 | N-[[4-Ethyl-5-[[5-(trifluoromethoxy)-1,3-benzoxazol-2-yl]methylsulfanyl]-1,2,4-triazol-3-yl]methyl]aniline | IC50 | 100.0 [1] |
 | 2-[4-(4-Fluorophenyl)piperazin-1-yl]-N-(1,3-thiazol-2-yl)acetamide | IC50 | 1000.0 [1] |
 | CID 71601847 | IC50 | 46.0 [1] |
 | 2-{[4-Allyl-5-(anilinomethyl)-4H-1,2,4-triazol-3-yl]sulfanyl}-N-(4-methoxyphenyl)acetamide | IC50 | 6600.0 [1] |
 | 2-(4-Phenylpiperazin-1-yl)-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)acetamide | IC50 | 280.0 [1] |
 | 2-[4-(4-Fluorophenyl)piperazin-1-yl]-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)acetamide | IC50 | 77.0 [1] |
 | N-(4,5-Dimethyl-1,3-thiazol-2-yl)-2-[4-(4-fluorophenyl)piperazin-1-yl]acetamide | IC50 | 430.0 [1] |
 | 2-[[5-(Anilinomethyl)-4-ethyl-1,2,4-triazol-3-yl]sulfanyl]-N-(6-propanoylpyridin-3-yl)acetamide | IC50 | 400.0 [1] |
 | 2-[[5-(Anilinomethyl)-4-ethyl-1,2,4-triazol-3-yl]sulfanyl]-N-methyl-N-(4-propanoylphenyl)acetamide | IC50 | 580.0 [1] |
 | 2-[[5-(Anilinomethyl)-4-ethyl-1,2,4-triazol-3-yl]sulfanyl]-N-ethyl-N-(4-propanoylphenyl)acetamide | IC50 | 1000.0 [1] |
 | Ethyl 1-[2-[[5-(anilinomethyl)-4-ethyl-1,2,4-triazol-3-yl]sulfanyl]acetyl]-3,4-dihydro-2H-quinoline-6-carboxylate | IC50 | 1000.0 [1] |
 | Ethyl 1-[2-[[5-(anilinomethyl)-4-ethyl-1,2,4-triazol-3-yl]sulfanyl]acetyl]-2,3-dihydroindole-5-carboxylate | IC50 | 1000.0 [1] |
 | Ethyl 4-[[2-[[5-(anilinomethyl)-4-ethyl-1,2,4-triazol-3-yl]sulfanyl]acetyl]amino]benzoate | IC50 | 330.0 [1] |
 | Ethyl 3-[[2-[[5-(anilinomethyl)-4-ethyl-1,2,4-triazol-3-yl]sulfanyl]acetyl]amino]benzoate | IC50 | 1000.0 [1] |
 | Methyl 4-[[2-[[5-(anilinomethyl)-4-ethyl-1,2,4-triazol-3-yl]sulfanyl]acetyl]amino]benzoate | IC50 | 540.0 [1] |
 | Tert-butyl 4-[[2-[[5-(anilinomethyl)-4-ethyl-1,2,4-triazol-3-yl]sulfanyl]acetyl]amino]benzoate | IC50 | 1000.0 [1] |
 | 4-[[2-[[5-(Anilinomethyl)-4-ethyl-1,2,4-triazol-3-yl]sulfanyl]acetyl]amino]benzoic acid | IC50 | 1000.0 [1] |
 | 4-[[2-[[5-(Anilinomethyl)-4-ethyl-1,2,4-triazol-3-yl]sulfanyl]acetyl]amino]-N-methylbenzamide | IC50 | 1000.0 [1] |
 | 4-[[2-[[5-(Anilinomethyl)-4-ethyl-1,2,4-triazol-3-yl]sulfanyl]acetyl]amino]-N,N-dimethylbenzamide | IC50 | 1000.0 [1] |
 | 4-[[2-[[5-(Anilinomethyl)-4-ethyl-1,2,4-triazol-3-yl]sulfanyl]acetyl]amino]-N-ethylbenzamide | IC50 | 1000.0 [1] |
 | 1-[2-[[5-(Anilinomethyl)-4-ethyl-1,2,4-triazol-3-yl]sulfanylmethyl]-1,3-benzoxazol-5-yl]propan-1-one | IC50 | 190.0 [1] |
 | Ethyl 2-[[5-(anilinomethyl)-4-ethyl-1,2,4-triazol-3-yl]sulfanylmethyl]-1,3-benzoxazole-5-carboxylate | IC50 | 680.0 [1] |
 | 1-[2-[[5-(Anilinomethyl)-4-ethyl-1,2,4-triazol-3-yl]sulfanylmethyl]-1,3-benzoxazol-6-yl]propan-1-one | IC50 | 900.0 [1] |
 | 1-[2-[[5-(Anilinomethyl)-4-ethyl-1,2,4-triazol-3-yl]sulfonylmethyl]-1,3-benzoxazol-5-yl]propan-1-one | IC50 | 1670.0 [1] |
 | 1-[2-[[5-(Anilinomethyl)-4-ethyl-1,2,4-triazol-3-yl]sulfanylmethyl]-1,3-benzoxazol-5-yl]propan-1-ol | IC50 | 1000.0 [1] |
 | (NZ)-N-[1-[2-[[5-(anilinomethyl)-4-ethyl-1,2,4-triazol-3-yl]sulfanylmethyl]-1,3-benzoxazol-5-yl]propylidene]hydroxylamine | IC50 | 260.0 [1] |
 | N-[[4-Ethyl-5-[[5-[(Z)-C-ethyl-N-methoxycarbonimidoyl]-1,3-benzoxazol-2-yl]methylsulfanyl]-1,2,4-triazol-3-yl]methyl]aniline | IC50 | 1000.0 [1] |
 | N-[[4-Ethyl-5-[[5-(trifluoromethyl)-1,3-benzoxazol-2-yl]methylsulfanyl]-1,2,4-triazol-3-yl]methyl]aniline | IC50 | 360.0 [1] |
 | 1-[2-[[5-(Anilinomethyl)-4-ethyl-1,2,4-triazol-3-yl]sulfanylmethyl]-1,3-benzoxazol-5-yl]-2-methylpropan-1-one | IC50 | 600.0 [1] |
 | N-(1,3-Benzothiazol-2-yl)-2-[4-(4-fluorophenyl)piperazin-1-yl]acetamide | IC50 | 490.0 [1] |
 | 2-[[5-(Anilinomethyl)-4-ethyl-1,2,4-triazol-3-yl]sulfanyl]-N-(4-methylsulfonylphenyl)acetamide | IC50 | 1000.0 [1] |
 | N-[[5-[(6-Chloro-1,3-benzoxazol-2-yl)methylsulfanyl]-4-ethyl-1,2,4-triazol-3-yl]methyl]aniline | IC50 | 1000.0 [1] |
 | N-[[4-Ethyl-5-[(5-ethyl-1,3-benzoxazol-2-yl)methylsulfanyl]-1,2,4-triazol-3-yl]methyl]aniline | IC50 | 1000.0 [1] |
 | N-[[4-Ethyl-5-[(5-methoxy-1,3-benzoxazol-2-yl)methylsulfanyl]-1,2,4-triazol-3-yl]methyl]aniline | IC50 | 1000.0 [1] |
 | 2-[[5-(Anilinomethyl)-4-ethyl-1,2,4-triazol-3-yl]sulfanyl]-N-(4-methoxyphenyl)acetamide | IC50 | 1000.0 [1] |
 | 2-[[5-(Anilinomethyl)-4-ethyl-1,2,4-triazol-3-yl]sulfanyl]-N-(4-chlorophenyl)acetamide | IC50 | 1000.0 [1] |
 | 2-[[5-(Anilinomethyl)-4-ethyl-1,2,4-triazol-3-yl]sulfanyl]-N-(4-propanoylphenyl)acetamide | IC50 | 400.0 [1] |
 | N-[[5-(1,3-Benzoxazol-2-ylmethylsulfanyl)-4-ethyl-1,2,4-triazol-3-yl]methyl]aniline | IC50 | 1000.0 [1] |
 | N-[[4-Ethyl-5-[(5-fluoro-1,3-benzoxazol-2-yl)methylsulfanyl]-1,2,4-triazol-3-yl]methyl]aniline | IC50 | 1000.0 [1] |
 | N-[[5-[(5-Chloro-1,3-benzoxazol-2-yl)methylsulfanyl]-4-ethyl-1,2,4-triazol-3-yl]methyl]aniline | IC50 | 1000.0 [1] |
 | 2-[[5-(Anilinomethyl)-4-ethyl-1,2,4-triazol-3-yl]sulfanyl]-N-phenylacetamide | IC50 | 1000.0 [1] |
 | N-(4-Acetylphenyl)-2-[[5-(anilinomethyl)-4-ethyl-1,2,4-triazol-3-yl]sulfanyl]acetamide | IC50 | 1000.0 [1] |
 | 2-[[5-(Anilinomethyl)-4-ethyl-1,2,4-triazol-3-yl]sulfanyl]-N-(4-benzoylphenyl)acetamide | IC50 | 1000.0 [1] |
 | N-[[4-Ethyl-5-[(5-methyl-1,3-benzoxazol-2-yl)methylsulfanyl]-1,2,4-triazol-3-yl]methyl]aniline | IC50 | 1000.0 [1] |
 | 2-[[5-(Anilinomethyl)-4-ethyl-1,2,4-triazol-3-yl]sulfanyl]-N-(4-cyanophenyl)acetamide | IC50 | 1000.0 [1] |
 | 2-[[5-(Anilinomethyl)-4-ethyl-1,2,4-triazol-3-yl]sulfanyl]-N-[4-(2-ethyltetrazol-5-yl)phenyl]acetamide | IC50 | 1000.0 [1] |
 | 2-[[5-(Anilinomethyl)-4-ethyl-1,2,4-triazol-3-yl]sulfanyl]-N-(4-butanoylphenyl)acetamide | IC50 | 230.0 [1] |
 | 2-[4-(4-Fluorophenyl)piperazin-1-yl]-N-(4,5,6,7-tetrahydro-1,3-benzoxazol-2-yl)acetamide | IC50 | 180.0 [1] |
 | N-(5,6-Dihydro-4H-cyclopenta[d][1,3]thiazol-2-yl)-2-[4-(4-fluorophenyl)piperazin-1-yl]acetamide | IC50 | 490.0 [1] |
 | 2-[4-(4-Fluorophenyl)piperazin-1-yl]-N-(5,6,7,8-tetrahydro-4H-cyclohepta[d][1,3]thiazol-2-yl)acetamide | IC50 | 120.0 [1] |
 | 2-[4-(4-Methylphenyl)piperazin-1-yl]-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)acetamide | IC50 | 250.0 [1] |
 | 2-[4-(3-Fluorophenyl)piperazin-1-yl]-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)acetamide | IC50 | 1000.0 [1] |
 | 2-(4-Benzoylpiperazin-1-yl)-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)acetamide | IC50 | 1000.0 [1] |
 | 2-(4-Cyclohexylpiperazin-1-yl)-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)acetamide | IC50 | 1000.0 [1] |
 | 2-(4-Pyridin-2-ylpiperazin-1-yl)-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)acetamide | IC50 | 200.0 [1] |
 | 2-(4-Pyridin-3-ylpiperazin-1-yl)-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)acetamide | IC50 | 1000.0 [1] |
 | 2-(4-Pyridin-4-ylpiperazin-1-yl)-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)acetamide | IC50 | 1000.0 [1] |
 | 2-(4-Pyrimidin-2-ylpiperazin-1-yl)-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)acetamide | IC50 | 1000.0 [1] |
 | N-(4,5,6,7-Tetrahydro-1,3-benzothiazol-2-yl)-2-[4-(1,3-thiazol-2-yl)piperazin-1-yl]acetamide | IC50 | 520.0 [1] |
 | 2-[4-(5-Fluoropyridin-2-yl)piperazin-1-yl]-N-(4,5,6,7-tetrahydro-1,3-benzoxazol-2-yl)acetamide | IC50 | 100.0 [1] |
 | 2-[4-(5-Fluoropyridin-2-yl)piperazin-1-yl]-N-methyl-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)acetamide | IC50 | 41.0 [1] |
 | N-Ethyl-2-[4-(5-fluoropyridin-2-yl)piperazin-1-yl]-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)acetamide | IC50 | 780.0 [1] |
 | 2-[4-(5-Fluoropyridin-2-yl)piperazin-1-yl]-1-(2-methylimidazo[1,2-a]pyridin-3-yl)ethanone | IC50 | 430.0 [1] |
 | 2-[4-(5-Fluoropyridin-2-yl)piperazin-1-yl]-1-imidazo[1,2-a]pyridin-3-ylethanone | IC50 | 130.0 [1] |
 | 2-[4-(5-Fluoropyridin-2-yl)piperazin-1-yl]-1-imidazo[1,5-a]pyridin-3-ylethanone | IC50 | 1000.0 [1] |
 | 2-[4-(5-Fluoropyridin-2-yl)piperazin-1-yl]-1-(1H-indazol-3-yl)ethanone | IC50 | 1000.0 [1] |
 | 2-[4-(5-Fluoropyridin-2-yl)piperazin-1-yl]-1-pyrazolo[1,5-a]pyridin-3-ylethanone | IC50 | 330.0 [1] |
 | 2-[4-(5-Fluoropyridin-2-yl)piperazin-1-yl]-1-(1H-indol-3-yl)ethanone | IC50 | 1000.0 [1] |
 | 1-(1-Benzofuran-3-yl)-2-[4-(5-fluoropyridin-2-yl)piperazin-1-yl]ethanone | IC50 | 470.0 [1] |
 | 2-[4-(5-Fluoropyridin-2-yl)piperazin-1-yl]-1-(2-methyl-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-3-yl)ethanone | IC50 | 190.0 [1] |
 | 2-[4-(5-Fluoropyridin-2-yl)piperazin-1-yl]-1-(5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-3-yl)ethanone | IC50 | 100.0 [1] |
 | 2-[4-(4-Fluorophenyl)piperazin-1-yl]-N-(5-methyl-4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)acetamide | IC50 | 26.0 [1] |
 | 1-(2-Methylimidazo[1,2-a]pyridine-3-yl)-2-(4-phenylpiperazino)ethanone | IC50 | 3000.0 [1] |
 | Ethyl 4-{[({5-[(benzylsulfanyl)methyl]-4-ethyl-4H-1,2,4-triazol-3-yl}sulfanyl)acetyl]amino}benzoate | IC50 | 7600.0 [1] |