| Levamisole | IC50 | 5000.0 [1], 20210.0 [2], 200000.0 [3], 400000.0 [4] |
| Phenylalanine | IC50 | 5000.0 [1], 80200.0 [2], 100000.0 [3] |
| 6-(1-Benzothiophen-2-yl)-5,6-dihydroimidazo[2,1-b][1,3]thiazole;hydrochloride | IC50 | 400000.0 [1] |
| 2-(5,6-Dihydroimidazo[2,1-b][1,3]thiazol-6-yl)-1-benzothiophen-5-amine;hydrochloride | IC50 | 400000.0 [1] |
| 6-(1-Benzothiophen-2-yl)-2,3,5,6-tetrahydroimidazo[2,1-b][1,3]thiazole;hydrochloride | IC50 | 400000.0 [1] |
| 6-(5-Nitro-1-benzothiophen-2-yl)-5,6-dihydroimidazo[2,1-b][1,3]thiazole | IC50 | 400000.0 [1] |
| Tryptophan | IC50 | 5000.0 [1] |
| Leucine | IC50 | 5000.0 [1] |
| Theophylline | IC50 | 5000.0 [1] |
| L-Homoarginine | IC50 | 5000.0 [1] |
| (S)-2-Amino-4-methylpentanamide | IC50 | 5000.0 [1] |
| 2,5-Dimethoxy-N-(3-quinolinyl)benzenesulfonamide | IC50 | 100000.0 [1] |
| 1-(3,4-Dihydroxyphenyl)-2-(1-imidazolyl)ethanone | IC50 | 30200.0 [1] |
| 1-(3,4-Dihydroxyphenyl)-2-[(4,6-dimethyl-2-pyrimidinyl)thio]ethanone | IC50 | 49500.0 [1] |
| CID 24790981 | IC50 | 100000.0 [1] |
| 3-Pyridinecarboxamide, 5-[[(5-chloro-2-methoxyphenyl)sulfonyl]amino]- | IC50 | 80000.0 [1] |
| N-(2,5-Dimethylphenyl)-2-[(2-oxo-3H-1,3-benzoxazol-6-yl)sulfonylamino]acetamide | IC50 | 27600.0 [1] |
| (3-Chloro-4-methyl-2-oxochromen-7-yl) 4-chloro-3-nitrobenzenesulfonate | IC50 | 4060.0 [1] |
| (3-Chloro-4-methyl-2-oxochromen-7-yl) ethanesulfonate | IC50 | 4180.0 [1] |
| (3-Cyano-4-methyl-2-oxochromen-7-yl) 4-nitrobenzenesulfonate | IC50 | 1110.0 [1] |
| (3-Cyano-4-methyl-2-oxochromen-7-yl) ethanesulfonate | IC50 | 4060.0 [1] |
| (3-Cyano-4-methyl-2-oxochromen-7-yl) butane-1-sulfonate | IC50 | 6290.0 [1] |
| (3-Cyano-4-methyl-2-oxochromen-7-yl) 4-chlorobenzenesulfonate | IC50 | 7030.0 [1] |
| (3-Chloro-4-methyl-2-oxochromen-7-yl) methanesulfonate | IC50 | 3580.0 [1] |
| (4-Methyl-8-nitro-2-oxochromen-7-yl) 4-chloro-3-nitrobenzenesulfonate | IC50 | 4650.0 [1] |
| (3-Cyano-4-methyl-2-oxochromen-7-yl) 3-nitrobenzenesulfonate | IC50 | 5160.0 [1] |
| [8-(2,5-Dichlorophenyl)sulfonyloxy-4-methyl-2-oxochromen-7-yl] 2,5-dichlorobenzenesulfonate | IC50 | 3210.0 [1] |
| (3-Cyano-4-methyl-2-oxochromen-7-yl) octane-1-sulfonate | IC50 | 2810.0 [1] |
| (3-Chloro-4-methyl-2-oxochromen-7-yl) butane-1-sulfonate | IC50 | 3220.0 [1] |
| (3-Cyano-4-methyl-2-oxochromen-7-yl) 4-propylbenzenesulfonate | IC50 | 4630.0 [1] |
| (3-Cyano-4-methyl-2-oxochromen-7-yl) 2,5-dichlorobenzenesulfonate | IC50 | 2260.0 [1] |
| (4-Methyl-8-nitro-2-oxochromen-7-yl) 4-octylbenzenesulfonate | IC50 | 3060.0 [1] |
| [4-Methyl-8-(4-nitrophenyl)sulfonyloxy-2-oxochromen-7-yl] 4-nitrobenzenesulfonate | IC50 | 4570.0 [1] |
| (8-Ethylsulfonyloxy-4-methyl-2-oxochromen-7-yl) ethanesulfonate | IC50 | 2870.0 [1] |
| (3-Chloro-4-methyl-2-oxochromen-7-yl) 2-nitrobenzenesulfonate | IC50 | 5490.0 [1] |
| (4-Methyl-8-octylsulfonyloxy-2-oxochromen-7-yl) octane-1-sulfonate | IC50 | 10300.0 [1] |
| [8-(4-Chlorophenyl)sulfonyloxy-4-methyl-2-oxochromen-7-yl] 4-chlorobenzenesulfonate | IC50 | 20600.0 [1] |
| (4-Methyl-2-oxochromen-7-yl) 4-chloro-3-nitrobenzenesulfonate | IC50 | 2720.0 [1] |
| (3-Cyano-4-methyl-2-oxochromen-7-yl) 4-methoxybenzenesulfonate | IC50 | 3590.0 [1] |
| (4-Methyl-2-oxochromen-7-yl) 2,4,5-trichlorobenzenesulfonate | IC50 | 1330.0 [1] |
| (3-Chloro-4-methyl-2-oxochromen-7-yl) 4-methoxybenzenesulfonate | IC50 | 2130.0 [1] |
| (3-Chloro-4-methyl-2-oxochromen-7-yl) octane-1-sulfonate | IC50 | 3120.0 [1] |
| (3-Chloro-4-methyl-2-oxochromen-7-yl) 4-chlorobenzenesulfonate | IC50 | 13100.0 [1] |
| [4-Methyl-2-oxo-8-(4-propylphenyl)sulfonyloxychromen-7-yl] 4-propylbenzenesulfonate | IC50 | 5950.0 [1] |
| 2-(3,4-Dimethylphenyl)-7-(trifluoromethyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one | IC50 | 1750.0 [1] |
| (3Z)-3-[(2-Methylphenyl)methylidene]-1,1-dioxo-1lambda6,2-benzothiazin-4-one | IC50 | 3750.0 [1] |
| 2-(Prop-2-enylamino)-7-(trifluoromethyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one | IC50 | 890.0 [1] |
| 2-(Butylamino)-7-(trifluoromethyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one | IC50 | 710.0 [1] |
| (3Z)-3-[(3-Fluorophenyl)methylidene]-1,1-dioxo-1lambda6,2-benzothiazin-4-one | IC50 | 9930.0 [1] |
| 2-[Amino(methyl)amino]-7-(trifluoromethyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one | IC50 | 2220.0 [1] |
| (3Z)-3-[(4-Chlorophenyl)methylidene]-1,1-dioxo-1lambda6,2-benzothiazin-4-one | IC50 | 4350.0 [1] |
| 2-(3-Fluorophenyl)-7-(trifluoromethyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one | IC50 | 740.0 [1] |
| 2-(3-Nitrophenyl)-7-(trifluoromethyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one | IC50 | 480.0 [1] |
| (3Z)-3-[(2-Bromophenyl)methylidene]-1,1-dioxo-1lambda6,2-benzothiazin-4-one | IC50 | 7430.0 [1] |
| (3Z)-3-[(4-Bromophenyl)methylidene]-1,1-dioxo-1lambda6,2-benzothiazin-4-one | IC50 | 3690.0 [1] |
| (3Z)-3-[(2,6-Difluorophenyl)methylidene]-1,1-dioxo-1lambda6,2-benzothiazin-4-one | IC50 | 10600.0 [1] |
| 2-(Pentylamino)-7-(trifluoromethyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one | IC50 | 760.0 [1] |
| 2-(2-Methoxyphenyl)-7-(trifluoromethyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one | IC50 | 100000.0 [1] |
| 2-(2-Fluorophenyl)-7-(trifluoromethyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one | IC50 | 100000.0 [1] |
| 2-(4-Ethoxyphenyl)-7-(trifluoromethyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one | IC50 | 790.0 [1] |
| 2-(Propylamino)-7-(trifluoromethyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one | IC50 | 310.0 [1] |
| 2-(4-Methylphenyl)-7-(trifluoromethyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one | IC50 | 360.0 [1] |
| 2-(4-Aminoanilino)-7-(trifluoromethyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one | IC50 | 710.0 [1] |
| 2-(4-Methoxyphenyl)-7-(trifluoromethyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one | IC50 | 480.0 [1] |
| 2-(4-Ethylphenyl)-7-(trifluoromethyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one | IC50 | 4550.0 [1] |
| (3Z)-3-[(3-Methoxyphenyl)methylidene]-1,1-dioxo-1lambda6,2-benzothiazin-4-one | IC50 | 1040.0 [1] |
| 2-(4-Propan-2-ylanilino)-7-(trifluoromethyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one | IC50 | 31500.0 [1] |
| (3Z)-3-[(3-Bromophenyl)methylidene]-1,1-dioxo-1lambda6,2-benzothiazin-4-one | IC50 | 2550.0 [1] |
| 2-Phenyl-7-(trifluoromethyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one | IC50 | 430.0 [1] |
| 2-(2-Ethoxyphenyl)-7-(trifluoromethyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one | IC50 | 100000.0 [1] |
| 2-(3-Phenylphenyl)-7-(trifluoromethyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one | IC50 | 1670.0 [1] |
| 2-[2-(Dimethylamino)ethylamino]-7-(trifluoromethyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one | IC50 | 3750.0 [1] |
| 2-[4-(Trifluoromethoxy)phenyl]-7-(trifluoromethyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one | IC50 | 240.0 [1] |
| (3Z)-3-[(2,4-Dichlorophenyl)methylidene]-1,1-dioxo-1lambda6,2-benzothiazin-4-one | IC50 | 4960.0 [1] |
| 2-(Dibutylamino)-7-(trifluoromethyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one | IC50 | 4630.0 [1] |
| 2-(3-Methoxyanilino)-7-(trifluoromethyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one | IC50 | 440.0 [1] |
| (3Z)-3-[(4-Fluorophenyl)methylidene]-1,1-dioxo-1lambda6,2-benzothiazin-4-one | IC50 | 3060.0 [1] |
| 3-[5-Oxo-7-(trifluoromethyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-2-yl]benzonitrile | IC50 | 1120.0 [1] |
| 2-(3,5-Dimethoxyphenyl)-7-(trifluoromethyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one | IC50 | 760.0 [1] |
| 2-(3,5-Dimethylphenyl)-7-(trifluoromethyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one | IC50 | 460.0 [1] |
| 2-(4-Ethoxyanilino)-7-(trifluoromethyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one | IC50 | 2020.0 [1] |
| 7-(Trifluoromethyl)-2-[3-(trifluoromethyl)phenyl]-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one | IC50 | 680.0 [1] |
| (3Z)-3-(3-Chlorobenzylidene)-2,3-dihydro-4H-1,2-benzothiazin-4-one 1,1-dioxide | IC50 | 3770.0 [1] |
| (3Z)-3-(3-Hydroxybenzylidene)-2,3-dihydro-4H-1,2-benzothiazin-4-one 1,1-dioxide | IC50 | 1210.0 [1] |
| (3Z)-3-(2-Methoxybenzylidene)-2,3-dihydro-4H-1,2-benzothiazin-4-one 1,1-dioxide | IC50 | 1240.0 [1] |
| (3-Chloro-4-methyl-2-oxochromen-7-yl) benzenesulfonate | IC50 | 5520.0 [1] |
| 1-(3,4-Dihydroxyphenyl)-2-(2-ethyl-1-imidazolyl)ethanone | IC50 | 100000.0 [1] |
| 1-(3,4-Dihydroxyphenyl)-2-(2-methyl-1-imidazolyl)ethanone | IC50 | 64600.0 [1] |
| 2-(Benzimidazol-1-yl)-1-(3,4-dihydroxyphenyl)ethanone | IC50 | 14800.0 [1] |
| 1-(3,4-Dihydroxyphenyl)-2-(2-methyl-1-benzimidazolyl)ethanone | IC50 | 100000.0 [1] |
| 1-(3,4-Dihydroxyphenyl)-2-(4-methyl-1-pyrazolyl)ethanone | IC50 | 53300.0 [1] |
| (4-Methyl-2-oxochromen-7-yl) 2-methyl-5-nitrobenzenesulfonate | IC50 | 3910.0 [1] |
| (3Z)-3-Benzylidene-1,1-dioxo-1lambda6,2-benzothiazin-4-one | IC50 | 1780.0 [1] |
| (3Z)-3-[(4-Methoxyphenyl)methylidene]-1,1-dioxo-1lambda6,2-benzothiazin-4-one | IC50 | 1530.0 [1] |