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Lymphocyte differentiation antigen CD38 Inhibitors (IC50, Ki)

Structure
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Compound Name
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Standard Type
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Standard Values (in nM)
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▼
2-Methyl-4-(2-fluoro-6-trifluoromethylbenzylamino)quinoline-8-carboxamideIC50510.0 [1]
1-Methyl-4-(oxan-4-ylamino)-6-(1,3-thiazol-5-yl)quinolin-2-oneIC5089.0 [1]
1-Methyl-4-(oxan-4-ylamino)-6-(1,3-thiazol-5-yl)quinolin-2-oneKi14.0 [1]
CD38 inhibitor 1IC507.3 [1]
CD38 inhibitor 1Ki0.3 [1]
4-[[4-(2-Methoxyethoxy)cyclohexyl]amino]-1,8-dimethyl-6-(1,3-thiazol-5-yl)quinolin-2-oneIC5010.0 [1]
4-[[4-(2-Methoxyethoxy)cyclohexyl]amino]-1,8-dimethyl-6-(1,3-thiazol-5-yl)quinolin-2-oneKi0.7 [1]
4-[(4-Methoxycyclohexyl)amino]-1,8-dimethyl-6-(1,3-thiazol-5-yl)quinolin-2-oneIC5015.0 [1]
4-[(4-Methoxycyclohexyl)amino]-1,8-dimethyl-6-(1,3-thiazol-5-yl)quinolin-2-oneKi0.45 [1]
4-[[6-(1,3-Thiazol-5-yl)quinazolin-4-yl]amino]cyclohexane-1-carboxylic acidIC50498.0 [1], 30200.0 [2]
1-[4-[[6-(1,3-Thiazol-5-yl)quinazolin-4-yl]amino]cyclohexyl]pyrrolidin-2-oneIC501960.0 [1], 8540.0 [2]
QuercetinIC5037900.0 [1]
ResveratrolIC50100000.0 [1]
LuteolinIC508200.0 [1]
MyricetinIC5024800.0 [1]
CyanidinIC5021800.0 [1]
3,3',4',5,5',7-HexahydroxyflavyliumIC5014600.0 [1]
PiceatannolIC50100000.0 [1]
Cyanidin 3-O-glucosideIC506300.0 [1]
FisetinidinIC5070300.0 [1]
DihydroquercetinIC50100000.0 [1]
MalvidinIC5017000.0 [1]
PelargonidinIC5016300.0 [1]
6-Chloro-2,3,4,9-tetrahydro-1H-carbazole-1-carboxamideIC50100000.0 [1]
PeonidinIC5020900.0 [1]
PetunidinIC5039200.0 [1]
L-EpicatechinIC50100000.0 [1]
QuercetagetinIC5048600.0 [1]
RobinetinIC5037900.0 [1]
6-Methyl-2,3,4,9-tetrahydro-1H-carbazole-1-carboxamideIC50100000.0 [1]
2-Chloro-5,6,7,8,9,10-hexahydrocyclohepta[b]indole-6-carboxamideIC50100000.0 [1]
2,3,4,9-Tetrahydro-1H-carbazole-1-carboxamideIC50100000.0 [1]
DiosmetinidinIC5032100.0 [1]
6-HydroxycyanidinIC5014200.0 [1]
(2R,3R,4S,5R,13R,14S,15R,16R)-3,4,8,10,14,15-Hexahydroxy-8,10-dioxo-7,9,11,25,26-pentaoxa-1,17,19,22-tetraza-8lambda5,10lambda5-diphosphapentacyclo[18.3.1.12,5.113,16.017,21]hexacosa-18,20,22-trien-24-oneIC50276000.0 [1]
4-(3-Chloro-4-fluoroanilino)-6-(1,3-thiazol-5-yl)quinoline-3-carboxamideIC501210.0 [1]
(2R,3R,4S,5R)-17-Bromo-3,4,8,10-tetrahydroxy-8,10-dioxo-7,9,11,24-tetraoxa-1,16,18,21-tetraza-8lambda5,10lambda5-diphosphatetracyclo[17.3.1.12,5.016,20]tetracosa-17,19,21-trien-23-oneIC5027000.0 [1]
(2R,3R,4S,5R)-17-Azido-3,4,8,10-tetrahydroxy-8,10-dioxo-7,9,11,24-tetraoxa-1,16,18,21-tetraza-8lambda5,10lambda5-diphosphatetracyclo[17.3.1.12,5.016,20]tetracosa-17,19,21-trien-23-oneIC506400.0 [1]
(2R,3R,4S,5R)-3,4,8,10-Tetrahydroxy-8,10-dioxo-7,9,11,24-tetraoxa-1,16,18,21-tetraza-8lambda5,10lambda5-diphosphatetracyclo[17.3.1.12,5.016,20]tetracosa-17,19,21-trien-23-oneIC5033000.0 [1]
(2R,3R,4S,5R)-17-Amino-3,4,8,10-tetrahydroxy-8,10-dioxo-7,9,11,24-tetraoxa-1,16,18,21-tetraza-8lambda5,10lambda5-diphosphatetracyclo[17.3.1.12,5.016,20]tetracosa-17,19,21-trien-23-oneIC503300.0 [1]
(2R,3R,4S,5R,13R,14S,15R,16R)-18-Bromo-3,4,8,10,14,15-hexahydroxy-8,10-dioxo-7,9,11,25,26-pentaoxa-1,17,19,22-tetraza-8lambda5,10lambda5-diphosphapentacyclo[18.3.1.12,5.113,16.017,21]hexacosa-18,20,22-trien-24-oneIC50158000.0 [1]
4-[[1-Ethyl-2-oxo-6-(1,3-thiazol-5-yl)quinolin-4-yl]amino]-N-methylcyclohexane-1-carboxamideIC5058.0 [1]
4-(Oxan-4-ylamino)-6-(1,3-thiazol-5-yl)-1H-quinolin-2-oneIC5061.0 [1]
8-Methyl-4-(oxan-4-ylamino)-6-(1,3-thiazol-5-yl)-1H-quinolin-2-oneIC5055.0 [1]
1,8-Dimethyl-4-(oxan-4-ylamino)-6-(1,3-thiazol-5-yl)quinolin-2-oneIC5052.0 [1]
4-[[4-(2-Methoxyethoxy)cyclohexyl]amino]-6-(1,3-thiazol-5-yl)-1H-quinolin-2-oneIC506.0 [1]
4-[[4-(2-Methoxyethoxy)cyclohexyl]amino]-8-methyl-6-(1,3-thiazol-5-yl)-1H-quinolin-2-oneIC503.9 [1]
1-Ethyl-4-[[4-(2-methoxyethoxy)cyclohexyl]amino]-6-(1,3-thiazol-5-yl)quinolin-2-oneIC5054.0 [1]
4-[(4-Methoxycyclohexyl)amino]-8-methyl-6-(1,3-thiazol-5-yl)-1H-quinolin-2-oneIC503.8 [1]
4-[(4-Methoxycyclohexyl)amino]-1-methyl-6-(1,3-thiazol-5-yl)quinolin-2-oneIC5013.0 [1]
4-[(4-Hydroxycyclohexyl)amino]-1-methyl-6-(1,3-thiazol-5-yl)quinolin-2-oneIC5014.0 [1]
4-Amino-1-methyl-6-(1,3-thiazol-5-yl)quinolin-2-oneIC5010773.0 [1]
N-(4-Methylsulfonylcyclohexyl)-6-(1,3-thiazol-5-yl)quinazolin-4-amineIC50959.0 [1]
N-Ethyl-6-(1,3-thiazol-5-yl)quinazolin-4-amineIC5011400.0 [1]
N-Propan-2-yl-6-(1,3-thiazol-5-yl)quinazolin-4-amineIC503350.0 [1]
N-Tert-butyl-6-(1,3-thiazol-5-yl)quinazolin-4-amineIC502300.0 [1]
2-[[6-(1,3-Thiazol-5-yl)quinazolin-4-yl]amino]ethanolIC5023400.0 [1]
N-(2-Methoxyethyl)-6-(1,3-thiazol-5-yl)quinazolin-4-amineIC5030200.0 [1]
N-(3-Chloro-4-fluorophenyl)-8-methoxy-6-(1,3-thiazol-5-yl)quinazolin-4-amineIC504710.0 [1]
4-[[8-Methoxy-6-(1,3-thiazol-5-yl)quinazolin-4-yl]amino]benzamideIC501160.0 [1]
N-(3-Chloro-4-fluorophenyl)-6-(1,3-thiazol-5-yl)-8-(trifluoromethyl)quinazolin-4-amineIC501590.0 [1]
4-[[6-(1,3-Thiazol-5-yl)-8-(trifluoromethyl)quinazolin-4-yl]amino]benzamideIC50263.0 [1]
N-(3-Chloro-4-fluorophenyl)-8-methyl-6-(1,3-thiazol-5-yl)quinazolin-4-amineIC50206.0 [1]
4-(3-Chloro-4-fluoroanilino)-8-methyl-6-(1,3-thiazol-5-yl)-1H-quinazolin-2-oneIC5028.0 [1]
4-[(4-Methoxycyclohexyl)amino]-8-methyl-6-(1,3-thiazol-5-yl)-1H-quinazolin-2-oneIC5026.0 [1]
4-[[4-(2-Methoxyethoxy)cyclohexyl]amino]-1-methyl-6-(1,3-thiazol-5-yl)quinazolin-2-oneIC5064.0 [1]
4-[(4-Methoxycyclohexyl)amino]-1-methyl-6-(1,3-thiazol-5-yl)quinazolin-2-oneIC5053.0 [1]
N-Methyl-4-[[2-methyl-6-(1,3-thiazol-5-yl)-8-(trifluoromethyl)quinazolin-4-yl]amino]cyclohexane-1-carboxamideIC5042.0 [1]
N-Methyl-4-[[8-methyl-6-(1,3-thiazol-5-yl)-2-(trifluoromethyl)quinazolin-4-yl]amino]cyclohexane-1-carboxamideIC50245.0 [1]
4-[[2,8-Dimethyl-6-(1,3-thiazol-5-yl)quinazolin-4-yl]amino]-N-methylcyclohexane-1-carboxamideIC5050.0 [1]
N-Methyl-4-[[2-oxo-6-(1,3-thiazol-5-yl)-1H-quinolin-4-yl]amino]cyclohexane-1-carboxamideIC503.4 [1]
N-Methyl-4-[[8-methyl-2-oxo-6-(1,3-thiazol-5-yl)-1H-quinolin-4-yl]amino]cyclohexane-1-carboxamideIC501.4 [1]
N-Methyl-4-[[1-methyl-2-oxo-6-(1,3-thiazol-5-yl)quinolin-4-yl]amino]cyclohexane-1-carboxamideIC504.8 [1]
4-[[1,8-Dimethyl-2-oxo-6-(1,3-thiazol-5-yl)quinolin-4-yl]amino]-N-methylcyclohexane-1-carboxamideIC505.3 [1]
N-(3-Chloro-4-fluorophenyl)-6-(1,3-thiazol-5-yl)quinolin-4-amineIC50298.0 [1]
N-Phenyl-6-(1,3-thiazol-5-yl)quinazolin-4-amineIC50840.0 [1]
N-(3-Chloro-4-fluorophenyl)-6-(1,3-thiazol-5-yl)quinazolin-4-amineIC501200.0 [1]
N-(4-Chlorophenyl)-6-(1,3-thiazol-5-yl)quinazolin-4-amineIC501320.0 [1]
N-(3-Chlorophenyl)-6-(1,3-thiazol-5-yl)quinazolin-4-amineIC50700.0 [1]
N-(2-Chlorophenyl)-6-(1,3-thiazol-5-yl)quinazolin-4-amineIC503610.0 [1]
N-(4-Fluorophenyl)-6-(1,3-thiazol-5-yl)quinazolin-4-amineIC502330.0 [1]
N-(3-Fluorophenyl)-6-(1,3-thiazol-5-yl)quinazolin-4-amineIC50970.0 [1]
N-(2-Fluorophenyl)-6-(1,3-thiazol-5-yl)quinazolin-4-amineIC504680.0 [1]
N-(4-Methylphenyl)-6-(1,3-thiazol-5-yl)quinazolin-4-amineIC501230.0 [1]
N-(3-Methylphenyl)-6-(1,3-thiazol-5-yl)quinazolin-4-amineIC501160.0 [1]
N-(2-Methylphenyl)-6-(1,3-thiazol-5-yl)quinazolin-4-amineIC5012800.0 [1]
6-(1,3-Thiazol-5-yl)-N-[3-(trifluoromethyl)phenyl]quinazolin-4-amineIC502150.0 [1]
4-[[6-(1,3-Thiazol-5-yl)quinazolin-4-yl]amino]benzenesulfonamideIC50700.0 [1]
N-[4-[[6-(1,3-Thiazol-5-yl)quinazolin-4-yl]amino]phenyl]methanesulfonamideIC50970.0 [1]
N-(3-Methylsulfonylphenyl)-6-(1,3-thiazol-5-yl)quinazolin-4-amineIC502690.0 [1]
4-[[6-(1,3-Thiazol-5-yl)quinazolin-4-yl]amino]benzamideIC50560.0 [1]
N-[4-(1,3-Oxazol-5-yl)phenyl]-6-(1,3-thiazol-5-yl)quinazolin-4-amineIC50840.0 [1]
N-(4-Imidazol-1-ylphenyl)-6-(1,3-thiazol-5-yl)quinazolin-4-amineIC50460.0 [1]
1-[4-[[6-(1,3-Thiazol-5-yl)quinazolin-4-yl]amino]phenyl]pyrrolidin-2-oneIC501460.0 [1]
N-Pyridin-2-yl-6-(1,3-thiazol-5-yl)quinazolin-4-amineIC5012300.0 [1]
N-Pyridin-3-yl-6-(1,3-thiazol-5-yl)quinazolin-4-amineIC503940.0 [1]
N-Pyridin-4-yl-6-(1,3-thiazol-5-yl)quinazolin-4-amineIC50950.0 [1]
N-Cyclopropyl-6-(1,3-thiazol-5-yl)quinazolin-4-amineIC507830.0 [1]
N-Cyclobutyl-6-(1,3-thiazol-5-yl)quinazolin-4-amineIC501930.0 [1]
N-Cyclopentyl-6-(1,3-thiazol-5-yl)quinazolin-4-amineIC50281.0 [1]
Items per page: 1 - 10 of 100
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References

This online tool may be cited as follows

MLA

"Quest Database™ Lymphocyte differentiation antigen CD38 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 22 Nov. 2024, https://www.aatbio.com/data-sets/lymphocyte-differentiation-antigen-cd38-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, November 22). Quest Database™ Lymphocyte differentiation antigen CD38 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/lymphocyte-differentiation-antigen-cd38-inhibitors-ic50-ki.
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