 | N-Oxalylglycine | IC50 | 1995.26 [1], 569000.0 [2] |
 | Pyridine-2,4-dicarboxylic acid | IC50 | 3300.0 [1], 7943.28 [2] |
 | 8-Hydroxy-5-quinolinecarboxylic acid | IC50 | 158.49 [1], 170.0 [2] |
 | Tranylcypromine hydrochloride | IC50 | 100000.0 [1] |
 | 3-[[2-Pyridin-2-Yl-6-(1,2,4,5-Tetrahydro-3-Benzazepin-3-Yl)pyrimidin-4-Yl]amino]propanoic Acid | IC50 | 39810.72 [1] |
 | 2-{5-[(4-Chloro-2-Methylphenyl)methoxy]-1h-Pyrazol-1-Yl}pyridine-4-Carboxylic Acid | IC50 | 2300.0 [1] |
 | 3-[[(1R)-6-(N-Methylanilino)-1,2,3,4-tetrahydronaphthalen-1-yl]methylamino]pyridine-4-carboxylic acid | IC50 | 4000.0 [1] |
 | Pyrido[3,4-d]pyrimidin-4(3H)-one | IC50 | 26200.0 [1] |
 | 2,2'-Bipyridine-4-carboxylic acid | IC50 | 1258.93 [1] |
 | 2-[1-[(3R)-1-Benzoylpiperidin-3-yl]triazol-4-yl]pyridine-4-carboxylic acid | IC50 | 100000.0 [1] |
 | 3-[5-[Butyl(methyl)amino]pentanoyl-hydroxyamino]propanoic acid | IC50 | 100000.0 [1] |
 | 3-[Hydroxy-[5-[methyl(pentyl)amino]pentanoyl]amino]propanoic acid | IC50 | 100000.0 [1] |
 | 3-[5-[Hexyl(methyl)amino]pentanoyl-hydroxyamino]propanoic acid | IC50 | 100000.0 [1] |
 | 3-[5-[Butyl(hexyl)amino]pentanoyl-hydroxyamino]propanoic acid | IC50 | 100000.0 [1] |
 | 3-[5-[Butyl(octyl)amino]pentanoyl-hydroxyamino]propanoic acid | IC50 | 100000.0 [1] |
 | 2-[1-(2-Phenylethyl)triazol-4-yl]pyridine-4-carboxylic acid | IC50 | 3162.28 [1] |
 | 2-[1-(2-Phenoxyethyl)triazol-4-yl]pyridine-4-carboxylic acid | IC50 | 10000.0 [1] |
 | 2-[1-(1-Ethoxycarbonylpiperidin-4-yl)triazol-4-yl]pyridine-4-carboxylic acid | IC50 | 19952.62 [1] |
 | 2-[1-(1-Propanoylpiperidin-4-yl)triazol-4-yl]pyridine-4-carboxylic acid | IC50 | 50118.72 [1] |
 | 2-[1-(1-Butanoylpiperidin-4-yl)triazol-4-yl]pyridine-4-carboxylic acid | IC50 | 100000.0 [1] |
 | 2-[1-(1-Benzoylpiperidin-4-yl)triazol-4-yl]pyridine-4-carboxylic acid | IC50 | 100000.0 [1] |
 | 2-[1-[1-(2-Phenylacetyl)piperidin-4-yl]triazol-4-yl]pyridine-4-carboxylic acid | IC50 | 31622.78 [1] |
 | 2-[1-[1-(3-Phenylpropanoyl)piperidin-4-yl]triazol-4-yl]pyridine-4-carboxylic acid | IC50 | 100000.0 [1] |
 | 2-[1-(1-Acetylazetidin-3-yl)triazol-4-yl]pyridine-4-carboxylic acid | IC50 | 50118.72 [1] |
 | 2-[1-(1-Propanoylazetidin-3-yl)triazol-4-yl]pyridine-4-carboxylic acid | IC50 | 100000.0 [1] |
 | 2-[1-(1-Butanoylazetidin-3-yl)triazol-4-yl]pyridine-4-carboxylic acid | IC50 | 100000.0 [1] |
 | 2-[1-(1-Benzoylazetidin-3-yl)triazol-4-yl]pyridine-4-carboxylic acid | IC50 | 31622.78 [1] |
 | 2-[1-[1-(2-Phenylacetyl)azetidin-3-yl]triazol-4-yl]pyridine-4-carboxylic acid | IC50 | 100000.0 [1] |
 | 2-[1-[1-(3-Phenylpropanoyl)azetidin-3-yl]triazol-4-yl]pyridine-4-carboxylic acid | IC50 | 100000.0 [1] |
 | 2-[1-(1-Butanoylpyrrolidin-3-yl)triazol-4-yl]pyridine-4-carboxylic acid | IC50 | 100000.0 [1] |
 | 2-[1-[1-(2-Phenylacetyl)pyrrolidin-3-yl]triazol-4-yl]pyridine-4-carboxylic acid | IC50 | 63095.73 [1] |
 | 2-[1-[1-(3-Phenylpropanoyl)pyrrolidin-3-yl]triazol-4-yl]pyridine-4-carboxylic acid | IC50 | 100000.0 [1] |
 | 2-[1-(1-Acetylpiperidin-3-yl)triazol-4-yl]pyridine-4-carboxylic acid | IC50 | 39810.72 [1] |
 | 2-[1-(1-Propanoylpiperidin-3-yl)triazol-4-yl]pyridine-4-carboxylic acid | IC50 | 63095.73 [1] |
 | 2-[1-(1-Butanoylpiperidin-3-yl)triazol-4-yl]pyridine-4-carboxylic acid | IC50 | 31622.78 [1] |
 | 2-[1-(1-Benzoylpiperidin-3-yl)triazol-4-yl]pyridine-4-carboxylic acid | IC50 | 50118.72 [1] |
 | 2-[1-[1-(2-Phenylacetyl)piperidin-3-yl]triazol-4-yl]pyridine-4-carboxylic acid | IC50 | 25118.86 [1] |
 | 2-[1-[1-(3-Phenylpropanoyl)piperidin-3-yl]triazol-4-yl]pyridine-4-carboxylic acid | IC50 | 50118.72 [1] |
 | 5-Chloro-7-[benzoylamino(3-methyl-2-thienyl)methyl]-8-quinolinol | IC50 | 191000.0 [1] |
 | Octyl 8-hydroxyquinoline-5-carboxylate | IC50 | 100000.0 [1] |
 | 2-[5-(2-Methoxyethanoylamino)-2-Oxidanyl-Phenyl]pyridine-4-Carboxylic Acid | IC50 | 11000.0 [1] |
 | 2-[5-[(5-Methyl-1,2-oxazol-3-yl)carbonylamino]-2-oxidanyl-phenyl]pyridine-4-carboxylic acid | IC50 | 5700.0 [1] |
 | 2-(5-Acetamido-2-Oxidanyl-Phenyl)pyridine-4-Carboxylic Acid | IC50 | 33000.0 [1] |
 | 2-[5-[(4-Hydroxyphenyl)carbonylamino]-2-Oxidanyl-Phenyl]pyridine-4-Carboxylic Acid | IC50 | 2300.0 [1] |
 | 2-[5-[2-(3-Methoxyphenyl)ethanoylamino]-2-Oxidanyl-Phenyl]pyridine-4-Carboxylic Acid | IC50 | 9000.0 [1] |
 | 8-[4-[2-[(4-Fluorophenyl)methyl-Methyl-Amino]ethyl]pyrazol-1-Yl]-3~{h}-Pyrido[3,4-D]pyrimidin-4-One | IC50 | 13900.0 [1] |
 | 8-[4-[2-[4-[(4-Chlorophenyl)methyl]piperidin-1-yl]ethyl]pyrazol-1-yl]-3H-pyrido[3,4-d]pyrimidin-4-one | IC50 | 4800.0 [1] |
 | 8-[4-[2-[4-(3,5-Dichlorophenyl)piperidin-1-yl]ethyl]pyrazol-1-yl]-3H-pyrido[3,4-d]pyrimidin-4-one | IC50 | 6100.0 [1] |
 | 8-[4-[2-[4-(3-Chlorophenyl)piperidin-1-yl]ethyl]pyrazol-1-yl]-3~{H}-pyrido[3,4-d]pyrimidin-4-one | IC50 | 5300.0 [1] |
 | 8-[4-[2-(4-Thiophen-2-ylpiperidin-1-yl)ethyl]pyrazol-1-yl]-3H-pyrido[3,4-d]pyrimidin-4-one | IC50 | 8300.0 [1] |
 | 4'-(Methoxycarbonyl)-[2,2'-bipyridine]-4-carboxylic acid | IC50 | 1100.0 [1] |
 | N-[[2-[[[2-[2-(Dimethylamino)ethyl-ethylamino]-2-oxoethyl]amino]methyl]pyridin-4-yl]methyl]-2,2,2-trifluoroacetamide | IC50 | 2500.0 [1] |
 | 2-[[4-(Diethylamino)butylamino]methyl]pyridine-4-carbaldehyde | IC50 | 2500.0 [1] |
 | 2-Hydrazinylpyrimidine-4-carboxylic acid | IC50 | 43000.0 [1] |
 | 2-(2h-1,2,3-Triazol-4-Yl)pyridine-4-Carboxylic Acid | IC50 | 19952.62 [1] |
 | 2-(2-Azanyl-1,3-Thiazol-4-Yl)pyridine-4-Carboxylic Acid | IC50 | 57.0 [1] |
 | 2-(1-Methyltriazol-4-yl)pyridine-4-carboxylic acid | IC50 | 25118.86 [1] |
 | 2-(1-Ethyltriazol-4-yl)pyridine-4-carboxylic acid | IC50 | 7943.28 [1] |
 | 2-[1-(3-Methylphenyl)triazol-4-yl]pyridine-4-carboxylic acid | IC50 | 7943.28 [1] |
 | 2-(1-Benzyltriazol-4-yl)pyridine-4-carboxylic acid | IC50 | 12589.25 [1] |
 | N-[4-[(1S,2R)-2-Aminocyclopropyl]phenyl]-8-hydroxyquinoline-5-carboxamide | IC50 | 31000.0 [1] |
 | 2-[4-[[4-[(1S,2R)-2-Aminocyclopropyl]phenyl]carbamoyl]pyridin-2-yl]pyridine-4-carboxylic acid | IC50 | 140.0 [1] |
 | N-[4-[4-[(1R,2S)-2-Aminocyclopropyl]anilino]-4-oxobutyl]-8-hydroxyquinoline-5-carboxamide | IC50 | 12000.0 [1] |
 | Methyl 2-[4-[[4-[(1S,2R)-2-aminocyclopropyl]phenyl]carbamoyl]pyridin-2-yl]pyridine-4-carboxylate | IC50 | 37000.0 [1] |
 | N-[6-[4-[(1R,2S)-2-Aminocyclopropyl]anilino]-6-oxohexyl]-8-hydroxyquinoline-5-carboxamide | IC50 | 9100.0 [1] |
 | N-[5-[4-[(1R,2S)-2-Aminocyclopropyl]anilino]-5-oxopentyl]-8-hydroxyquinoline-5-carboxamide | IC50 | 9700.0 [1] |