4-oneIC5080.0 [1]
8-[[(Phenylmethyl)amino]methyl]-1~{h}-Pyrido[3,4-D]pyrimidin-4-OneIC5015600.0 [1]
8-[4-(2-Hydroxyethyl)pyrazol-1-yl]-3H-pyrido[3,4-d]pyrimidin-4-oneIC5021800.0 [1]
2-[1-(Cyclohexylmethyl)pyrazol-4-yl]oxy-3H-pyrido[3,4-d]pyrimidin-4-oneIC50630.96 [1]
2-(1-Cyclopentylpyrazol-4-yl)oxy-3H-pyrido[3,4-d]pyrimidin-4-oneIC50794.33 [1]
2-(6-Propan-2-ylpyridin-3-yl)oxy-3H-pyrido[3,4-d]pyrimidin-4-oneIC501584.89 [1]
2-(4-Chloro-3-hydroxyphenoxy)-3H-pyrido[3,4-d]pyrimidin-4-oneIC50398.11 [1]
2-(1-Benzylpyrazol-4-yl)oxy-3H-pyrido[2,3-d]pyrimidin-4-oneIC50100000.0 [1]
8-(1H-Pyrazol-5-yl)-3H-pyrido[3,4-d]pyrimidin-4-oneIC506900.0 [1]
8-[4-(2-Pyrrolidin-1-ylethyl)pyrazol-1-yl]-3H-pyrido[3,4-d]pyrimidin-4-oneIC501400.0 [1]
8-[4-(2-Piperidin-1-ylethyl)pyrazol-1-yl]-3H-pyrido[3,4-d]pyrimidin-4-oneIC501800.0 [1]
8-[4-[2-[(3,4-Dichlorophenyl)methyl-methylamino]ethyl]pyrazol-1-yl]-3H-pyrido[3,4-d]pyrimidin-4-oneIC50390.0 [1]
Items per page: 1 - 10 of 100
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References

This online tool may be cited as follows

MLA

"Quest Database™ Lysine-specific demethylase 4A Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 22 Feb. 2025, https://www.aatbio.com/data-sets/lysine-specific-demethylase-4a-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2025, February 22). Quest Database™ Lysine-specific demethylase 4A Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/lysine-specific-demethylase-4a-inhibitors-ic50-ki.
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