L-type amino acid transporter 1 Inhibitors (IC50, Ki)

Structure ▲ ▼	Compound Name ▲ ▼	Standard Type ▲ ▼	Standard Values (in nM) ▲ ▼
	(S)-2-Amino-3-biphenyl-3-yl-propionic acid	IC50	6600.0 [1]
	(2S)-2-Amino-3-(3-benzylphenyl)propanoic acid	IC50	7300.0 [1]
	Tyrosine	IC50	68000.0 [1]
	Tryptophan	IC50	160000.0 [1]
	Leucine	IC50	85000.0 [1]
	Histidine	IC50	20000.0 [1]
	Phenylalanine	IC50	69000.0 [1]
	D-Tryptophan	IC50	380000.0 [1]
	Methionine	IC50	170000.0 [1]
	D-Methionine	IC50	120000.0 [1]
	Valine	IC50	68000.0 [1]
	l-Isoleucine	IC50	140000.0 [1]
	D-Leucine	IC50	220000.0 [1]
	1-Methyl-L-histidine	IC50	190000.0 [1]
	3-Hydroxy-L-phenylalanine	IC50	130000.0 [1]
	alpha-Methyl-L-phenylalanine	IC50	130000.0 [1]
	D-Phenylalanine	IC50	46000.0 [1]
	(S)-2-Amino-3-cyclohexylpropanoic acid	IC50	200000.0 [1]
	D-Histidine	IC50	460000.0 [1]
	D-Alloisoleucine	IC50	3000000.0 [1]
	D-Tyrosine	IC50	380000.0 [1]
	D-Valine	IC50	50000000.0 [1]
	3-(3-Pyridyl)-L-alanine	IC50	69000.0 [1]
	(S)-2-Amino-3-(1-benzyl-1H-imidazol-4-yl)propanoic acid	IC50	170000.0 [1]
	(R)-2-Amino-2-methyl-3-phenylpropanoic acid	IC50	810000.0 [1]
	m-Acetylphenylalanine	IC50	92000.0 [1]
	alpha-Benzyl-D-methionine	IC50	240000.0 [1]
	(S)-2-Amino-3-(3-(aminomethyl)phenyl)propanoic acid	IC50	470000.0 [1]
	4-(Methoxycarbonyl)-L-phenylalanine	IC50	260000.0 [1]
	(S)-2-Amino-3-(3-aminophenyl)propanoic acid	IC50	101000.0 [1]
	3-(4-Pyridyl)-L-alanine	IC50	100000.0 [1]
	(R)-2-Amino-3-cyclohexylpropanoic acid	IC50	260000.0 [1]
	(2S)-2-Amino-3-[3-(2-hydroxyethoxycarbonyl)phenyl]propanoic acid	IC50	29000.0 [1]
	3-[(2S)-2-Amino-2-carboxyethyl]-5-methylbenzoic acid	IC50	680000.0 [1]
	(2S)-2-Amino-3-[3-(2-methoxy-2-oxoethyl)phenyl]propanoic acid	IC50	76000.0 [1]
	(2S)-2-Amino-3-(3-methoxycarbonyl-5-methylphenyl)propanoic acid	IC50	95000.0 [1]
	(2R)-2-Amino-3-(3-methoxycarbonylphenyl)propanoic acid	IC50	150000.0 [1]
	(2S)-2-Amino-3-[3-(methylcarbamoyl)phenyl]propanoic acid	IC50	96000.0 [1]
	3-Methoxycarbonyl-L-phenylalanine	IC50	36000.0 [1]
	3-[(2S)-2-Amino-2-carboxyethyl]benzoic acid	IC50	130000.0 [1]
	3-(2-Pyridyl)-L-alanine	IC50	160000.0 [1]
	(2S)-2-Amino-3-(3-benzyl-4-hydroxyphenyl)propanoic acid	IC50	9100.0 [1]
	(2S)-2-Amino-3-[3-[(2-methylpropan-2-yl)oxycarbonyl]phenyl]propanoic acid	IC50	17000.0 [1]
	3-(Hydroxymethyl)-phenylalanine	IC50	83000.0 [1]
	(2S)-3-(3-Acetamidophenyl)-2-aminopropanoic acid	IC50	110000.0 [1]

Entire TableStructureCompound NameStandard TypeStandard Values (in nM)

Items per page: 510All1 - 10 of 45 ⟨⟩

---

---

References

This online tool may be cited as follows

MLA	"Quest Database™ L-type amino acid transporter 1 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 20 Feb. 2025, https://www.aatbio.com/data-sets/l-type-amino-acid-transporter-1-inhibitors-ic50-ki.
APA	AAT Bioquest, Inc. (2025, February 20). Quest Database™ L-type amino acid transporter 1 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/l-type-amino-acid-transporter-1-inhibitors-ic50-ki.
BibTeX	EndNote	RefMan