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Kallikrein 7 Inhibitors (IC50, Ki)

Structure
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Compound Name
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Standard Type
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Standard Values (in nM)
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4-[4-(4-Hydroxy-phenyl)-phthalazin-1-ylamino]-N-methyl-benzamideIC5066000.0 [1]
4-[4-(4-Hydroxy-phenyl)-phthalazin-1-ylamino]-N-methyl-benzamideKi50000.0 [1], 166000.0 [2]
3-[[2-[(6R)-6-[(5-Chloro-2-methoxyphenyl)methyl]-3-(2,2-dimethylhydrazinyl)-7-oxo-5,6-dihydro-2H-1,4-diazepin-1-yl]acetyl]amino]benzoic acid;hydrochlorideIC501900.0 [1]
8,8'-Paepalantine dimerIC50112400.0 [1]
8,8'-Paepalantine dimerKi12200.0 [1]
2-[(6-Amino-1H-benzimidazol-2-yl)sulfanylmethyl]-3-[3-(trifluoromethyl)phenyl]quinazolin-4-oneIC5025000.0 [1]
2-[(6-Amino-1H-benzimidazol-2-yl)sulfanylmethyl]-3-[3-(trifluoromethyl)phenyl]quinazolin-4-oneKi15000.0 [1], 44000.0 [2]
2-[4-[(Z)-2-Cyano-3-(3-ethoxyanilino)-3-oxoprop-1-enyl]-2-methoxyphenoxy]acetic acidIC50113000.0 [1]
2-[4-[(Z)-2-Cyano-3-(3-ethoxyanilino)-3-oxoprop-1-enyl]-2-methoxyphenoxy]acetic acidKi95000.0 [1], 140000.0 [2]
(Z)-2-Cyano-3-(4-hydroxy-3-methoxyphenyl)-N-(4-methoxyphenyl)prop-2-enamideIC5090000.0 [1]
(Z)-2-Cyano-3-(4-hydroxy-3-methoxyphenyl)-N-(4-methoxyphenyl)prop-2-enamideKi72000.0 [1], 164000.0 [2]
(5E)-5-[(3,4-Dimethoxyphenyl)methylidene]-3-[(5-fluoro-2-methylanilino)methyl]-1,3-thiazolidine-2,4-dioneIC50106000.0 [1]
(5E)-5-[(3,4-Dimethoxyphenyl)methylidene]-3-[(5-fluoro-2-methylanilino)methyl]-1,3-thiazolidine-2,4-dioneKi83000.0 [1], 166000.0 [2]
(Z)-2-(1H-Benzimidazol-2-yl)-3-[3-methoxy-4-(2-morpholin-4-yl-2-oxoethoxy)phenyl]prop-2-enenitrileIC5083000.0 [1]
(Z)-2-(1H-Benzimidazol-2-yl)-3-[3-methoxy-4-(2-morpholin-4-yl-2-oxoethoxy)phenyl]prop-2-enenitrileKi55000.0 [1], 131000.0 [2]
(2Z)-2-Cyano-3-(4-hydroxy-3-methoxyphenyl)-N-(4-hydroxyphenyl)prop-2-enamideIC50107000.0 [1]
(2Z)-2-Cyano-3-(4-hydroxy-3-methoxyphenyl)-N-(4-hydroxyphenyl)prop-2-enamideKi70000.0 [1], 129000.0 [2]
(Z)-2-Cyano-3-(3-ethoxy-4-hydroxyphenyl)-N-(4-hydroxyphenyl)prop-2-enamideIC5094000.0 [1]
(Z)-2-Cyano-3-(3-ethoxy-4-hydroxyphenyl)-N-(4-hydroxyphenyl)prop-2-enamideKi75000.0 [1], 152000.0 [2]
PaepalantineIC50165800.0 [1]
PaepalantineKi70700.0 [1]
VioxanthinIC50135300.0 [1]
VioxanthinKi37200.0 [1]
2-[(6R)-6-[(5-Chloro-2-methoxyphenyl)methyl]-3-(2,2-dimethylhydrazinyl)-7-oxo-5,6-dihydro-2H-1,4-diazepin-1-yl]-N-(3-methylsulfonylphenyl)acetamideIC50820.0 [1]
2-[(6R)-6-[(5-Chloro-2-methoxyphenyl)methyl]-3-(2,2-dimethylhydrazinyl)-7-oxo-5,6-dihydro-2H-1,4-diazepin-1-yl]-N-[3-(1-methylpyrazol-4-yl)phenyl]acetamideIC50520.0 [1]
(2S)-2-[(6R)-6-[(5-Chloro-2-methoxyphenyl)methyl]-3-(2,2-dimethylhydrazinyl)-7-oxo-5,6-dihydro-2H-1,4-diazepin-1-yl]-N-[3-(1-methylpyrazol-4-yl)phenyl]propanamideIC5058.0 [1]
(13S)-13-Benzyl-11-(2-methylphenyl)-2,8,10,12-tetrazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7,11-pentaen-14-oneIC5057000.0 [1]
(13S)-13-Benzyl-11-(2-methylphenyl)-2,8,10,12-tetrazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7,11-pentaen-14-oneKi50600.0 [1]
(13S)-13-Benzyl-11-(3,4-dimethoxyphenyl)-2,8,10,12-tetrazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7,11-pentaen-14-oneIC5033500.0 [1]
(13S)-13-Benzyl-11-(3,4-dimethoxyphenyl)-2,8,10,12-tetrazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7,11-pentaen-14-oneKi27000.0 [1]
N-[(Z)-3-[[(3S,3Ar,6R,6aS)-6-phenylmethoxy-2,3,3a,5,6,6a-hexahydrofuro[3,2-b]furan-3-yl]amino]-3-oxo-1-thiophen-2-ylprop-1-en-2-yl]benzamideIC5013300.0 [1]
N-[(Z)-3-[[(3S,3Ar,6R,6aS)-6-phenylmethoxy-2,3,3a,5,6,6a-hexahydrofuro[3,2-b]furan-3-yl]amino]-3-oxo-1-thiophen-2-ylprop-1-en-2-yl]benzamideKi1800.0 [1]
N-[(Z)-3-[[(3R,3Ar,6R,6aS)-6-phenylmethoxy-2,3,3a,5,6,6a-hexahydrofuro[3,2-b]furan-3-yl]amino]-1-(1,3-benzodioxol-5-yl)-3-oxoprop-1-en-2-yl]benzamideIC50205200.0 [1]
N-[(Z)-3-[[(3R,3Ar,6R,6aS)-6-phenylmethoxy-2,3,3a,5,6,6a-hexahydrofuro[3,2-b]furan-3-yl]amino]-1-(1,3-benzodioxol-5-yl)-3-oxoprop-1-en-2-yl]benzamideKi80300.0 [1]
N-[(Z)-3-[[(3R,3Ar,6R,6aS)-6-phenylmethoxy-2,3,3a,5,6,6a-hexahydrofuro[3,2-b]furan-3-yl]amino]-3-oxo-1-pyridin-3-ylprop-1-en-2-yl]benzamideIC50195800.0 [1]
N-[(Z)-3-[[(3R,3Ar,6R,6aS)-6-phenylmethoxy-2,3,3a,5,6,6a-hexahydrofuro[3,2-b]furan-3-yl]amino]-3-oxo-1-pyridin-3-ylprop-1-en-2-yl]benzamideKi75100.0 [1]
(Z)-N-[(3R,3Ar,6R,6aS)-6-phenylmethoxy-2,3,3a,5,6,6a-hexahydrofuro[3,2-b]furan-3-yl]-2-acetamido-3-thiophen-2-ylprop-2-enamideIC50160500.0 [1]
(Z)-N-[(3R,3Ar,6R,6aS)-6-phenylmethoxy-2,3,3a,5,6,6a-hexahydrofuro[3,2-b]furan-3-yl]-2-acetamido-3-thiophen-2-ylprop-2-enamideKi77400.0 [1]
Benzyl (2S)-2-[[(2S)-1-[[(3R,3aR,6R,6aR)-3-phenylmethoxy-2,3,3a,5,6,6a-hexahydrofuro[3,2-b]furan-6-yl]oxy]-1-oxo-3-phenylpropan-2-yl]carbamoyl]pyrrolidine-1-carboxylateIC5019600.0 [1]
Benzyl (2S)-2-[[(2S)-1-[[(3R,3aR,6R,6aR)-3-phenylmethoxy-2,3,3a,5,6,6a-hexahydrofuro[3,2-b]furan-6-yl]oxy]-1-oxo-3-phenylpropan-2-yl]carbamoyl]pyrrolidine-1-carboxylateKi2800.0 [1]
Tert-butyl N-[(2S)-1-[[(3S,3aR,6R,6aS)-6-phenylmethoxy-2,3,3a,5,6,6a-hexahydrofuro[3,2-b]furan-3-yl]amino]-3-[1-(4-methylphenyl)sulfonylimidazol-4-yl]-1-oxopropan-2-yl]carbamateIC5027800.0 [1]
Tert-butyl N-[(2S)-1-[[(3S,3aR,6R,6aS)-6-phenylmethoxy-2,3,3a,5,6,6a-hexahydrofuro[3,2-b]furan-3-yl]amino]-3-[1-(4-methylphenyl)sulfonylimidazol-4-yl]-1-oxopropan-2-yl]carbamateKi4400.0 [1]
Benzyl N-[(5S)-6-[[(3S,3aR,6R,6aS)-6-phenylmethoxy-2,3,3a,5,6,6a-hexahydrofuro[3,2-b]furan-3-yl]amino]-5-[(2-methylpropan-2-yl)oxycarbonylamino]-6-oxohexyl]carbamateIC5023600.0 [1]
Benzyl N-[(5S)-6-[[(3S,3aR,6R,6aS)-6-phenylmethoxy-2,3,3a,5,6,6a-hexahydrofuro[3,2-b]furan-3-yl]amino]-5-[(2-methylpropan-2-yl)oxycarbonylamino]-6-oxohexyl]carbamateKi2900.0 [1]
2-O-[(3R,3Ar,6R,6aR)-3-phenylmethoxy-2,3,3a,5,6,6a-hexahydrofuro[3,2-b]furan-6-yl] 1-O-tert-butyl (2S)-pyrrolidine-1,2-dicarboxylateIC5024400.0 [1]
2-O-[(3R,3Ar,6R,6aR)-3-phenylmethoxy-2,3,3a,5,6,6a-hexahydrofuro[3,2-b]furan-6-yl] 1-O-tert-butyl (2S)-pyrrolidine-1,2-dicarboxylateKi15600.0 [1]
Tert-butyl N-[(2R)-1-[[(3S,3aR,6R,6aS)-6-phenylmethoxy-2,3,3a,5,6,6a-hexahydrofuro[3,2-b]furan-3-yl]amino]-5-[bis(phenylmethoxycarbonylamino)methylideneamino]-1-oxopentan-2-yl]carbamateIC5016900.0 [1]
Tert-butyl N-[(2R)-1-[[(3S,3aR,6R,6aS)-6-phenylmethoxy-2,3,3a,5,6,6a-hexahydrofuro[3,2-b]furan-3-yl]amino]-5-[bis(phenylmethoxycarbonylamino)methylideneamino]-1-oxopentan-2-yl]carbamateKi2400.0 [1]
[(3R,3Ar,6R,6aR)-3-phenylmethoxy-2,3,3a,5,6,6a-hexahydrofuro[3,2-b]furan-6-yl] (2R)-2-[(2-methylpropan-2-yl)oxycarbonylamino]-3-phenylmethoxypropanoateIC5016000.0 [1]
[(3R,3Ar,6R,6aR)-3-phenylmethoxy-2,3,3a,5,6,6a-hexahydrofuro[3,2-b]furan-6-yl] (2R)-2-[(2-methylpropan-2-yl)oxycarbonylamino]-3-phenylmethoxypropanoateKi2300.0 [1]
[(3R,3Ar,6R,6aR)-3-phenylmethoxy-2,3,3a,5,6,6a-hexahydrofuro[3,2-b]furan-6-yl] (2S)-2-[(2-methylpropan-2-yl)oxycarbonylamino]-4-methylsulfanylbutanoateIC5028700.0 [1]
[(3R,3Ar,6R,6aR)-3-phenylmethoxy-2,3,3a,5,6,6a-hexahydrofuro[3,2-b]furan-6-yl] (2S)-2-[(2-methylpropan-2-yl)oxycarbonylamino]-4-methylsulfanylbutanoateKi18400.0 [1]
[(3R,3Ar,6R,6aR)-3-phenylmethoxy-2,3,3a,5,6,6a-hexahydrofuro[3,2-b]furan-6-yl] (2S)-2-[(2-methylpropan-2-yl)oxycarbonylamino]-6-(phenylmethoxycarbonylamino)hexanoateIC5013700.0 [1]
[(3R,3Ar,6R,6aR)-3-phenylmethoxy-2,3,3a,5,6,6a-hexahydrofuro[3,2-b]furan-6-yl] (2S)-2-[(2-methylpropan-2-yl)oxycarbonylamino]-6-(phenylmethoxycarbonylamino)hexanoateKi1400.0 [1]
Benzyl (2R)-2-[[(3S,3aR,6R,6aS)-6-phenylmethoxy-2,3,3a,5,6,6a-hexahydrofuro[3,2-b]furan-3-yl]carbamoyl]pyrrolidine-1-carboxylateIC5023600.0 [1]
Benzyl (2R)-2-[[(3S,3aR,6R,6aS)-6-phenylmethoxy-2,3,3a,5,6,6a-hexahydrofuro[3,2-b]furan-3-yl]carbamoyl]pyrrolidine-1-carboxylateKi15100.0 [1]
Benzyl N-[(2S)-1-[[(2R)-1-[[(3S,3aR,6R,6aS)-6-phenylmethoxy-2,3,3a,5,6,6a-hexahydrofuro[3,2-b]furan-3-yl]amino]-1-oxo-3-phenylpropan-2-yl]amino]-3-methyl-1-oxobutan-2-yl]carbamateIC5056600.0 [1]
Benzyl N-[(2S)-1-[[(2R)-1-[[(3S,3aR,6R,6aS)-6-phenylmethoxy-2,3,3a,5,6,6a-hexahydrofuro[3,2-b]furan-3-yl]amino]-1-oxo-3-phenylpropan-2-yl]amino]-3-methyl-1-oxobutan-2-yl]carbamateKi3800.0 [1]
2-O-[(3R,3Ar,6R,6aR)-3-phenylmethoxy-2,3,3a,5,6,6a-hexahydrofuro[3,2-b]furan-6-yl] 1-O-benzyl (2R)-pyrrolidine-1,2-dicarboxylateIC5016600.0 [1]
2-O-[(3R,3Ar,6R,6aR)-3-phenylmethoxy-2,3,3a,5,6,6a-hexahydrofuro[3,2-b]furan-6-yl] 1-O-benzyl (2R)-pyrrolidine-1,2-dicarboxylateKi1900.0 [1]
1-O-[(3R,3Ar,6R,6aR)-3-phenylmethoxy-2,3,3a,5,6,6a-hexahydrofuro[3,2-b]furan-6-yl] 4-O-benzyl (2S)-2-[(2-methylpropan-2-yl)oxycarbonylamino]butanedioateIC5010200.0 [1]
1-O-[(3R,3Ar,6R,6aR)-3-phenylmethoxy-2,3,3a,5,6,6a-hexahydrofuro[3,2-b]furan-6-yl] 4-O-benzyl (2S)-2-[(2-methylpropan-2-yl)oxycarbonylamino]butanedioateKi1300.0 [1]
Gabexate mesylateIC5020400.0 [1]
(5-Amino-3-pyridin-3-yl-1,2,4-triazol-1-yl)-(4-methylphenyl)methanoneIC5040.0 [1]
(3-Amino-[1,2,4]triazol-4-yl)-(4-methoxy-phenyl)-methanoneIC50610.0 [1]
1-(4-Chlorobenzoyl)-3-pyridin-3-yl-1H-1,2,4-triazol-5-amineIC50220.0 [1]
1-Benzoyl-3-(4-chlorophenyl)-5-(methylthio)-1H-1,2,4-triazoleIC50660.0 [1]
1-(3,4-Dimethoxybenzoyl)-3-phenyl-1H-1,2,4-triazol-5-amineIC50230.0 [1]
Methyl (S)-2-((2-((3-(trifluoromethoxy)phenyl)carbamoyl)pyrrolidine-1-carboxamido)-methyl)benzoateIC509000.0 [1]
2-[(1R,4S,7S,13S,19S,22S,25S,28S,31R,34S,40S,43S,49S)-49-(2-Amino-2-oxoethyl)-4,19-bis[(2S)-butan-2-yl]-25-[3-(diaminomethylideneamino)propyl]-28,34-bis[(1R)-1-hydroxyethyl]-22-(hydroxymethyl)-3,6,12,18,21,24,27,30,33,36,39,42,48,51-tetradecaoxo-53,54-dithia-2,5,11,17,20,23,26,29,32,35,38,41,47,50-tetradecazapentacyclo[29.20.4.07,11.013,17.043,47]pentapentacontan-40-yl]acetamideKi16.8 [1]
CID 38335241IC5073000.0 [1]
8-[(2R,3S)-5,7-Dihydroxy-2-(4-hydroxyphenyl)-4-oxo-2,3-dihydrochromen-3-yl]-2-(3,4-dihydroxyphenyl)-5,7-dihydroxy-2,3-dihydrochromen-4-oneIC5015000.0 [1]
(13S)-13-Benzyl-11-(4-methylphenyl)-2,8,10,12-tetrazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7,11-pentaen-14-oneIC5068000.0 [1]
(13S)-13-Benzyl-11-(4-methoxyphenyl)-2,8,10,12-tetrazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7,11-pentaen-14-oneIC5072000.0 [1]
N-[(Z)-3-[[(3R,3Ar,6R,6aS)-6-phenylmethoxy-2,3,3a,5,6,6a-hexahydrofuro[3,2-b]furan-3-yl]amino]-3-oxo-1-thiophen-2-ylprop-1-en-2-yl]benzamideKi1800.0 [1]
(13R)-13-Benzyl-11-(2-methylphenyl)-2,8,10,12-tetrazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7,11-pentaen-14-oneIC5095900.0 [1]
(13S)-13-Benzyl-11-(2,4-dimethylphenyl)-2,8,10,12-tetrazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7,11-pentaen-14-oneIC5083900.0 [1]
(13S)-13-Benzyl-11-(2,5-dimethoxyphenyl)-2,8,10,12-tetrazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7,11-pentaen-14-oneIC5080900.0 [1]
(13S)-13-Benzyl-11-(3,4,5-trimethoxyphenyl)-2,8,10,12-tetrazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7,11-pentaen-14-oneIC5055700.0 [1]
(13S)-13-Benzyl-11-(3-hydroxyphenyl)-2,8,10,12-tetrazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7,11-pentaen-14-oneIC50124800.0 [1]
N-[(2S)-1-(2-Aminoimidazo[1,2-a]pyridin-3-yl)-1-oxo-3-phenylpropan-2-yl]-2-methylbenzamideIC50135400.0 [1]
N-[(2S)-1-(2-Aminoimidazo[1,2-a]pyridin-3-yl)-1-oxo-3-phenylpropan-2-yl]-2-phenylacetamideIC50149200.0 [1]
2-[(1R,4S,7S,13S,19S,22S,25S,28S,31R,34S,40S,43S,49S)-19,49-Bis(2-amino-2-oxoethyl)-4-[(2S)-butan-2-yl]-25-[3-(diaminomethylideneamino)propyl]-28,34-bis[(1R)-1-hydroxyethyl]-22-(hydroxymethyl)-3,6,12,18,21,24,27,30,33,36,39,42,48,51-tetradecaoxo-53,54-dithia-2,5,11,17,20,23,26,29,32,35,38,41,47,50-tetradecazapentacyclo[29.20.4.07,11.013,17.043,47]pentapentacontan-40-yl]acetamideKi0.8 [1]
2-[[(3S,3Ar,6S,6aR)-6-[[1-(cyclohexylamino)-2-methyl-1-oxopropan-2-yl]-[2-(4-hydroxyphenyl)acetyl]amino]-2,3,3a,5,6,6a-hexahydrofuro[3,2-b]furan-3-yl]-[2-(4-hydroxyphenyl)acetyl]amino]-N-cyclohexyl-2-methylpropanamideIC50133000.0 [1]
N-[(3S,3Ar,6R,6aS)-6-phenylmethoxy-2,3,3a,5,6,6a-hexahydrofuro[3,2-b]furan-3-yl]-N-[1-(cyclohexylamino)-2-methyl-1-oxopropan-2-yl]benzamideIC50572000.0 [1]
2-[[(3S,3Ar,6R,6aS)-6-phenylmethoxy-2,3,3a,5,6,6a-hexahydrofuro[3,2-b]furan-3-yl]-[2-(4-fluorophenyl)acetyl]amino]-N-cyclohexyl-2-methylpropanamideIC50185000.0 [1]
2-[[(3S,3Ar,6R,6aS)-6-phenylmethoxy-2,3,3a,5,6,6a-hexahydrofuro[3,2-b]furan-3-yl]-[2-(4-hydroxyphenyl)acetyl]amino]-N-cyclohexyl-2-methylpropanamideIC50249000.0 [1]
2-[[(3S,3Ar,6R,6aS)-6-phenylmethoxy-2,3,3a,5,6,6a-hexahydrofuro[3,2-b]furan-3-yl]-[2-(4-methoxyphenyl)acetyl]amino]-N-cyclohexyl-2-methylpropanamideIC50272000.0 [1]
[2-[(3,5-Dimethyl-1-phenylpyrazol-4-yl)amino]-2-oxoethyl] 2-(6-carbamimidoyl-2-methyl-1H-indol-3-yl)acetateIC50500.0 [1]
(3S)-7-Methoxy-3-methyl-8-[(3S)-5,9,10-trihydroxy-7-methoxy-3-methyl-1-oxo-3,4-dihydrobenzo[g]isochromen-8-yl]-3,4-dihydrobenzo[g]isochromene-1,5,6,9,10-pentoneKi12200.0 [1]
2-[(1R,4S,7S,13S,19S,22S,25S,31R,34S,40S,43S,49S)-25,49-Dibenzyl-4,19-bis[(2S)-butan-2-yl]-28-butyl-34-[(1R)-1-hydroxyethyl]-22-(hydroxymethyl)-3,6,12,18,21,24,27,30,33,36,39,42,48,51-tetradecaoxo-53,54-dithia-2,5,11,17,20,23,26,29,32,35,38,41,47,50-tetradecazapentacyclo[29.20.4.07,11.013,17.043,47]pentapentacontan-40-yl]acetamideKi69.0 [1]
2-[(1R,4S,7S,13S,19S,22S,25S,31R,34S,40S,43S,49S)-40-(2-Amino-2-oxoethyl)-25,49-dibenzyl-4-[(2S)-butan-2-yl]-28-butyl-34-[(1R)-1-hydroxyethyl]-22-(hydroxymethyl)-3,6,12,18,21,24,27,30,33,36,39,42,48,51-tetradecaoxo-53,54-dithia-2,5,11,17,20,23,26,29,32,35,38,41,47,50-tetradecazapentacyclo[29.20.4.07,11.013,17.043,47]pentapentacontan-19-yl]acetic acidKi130.0 [1]
2-[(1R,4S,7S,13S,19S,22S,25S,31R,34S,40S,43S,49S)-40-(2-Amino-2-oxoethyl)-49-benzyl-4-[(2S)-butan-2-yl]-28-butyl-25-[[4-(diaminomethylideneamino)phenyl]methyl]-34-[(1R)-1-hydroxyethyl]-22-(hydroxymethyl)-3,6,12,18,21,24,27,30,33,36,39,42,48,51-tetradecaoxo-53,54-dithia-2,5,11,17,20,23,26,29,32,35,38,41,47,50-tetradecazapentacyclo[29.20.4.07,11.013,17.043,47]pentapentacontan-19-yl]acetic acidKi740.0 [1]
Methyl (2S)-1-[(2R)-2-[[(2S)-2-[[(2S)-2-[[2-[[(2S)-1-[(2R,3S)-2-hydroxy-3-methylpentanoyl]pyrrolidine-2-carbonyl]amino]acetyl]-methylamino]-4-methylpentanoyl]amino]propanoyl]-methylamino]-3-phenylpropanoyl]pyrrolidine-2-carboxylateIC5022100.0 [1]
Methyl (2S)-1-[(2R)-2-[methyl-[(2S)-2-[[(2S)-4-methyl-2-[methyl-[2-[[(2S)-1-[(2R,3S)-3-methyl-2-[(E)-3-phenylprop-2-enoyl]oxypentanoyl]pyrrolidine-2-carbonyl]amino]acetyl]amino]pentanoyl]amino]propanoyl]amino]-3-phenylpropanoyl]pyrrolidine-2-carboxylateIC5018900.0 [1]
2-[6-[(2-Chloro-6-cyanophenyl)methyl]-3-(2,2-dimethylhydrazinyl)-7-oxo-5,6-dihydro-2H-1,4-diazepin-1-yl]-N-[3-(1-methylpyrazol-4-yl)phenyl]acetamideIC5011000.0 [1]
2-[6-[(2-Chloro-6-fluorophenyl)methyl]-3-(2,2-dimethylhydrazinyl)-7-oxo-5,6-dihydro-2H-1,4-diazepin-1-yl]-N-[3-(1-methylpyrazol-4-yl)phenyl]acetamideIC50940.0 [1]
2-[3-(2,2-Dimethylhydrazinyl)-6-[(2-fluoro-6-methoxyphenyl)methyl]-7-oxo-5,6-dihydro-2H-1,4-diazepin-1-yl]-N-[3-(1-methylpyrazol-4-yl)phenyl]acetamideIC506800.0 [1]
2-[3-(2,2-Dimethylhydrazinyl)-6-[[2-fluoro-6-(trifluoromethyl)phenyl]methyl]-7-oxo-5,6-dihydro-2H-1,4-diazepin-1-yl]-N-[3-(1-methylpyrazol-4-yl)phenyl]acetamideIC502700.0 [1]
2-[6-[(2-Chloro-6-methylphenyl)methyl]-3-(2,2-dimethylhydrazinyl)-7-oxo-5,6-dihydro-2H-1,4-diazepin-1-yl]-N-[3-(1-methylpyrazol-4-yl)phenyl]acetamideIC501500.0 [1]
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References

This online tool may be cited as follows

MLA

"Quest Database™ Kallikrein 7 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 21 Feb. 2025, https://www.aatbio.com/data-sets/kallikrein-7-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2025, February 21). Quest Database™ Kallikrein 7 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/kallikrein-7-inhibitors-ic50-ki.
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